Page last updated: 2024-09-04

olmesartan and enalapril

olmesartan has been researched along with enalapril in 7 studies

Compound Research Comparison

Studies
(olmesartan)
Trials
(olmesartan)
Recent Studies (post-2010)
(olmesartan)
Studies
(enalapril)
Trials
(enalapril)
Recent Studies (post-2010) (enalapril)
8411855546,3111,924859

Protein Interaction Comparison

ProteinTaxonomyolmesartan (IC50)enalapril (IC50)
Angiotensin-converting enzyme Homo sapiens (human)0.3536
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)2.7083
Type-2 angiotensin II receptorRattus norvegicus (Norway rat)1.2
Angiotensin-converting enzymeRattus norvegicus (Norway rat)0.14
Angiotensin-converting enzyme 2 Homo sapiens (human)0.14

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (42.86)29.6817
2010's4 (57.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andricopulo, AD; Moda, TL; Montanari, CA1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Carl-McGrath, S; Ebert, MP; Lendeckel, U; Röcken, C1
Agabiti-Rosei, E; Assanelli, D; Boari, GE; De Ciuceis, C; Favero, G; Flati, V; Martinotti, S; Paiardi, S; Pasini, E; Platto, C; Porteri, E; Rezzani, R; Rizzoni, D; Rodella, LF; Speca, S; Toniato, E1
Carvalho-Tavares, J; Castro-Faria Neto, H; Estato, V; Freitas, FS; Lessa, MA; Obadia, N; Reis, P; Tibiriçá, E1
Angeloni, E; Lombardo, P; Pirelli, M; Refice, S; Vitaterna, A1
Fukuda, K; Iwanaga, S; Mahara, K; Murata, M; Tsugu, T1

Reviews

2 review(s) available for olmesartan and enalapril

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
Long-Term Survival on Medical Therapy Alone after Blunt-Trauma Aortic Regurgitation: Report of a New Case with Summary of 95 Others.
    Texas Heart Institute journal, 2016, Volume: 43, Issue:5

    Topics: Accidents, Traffic; Adolescent; Adult; Aged; Aged, 80 and over; Angiotensin II Type 1 Receptor Blockers; Angiotensin-Converting Enzyme Inhibitors; Aortic Valve; Aortic Valve Insufficiency; Drug Therapy, Combination; Echocardiography, Doppler, Color; Echocardiography, Transesophageal; Enalapril; Female; Heart Injuries; Humans; Imidazoles; Male; Middle Aged; Survivors; Tetrazoles; Time Factors; Treatment Outcome; Wounds, Nonpenetrating; Young Adult

2016

Other Studies

5 other study(ies) available for olmesartan and enalapril

ArticleYear
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Expression of the local angiotensin II system in gastric cancer may facilitate lymphatic invasion and nodal spread.
    Cancer biology & therapy, 2007, Volume: 6, Issue:8

    Topics: Adult; Aged; Aged, 80 and over; Angiotensin II Type 2 Receptor Blockers; Apoptosis; Cell Line, Tumor; Cell Movement; Cell Proliferation; Enalapril; Female; Gene Expression Regulation, Neoplastic; Genotype; Humans; Imidazoles; Immunohistochemistry; Lymphatic Metastasis; Male; Middle Aged; Neoplasm Invasiveness; Peptidyl-Dipeptidase A; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Reverse Transcriptase Polymerase Chain Reaction; Stomach Neoplasms; Tetrazoles

2007
Angiotensin receptor blockers improve insulin signaling and prevent microvascular rarefaction in the skeletal muscle of spontaneously hypertensive rats.
    Journal of hypertension, 2008, Volume: 26, Issue:8

    Topics: Adaptor Proteins, Signal Transducing; Angiotensin II Type 1 Receptor Blockers; Angiotensin-Converting Enzyme Inhibitors; Animals; Capillaries; Enalapril; Glucose Transporter Type 4; Hypertension; Imidazoles; Insulin; Insulin Receptor Substrate Proteins; Insulin Resistance; Male; Myocardium; Quadriceps Muscle; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Insulin; Renin-Angiotensin System; Signal Transduction; Tetrazoles; Transcription Factors

2008
Blockade of the renin-angiotensin system improves cerebral microcirculatory perfusion in diabetic hypertensive rats.
    Microvascular research, 2013, Volume: 87

    Topics: Angiotensin II Type 1 Receptor Blockers; Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Arterial Pressure; Blood Glucose; Brain; Capillaries; Cerebrovascular Circulation; Cerebrovascular Disorders; Coronary Circulation; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Diet, High-Fat; Enalapril; Heart Ventricles; Hypertension; Imidazoles; Insulin; Leukocyte Rolling; Male; Microcirculation; Microscopy, Fluorescence; Microscopy, Video; Muscle, Skeletal; Oxidative Stress; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Renin-Angiotensin System; Streptozocin; Tetrazoles

2013
Single-pill combination therapy in the initial treatment of marked hypertension: a propensity-matched analysis.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2015, Volume: 37, Issue:5

    Topics: Amlodipine; Antihypertensive Agents; Benzimidazoles; Benzoates; Blood Pressure; Dihydropyridines; Dose-Response Relationship, Drug; Drug Combinations; Enalapril; Female; Humans; Hydrochlorothiazide; Hypertension; Imidazoles; Male; Middle Aged; Perindopril; Propensity Score; Ramipril; Retrospective Studies; Risk Factors; Telmisartan; Tetrazoles

2015