Page last updated: 2024-09-04

olmesartan and pioglitazone

olmesartan has been researched along with pioglitazone in 5 studies

Compound Research Comparison

Studies
(olmesartan)
Trials
(olmesartan)
Recent Studies (post-2010)
(olmesartan)
Studies
(pioglitazone)
Trials
(pioglitazone)
Recent Studies (post-2010) (pioglitazone)
8411855544,3388242,277

Protein Interaction Comparison

ProteinTaxonomyolmesartan (IC50)pioglitazone (IC50)
CDGSH iron-sulfur domain-containing protein 1Rattus norvegicus (Norway rat)1
Bile salt export pumpRattus norvegicus (Norway rat)2
Peroxisome proliferator-activated receptor gammaRattus norvegicus (Norway rat)0.7
Bile salt export pumpHomo sapiens (human)0.337
Carbonic anhydrase 2Homo sapiens (human)0.114
Steryl-sulfataseHomo sapiens (human)0.8
Peroxisome proliferator-activated receptor alphaMus musculus (house mouse)1.15
Amine oxidase [flavin-containing] BHomo sapiens (human)0.298
Peroxisome proliferator-activated receptor gammaHomo sapiens (human)3.0379
Peroxisome proliferator-activated receptor gammaMus musculus (house mouse)0.7
CDGSH iron-sulfur domain-containing protein 2Homo sapiens (human)4.8
CDGSH iron-sulfur domain-containing protein 1Homo sapiens (human)8.65

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Ekins, S; Williams, AJ; Xu, JJ1
Honda, K; Izumi, T; Miyaji, Y; Nakayama, S; Okazaki, O; Okudaira, N; Shiosakai, K; Sugiyama, D; Suzuki, W; Takakusa, H; Watanabe, A1
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY1
Gust, R; Obexer, P; Salcher, S; Schoepf, AM1
Bhaumik, U; Chakraborty, US; Chatterjee, B; Pal, TK; Roy, B; Sarkar, AK; Sengupta, P1

Other Studies

5 other study(ies) available for olmesartan and pioglitazone

ArticleYear
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Combination of GSH trapping and time-dependent inhibition assays as a predictive method of drugs generating highly reactive metabolites.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:7

    Topics: Glutathione; Pharmacology; Sulfur Radioisotopes

2011
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
    Chemical research in toxicology, 2012, Oct-15, Volume: 25, Issue:10

    Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding

2012
Identification and development of non-cytotoxic cell death modulators: Impact of sartans and derivatives on PPARĪ³ activation and on growth of imatinib-resistant chronic myelogenous leukemia cells.
    European journal of medicinal chemistry, 2020, Jun-01, Volume: 195

    Topics: Animals; Cell Death; Cell Proliferation; Chlorocebus aethiops; COS Cells; Drug Design; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; PPAR gamma; Structure-Activity Relationship; Telmisartan

2020
Development and validation of an LC-ESI-MS/MS method for simultaneous quantitation of olmesartan and pioglitazone in rat plasma and its pharmacokinetic application.
    Biomedical chromatography : BMC, 2010, Volume: 24, Issue:12

    Topics: Angiotensin II Type 1 Receptor Blockers; Animals; Chromatography, High Pressure Liquid; Imidazoles; Male; Pioglitazone; Rats; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Tetrazoles; Thiazolidinediones

2010