Page last updated: 2024-09-02

opc 21268 and l 368899

opc 21268 has been researched along with l 368899 in 3 studies

Compound Research Comparison

Studies
(opc 21268)
Trials
(opc 21268)
Recent Studies (post-2010)
(opc 21268)
Studies
(l 368899)
Trials
(l 368899)
Recent Studies (post-2010) (l 368899)
1333646030
13336604

Protein Interaction Comparison

ProteinTaxonomyopc 21268 (IC50)l 368899 (IC50)
Vasopressin V1a receptorRattus norvegicus (Norway rat)0.37
Oxytocin receptorRattus norvegicus (Norway rat)0.0089
Vasopressin V2 receptor Rattus norvegicus (Norway rat)0.57

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Honda, K; Ikeda, K; Onaka, T; Yamashita, T1
Harrell, CM; Jasper, JR; O'Brien, JA; Pettibone, DJ1
Borthwick, AD1

Other Studies

3 other study(ies) available for opc 21268 and l 368899

ArticleYear
Facilitative role of endogenous oxytocin in noradrenaline release in the rat supraoptic nucleus.
    The European journal of neuroscience, 2003, Volume: 18, Issue:11

    Topics: Analysis of Variance; Animals; Antidiuretic Hormone Receptor Antagonists; Brain Chemistry; Camphanes; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; Electroshock; Fear; Male; Microdialysis; Norepinephrine; Oxytocin; Piperazines; Piperidines; Potassium; Quinolones; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Oxytocin; Stimulation, Chemical; Supraoptic Nucleus; Synaptosomes

2003
Characterization of the human oxytocin receptor stably expressed in 293 human embryonic kidney cells.
    Life sciences, 1995, Volume: 57, Issue:24

    Topics: Arginine Vasopressin; Cell Line; Drug Tolerance; Embryo, Mammalian; Female; Gene Expression; Guanine Nucleotides; Humans; Hydrolysis; Kidney; Myometrium; Oxytocin; Phosphatidylinositols; Receptors, Oxytocin; Recombinant Proteins; Transfection; Tritium

1995
Oral oxytocin antagonists.
    Journal of medicinal chemistry, 2010, Sep-23, Volume: 53, Issue:18

    Topics: Administration, Oral; Animals; Biological Availability; Camphor; Humans; Indoles; Oxytocin; Piperazines; Piperidines; Protein Conformation; Pyrrolidines; Receptors, Oxytocin; Sulfonamides; Triazoles

2010