ondansetron and piperidines

ondansetron has been researched along with piperidines in 60 studies

Research

Studies (60)

TimeframeStudies, this research(%)All Research%
pre-19902 (3.33)18.7374
1990's17 (28.33)18.2507
2000's24 (40.00)29.6817
2010's17 (28.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G1
Dreteler, GH; Saxena, PR; Wouters, W1
Galligan, JJ; North, RA; Tonini, M1
Hewson, G; Hill, RG; Hughes, J; Leighton, GE1
Sussman, N1
Cesana, R; Donetti, A; Ladinsky, H; Rizzi, CA; Sagrada, A; Schiantarelli, P; Schiavi, GB; Schiavone, A1
Güller, R; Jost, G; Reichlin, B1
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M1
Coupar, IM; McLean, PG1
Jordan, CC; Naylor, RJ; Rudd, JA1
Hirata, T; Kato, S; Nishiwaki, H; Takeuchi, K1
Kadowaki, M; Kontoh, A; Nagakura, Y; Shimomura, K; Tokita, K; Tomoi, M1
González, AA; Puig, MM1
Kamato, T; Miyata, K; Nagakura, Y; Yamano, M1
Kaisar, M; Naylor, RJ; Tuladhar, BR1
McAllister, KH; Pratt, JA1
Gardner, C; Perren, M1
De Miguel, E; Gomez-de-Segura, IA; Grande, AG1
Choudhury, I; Robichaud, A; Rodger, IW; Tattersall, FD1
Clemes, SA; House, F; Palmer, JL; Reid, K; Somal, HS; Stott, JR; Troakes, C; Wright, RJ1
Berggreen, P; Ersbøll, AK; Grøndahl, ML; Hansen, MB; Maltbaek, JS; Skadhauge, E; Thorbøll, JE1
Black, LS; D'Angelo, R; Dalby, PL; Gesztesi, Z; MacLean, D; Scuderi, PE; Wender, RH; White, PF; Wright, W1
Hollywood, MA; McHale, NG; Thornbury, KD1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Alsasua, A; Benhamú, B; Girón, R; López-Rodríguez, ML; Martín, MI; Pascual, D1
Burton, P; Kwiatkowska, M; Mechoulam, R; Parker, LA1
Abdalla, M; Apfel, CC; Biedler, A; Danner, K; Jokela, R; Kerger, H; Korttila, K; Kredel, M; Pocock, SJ; Roewer, N; Sessler, DI; Trenkler, S; Turan, A; Vedder, I; Zernak, C1
Kan, KK; Lai, HW; Lau, AH; Ngan, MP; Rudd, JA; Wai, MK; Yew, DT1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1
Apfel, CC; Bacher, A; Biedler, A; Danner, K; Danzeisen, O; Eberhart, LH; Forst, H; Frings, G; Fritz, G; Goebel, A; Hergert, M; Hopf, HB; Kerger, H; Kranke, P; Lange, M; Mertzlufft, F; Motsch, J; Paura, A; Roewer, N; Schneider, E; Stoecklein, K; Wermelt, J; Zernak, C1
Filip, M; Frankowska, M; Göthert, M; Przegaliński, E1
Furuya, T; Nohara, K; Yamamoto, K; Yamatodani, A1
Lau, AH; Rudd, JA; Yew, DT1
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS1
Nylander, O; Pihl, L1
Andrews, PL; Cole, N; Liu, YL; Malik, NM; Sanger, GJ1
Komada, T; Yano, S1
Camblor, E; Fernández, R; Janeiro, M; Núñez, D1
Amano, T; Ariga, H; Ishida, T; Kimura, T; Matsueda, K; Tajiri, H; Torii, A; Uehara, H; Yamato, S1
Adams, L; Blum, R; Johnson, B; Lates, C; Lebowitz, P; Lu, E; Zhang, K1
Bandekar, RR; Dediu, M; Grunberg, SM; Ramlau, R; Roila, F; Rolski, J; Russo, MW1
Apornwirat, W; Aziz, Z; Grunberg, SM; Guckert, M; Herrstedt, J; Levin, J; Ranganathan, S; Roila, F; Russo, MW; Shaharyar, A; Van Belle, S1
Albert, I; Arpornwirat, W; Bandekar, RR; Grunberg, SM; Hansen, VL; Levin, J1
Blackburn, LM; Gridelli, C; Haiderali, AM; Lykopoulos, K; Russo, MW1
Blackburn, L; Chung, F; Johnson, B; Kutsogiannis, DJ; Lane, SR; Levin, J; Pergolizzi, JV; Singla, NK; Singla, SK1
Adams, LM; Bauman, J; Dandamudi, UB; Gartner, E; Hohl, R; Johnson, B; Lewis, LD; Morris, S; Murray, S; Webb, RT1
Abissi, CJ; Hunt, CM; Papay, JI; Rich, DS; Russo, MW1
Anixter, MB1
Altorjay, A; Aqua, K; Blackburn, LM; Chinachoit, T; Kett, A; Lane, S; Levin, J; Melson, T; Pergolizzi, JV1
Dube, P; Hesketh, PJ; Kopp, M; Lane, S; Levin, J; Makhson, A; Moiseyenko, V; Rosati, G; Russo, M; Wright, O1
Ashton, JC; Jain, S; Mandhane, S; Nayak, P; Rajamannar, T; Soni, D1
Cui, R; Dong, X; Li, B; Liu, C; Lv, J; Shao, D; Song, Y; Sun, Z; Wang, L; Wang, P; Zhang, X; Zhao, J; Zhou, Y1
Chan, SW; Lin, G; Lu, Z; Rudd, JA; Yeung, CK; Yew, DT1
Brigandi, RA; Dalby, PL; Eberhart, LH; Johnson, BM; Kranke, P; Noble, R; Novikova, E; Russ, SF; Thompson, JP1
Gencer, A; Gunduz, O; Ulugol, A1
Fukuta, K; Hamaguchi, E; Kakuta, N; Kawanishi, R; Kume, K; Soga, T; Tanaka, K; Tsutsumi, R; Tsutsumi, YM1
Kurosawa, N; Seki, K; Shimizu, K1
Bataille, A; Charmeau, A; Chazot, T; Diemunsch, P; Fischler, M; Le Guen, M; Léger, P; Lemedioni, P; Letourneulx, JF; Liu, N1
Amatucci, C; Illuminati, G; Palumbo, P; Pulli, VT; Tellan, G; Usai, S; Vietri, F1
Fernandes, PD; Giorno, TBS; Moreira, IGDS; Rezende, CM1

