Page last updated: 2024-09-03

omega-n-methylarginine and propranolol

omega-n-methylarginine has been researched along with propranolol in 20 studies

Compound Research Comparison

Studies
(omega-n-methylarginine)
Trials
(omega-n-methylarginine)
Recent Studies (post-2010)
(omega-n-methylarginine)
Studies
(propranolol)
Trials
(propranolol)
Recent Studies (post-2010) (propranolol)
4,41134433633,3103,4063,218

Protein Interaction Comparison

ProteinTaxonomyomega-n-methylarginine (IC50)propranolol (IC50)
Beta-1 adrenergic receptor Cavia porcellus (domestic guinea pig)0.0347
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.294
Cytochrome P450 1A2Homo sapiens (human)4
Beta-2 adrenergic receptorHomo sapiens (human)0.0114
Beta-1 adrenergic receptorHomo sapiens (human)0.0575
5-hydroxytryptamine receptor 1AHomo sapiens (human)3.9811
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.012
Cytochrome P450 2D6Homo sapiens (human)2.9706
Beta-3 adrenergic receptorHomo sapiens (human)0.0493
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0288
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.012
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0827
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0288
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.012
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.466
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.294
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.243
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0288
Sodium-dependent serotonin transporterHomo sapiens (human)0.38
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.342
5-hydroxytryptamine receptor 6Homo sapiens (human)3.065
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0288
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)2.828
Sodium channel protein type 5 subunit alphaHomo sapiens (human)2.1
Sodium/bile acid cotransporterHomo sapiens (human)5.5
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0288
GABA theta subunitRattus norvegicus (Norway rat)0.0288
Sigma non-opioid intracellular receptor 1Homo sapiens (human)2.87
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0288

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (60.00)18.2507
2000's7 (35.00)29.6817
2010's1 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, PJ; Crawley, DE; Evans, TW; Liu, SF1
Kobayashi, D; Okabe, E; Ozono, S; Todoki, K1
Demedts, MG; Pype, JL; Verleden, GM1
Leblanc, PH; Robinson, NE; Wang, Z; Yu, M1
Bayguinov, O; Sanders, KM1
Anfossi, G; Cavalot, F; Hahn, AW; Massucco, P; Mattiello, L; Mularoni, EM; Trovati, M1
Chang, PC; van Veen, S1
Hucks, D; Priest, RM; Ward, JP1
Choate, JK; Paterson, DJ; Sears, CE1
Hayashi, H; Sanae, F1
Bohrer, A; Hsu, FF; Ma, Z; Ramanadham, S; Turk, J1
Brennan, AJ; Campbell, KB; Harding, JW; Slinker, BK; Wu, Y1
Halliwill, JR; Joyner, MJ; Minson, CT; Nauss, LA; Reed, AS; Torp, KD; Tschakovsky, ME1
Brett, SE; Chowienczyk, PJ; Coltart, DJ; Kneale, BJ; Ritter, JM1
Hiraga, H; Okubo, T; Okumura, K; Suto, N; Yamamoto, T; Yoshida, IM1
Duplain, H; Lepori, M; Nicod, P; Sartori, C; Scherrer, U1
D'Agostino, B; Falciani, M; Filippelli, A; Mazzeo, F; Nobili, B; Rinaldi, B; Rossi, F; Rossi, S1
Colledge, WH; Grace, AA; Joseph, SS; Kaumann, AJ; Lynham, JA; Molenaar, P1
Ardilouze, JL; Currie, JM; Fielding, BA; Frayn, KN; Karpe, F1
Crecelius, AR; Dinenno, FA; Hearon, CM; Kirby, BS; Larson, DG; Luckasen, GJ1

Trials

3 trial(s) available for omega-n-methylarginine and propranolol

ArticleYear
Prostaglandins and nitric oxide mediate insulin-induced vasodilation in the human forearm.
    Cardiovascular research, 1997, Volume: 34, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Forearm; Humans; Indomethacin; Insulin; Isoproterenol; Male; Nitric Oxide Synthase; omega-N-Methylarginine; Propranolol; Vascular Resistance; Vasodilation

1997
Interaction between cholinergic and nitrergic vasodilation: a novel mechanism of blood pressure control.
    Cardiovascular research, 2001, Volume: 51, Issue:4

    Topics: Adrenergic beta-Antagonists; Adult; Arginine; Atropine; Cardiac Output; Enzyme Inhibitors; Female; Hemodynamics; Humans; Leg; Male; Muscarinic Antagonists; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Propranolol; Regional Blood Flow; Statistics, Nonparametric; Vasoconstrictor Agents

2001
Contracting human skeletal muscle maintains the ability to blunt α1 -adrenergic vasoconstriction during KIR channel and Na(+) /K(+) -ATPase inhibition.
    The Journal of physiology, 2015, Jun-15, Volume: 593, Issue:12

