ondansetron has been researched along with piperidines in 60 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (3.33) | 18.7374 |
1990's | 17 (28.33) | 18.2507 |
2000's | 24 (40.00) | 29.6817 |
2010's | 17 (28.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G | 1 |
Dreteler, GH; Saxena, PR; Wouters, W | 1 |
Galligan, JJ; North, RA; Tonini, M | 1 |
Hewson, G; Hill, RG; Hughes, J; Leighton, GE | 1 |
Sussman, N | 1 |
Cesana, R; Donetti, A; Ladinsky, H; Rizzi, CA; Sagrada, A; Schiantarelli, P; Schiavi, GB; Schiavone, A | 1 |
Güller, R; Jost, G; Reichlin, B | 1 |
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M | 1 |
Coupar, IM; McLean, PG | 1 |
Jordan, CC; Naylor, RJ; Rudd, JA | 1 |
Hirata, T; Kato, S; Nishiwaki, H; Takeuchi, K | 1 |
Kadowaki, M; Kontoh, A; Nagakura, Y; Shimomura, K; Tokita, K; Tomoi, M | 1 |
González, AA; Puig, MM | 1 |
Kamato, T; Miyata, K; Nagakura, Y; Yamano, M | 1 |
Kaisar, M; Naylor, RJ; Tuladhar, BR | 1 |
McAllister, KH; Pratt, JA | 1 |
Gardner, C; Perren, M | 1 |
De Miguel, E; Gomez-de-Segura, IA; Grande, AG | 1 |
Choudhury, I; Robichaud, A; Rodger, IW; Tattersall, FD | 1 |
Clemes, SA; House, F; Palmer, JL; Reid, K; Somal, HS; Stott, JR; Troakes, C; Wright, RJ | 1 |
Berggreen, P; Ersbøll, AK; Grøndahl, ML; Hansen, MB; Maltbaek, JS; Skadhauge, E; Thorbøll, JE | 1 |
Black, LS; D'Angelo, R; Dalby, PL; Gesztesi, Z; MacLean, D; Scuderi, PE; Wender, RH; White, PF; Wright, W | 1 |
Hollywood, MA; McHale, NG; Thornbury, KD | 1 |
Naylor, RJ; Tuladhar, BR; Womack, MD | 1 |
Alsasua, A; Benhamú, B; Girón, R; López-Rodríguez, ML; Martín, MI; Pascual, D | 1 |
Burton, P; Kwiatkowska, M; Mechoulam, R; Parker, LA | 1 |
Abdalla, M; Apfel, CC; Biedler, A; Danner, K; Jokela, R; Kerger, H; Korttila, K; Kredel, M; Pocock, SJ; Roewer, N; Sessler, DI; Trenkler, S; Turan, A; Vedder, I; Zernak, C | 1 |
Kan, KK; Lai, HW; Lau, AH; Ngan, MP; Rudd, JA; Wai, MK; Yew, DT | 1 |
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C | 1 |
Apfel, CC; Bacher, A; Biedler, A; Danner, K; Danzeisen, O; Eberhart, LH; Forst, H; Frings, G; Fritz, G; Goebel, A; Hergert, M; Hopf, HB; Kerger, H; Kranke, P; Lange, M; Mertzlufft, F; Motsch, J; Paura, A; Roewer, N; Schneider, E; Stoecklein, K; Wermelt, J; Zernak, C | 1 |
Filip, M; Frankowska, M; Göthert, M; Przegaliński, E | 1 |
Furuya, T; Nohara, K; Yamamoto, K; Yamatodani, A | 1 |
Lau, AH; Rudd, JA; Yew, DT | 1 |
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS | 1 |
Nylander, O; Pihl, L | 1 |
Andrews, PL; Cole, N; Liu, YL; Malik, NM; Sanger, GJ | 1 |
Komada, T; Yano, S | 1 |
Camblor, E; Fernández, R; Janeiro, M; Núñez, D | 1 |
Amano, T; Ariga, H; Ishida, T; Kimura, T; Matsueda, K; Tajiri, H; Torii, A; Uehara, H; Yamato, S | 1 |
Adams, L; Blum, R; Johnson, B; Lates, C; Lebowitz, P; Lu, E; Zhang, K | 1 |