Reviews

1 review(s) available for ondansetron and piperidines

ArticleYear
The potential benefits of serotonin receptor-specific agents.
    The Journal of clinical psychiatry, 1994, Volume: 55 Suppl

    Topics: Antidepressive Agents; Buspirone; Depressive Disorder; Humans; Isoxazoles; Ondansetron; Piperazines; Piperidines; Receptors, Serotonin; Risperidone; Selective Serotonin Reuptake Inhibitors; Serotonin; Sumatriptan; Triazoles

1994

Trials

18 trial(s) available for ondansetron and piperidines

ArticleYear
[Colonic preparation with sodium phosphate. Prospective, randomized, placebo-controlled double blind study with various antiemetics].
    Schweizerische medizinische Wochenschrift, 1996, Aug-06, Volume: 126, Issue:31-32

    Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Cathartics; Cisapride; Colonoscopy; Double-Blind Method; Female; Humans; Male; Metoclopramide; Middle Aged; Nausea; Ondansetron; Phosphates; Piperidines; Prospective Studies; Vomiting

1996
Comparison of the neurokinin-1 antagonist GR205171, alone and in combination with the 5-HT3 antagonist ondansetron, hyoscine and placebo in the prevention of motion-induced nausea in man.
    British journal of clinical pharmacology, 2000, Volume: 50, Issue:1