    Topics: Adenosine; Adult; Barium Compounds; Brachial Artery; Chlorides; Exercise; Female; Forearm; Hand Strength; Humans; Ketorolac; Male; Muscle Contraction; Muscle, Skeletal; omega-N-Methylarginine; Ouabain; Potassium Channels, Inwardly Rectifying; Propranolol; Receptors, Adrenergic, alpha-1; Regional Blood Flow; Sodium-Potassium-Exchanging ATPase; Vasoconstriction; Young Adult

2015

Other Studies

17 other study(ies) available for omega-n-methylarginine and propranolol

ArticleYear
Endothelium-dependent nonadrenergic, noncholinergic neural relaxation in guinea pig pulmonary artery.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Acetamides; Adenosine Triphosphate; Animals; Arginine; Atropine; Autonomic Nervous System; Capsaicin; Chymotrypsin; Drug Interactions; Endothelium, Vascular; Guinea Pigs; In Vitro Techniques; Indomethacin; Lipoxygenase Inhibitors; Male; Muscle Contraction; Muscle, Smooth, Vascular; omega-N-Methylarginine; Phenyl Ethers; Propranolol; Prostaglandin Endoperoxides, Synthetic; Pulmonary Artery; Vasoactive Intestinal Peptide

1992
Calcitonin gene-related peptide mediated neurogenic vasorelaxation in the isolated canine lingual artery.
    Japanese journal of pharmacology, 1995, Volume: 67, Issue:4

    Topics: Animals; Arginine; Benzopyrans; Calcitonin Gene-Related Peptide; Capsaicin; Cromakalim; Dogs; Electric Stimulation; Female; Glyburide; Humans; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; omega-N-Methylarginine; Peptide Fragments; Potassium Channel Blockers; Potassium Channels; Propranolol; Pyrroles; Substance P; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Vasoconstriction; Vasodilator Agents

1995
Furosemide and bumetanide, but not nedocromil sodium, modulate nonadrenergic relaxation in guinea pig trachea in vitro.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Animals; Arginine; Atropine; Bumetanide; Chymotrypsin; Drug Therapy, Combination; Electric Stimulation; Female; Furosemide; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Nedocromil; Nitric Oxide; Nitroprusside; omega-N-Methylarginine; Premedication; Propranolol; Trachea; Vasoactive Intestinal Peptide

1994
Inhibitory nerve distribution and mediation of NANC relaxation by nitric oxide in horse airways.
    Journal of applied physiology (Bethesda, Md. : 1985), 1994, Volume: 76, Issue:1

    Topics: Animals; Arginine; Atropine; Autonomic Nervous System; Bronchi; Electric Stimulation; Horses; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; omega-N-Methylarginine; Parasympathetic Nervous System; Propranolol; Respiratory Physiological Phenomena; Respiratory System; Trachea

1994
Role of nitric oxide as an inhibitory neurotransmitter in the canine pyloric sphincter.
    The American journal of physiology, 1993, Volume: 264, Issue:5 Pt 1

    Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Arginine; Cyclic GMP; Dogs; Duodenum; Electric Stimulation; Female; Gastric Mucosa; In Vitro Techniques; Intercellular Junctions; Intestinal Mucosa; Male; Membrane Potentials; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; omega-N-Methylarginine; Oxyhemoglobins; Phentolamine; Propranolol; Purinones; Pylorus; Stomach; Tetrodotoxin

1993
Studies on the influence of insulin on cyclic adenosine monophosphate in human vascular smooth muscle cells: dependence on cyclic guanosine monophosphate and modulation of catecholamine effects.
    Diabetologia, 1996, Volume: 39, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Analysis of Variance; Arterioles; Cells, Cultured; Cyclic AMP; Cyclic GMP; Epinephrine; Humans; Insulin; Isoproterenol; Kinetics; Methylene Blue; Muscle, Smooth, Vascular; Norepinephrine; omega-N-Methylarginine; Propranolol; Receptors, Adrenergic, beta; Recombinant Proteins; Yohimbine

1996
Noradrenaline, beta-adrenoceptor mediated vasorelaxation and nitric oxide in large and small pulmonary arteries of the rat.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Dinoprost; Dose-Response Relationship, Drug; Isoproterenol; Male; Nitric Oxide; Nitric Oxide Synthase; Norepinephrine; omega-N-Methylarginine; Oxytocics; Propanolamines; Propranolol; Pulmonary Artery; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasoconstriction; Vasoconstrictor Agents; Vasodilation

1997
Effect of nitric oxide synthase inhibition on the sympatho-vagal contol of heart rate.
    Journal of the autonomic nervous system, 1998, Aug-27, Volume: 73, Issue:1