Bandekar, RR; Dediu, M; Grunberg, SM; Ramlau, R; Roila, F; Rolski, J; Russo, MW | 1 |
Apornwirat, W; Aziz, Z; Grunberg, SM; Guckert, M; Herrstedt, J; Levin, J; Ranganathan, S; Roila, F; Russo, MW; Shaharyar, A; Van Belle, S | 1 |
Albert, I; Arpornwirat, W; Bandekar, RR; Grunberg, SM; Hansen, VL; Levin, J | 1 |
Blackburn, LM; Gridelli, C; Haiderali, AM; Lykopoulos, K; Russo, MW | 1 |
Blackburn, L; Chung, F; Johnson, B; Kutsogiannis, DJ; Lane, SR; Levin, J; Pergolizzi, JV; Singla, NK; Singla, SK | 1 |
Adams, LM; Bauman, J; Dandamudi, UB; Gartner, E; Hohl, R; Johnson, B; Lewis, LD; Morris, S; Murray, S; Webb, RT | 1 |
Abissi, CJ; Hunt, CM; Papay, JI; Rich, DS; Russo, MW | 1 |
Anixter, MB | 1 |
Altorjay, A; Aqua, K; Blackburn, LM; Chinachoit, T; Kett, A; Lane, S; Levin, J; Melson, T; Pergolizzi, JV | 1 |
Dube, P; Hesketh, PJ; Kopp, M; Lane, S; Levin, J; Makhson, A; Moiseyenko, V; Rosati, G; Russo, M; Wright, O | 1 |
Ashton, JC; Jain, S; Mandhane, S; Nayak, P; Rajamannar, T; Soni, D | 1 |
Cui, R; Dong, X; Li, B; Liu, C; Lv, J; Shao, D; Song, Y; Sun, Z; Wang, L; Wang, P; Zhang, X; Zhao, J; Zhou, Y | 1 |
Chan, SW; Lin, G; Lu, Z; Rudd, JA; Yeung, CK; Yew, DT | 1 |
Brigandi, RA; Dalby, PL; Eberhart, LH; Johnson, BM; Kranke, P; Noble, R; Novikova, E; Russ, SF; Thompson, JP | 1 |
Gencer, A; Gunduz, O; Ulugol, A | 1 |
Fukuta, K; Hamaguchi, E; Kakuta, N; Kawanishi, R; Kume, K; Soga, T; Tanaka, K; Tsutsumi, R; Tsutsumi, YM | 1 |
Kurosawa, N; Seki, K; Shimizu, K | 1 |
Bataille, A; Charmeau, A; Chazot, T; Diemunsch, P; Fischler, M; Le Guen, M; Léger, P; Lemedioni, P; Letourneulx, JF; Liu, N | 1 |
Amatucci, C; Illuminati, G; Palumbo, P; Pulli, VT; Tellan, G; Usai, S; Vietri, F | 1 |
Fernandes, PD; Giorno, TBS; Moreira, IGDS; Rezende, CM | 1 |
1 review(s) available for ondansetron and piperidines
Article | Year |
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The potential benefits of serotonin receptor-specific agents.
Topics: Antidepressive Agents; Buspirone; Depressive Disorder; Humans; Isoxazoles; Ondansetron; Piperazines; Piperidines; Receptors, Serotonin; Risperidone; Selective Serotonin Reuptake Inhibitors; Serotonin; Sumatriptan; Triazoles | 1994 |
18 trial(s) available for ondansetron and piperidines
Article | Year |
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[Colonic preparation with sodium phosphate. Prospective, randomized, placebo-controlled double blind study with various antiemetics].
Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Cathartics; Cisapride; Colonoscopy; Double-Blind Method; Female; Humans; Male; Metoclopramide; Middle Aged; Nausea; Ondansetron; Phosphates; Piperidines; Prospective Studies; Vomiting | 1996 |
Comparison of the neurokinin-1 antagonist GR205171, alone and in combination with the 5-HT3 antagonist ondansetron, hyoscine and placebo in the prevention of motion-induced nausea in man.