    Topics: Adolescent; Adult; Antiemetics; Cross-Over Studies; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Motion Sickness; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Scopolamine; Serotonin Antagonists; Tetrazoles

2000
Substance P (Neurokinin-1) antagonist prevents postoperative vomiting after abdominal hysterectomy procedures.
    Anesthesiology, 2000, Volume: 93, Issue:4

    Topics: Administration, Oral; Adult; Antiemetics; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hysterectomy; Injections, Intravenous; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Placebos; Postoperative Nausea and Vomiting; Preanesthetic Medication; Risk Factors; Serotonin Antagonists; Substance P

2000
A factorial trial of six interventions for the prevention of postoperative nausea and vomiting.
    The New England journal of medicine, 2004, Jun-10, Volume: 350, Issue:24

    Topics: Anesthesia, General; Anesthesia, Intravenous; Anesthesia, Local; Anesthetics, Intravenous; Antiemetics; Dexamethasone; Droperidol; Drug Therapy, Combination; Factor Analysis, Statistical; Female; Fentanyl; Humans; Logistic Models; Male; Multivariate Analysis; Nitrogen; Nitrous Oxide; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Premedication; Propofol; Remifentanil; Single-Blind Method

2004
[A factorial trial of six interventions for the prevention of postoperative nausea and vomiting].
    Der Anaesthesist, 2005, Volume: 54, Issue:3

    Topics: Analgesics, Opioid; Anesthetics, Inhalation; Anesthetics, Intravenous; Antiemetics; Clinical Protocols; Dexamethasone; Droperidol; Drug Therapy, Combination; Female; Fentanyl; Humans; Male; Odds Ratio; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Propofol; Remifentanil; Research Design; Risk

2005
Impact of casopitant, a novel NK-1 antagonist, on the pharmacokinetics of ondansetron and dexamethasone.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2009, Volume: 17, Issue:9

    Topics: Adolescent; Adult; Antiemetics; Dexamethasone; Drug Therapy, Combination; Drug-Related Side Effects and Adverse Reactions; Female; Humans; Male; Middle Aged; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Vomiting; Young Adult

2009
Randomized, double-blind, dose-ranging trial of the oral neurokinin-1 receptor antagonist casopitant mesylate for the prevention of cisplatin-induced nausea and vomiting.
    Annals of oncology : official journal of the European Society for Medical Oncology, 2009, Volume: 20, Issue:11

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nausea; Neoplasms; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Receptors, Neurokinin-1; Vomiting

2009
Phase III trial of casopitant, a novel neurokinin-1 receptor antagonist, for the prevention of nausea and vomiting in patients receiving moderately emetogenic chemotherapy.
    Journal of clinical oncology : official journal of the American Society of Clinical Oncology, 2009, Nov-10, Volume: 27, Issue:32

    Topics: Administration, Oral; Alopecia; Anthracyclines; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Constipation; Cyclophosphamide; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Headache; Humans; Injections, Intravenous; Kaplan-Meier Estimate; Male; Middle Aged; Nausea; Neoplasms; Neurokinin-1 Receptor Antagonists; Neutropenia; Ondansetron; Piperazines; Piperidines; Treatment Outcome; Vomiting

2009
Phase 2 trial results with the novel neurokinin-1 receptor antagonist casopitant in combination with ondansetron and dexamethasone for the prevention of chemotherapy-induced nausea and vomiting in cancer patients receiving moderately emetogenic chemothera
    Cancer, 2009, Dec-15, Volume: 115, Issue:24

    Topics: Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Dexamethasone; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Middle Aged; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Vomiting

2009
Casopitant improves the quality of life in patients receiving highly emetogenic chemotherapy.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2010, Volume: 18, Issue:11

    Topics: Activities of Daily Living; Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nausea; Neoplasms; Ondansetron; Piperazines; Piperidines; Quality of Life; Surveys and Questionnaires; Vomiting; Young Adult