    Topics: Adrenergic Fibers; Animals; Arginine; Enzyme Inhibitors; Guinea Pigs; Heart Atria; Heart Rate; Indazoles; Isoproterenol; Male; Neural Inhibition; Nitric Oxide Synthase; Nitroarginine; omega-N-Methylarginine; Polymethacrylic Acids; Propranolol; Rabbits; Sympatholytics; Sympathomimetics; Vagus Nerve

1998
Effects of adrenergic and nitrergic blockade on theophylline-induced increase in peripheral blood flow in rat ear.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:3

    Topics: Acetylcholine; Adrenergic Agents; Animals; Atropine; Blood Pressure; Ear; Enzyme Inhibitors; Heart Rate; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitroarginine; omega-N-Methylarginine; Propranolol; Rats; Rats, Wistar; Regional Blood Flow; Reserpine; Theophylline

1998
Studies of the role of group VI phospholipase A2 in fatty acid incorporation, phospholipid remodeling, lysophosphatidylcholine generation, and secretagogue-induced arachidonic acid release in pancreatic islets and insulinoma cells.
    The Journal of biological chemistry, 1999, May-14, Volume: 274, Issue:20

    Topics: Animals; Arachidonic Acid; Cricetinae; Enzyme Inhibitors; Ethylmaleimide; Fatty Acids; Group VI Phospholipases A2; Insulinoma; Interleukin-1; Islets of Langerhans; Lysophosphatidylcholines; Male; Naphthalenes; omega-N-Methylarginine; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Phospholipids; Propranolol; Pyrones; Rats; Rats, Sprague-Dawley; Tumor Cells, Cultured

1999
Angiotensin IV has mixed effects on left ventricle systolic function and speeds relaxation.
    Cardiovascular research, 1999, Volume: 42, Issue:3

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Animals; Linear Models; Male; Nitric Oxide Synthase; omega-N-Methylarginine; Perfusion; Propranolol; Rabbits; Random Allocation; Receptors, Angiotensin; Systole; Ventricular Function, Left

1999
Skeletal muscle vasodilatation during sympathoexcitation is not neurally mediated in humans.
    The Journal of physiology, 2000, May-15, Volume: 525 Pt 1

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Blood Pressure; Epinephrine; Female; Forearm; Hand; Humans; Male; Muscle Fatigue; Muscle, Skeletal; Nitric Oxide; omega-N-Methylarginine; Plethysmography; Propranolol; Regional Blood Flow; Stellate Ganglion; Sympathetic Nervous System; Vasoconstriction; Vasodilation

2000
Gender differences in sensitivity to adrenergic agonists of forearm resistance vasculature.
    Journal of the American College of Cardiology, 2000, Volume: 36, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Albuterol; Blood Flow Velocity; Brachial Artery; Enzyme Inhibitors; Female; Forearm; Humans; Injections, Intra-Arterial; Male; Nitric Oxide Synthase; Nitroprusside; Norepinephrine; omega-N-Methylarginine; Plethysmography; Propranolol; Receptors, Adrenergic, beta-2; Reference Values; Sex Characteristics; Substance P; Vascular Resistance; Vasodilation; Vasodilator Agents; Verapamil

2000
Nitric oxide donor FK409 and 8-bromoguanosine-cyclic monophosphate attenuate cardiac contractility assessed by Emax.
    Fundamental & clinical pharmacology, 2001, Volume: 15, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Coronary Circulation; Cyclic GMP; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Myocardial Contraction; Myocardium; Nitric Oxide Donors; Nitro Compounds; omega-N-Methylarginine; Papaverine; Propranolol; Vasodilation; Vasodilator Agents; Ventricular Function, Left

2001
Effects of nebivolol on human platelet aggregation.
    Journal of cardiovascular pharmacology, 2001, Volume: 38, Issue:6

    Topics: Adenosine Diphosphate; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Arginine; Benzopyrans; Blood Platelets; Carbazoles; Carvedilol; Collagen; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Ethanolamines; Humans; Male; Nebivolol; Nitric Oxide Synthase; omega-N-Methylarginine; Platelet Aggregation; Platelet Aggregation Inhibitors; Propanolamines; Propranolol; Vasodilator Agents

2001
Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Animals; Binding Sites; CHO Cells; Cricetinae; Cyclic AMP; Drug Interactions; Drug Resistance; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; omega-N-Methylarginine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Recombinant Proteins; Stereoisomerism; Sympathomimetics

2003
Nitric oxide and beta-adrenergic stimulation are major regulators of preprandial and postprandial subcutaneous adipose tissue blood flow in humans.
    Circulation, 2004, Jan-06, Volume: 109, Issue:1

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Eating; Female; Glucose; Humans; Infusions, Parenteral; Male; Middle Aged; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Phentolamine; Propranolol; Receptors, Adrenergic, beta; Regional Blood Flow; Xenon Radioisotopes; Yohimbine

2004