ondansetron and bemesetron

ondansetron has been researched along with bemesetron in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.78)18.7374
1990's31 (86.11)18.2507
2000's4 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD1
Baker, R; Beer, M; Herbert, R; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, GI; Swain, CJ1
Bradley, G; Coleman, J; Rhodes, KF; Taylor, A; Ward, TJ; White, JC1
Bloomquist, W; Cohen, ML; Lacefield, WB; Pfeifer, W; Robertson, DW; Simon, RL1
Baker, R; Beer, M; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, G; Swain, CJ; Watling, K1
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT1
Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC1
Bermudez, J; Fake, CS; Joiner, GF; Joiner, KA; King, FD; Miner, WD; Sanger, GJ1
Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG1
Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Cervo, L; Dalla Valle, F; Fracasso, C; Gemma, S; Goegan, M; Greco, G; Hamon, M; Mennini, T; Morelli, E; Nacci, V; Novellino, E1
Adrien, J; Franc, B; Haj-Dahmane, S; Hamon, M; Jolas, T; Lanfumey, L; Tissier, MH1
Higgins, GA; Joharchi, N; Nguyen, P; Sellers, EM2
Moser, PC1
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
Gifford, AN; Johnson, KM; Yi, SJ1
Gandara, DR; Hesketh, PJ1
Surprenant, A; Vanner, S1
Dyche, J; Giordano, J1
Bountra, C; Dale, TJ; Freeman, AJ; Gardner, CJ; Twissell, DJ1
Allison, K; Arnold, B; Greenshaw, AJ; Ivanová, S; Paetsch, PR; Paslawski, T1
Gietzen, DW; Rogers, QR; Terry-Nathan, VR1
Corrigall, WA; Higgins, GA; Sellers, EM; Wang, Y1
Gietzen, DW; Jiang, JC1
Barrett, JE; Critchett, D; Hu, W; Sokol, PT; Solomon, AJ; Toral, J; Ziai, MR1
Aulakh, CS; Mazzola-Pomietto, P; Murphy, DL1
Cervo, L; Pozzi, L; Samanin, R1
Cottrell, GA; Green, KA; Lambert, JJ1
González, AA; Puig, MM1
Del Río, J; Díez-Ariza, M; Lasheras, B; Ramírez, MJ1
Maksay, G1
Saederup, E; Squires, RF1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Frys, KA; Kalivas, PW; Szumlinski, KK1
De Deurwaerdère, P; Moison, D; Porras, G; Spampinato, U1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1

Reviews

1 review(s) available for ondansetron and bemesetron

ArticleYear
The vomiting reflex and the role of 5-HT3 receptors.
    Anti-cancer drugs, 1993, Volume: 4 Suppl 2

    Topics: Afferent Pathways; Animals; Antiemetics; Antineoplastic Agents; Brain Stem; Chemoreceptor Cells; Ferrets; Humans; Ion Channels; Ondansetron; Postoperative Complications; Radiotherapy; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Solitary Nucleus; Tropanes; Vagus Nerve; Vestibule, Labyrinth; Vomiting

1993

Other Studies

35 other study(ies) available for ondansetron and bemesetron

ArticleYear
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction

1992
Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).
    Journal of medicinal chemistry, 1992, Mar-20, Volume: 35, Issue:6

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Oxazoles; Rats; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction

1992
Novel antagonists of the 5-HT3 receptor. Synthesis and structure-activity relationships of (2-alkoxybenzoyl)ureas.
    Journal of medicinal chemistry, 1992, May-01, Volume: 35, Issue:9

    Topics: Animals; Benzoates; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Rats; Rats, Inbred Strains; Serotonin Antagonists; Structure-Activity Relationship; Urea; Vagus Nerve; X-Ray Diffraction

1992
Zatosetron, a potent, selective, and long-acting 5HT3 receptor antagonist: synthesis and structure-activity relationships.
    Journal of medicinal chemistry, 1992, Jan-24, Volume: 35, Issue:2

    Topics: Animals; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Guinea Pigs; Heart Rate; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Inbred Strains; Serotonin Antagonists; Structure-Activity Relationship; Tropisetron