2010
Phase II study to evaluate the safety and efficacy of the oral neurokinin-1 receptor antagonist casopitant (GW679769) administered with ondansetron for the prevention of postoperative and postdischarge nausea and vomiting in high-risk patients.
    Anesthesiology, 2010, Volume: 113, Issue:1

    Topics: Administration, Oral; Adolescent; Adult; Anesthesia, General; Antiemetics; Cholecystectomy, Laparoscopic; Constipation; Dizziness; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Female; Gynecologic Surgical Procedures; Headache; Humans; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Postoperative Nausea and Vomiting; Risk Factors; Treatment Outcome; Young Adult

2010
Lack of effect of casopitant on the pharmacokinetics of docetaxel in patients with cancer.
    Cancer chemotherapy and pharmacology, 2011, Volume: 67, Issue:4

    Topics: Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Area Under Curve; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Dexamethasone; Docetaxel; Drug Therapy, Combination; Enzyme Inhibitors; Female; Humans; Least-Squares Analysis; Leukocyte Count; Male; Middle Aged; Neoplasms; Neurokinin-1 Receptor Antagonists; Neutrophils; Ondansetron; Piperazines; Piperidines; Taxoids

2011
The evaluation of drug rechallenge: the casopitant Phase III program.
    Regulatory toxicology and pharmacology : RTP, 2010, Volume: 58, Issue:3

    Topics: Administration, Oral; Antiemetics; Antineoplastic Agents; Dexamethasone; Dose-Response Relationship, Drug; Female; Humans; Male; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Serotonin Antagonists; Vomiting

2010
Casopitant and ondansetron for postoperative nausea and vomiting prevention in women at high risk for emesis: a phase 3 study.
    Archives of surgery (Chicago, Ill. : 1960), 2011, Volume: 146, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Dose-Response Relationship, Drug; Double-Blind Method; Female; Follow-Up Studies; Humans; Incidence; Injections, Intravenous; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Postoperative Care; Postoperative Nausea and Vomiting; Retrospective Studies; Risk Factors; Treatment Outcome; United States; Young Adult

2011
Single-dose intravenous casopitant in combination with ondansetron and dexamethasone for the prevention of oxaliplatin-induced nausea and vomiting: a multicenter, randomized, double-blind, active-controlled, two arm, parallel group study.
    Supportive care in cancer : official journal of the Multinational Association of Supportive Care in Cancer, 2012, Volume: 20, Issue:7

    Topics: Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Area Under Curve; Colorectal Neoplasms; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Infusions, Intravenous; Male; Middle Aged; Nausea; Ondansetron; Organoplatinum Compounds; Oxaliplatin; Piperazines; Piperidines; Time Factors; Treatment Outcome; Vomiting

2012
Comparison of vestipitant with ondansetron for the treatment of breakthrough postoperative nausea and vomiting after failed prophylaxis with ondansetron.
    British journal of anaesthesia, 2015, Volume: 114, Issue:3

    Topics: Adult; Aged; Antiemetics; Dose-Response Relationship, Drug; Female; Fluorobenzenes; Humans; Male; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Single-Blind Method; Treatment Failure; Treatment Outcome; Young Adult

2015
Fosaprepitant versus ondansetron for the prevention of postoperative nausea and vomiting in patients who undergo gynecologic abdominal surgery with patient-controlled epidural analgesia: a prospective, randomized, double-blind study.
    Journal of anesthesia, 2015, Volume: 29, Issue:5

    Topics: Adult; Analgesia, Epidural; Analgesia, Patient-Controlled; Analgesics, Opioid; Androstanols; Antiemetics; Double-Blind Method; Female; Fentanyl; Gynecologic Surgical Procedures; Humans; Middle Aged; Morpholines; Ondansetron; Pain; Piperidines; Postoperative Nausea and Vomiting; Postoperative Period; Prospective Studies; Remifentanil; Rocuronium

