Page last updated: 2024-09-04

olmesartan and tacrolimus

olmesartan has been researched along with tacrolimus in 4 studies

Compound Research Comparison

Studies
(olmesartan)
Trials
(olmesartan)
Recent Studies (post-2010)
(olmesartan)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
84118555417,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomyolmesartan (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Andricopulo, AD; Moda, TL; Montanari, CA1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Al-Harbi, MM; Al-Harbi, NO; Alabidy, AD; Almukhallafi, AF; Imam, F; Iqbal, M; Nadeem, A; Sayed-Ahmed, MM1
Al-Harbi, MM; Al-Harbi, NO; Al-Hosaini, KA; Bahashwan, S; Imam, F; Iqbal, M; Nadeem, A; Rahman, S1

Other Studies

4 other study(ies) available for olmesartan and tacrolimus

ArticleYear
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Olmesartan attenuates tacrolimus-induced biochemical and ultrastructural changes in rat kidney tissue.
    BioMed research international, 2014, Volume: 2014

    Topics: Angiotensin II Type 1 Receptor Blockers; Animals; Calcineurin Inhibitors; Imidazoles; Kidney Diseases; Kidney Tubules, Proximal; Male; Mitochondria; Podocytes; Rats; Rats, Wistar; Tacrolimus; Tetrazoles

2014
Protection against tacrolimus-induced cardiotoxicity in rats by olmesartan and aliskiren.
    Toxicology mechanisms and methods, 2014, Volume: 24, Issue:9

    Topics: Amides; Animals; Fumarates; Heart; Imidazoles; Immunosuppressive Agents; Male; Myocardium; Rats; Rats, Wistar; Tacrolimus; Tetrazoles

2014