ondansetron has been researched along with zacopride in 33 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (9.09) | 18.7374 |
1990's | 28 (84.85) | 18.2507 |
2000's | 2 (6.06) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Airey, JE; Campbell, HF; Darkes, P; Fitzpatrick, LR; Klein, S; Neuenschwander, K; Pendley, CE; Powers, M; Schnapper, M; Youssefyeh, RD | 1 |
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD | 1 |
Bradley, G; Coleman, J; Rhodes, KF; Taylor, A; Ward, TJ; White, JC | 1 |
McLean, S; Nagel, AA; Rizzi, JP; Rosen, T; Seeger, T | 1 |
Bryce, D; Chalabi, PM; Furman, J; Guarino, KJ; Ives, JL; McLean, S; Nagel, AA; Rosen, T; Roth, RW; Seeger, TF | 1 |
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT | 1 |
McDonough, JR; McLean, DB; Mele, PC; O'Halloran, KP | 1 |
Fink-Jensen, A; Hansen, JB; Honoré, T; Jacobsen, P; Judge, ME; Olney, J; Turski, L | 1 |
Barnes, NM; Cheng, CH; Costall, B; Ge, J; Kelly, ME; Naylor, RJ | 1 |
Barnes, NM; Cheng, CH; Costall, B; Ge, J; Naylor, RJ | 1 |
Adrien, J; Franc, B; Haj-Dahmane, S; Hamon, M; Jolas, T; Lanfumey, L; Tissier, MH | 1 |
Gozlan, H; Martin, P; Puech, AJ | 1 |
Andrews, PL; Bhandari, P | 1 |
Chen, JP; Gardner, EL; van Praag, HM | 1 |
Middlefell, VC; Price, TL | 1 |
Gandara, DR; Hesketh, PJ | 1 |
Coffman, WJ; Cohen, ML; Wilson, H | 1 |
Bloomquist, W; Cohen, ML; Gidda, JS; Lacefield, W | 1 |
Barnes, JM; Barnes, NM; Costall, B; Naylor, RJ; Tyers, MB | 1 |
File, SE; Johnston, AL | 1 |
Cheng, CH; Costall, B; Ge, J; Naylor, RJ | 1 |
Anthony, EW; Nevins, ME | 1 |
Daniels, S; Eglen, RM; Fontana, DJ; Khabbaz, M; Kilfoil, T; Lee, CH; Wong, EH | 1 |
Gozlan, H; Hamon, M; Kidd, FJ; Levy, JC; Nielsen, M | 1 |
Barnes, JM; Barnes, NM | 1 |
Barrett, JE; Critchett, D; Hu, W; Sokol, PT; Solomon, AJ; Toral, J; Ziai, MR | 1 |
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M | 1 |
Dahl, SG; Junien, JL; Langlois, A; Pascaud, X; Rivière, PJ | 1 |
Callera, JC; Hamon, M; Laguzzi, R; Machado, BH; Sévoz, C | 1 |
Alcalde, AI; Rodríguez-Yoldi, MC; Rodríguez-Yoldi, MJ; Salvador, MT | 1 |
Saederup, E; Squires, RF | 1 |
Allan, AM; Girasa, KA; McKenzie-Quirk, SD; Miczek, KA | 1 |
Dukat, M; Wesołowska, A | 1 |
33 other study(ies) available for ondansetron and zacopride
Article | Year |
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Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.
Topics: Animals; Antiemetics; Benzamides; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Male; Metoclopramide; Molecular Structure; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting | 1992 |
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction | 1992 |
Novel antagonists of the 5-HT3 receptor. Synthesis and structure-activity relationships of (2-alkoxybenzoyl)ureas.
Topics: Animals; Benzoates; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Rats; Rats, Inbred Strains; Serotonin Antagonists; Structure-Activity Relationship; Urea; Vagus Nerve; X-Ray Diffraction | 1992 |
An initial three-component pharmacophore for specific serotonin-3 receptor ligands.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Computer Graphics; Computer Simulation; Imidazoles; In Vitro Techniques; Indoles; Ligands; Mice; Models, Molecular; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Thiazoles; Tropisetron | 1990 |
Synthesis, in vitro binding profile, and central nervous system penetrability of the highly potent 5-HT3 receptor antagonist [3H]-4-(2-methoxyphenyl)-2-[4(5)-methyl-5(4)-imidazolylmethyl]thiazole.