2015
Impact of a prophylactic combination of dexamethasone-ondansetron on postoperative nausea and vomiting in obese adult patients undergoing laparoscopic sleeve gastrectomy during closed-loop propofol-remifentanil anaesthesia: A randomised double-blind place
    European journal of anaesthesiology, 2016, Volume: 33, Issue:12

    Topics: Adult; Anesthesia, General; Anesthetics, Intravenous; Dexamethasone; Double-Blind Method; Female; Gastrectomy; Humans; Laparoscopy; Male; Middle Aged; Monitoring, Intraoperative; Obesity; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Pre-Exposure Prophylaxis; Propofol; Remifentanil

2016

Other Studies

41 other study(ies) available for ondansetron and piperidines

ArticleYear
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
    Journal of neural transmission. General section, 1990, Volume: 82, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes

1990
Comparison of the cardiovascular effects of the 5-HT1A receptor agonist flesinoxan with that of 8-OH-DPAT in the rat.
    European journal of pharmacology, 1990, May-16, Volume: 180, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Antihypertensive Agents; Atropine; Blood Pressure; Decerebrate State; Heart Rate; Hemodynamics; Imidazoles; In Vitro Techniques; Male; Naphthalenes; Ondansetron; Piperazines; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tetrahydronaphthalenes

1990
Effects of cisapride on cholinergic neurotransmission and propulsive motility in the guinea pig ileum.
    Gastroenterology, 1989, Volume: 96, Issue:5 Pt 1

    Topics: Acetylcholine; Animals; Cisapride; Gastrointestinal Motility; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Indoles; Membrane Potentials; Ondansetron; Peristalsis; Piperidines; Serotonin; Serotonin Antagonists; Synapses; Synaptic Transmission; Tropisetron

1989
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1988
Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:4

    Topics: Animals; Anti-Ulcer Agents; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dogs; Dose-Response Relationship, Drug; Female; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle Denervation; Neostriatum; Ondansetron; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Swine; Tumor Cells, Cultured

1994
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
    European journal of pharmacology, 1996, Sep-05, Volume: 311, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1996
Characterisation of a postjunctional 5-ht7-like and a prejunctional 5-HT3 receptor mediating contraction of rat isolated jejunum.
    European journal of pharmacology, 1996, Sep-26, Volume: 312, Issue:2

    Topics: Animals; Atropine; Benzamides; Dose-Response Relationship, Drug; In Vitro Techniques; Jejunum; Male; Methysergide; Monoamine Oxidase Inhibitors; Muscle Contraction; Ondansetron; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrodotoxin

1996
The action of the NK1 tachykinin receptor antagonist, CP 99,994, in antagonizing the acute and delayed emesis induced by cisplatin in the ferret.
    British journal of pharmacology, 1996, Volume: 119, Issue:5

    Topics: Animals; Antineoplastic Agents; Cisplatin; Ferrets; Male; Neurokinin-1 Receptor Antagonists; Ondansetron; Pharmaceutical Vehicles; Piperidines; Vomiting

1996
Gastric motility and mucosal ulcerogenic responses induced by prokinetic drugs in rats under prostaglandin-deficient conditions.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:2

    Topics: Animals; Cisapride; Dose-Response Relationship, Drug; Gastric Acid; Gastric Emptying; Gastric Mucosa; Gastrointestinal Agents; Gastrointestinal Motility; Indomethacin; Male; Metoclopramide; Ondansetron; Piperidines; Prostaglandin Antagonists; Prostaglandins; Rats; Rats, Sprague-Dawley; Stomach; Stomach Ulcer

1997
Combined blockade of 5-HT3- and 5-HT4-serotonin receptors inhibits colonic functions in conscious rats and mice.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: 4-Aminobenzoic Acid; Animals; Colon; Dioxanes; Male; Mice; Ondansetron; para-Aminobenzoates; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists

1997
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron

1997
Effects of gastroprokinetic agents on gastroparesis in streptozotocin-induced diabetic rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: Animals; Benzamides; Benzimidazoles; Blood Glucose; Cisapride; Diabetes Mellitus, Experimental; Gastric Emptying; Gastrointestinal Motility; Gastroparesis; Granisetron; Male; Morpholines; Ondansetron; Piperidines; Pyrroles; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Vagotomy

1997
Evidence for a 5-HT3 receptor involvement in the facilitation of peristalsis on mucosal application of 5-HT in the guinea pig isolated ileum.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: Animals; Dioxanes; Female; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methiothepin; Mucous Membrane; Ondansetron; Peristalsis; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists

1997
GR205171 blocks apomorphine and amphetamine-induced conditioned taste aversions.
    European journal of pharmacology, 1998, Jul-24, Volume: 353, Issue:2-3

    Topics: Amphetamines; Animals; Apomorphine; Avoidance Learning; Conditioning, Classical; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Taste; Tetrazoles

1998
Inhibition of anaesthetic-induced emesis by a NK1 or 5-HT3 receptor antagonist in the house musk shrew, Suncus murinus.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: Anesthesia; Animals; Halothane; Humans; Male; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Shrews; Tetrazoles; Vomiting

1998
Antiemetic effects of Lerisetron in radiation-induced emesis in the dog.
    Acta oncologica (Stockholm, Sweden), 1998, Volume: 37, Issue:7-8

    Topics: Animals; Antiemetics; Benzimidazoles; Cobalt Radioisotopes; Dogs; Drug Administration Schedule; Ondansetron; Piperidines; Radiotherapy; Serotonin Antagonists; Vomiting

1998
Emesis induced by inhibitors of type IV cyclic nucleotide phosphodiesterase (PDE IV) in the ferret.
    Neuropharmacology, 1999, Volume: 38, Issue:2

    Topics: Animals; Antiemetics; Dose-Response Relationship, Drug; Emetics; Ferrets; Indoles; Molecular Structure; Nitrobenzenes; Ondansetron; Phenylurea Compounds; Phosphodiesterase Inhibitors; Piperidines; Pyridines; Pyrrolidinones; Quinolones; Rolipram; Stereoisomerism; Time Factors; Vomiting

1999
Regional differences in neurogenic signal transduction pathway of cholera toxin-induced fluid, electrolyte and serotonin accumulation in the porcine jejunum.
    Pharmacology & toxicology, 2000, Volume: 86, Issue:6

    Topics: Animals; Body Fluids; Cholera Toxin; Dose-Response Relationship, Drug; Electrolytes; Female; Hexamethonium; Jejunum; Nicotinic Antagonists; Ondansetron; Piperidines; Receptors, Neurokinin-1; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Signal Transduction; Substance P; Swine

2000
5-HT inhibits spontaneous contractility of isolated sheep mesenteric lymphatics via activation of 5-HT(4) receptors.
    Microvascular research, 2000, Volume: 60, Issue:3

    Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Isometric Contraction; Lymphatic System; Methysergide; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sheep

2000
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
New benzimidazole derivatives: selective and orally active 5-HT3 receptor antagonists.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: 5-Hydroxytryptophan; Administration, Oral; Animals; Aza Compounds; Behavior, Animal; Benzimidazoles; Carbachol; Diarrhea; Dose-Response Relationship, Drug; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Injections, Intraperitoneal; Injections, Intravenous; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Piperidines; Propane; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Serotonin; Serotonin Antagonists

2003
A comparative analysis of the potential of cannabinoids and ondansetron to suppress cisplatin-induced emesis in the Suncus murinus (house musk shrew).
    Psychopharmacology, 2004, Volume: 174, Issue:2

    Topics: Animals; Antiemetics; Antineoplastic Agents; Cannabinoids; Cisplatin; Dose-Response Relationship, Drug; Dronabinol; Drug Therapy, Combination; Female; Lithium; Male; Ondansetron; Piperidines; Psychotropic Drugs; Pyrazoles; Rimonabant; Shrews; Vomiting