Topics: Adolescent; Adult; Antiemetics; Cross-Over Studies; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Motion Sickness; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Scopolamine; Serotonin Antagonists; Tetrazoles | 2000 |
Substance P (Neurokinin-1) antagonist prevents postoperative vomiting after abdominal hysterectomy procedures.
Topics: Administration, Oral; Adult; Antiemetics; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hysterectomy; Injections, Intravenous; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Placebos; Postoperative Nausea and Vomiting; Preanesthetic Medication; Risk Factors; Serotonin Antagonists; Substance P | 2000 |
A factorial trial of six interventions for the prevention of postoperative nausea and vomiting.
Topics: Anesthesia, General; Anesthesia, Intravenous; Anesthesia, Local; Anesthetics, Intravenous; Antiemetics; Dexamethasone; Droperidol; Drug Therapy, Combination; Factor Analysis, Statistical; Female; Fentanyl; Humans; Logistic Models; Male; Multivariate Analysis; Nitrogen; Nitrous Oxide; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Premedication; Propofol; Remifentanil; Single-Blind Method | 2004 |
[A factorial trial of six interventions for the prevention of postoperative nausea and vomiting].
Topics: Analgesics, Opioid; Anesthetics, Inhalation; Anesthetics, Intravenous; Antiemetics; Clinical Protocols; Dexamethasone; Droperidol; Drug Therapy, Combination; Female; Fentanyl; Humans; Male; Odds Ratio; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Propofol; Remifentanil; Research Design; Risk | 2005 |
Impact of casopitant, a novel NK-1 antagonist, on the pharmacokinetics of ondansetron and dexamethasone.
Topics: Adolescent; Adult; Antiemetics; Dexamethasone; Drug Therapy, Combination; Drug-Related Side Effects and Adverse Reactions; Female; Humans; Male; Middle Aged; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Vomiting; Young Adult | 2009 |
Randomized, double-blind, dose-ranging trial of the oral neurokinin-1 receptor antagonist casopitant mesylate for the prevention of cisplatin-induced nausea and vomiting.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nausea; Neoplasms; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Receptors, Neurokinin-1; Vomiting | 2009 |
Phase III trial of casopitant, a novel neurokinin-1 receptor antagonist, for the prevention of nausea and vomiting in patients receiving moderately emetogenic chemotherapy.
Topics: Administration, Oral; Alopecia; Anthracyclines; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Constipation; Cyclophosphamide; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Headache; Humans; Injections, Intravenous; Kaplan-Meier Estimate; Male; Middle Aged; Nausea; Neoplasms; Neurokinin-1 Receptor Antagonists; Neutropenia; Ondansetron; Piperazines; Piperidines; Treatment Outcome; Vomiting | 2009 |
Phase 2 trial results with the novel neurokinin-1 receptor antagonist casopitant in combination with ondansetron and dexamethasone for the prevention of chemotherapy-induced nausea and vomiting in cancer patients receiving moderately emetogenic chemothera
Topics: Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Dexamethasone; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Middle Aged; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Vomiting | 2009 |
Casopitant improves the quality of life in patients receiving highly emetogenic chemotherapy.
Topics: Activities of Daily Living; Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nausea; Neoplasms; Ondansetron; Piperazines; Piperidines; Quality of Life; Surveys and Questionnaires; Vomiting; Young Adult | 2010 |
Phase II study to evaluate the safety and efficacy of the oral neurokinin-1 receptor antagonist casopitant (GW679769) administered with ondansetron for the prevention of postoperative and postdischarge nausea and vomiting in high-risk patients.
Topics: Administration, Oral; Adolescent; Adult; Anesthesia, General; Antiemetics; Cholecystectomy, Laparoscopic; Constipation; Dizziness; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Female; Gynecologic Surgical Procedures; Headache; Humans; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Postoperative Nausea and Vomiting; Risk Factors; Treatment Outcome; Young Adult | 2010 |
Lack of effect of casopitant on the pharmacokinetics of docetaxel in patients with cancer.