1992
Novel 5-HT3 antagonists. Indole oxadiazoles.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Electrochemistry; Indicators and Reagents; Indoles; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tropisetron

1991
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes

1990
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1990
5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:7

    Topics: Animals; Antiemetics; Carboxylic Acids; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Indicators and Reagents; Indolizines; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Muscle Contraction; Muscle, Smooth; Pyrazoles; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

1990
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
    Journal of medicinal chemistry, 1998, Jan-29, Volume: 41, Issue:3

    Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

1998
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Blood-Brain Barrier; Brain; Guanidine; Guinea Pigs; Hybrid Cells; In Vitro Techniques; Ligands; Male; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

1999
Central action of 5-HT3 receptor ligands in the regulation of sleep-wakefulness and raphe neuronal activity in the rat.
    Neuropharmacology, 1992, Volume: 31, Issue:6

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electrophysiology; Indoles; Male; Neurons; Ondansetron; Propranolol; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Sleep; Time Factors; Tropanes; Tropisetron; Wakefulness

1992
Effect of the 5-HT3 receptor antagonists, MDL72222 and ondansetron on morphine place conditioning.
    Psychopharmacology, 1992, Volume: 106, Issue:3

    Topics: Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Imidazoles; Male; Morphine; Ondansetron; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tropanes

1992
The effect of 5-HT3 receptor antagonists on the discriminative stimulus effects of amphetamine.
    European journal of pharmacology, 1992, Mar-03, Volume: 212, Issue:2-3

    Topics: Amphetamine; Animals; Discrimination Learning; Imidazoles; Indoles; Male; Ondansetron; Quinolizines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tropanes; Tropisetron

1992
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
Effect of cocaine and 5-HT3 receptor antagonists on 5-HT-induced [3H]dopamine release from rat striatal synaptosomes.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: Animals; Calcium; Cocaine; Corpus Striatum; Dopamine; Female; Imidazoles; Lysergic Acid Diethylamide; Nomifensine; Ondansetron; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Synaptosomes; Tropanes

1991
Effects of 5-HT3 receptor antagonists on behavioural measures of naloxone-precipitated opioid withdrawal.
    Psychopharmacology, 1991, Volume: 105, Issue:3

    Topics: Animals; Behavior, Animal; Chlordiazepoxide; Conditioning, Operant; Drug Implants; Imidazoles; Male; Morphine Dependence; Naloxone; Ondansetron; Pyrimidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Substance Withdrawal Syndrome; Tropanes

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Effects of 5-HT3 receptor antagonists on 5-HT and nicotinic depolarizations in guinea-pig submucosal neurones.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: Acetylcholine; Animals; Cocaine; Curare; Electric Stimulation; Ganglionic Stimulants; Gastric Mucosa; Guinea Pigs; Hexamethonium Compounds; Imidazoles; In Vitro Techniques; Indoles; Iontophoresis; Neuromuscular Depolarizing Agents; Ondansetron; Receptors, Nicotinic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1990
Differential analgesic actions of serotonin 5-HT3 receptor antagonists in the mouse.
    Neuropharmacology, 1989, Volume: 28, Issue:4

    Topics: Analgesics; Animals; Imidazoles; Indoles; Injections, Intraventricular; Male; Mice; Mice, Inbred C3H; Naloxone; Nociceptors; Ondansetron; Pain Measurement; Reaction Time; Serotonin Antagonists; Tropanes; Tropisetron

1989
5HT3 receptor antagonists do not block nicotine induced hyperactivity in rats.
    Psychopharmacology, 1995, Volume: 119, Issue:2

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Granisetron; Haloperidol; Indoles; Male; Motor Activity; Nicotine; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Time Factors; Tropanes; Tropisetron

1995
Serotonin3 antagonists block aversion to saccharin in an amino acid-imbalanced diet.
    The American journal of physiology, 1995, Volume: 268, Issue:5 Pt 2

    Topics: Amino Acids; Animals; Avoidance Learning; Conditioning, Psychological; Diet; Eating; Food Preferences; Indoles; Male; Ondansetron; Rats; Rats, Sprague-Dawley; Saccharin; Serotonin Antagonists; Tropanes; Tropisetron