2004
Action of ondansetron and CP-99,994 to modify behavior and antagonize cisplatin-induced emesis in the ferret.
    European journal of pharmacology, 2005, Jan-04, Volume: 506, Issue:3

    Topics: Animals; Antiemetics; Behavior, Animal; Cisplatin; Ferrets; Male; Ondansetron; Piperidines; Vomiting

2005
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005
WIN 55,212-2-induced reduction of cocaine hyperlocomotion: possible inhibition of 5-HT(3) receptor function.
    European journal of pharmacology, 2005, Jul-04, Volume: 517, Issue:1-2

    Topics: Animals; Benzoxazines; Cocaine; Dose-Response Relationship, Drug; Male; Morpholines; Motor Activity; Naphthalenes; Ondansetron; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Rimonabant; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists

2005
Ondansetron, dexamethasone and an NK1 antagonist block radiation sickness in mice.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 82, Issue:1

    Topics: Animals; Antiemetics; Dexamethasone; Drug Therapy, Combination; Male; Mice; Mice, Inbred ICR; Neurokinin-1 Receptor Antagonists; Ondansetron; Pica; Piperidines; Radiation Injuries; Serotonin Antagonists

2005
Action of ondansetron and CP-99,994 on cisplatin-induced emesis and locomotor activity in Suncus murinus (house musk shrew).
    Behavioural pharmacology, 2005, Volume: 16, Issue:8

    Topics: Animals; Antineoplastic Agents; Behavior, Animal; Cisplatin; Female; Motor Activity; Ondansetron; Piperidines; Serotonin Receptor Agonists; Shrews; Vomiting

2005
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:2

    Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors

2006
Luminal hypotonicity increases duodenal mucosal permeability by a mechanism involving 5-hydroxytryptamine.
    Acta physiologica (Oxford, England), 2006, Volume: 186, Issue:1

    Topics: Anesthetics, Local; Animals; Cyclooxygenase Inhibitors; Duodenum; Granisetron; Indoles; Indomethacin; Intestinal Mucosa; Lidocaine; Male; Ondansetron; Osmotic Pressure; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Tetrodotoxin; Tropisetron

2006
Differential effects of dexamethasone, ondansetron and a tachykinin NK1 receptor antagonist (GR205171) on cisplatin-induced changes in behaviour, food intake, pica and gastric function in rats.
    European journal of pharmacology, 2007, Jan-26, Volume: 555, Issue:2-3

    Topics: Animals; Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Eating; Gastric Emptying; Male; Motor Activity; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Pica; Piperidines; Rats; Rats, Wistar; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Tetrazoles

2007
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2007
[Narcolepsy and anesthesia].
    Revista espanola de anestesiologia y reanimacion, 2007, Volume: 54, Issue:3

    Topics: Analgesia, Epidural; Anesthesia, Intravenous; Antiemetics; Benzhydryl Compounds; Chemical and Drug Induced Liver Injury; Clomipramine; Contraindications; Humans; Hypnotics and Sedatives; Intracellular Signaling Peptides and Proteins; Intraoperative Complications; Kidney Pelvis; Modafinil; Narcolepsy; Neuropeptides; Ondansetron; Orexins; Pain, Postoperative; Piperidines; Preanesthetic Medication; Propofol; Remifentanil; Ureteral Obstruction

2007
Urocortin I is present in the enteric nervous system and exerts an excitatory effect via cholinergic and serotonergic pathways in the rat colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 293, Issue:4

    Topics: Animals; Atropine; Colon; Corticotropin-Releasing Hormone; Dioxanes; Electric Stimulation; Enteric Nervous System; Gastrointestinal Motility; Hexamethonium; Immunohistochemistry; Male; NG-Nitroarginine Methyl Ester; Ondansetron; Peptide Fragments; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Tetrodotoxin; Urocortins