Topics: Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry; Glioma; Imidazoles; Mice; Molecular Structure; Neuroblastoma; Serotonin Antagonists; Thiazoles; Tumor Cells, Cultured | 1990 |
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes | 1990 |
Cisplatin-induced conditioned taste aversion: attenuation by dexamethasone but not zacopride or GR38032F.
Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cisplatin; Dexamethasone; Dose-Response Relationship, Drug; Lithium; Lithium Chloride; Male; Ondansetron; Rats; Rats, Inbred Strains; Serotonin Antagonists; Taste Disorders | 1992 |
Inhibition of cisplatin-induced emesis in ferrets by the non-NMDA receptor antagonists NBQX and CNQX.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Exploratory Behavior; Ferrets; Imidazoles; Male; Ondansetron; Quinoxalines; Receptors, Amino Acid; Receptors, Cell Surface; Serotonin Antagonists; Vomiting | 1992 |
Profiles of interaction of R(+)/S(-)-zacopride and anxiolytic agents in a mouse model.
Topics: Animals; Anti-Anxiety Agents; Antiemetics; Behavior, Animal; Benzamides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlordiazepoxide; Fenclonine; Granisetron; Indazoles; Male; Mice; Neurotransmitter Agents; Ondansetron; Receptors, Cholecystokinin; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereoisomerism | 1992 |
Differential modulation of extracellular levels of 5-hydroxytryptamine in the rat frontal cortex by (R)- and (S)-zacopride.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Buspirone; Diazepam; Dose-Response Relationship, Drug; Frontal Lobe; Hydroxyindoleacetic Acid; Male; Ondansetron; Rats; Serotonin; Serotonin Antagonists; Stereoisomerism | 1992 |
Central action of 5-HT3 receptor ligands in the regulation of sleep-wakefulness and raphe neuronal activity in the rat.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electrophysiology; Indoles; Male; Neurons; Ondansetron; Propranolol; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Sleep; Time Factors; Tropanes; Tropisetron; Wakefulness | 1992 |
5-HT3 receptor antagonists reverse helpless behaviour in rats.
Topics: Analysis of Variance; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Depression; Disease Models, Animal; Helplessness, Learned; Imidazoles; Indoles; Male; Ondansetron; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tropisetron | 1992 |
Preliminary evidence for the involvement of the putative 5-HT4 receptor in zacopride- and copper sulphate-induced vomiting in the ferret.
Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Copper; Copper Sulfate; Female; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Loperamide; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting | 1991 |
Activation of 5-HT3 receptor by 1-phenylbiguanide increases dopamine release in the rat nucleus accumbens.
Topics: 3,4-Dihydroxyphenylacetic Acid; 5,7-Dihydroxytryptamine; Animals; Benzamides; Biguanides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Denervation; Dopamine; Homovanillic Acid; Hydroxyindoleacetic Acid; Hypoglycemic Agents; Imidazoles; In Vitro Techniques; Male; Nucleus Accumbens; Ondansetron; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1991 |
5-HT3 receptor agonism may be responsible for the emetic effects of zacopride in the ferret.
Topics: Anesthesia; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Emetics; Female; Ferrets; Imidazoles; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism | 1991 |
Serotonin antagonists: a new class of antiemetic agents.
Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting | 1991 |
5-Hydroxytryptamine3 receptors mediate tachycardia in conscious instrumented dogs.
Topics: Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Ergolines; Heart Rate; Hexamethonium; Hexamethonium Compounds; Imidazoles; Indoles; Male; Ondansetron; Receptors, Serotonin; Serotonin; Tropisetron | 1990 |
Comparison of the 5-HT3 receptor antagonist properties of ICS 205-930, GR38032F and zacopride.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbachol; Cisplatin; Guinea Pigs; Heart Rate; Imidazoles; In Vitro Techniques; Indoles; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting | 1989 |
5-HT3 receptors mediate inhibition of acetylcholine release in cortical tissue.
Topics: Acetylcholine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Female; Imidazoles; Metoclopramide; Ondansetron; Potassium; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1989 |
Lack of effects of 5HT3 receptor antagonists in the social interaction and elevated plus-maze tests of anxiety in the rat.