1995
Influence of 5-HT3 receptor antagonists and the indirect 5-HT agonist, dexfenfluramine, on heroin self-administration in rats.
    Psychopharmacology, 1994, Volume: 114, Issue:4

    Topics: Animals; Conditioning, Operant; Fenfluramine; Food; Heroin; Infusions, Intravenous; Male; Naloxone; Ondansetron; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

1994
Anorectic response to amino acid imbalance: a selective serotonin3 effect?
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:1

    Topics: Amino Acids; Animals; Diet; Eating; Food Preferences; Indoles; Isoleucine; Male; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1994
5-HT3 receptor-independent inhibition of the depolarization-induced 86Rb efflux from human neuroblastoma cells, TE671, by ondansetron.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:7

    Topics: Anti-Anxiety Agents; Benzamides; Benzofurans; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypoglycemic Agents; Indazoles; Indoles; Neuroblastoma; Neurotoxins; Ondansetron; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Rubidium Radioisotopes; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tropanes; Tropisetron; Tumor Cells, Cultured

1995
Temperature, food intake, and locomotor activity effects of a 5-HT3 receptor agonist and two 5-HT3 receptor antagonists in rats.
    Psychopharmacology, 1995, Volume: 121, Issue:4

    Topics: Animals; Biguanides; Body Temperature; Dose-Response Relationship, Drug; Eating; Locomotion; Male; Ondansetron; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

1995
5-HT3 receptor antagonists do not modify cocaine place conditioning or the rise in extracellular dopamine in the nucleus accumbens of rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 55, Issue:1

    Topics: Animals; Cocaine; Conditioning, Operant; Dopamine; Dopamine Uptake Inhibitors; Extracellular Space; Indoles; Male; Microdialysis; Nucleus Accumbens; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Tropanes; Tropisetron

1996
Ligand-gated ion channels opened by 5-HT in molluscan neurones.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Calcium; Convulsants; Dose-Response Relationship, Drug; Electrophysiology; GTP-Binding Proteins; Helix, Snails; Ion Channel Gating; Ion Channels; Ketanserin; Neurons; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Strychnine; Tropanes

1996
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron

1997
Differential interaction between 5-HT3 receptors and GABAergic neurons inhibiting acetylcholine release in rat entorhinal cortex slices.
    Brain research, 1998, Aug-10, Volume: 801, Issue:1-2

    Topics: Acetylcholine; Animals; Barium; Bicuculline; Chloride Channels; Culture Techniques; Entorhinal Cortex; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neurons; Ondansetron; Perfusion; Potassium Channel Blockers; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Tetraethylammonium; Tropanes

1998
Bidirectional allosteric modulation of strychnine-sensitive glycine receptors by tropeines and 5-HT3 serotonin receptor ligands.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: Allosteric Regulation; Animals; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Glycine; Granisetron; Indoles; Ligands; Male; Medulla Oblongata; Ondansetron; Pons; Rats; Rats, Wistar; Receptors, Glycine; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Strychnine; Tropanes; Tropisetron; Tubocurarine

1998
Clozapine's antipsychotic effects do not depend on blockade of 5-HT3 receptors.
    Neurochemical research, 1999, Volume: 24, Issue:5

    Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; Drug Interactions; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Ondansetron; Quinacrine; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Sulfur Radioisotopes; Tropanes

1999
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
Pretreatment with serotonin 5-HT(3) receptor antagonists produces no observable blockade of long-term motor sensitization to cocaine in rats.
    Psychopharmacology, 2003, Volume: 165, Issue:4

    Topics: Anesthetics, Local; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Fluphenazine; Injections; Male; Motor Activity; Ondansetron; Oxazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Tropanes

2003
Conditional involvement of striatal serotonin3 receptors in the control of in vivo dopamine outflow in the rat striatum.
    The European journal of neuroscience, 2003, Volume: 17, Issue:4

    Topics: Amphetamine; Analgesics, Opioid; Animals; Brain Chemistry; Central Nervous System Stimulants; Chromatography, High Pressure Liquid; Citalopram; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Interactions; Electrochemistry; Haloperidol; Male; Microdialysis; Morphine; Ondansetron; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT3 Receptor Antagonists; Tropanes

2003
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005