2007
Why no casopitant-only arm?
    Anesthesiology, 2011, Volume: 114, Issue:1

    Topics: Antiemetics; Dose-Response Relationship, Drug; Drug Therapy, Combination; Humans; Ondansetron; Piperazines; Piperidines; Postoperative Nausea and Vomiting; Treatment Outcome

2011
Induction of glucose intolerance by acute administration of rimonabant.
    Pharmacology, 2012, Volume: 89, Issue:5-6

    Topics: Administration, Oral; Animals; Benzoxazines; Blood Glucose; Dopamine Antagonists; Eating; Fenclonine; Glucose; Glucose Intolerance; Haloperidol; Hepatocytes; Infusions, Intraventricular; Insulin; Male; Mice; Morpholines; Naphthalenes; Ondansetron; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Dopamine; Receptors, Serotonin; Rimonabant; Serotonin Antagonists

2012
The anticonvulsant effects of SR 57227 on pentylenetetrazole-induced seizure in mice.
    PloS one, 2014, Volume: 9, Issue:4

    Topics: Animals; Anticonvulsants; gamma-Aminobutyric Acid; Hippocampus; Male; Mice, Inbred ICR; Ondansetron; Pentylenetetrazole; Piperidines; Proto-Oncogene Proteins c-fos; Seizures; Survival Analysis

2014
The differential antiemetic properties of GLP-1 receptor antagonist, exendin (9-39) in Suncus murinus (house musk shrew).
    Neuropharmacology, 2014, Volume: 83

    Topics: Animals; Antiemetics; Brain; Exenatide; Glucagon-Like Peptide-1 Receptor; Male; Ondansetron; Peptide Fragments; Peptides; Piperidines; Proto-Oncogene Proteins c-fos; Receptors, Glucagon; Shrews; Venoms; Vomiting

2014
Involvement of Descending Serotonergic and Noradrenergic Systems and their Spinal Receptor Subtypes in the Antinociceptive Effect of Dipyrone.
    Drug research, 2015, Volume: 65, Issue:12

    Topics: 5,7-Dihydroxytryptamine; Adrenergic Neurons; Analgesics; Animals; Dipyrone; Dose-Response Relationship, Drug; Injections, Spinal; Ketanserin; Mice; Ondansetron; Oxidopamine; Pain Measurement; Piperidines; Prazosin; Propranolol; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonergic Neurons; Spinal Cord; Sulfonamides; Yohimbine

2015
The role of the AMPA receptor and 5-HT(3) receptor on aggressive behavior and depressive-like symptoms in chronic social isolation-reared mice.
    Physiology & behavior, 2016, Jan-01, Volume: 153

    Topics: Aggression; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amygdala; Animals; Depression; Food Preferences; Glutamate Decarboxylase; Hypothalamus; Injections, Intraperitoneal; Male; Mice; Microinjections; Motor Activity; Neurons; Ondansetron; Piperidines; Quinoxalines; Receptors, AMPA; Receptors, Serotonin, 5-HT3; Social Isolation

2016
Postoperative nausea and vomiting (PONV) in outpatient repair of inguinal hernia.
    Annali italiani di chirurgia, 2018, Volume: 89

    Topics: Adjuvants, Anesthesia; Adolescent; Adult; Aged; Aged, 80 and over; Analgesics, Opioid; Anesthesia, Local; Antiemetics; Deep Sedation; Dexamethasone; Female; Fentanyl; Hernia, Inguinal; Herniorrhaphy; Humans; Male; Middle Aged; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Preanesthetic Medication; Propofol; Remifentanil; Retrospective Studies; Young Adult

2018
New
    Scientific reports, 2018, 07-03, Volume: 8, Issue:1

    Topics: Analgesics; Animals; Behavior, Animal; Capsaicin; Coffee; Disease Models, Animal; Female; Formaldehyde; Glutamic Acid; Hot Temperature; Hyperalgesia; Male; Mice; Naloxone; Narcotic Antagonists; Ondansetron; Pain; Pain Measurement; Piperidines; Pyrazoles; Serotonin

2018