Topics: Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Area Under Curve; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Dexamethasone; Docetaxel; Drug Therapy, Combination; Enzyme Inhibitors; Female; Humans; Least-Squares Analysis; Leukocyte Count; Male; Middle Aged; Neoplasms; Neurokinin-1 Receptor Antagonists; Neutrophils; Ondansetron; Piperazines; Piperidines; Taxoids | 2011 |
The evaluation of drug rechallenge: the casopitant Phase III program.
Topics: Administration, Oral; Antiemetics; Antineoplastic Agents; Dexamethasone; Dose-Response Relationship, Drug; Female; Humans; Male; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Serotonin Antagonists; Vomiting | 2010 |
Casopitant and ondansetron for postoperative nausea and vomiting prevention in women at high risk for emesis: a phase 3 study.
Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Dose-Response Relationship, Drug; Double-Blind Method; Female; Follow-Up Studies; Humans; Incidence; Injections, Intravenous; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperazines; Piperidines; Postoperative Care; Postoperative Nausea and Vomiting; Retrospective Studies; Risk Factors; Treatment Outcome; United States; Young Adult | 2011 |
Single-dose intravenous casopitant in combination with ondansetron and dexamethasone for the prevention of oxaliplatin-induced nausea and vomiting: a multicenter, randomized, double-blind, active-controlled, two arm, parallel group study.
Topics: Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Area Under Curve; Colorectal Neoplasms; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Infusions, Intravenous; Male; Middle Aged; Nausea; Ondansetron; Organoplatinum Compounds; Oxaliplatin; Piperazines; Piperidines; Time Factors; Treatment Outcome; Vomiting | 2012 |
Comparison of vestipitant with ondansetron for the treatment of breakthrough postoperative nausea and vomiting after failed prophylaxis with ondansetron.
Topics: Adult; Aged; Antiemetics; Dose-Response Relationship, Drug; Female; Fluorobenzenes; Humans; Male; Middle Aged; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Single-Blind Method; Treatment Failure; Treatment Outcome; Young Adult | 2015 |
Fosaprepitant versus ondansetron for the prevention of postoperative nausea and vomiting in patients who undergo gynecologic abdominal surgery with patient-controlled epidural analgesia: a prospective, randomized, double-blind study.
Topics: Adult; Analgesia, Epidural; Analgesia, Patient-Controlled; Analgesics, Opioid; Androstanols; Antiemetics; Double-Blind Method; Female; Fentanyl; Gynecologic Surgical Procedures; Humans; Middle Aged; Morpholines; Ondansetron; Pain; Piperidines; Postoperative Nausea and Vomiting; Postoperative Period; Prospective Studies; Remifentanil; Rocuronium | 2015 |
Impact of a prophylactic combination of dexamethasone-ondansetron on postoperative nausea and vomiting in obese adult patients undergoing laparoscopic sleeve gastrectomy during closed-loop propofol-remifentanil anaesthesia: A randomised double-blind place
Topics: Adult; Anesthesia, General; Anesthetics, Intravenous; Dexamethasone; Double-Blind Method; Female; Gastrectomy; Humans; Laparoscopy; Male; Middle Aged; Monitoring, Intraoperative; Obesity; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Pre-Exposure Prophylaxis; Propofol; Remifentanil | 2016 |
41 other study(ies) available for ondansetron and piperidines
Article | Year |
---|---|
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes | 1990 |
Comparison of the cardiovascular effects of the 5-HT1A receptor agonist flesinoxan with that of 8-OH-DPAT in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Antihypertensive Agents; Atropine; Blood Pressure; Decerebrate State; Heart Rate; Hemodynamics; Imidazoles; In Vitro Techniques; Male; Naphthalenes; Ondansetron; Piperazines; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
Effects of cisapride on cholinergic neurotransmission and propulsive motility in the guinea pig ileum.
Topics: Acetylcholine; Animals; Cisapride; Gastrointestinal Motility; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Indoles; Membrane Potentials; Ondansetron; Peristalsis; Piperidines; Serotonin; Serotonin Antagonists; Synapses; Synaptic Transmission; Tropisetron | 1989 |
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors.
Topics: Animals; Anti-Ulcer Agents; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dogs; Dose-Response Relationship, Drug; Female; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle Denervation; Neostriatum; Ondansetron; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Swine; Tumor Cells, Cultured | 1994 |
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1996 |
Characterisation of a postjunctional 5-ht7-like and a prejunctional 5-HT3 receptor mediating contraction of rat isolated jejunum.