Topics: Animals; Anxiety; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlordiazepoxide; Granisetron; Imidazoles; Indazoles; Male; Motor Activity; Ondansetron; Rats; Serotonin Antagonists; Social Behavior | 1989 |
The profiles of interaction of yohimbine with anxiolytic and putative anxiolytic agents to modify 5-HT release in the frontal cortex of freely-moving rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Clonidine; Dialysis; Diazepam; Drug Interactions; Extracellular Space; Frontal Lobe; Hydroxyindoleacetic Acid; Male; Ondansetron; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Yohimbine | 1993 |
Antagonists at the serotonin-3 receptor can reduce the fear-potentiated startle response in the rat: evidence for different types of anxiolytic activity?
Topics: Animals; Anti-Anxiety Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Buspirone; Diazepam; Fear; Granisetron; Male; Ondansetron; Rats; Reflex, Startle; Serotonin Antagonists | 1994 |
Comparison of potencies of 5-HT3 receptor antagonists at inhibiting aversive behavior to illumination and the von Bezold-Jarisch reflex in the mouse.
Topics: Animals; Behavior, Animal; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Granisetron; Heart Rate; Lighting; Mice; Motor Activity; Ondansetron; Reflex; Serotonin Antagonists; Stereoisomerism | 1994 |
Characterisation of the non-5-HT3 high-affinity 'R' binding site for (R)-zacopride in brain and other tissues.
Topics: Aged; Aged, 80 and over; Animals; Benzamides; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Female; Glioma; Hippocampus; Humans; Male; Mianserin; Ondansetron; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord; Stereoisomerism; Tissue Distribution; Tumor Cells, Cultured | 1993 |
Differential binding characteristics of agonists at 5-HT3 receptor recognition sites in NG108-15 neuroblastoma-glioma cells labelled by [3H]-(S)-zacopride and [3H]granisetron.
Topics: Animals; Benzamides; Biguanides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Glioma; Granisetron; Indazoles; Kinetics; Neuroblastoma; Ondansetron; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 1993 |
5-HT3 receptor-independent inhibition of the depolarization-induced 86Rb efflux from human neuroblastoma cells, TE671, by ondansetron.
Topics: Anti-Anxiety Agents; Benzamides; Benzofurans; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypoglycemic Agents; Indazoles; Indoles; Neuroblastoma; Neurotoxins; Ondansetron; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Rubidium Radioisotopes; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tropanes; Tropisetron; Tumor Cells, Cultured | 1995 |
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1996 |
Response heterogeneity of 5-HT3 receptor antagonists in a rat visceral hypersensitivity model.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Colon; Granisetron; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Pain; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Tropisetron | 1996 |
Role of serotonin3 receptors in the nucleus tractus solitarii on the carotid chemoreflex.
Topics: Animals; Atropine; Benzamides; Biguanides; Brain Mapping; Bridged Bicyclo Compounds, Heterocyclic; Carotid Body; Chemoreceptor Cells; Heart Rate; Kynurenic Acid; Male; Microinjections; Ondansetron; Potassium Cyanide; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Respiration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Sympathetic Nervous System; Tidal Volume; Vagus Nerve | 1997 |
5-HT receptor subtypes involved in the serotonin-induced inhibition of L-leucine absorption in rabbit jejunum.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Indoles; Intestinal Absorption; Jejunum; Leucine; Male; Ondansetron; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides | 1997 |
Clozapine's antipsychotic effects do not depend on blockade of 5-HT3 receptors.
Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; Drug Interactions; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Ondansetron; Quinacrine; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Sulfur Radioisotopes; Tropanes | 1999 |
5-HT(3) receptors, alcohol and aggressive behavior in mice.
Topics: Aggression; Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Ethanol; Male; Mice; Ondansetron; Receptors, Serotonin, 5-HT3; Serotonin Antagonists | 2005 |
Antinociception: mechanistic studies on the action of MD-354 and clonidine. Part 1. The 5-HT3 component.
Topics: Analgesics; Animals; Behavior, Animal; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Clonidine; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Indoles; Male; Mice; Mice, Inbred ICR; Models, Animal; Motor Activity; Ondansetron; Pain; Pain Measurement; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Time Factors; Tropisetron | 2005 |