Topics: Animals; Atropine; Benzamides; Dose-Response Relationship, Drug; In Vitro Techniques; Jejunum; Male; Methysergide; Monoamine Oxidase Inhibitors; Muscle Contraction; Ondansetron; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrodotoxin | 1996 |
The action of the NK1 tachykinin receptor antagonist, CP 99,994, in antagonizing the acute and delayed emesis induced by cisplatin in the ferret.
Topics: Animals; Antineoplastic Agents; Cisplatin; Ferrets; Male; Neurokinin-1 Receptor Antagonists; Ondansetron; Pharmaceutical Vehicles; Piperidines; Vomiting | 1996 |
Gastric motility and mucosal ulcerogenic responses induced by prokinetic drugs in rats under prostaglandin-deficient conditions.
Topics: Animals; Cisapride; Dose-Response Relationship, Drug; Gastric Acid; Gastric Emptying; Gastric Mucosa; Gastrointestinal Agents; Gastrointestinal Motility; Indomethacin; Male; Metoclopramide; Ondansetron; Piperidines; Prostaglandin Antagonists; Prostaglandins; Rats; Rats, Sprague-Dawley; Stomach; Stomach Ulcer | 1997 |
Combined blockade of 5-HT3- and 5-HT4-serotonin receptors inhibits colonic functions in conscious rats and mice.
Topics: 4-Aminobenzoic Acid; Animals; Colon; Dioxanes; Male; Mice; Ondansetron; para-Aminobenzoates; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists | 1997 |
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron | 1997 |
Effects of gastroprokinetic agents on gastroparesis in streptozotocin-induced diabetic rats.
Topics: Animals; Benzamides; Benzimidazoles; Blood Glucose; Cisapride; Diabetes Mellitus, Experimental; Gastric Emptying; Gastrointestinal Motility; Gastroparesis; Granisetron; Male; Morpholines; Ondansetron; Piperidines; Pyrroles; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Vagotomy | 1997 |
Evidence for a 5-HT3 receptor involvement in the facilitation of peristalsis on mucosal application of 5-HT in the guinea pig isolated ileum.
Topics: Animals; Dioxanes; Female; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methiothepin; Mucous Membrane; Ondansetron; Peristalsis; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists | 1997 |
GR205171 blocks apomorphine and amphetamine-induced conditioned taste aversions.
Topics: Amphetamines; Animals; Apomorphine; Avoidance Learning; Conditioning, Classical; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Taste; Tetrazoles | 1998 |
Inhibition of anaesthetic-induced emesis by a NK1 or 5-HT3 receptor antagonist in the house musk shrew, Suncus murinus.
Topics: Anesthesia; Animals; Halothane; Humans; Male; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Shrews; Tetrazoles; Vomiting | 1998 |
Antiemetic effects of Lerisetron in radiation-induced emesis in the dog.
Topics: Animals; Antiemetics; Benzimidazoles; Cobalt Radioisotopes; Dogs; Drug Administration Schedule; Ondansetron; Piperidines; Radiotherapy; Serotonin Antagonists; Vomiting | 1998 |
Emesis induced by inhibitors of type IV cyclic nucleotide phosphodiesterase (PDE IV) in the ferret.
Topics: Animals; Antiemetics; Dose-Response Relationship, Drug; Emetics; Ferrets; Indoles; Molecular Structure; Nitrobenzenes; Ondansetron; Phenylurea Compounds; Phosphodiesterase Inhibitors; Piperidines; Pyridines; Pyrrolidinones; Quinolones; Rolipram; Stereoisomerism; Time Factors; Vomiting | 1999 |
Regional differences in neurogenic signal transduction pathway of cholera toxin-induced fluid, electrolyte and serotonin accumulation in the porcine jejunum.
Topics: Animals; Body Fluids; Cholera Toxin; Dose-Response Relationship, Drug; Electrolytes; Female; Hexamethonium; Jejunum; Nicotinic Antagonists; Ondansetron; Piperidines; Receptors, Neurokinin-1; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Signal Transduction; Substance P; Swine | 2000 |
5-HT inhibits spontaneous contractility of isolated sheep mesenteric lymphatics via activation of 5-HT(4) receptors.
Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Isometric Contraction; Lymphatic System; Methysergide; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sheep | 2000 |
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron | 2000 |
New benzimidazole derivatives: selective and orally active 5-HT3 receptor antagonists.
Topics: 5-Hydroxytryptophan; Administration, Oral; Animals; Aza Compounds; Behavior, Animal; Benzimidazoles; Carbachol; Diarrhea; Dose-Response Relationship, Drug; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Injections, Intraperitoneal; Injections, Intravenous; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Piperidines; Propane; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Serotonin; Serotonin Antagonists | 2003 |
A comparative analysis of the potential of cannabinoids and ondansetron to suppress cisplatin-induced emesis in the Suncus murinus (house musk shrew).
Topics: Animals; Antiemetics; Antineoplastic Agents; Cannabinoids; Cisplatin; Dose-Response Relationship, Drug; Dronabinol; Drug Therapy, Combination; Female; Lithium; Male; Ondansetron; Piperidines; Psychotropic Drugs; Pyrazoles; Rimonabant; Shrews; Vomiting | 2004 |
Action of ondansetron and CP-99,994 to modify behavior and antagonize cisplatin-induced emesis in the ferret.
Topics: Animals; Antiemetics; Behavior, Animal; Cisplatin; Ferrets; Male; Ondansetron; Piperidines; Vomiting | 2005 |
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting | 2005 |
WIN 55,212-2-induced reduction of cocaine hyperlocomotion: possible inhibition of 5-HT(3) receptor function.
Topics: Animals; Benzoxazines; Cocaine; Dose-Response Relationship, Drug; Male; Morpholines; Motor Activity; Naphthalenes; Ondansetron; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Rimonabant; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists | 2005 |
Ondansetron, dexamethasone and an NK1 antagonist block radiation sickness in mice.
Topics: Animals; Antiemetics; Dexamethasone; Drug Therapy, Combination; Male; Mice; Mice, Inbred ICR; Neurokinin-1 Receptor Antagonists; Ondansetron; Pica; Piperidines; Radiation Injuries; Serotonin Antagonists | 2005 |
Action of ondansetron and CP-99,994 on cisplatin-induced emesis and locomotor activity in Suncus murinus (house musk shrew).
Topics: Animals; Antineoplastic Agents; Behavior, Animal; Cisplatin; Female; Motor Activity; Ondansetron; Piperidines; Serotonin Receptor Agonists; Shrews; Vomiting | 2005 |
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors | 2006 |
Luminal hypotonicity increases duodenal mucosal permeability by a mechanism involving 5-hydroxytryptamine.
Topics: Anesthetics, Local; Animals; Cyclooxygenase Inhibitors; Duodenum; Granisetron; Indoles; Indomethacin; Intestinal Mucosa; Lidocaine; Male; Ondansetron; Osmotic Pressure; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Tetrodotoxin; Tropisetron | 2006 |
Differential effects of dexamethasone, ondansetron and a tachykinin NK1 receptor antagonist (GR205171) on cisplatin-induced changes in behaviour, food intake, pica and gastric function in rats.
Topics: Animals; Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Eating; Gastric Emptying; Male; Motor Activity; Nausea; Neurokinin-1 Receptor Antagonists; Ondansetron; Pica; Piperidines; Rats; Rats, Wistar; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Tetrazoles | 2007 |
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin | 2007 |
[Narcolepsy and anesthesia].
Topics: Analgesia, Epidural; Anesthesia, Intravenous; Antiemetics; Benzhydryl Compounds; Chemical and Drug Induced Liver Injury; Clomipramine; Contraindications; Humans; Hypnotics and Sedatives; Intracellular Signaling Peptides and Proteins; Intraoperative Complications; Kidney Pelvis; Modafinil; Narcolepsy; Neuropeptides; Ondansetron; Orexins; Pain, Postoperative; Piperidines; Preanesthetic Medication; Propofol; Remifentanil; Ureteral Obstruction | 2007 |
Urocortin I is present in the enteric nervous system and exerts an excitatory effect via cholinergic and serotonergic pathways in the rat colon.
Topics: Animals; Atropine; Colon; Corticotropin-Releasing Hormone; Dioxanes; Electric Stimulation; Enteric Nervous System; Gastrointestinal Motility; Hexamethonium; Immunohistochemistry; Male; NG-Nitroarginine Methyl Ester; Ondansetron; Peptide Fragments; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Tetrodotoxin; Urocortins | 2007 |
Why no casopitant-only arm?
Topics: Antiemetics; Dose-Response Relationship, Drug; Drug Therapy, Combination; Humans; Ondansetron; Piperazines; Piperidines; Postoperative Nausea and Vomiting; Treatment Outcome | 2011 |
Induction of glucose intolerance by acute administration of rimonabant.
Topics: Administration, Oral; Animals; Benzoxazines; Blood Glucose; Dopamine Antagonists; Eating; Fenclonine; Glucose; Glucose Intolerance; Haloperidol; Hepatocytes; Infusions, Intraventricular; Insulin; Male; Mice; Morpholines; Naphthalenes; Ondansetron; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Dopamine; Receptors, Serotonin; Rimonabant; Serotonin Antagonists | 2012 |
The anticonvulsant effects of SR 57227 on pentylenetetrazole-induced seizure in mice.
Topics: Animals; Anticonvulsants; gamma-Aminobutyric Acid; Hippocampus; Male; Mice, Inbred ICR; Ondansetron; Pentylenetetrazole; Piperidines; Proto-Oncogene Proteins c-fos; Seizures; Survival Analysis | 2014 |
The differential antiemetic properties of GLP-1 receptor antagonist, exendin (9-39) in Suncus murinus (house musk shrew).
Topics: Animals; Antiemetics; Brain; Exenatide; Glucagon-Like Peptide-1 Receptor; Male; Ondansetron; Peptide Fragments; Peptides; Piperidines; Proto-Oncogene Proteins c-fos; Receptors, Glucagon; Shrews; Venoms; Vomiting | 2014 |
Involvement of Descending Serotonergic and Noradrenergic Systems and their Spinal Receptor Subtypes in the Antinociceptive Effect of Dipyrone.
Topics: 5,7-Dihydroxytryptamine; Adrenergic Neurons; Analgesics; Animals; Dipyrone; Dose-Response Relationship, Drug; Injections, Spinal; Ketanserin; Mice; Ondansetron; Oxidopamine; Pain Measurement; Piperidines; Prazosin; Propranolol; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonergic Neurons; Spinal Cord; Sulfonamides; Yohimbine | 2015 |
The role of the AMPA receptor and 5-HT(3) receptor on aggressive behavior and depressive-like symptoms in chronic social isolation-reared mice.
Topics: Aggression; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amygdala; Animals; Depression; Food Preferences; Glutamate Decarboxylase; Hypothalamus; Injections, Intraperitoneal; Male; Mice; Microinjections; Motor Activity; Neurons; Ondansetron; Piperidines; Quinoxalines; Receptors, AMPA; Receptors, Serotonin, 5-HT3; Social Isolation | 2016 |
Postoperative nausea and vomiting (PONV) in outpatient repair of inguinal hernia.
Topics: Adjuvants, Anesthesia; Adolescent; Adult; Aged; Aged, 80 and over; Analgesics, Opioid; Anesthesia, Local; Antiemetics; Deep Sedation; Dexamethasone; Female; Fentanyl; Hernia, Inguinal; Herniorrhaphy; Humans; Male; Middle Aged; Ondansetron; Piperidines; Postoperative Nausea and Vomiting; Preanesthetic Medication; Propofol; Remifentanil; Retrospective Studies; Young Adult | 2018 |
New
Topics: Analgesics; Animals; Behavior, Animal; Capsaicin; Coffee; Disease Models, Animal; Female; Formaldehyde; Glutamic Acid; Hot Temperature; Hyperalgesia; Male; Mice; Naloxone; Narcotic Antagonists; Ondansetron; Pain; Pain Measurement; Piperidines; Pyrazoles; Serotonin | 2018 |