ns 2028 and oxadiazoles

ns 2028 has been researched along with oxadiazoles in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (16.67)18.2507
2000's13 (43.33)29.6817
2010's11 (36.67)24.3611
2020's1 (3.33)2.80

Authors

AuthorsStudies
Axelsson, O; Bang, L; Busse, R; Drejer, J; Moldt, P; Mülsch, A; Nielsen-Kudsk, JE; Olesen, SP1
Brüne, B; Callsen, D; Pfeilschifter, J1
Aldershvile, J; Bauersachs, J; Busse, R; Fleming, I; Schäfer, A; Scholz, D1
Aldershvile, J; Bang, L; Boesgaard, S; Gruhn, N; Nielsen-Kudsk, JE; Olesen, SP; Theilgaard, SA1
Aldershvile, J; Bang, L; Boesgaard, S; Nielsen-Kudsk, JE; Vejlstrup, NG1
Brüne, B; Fandrey, J; Sandau, KB1
Kellum, JM; Stoner, MC1
Trakranrungsie, N; Will, JA1
Fujimura, S; Hisa, H; Nakamura, K; Satoh, S; Suzuki-Kusaba, M; Tanioka, H; Yoshida, M1
Furneaux, H; Kloss, S; Mülsch, A1
Chan, SL; Fiscus, RR1
Busse, R; Fleming, I; Randriamboavonjy, V; Schrader, J1
Berg, A; Ericson, AC; Grenegård, M; Redéen, S; Sjöstrand, SE1
Fung, YK; Liu, X; Pahan, K; Roy, A1
Jang, Y; Mueller, RA; Norfleet, EA; Wang, H; Xi, J; Xu, Z1
Detmar, M; Drinnenberg, I; Huggenberger, R; Kajiya, K; Ma, B1
Haramis, G; Koutsilieris, M; Papapetropoulos, A; Pyriochou, A; Roussos, C; Zhou, Z1
Dombkowski, RA; Gao, Y; Motterlini, R; Olson, KR; Whitfield, NL1
Filippi, S; Giannis, A; Loutrari, H; Morbidelli, L; Papapetropoulos, A; Pyriochou, A; Roussos, C; Stössel, A; Vasileiadis, I; Waltenberger, J; Zhou, Z; Ziche, M1
Au, AL; Félétou, M; Kwan, YW; Leung, SW; Liang, CF; Man, RY; Ng, KF; Vanhoutte, PM1
Ahtesham, AK; Akaike, T; Ida, T; Ihara, H; Kasamatsu, S; Kunieda, K; Okamoto, T; Sawa, T1
Buck, J; Hess, KC; Levin, LR; Ramos-Espiritu, LS1
Hoffmann, C; Hoffmann, LS; Keim, Y; Schmidt, HH; Schmidt, PM; Stasch, JP1
Meng, Z; Zhang, Q1
Bilzer, M; Gerbes, AL; Gmelin, L; Göke, B; Steib, CJ1
Friebe, A; Gambaryan, S; Groneberg, D; Lies, B1
Fang, F; Liu, X; Pan, M; Qu, J; Tao, Y; Wu, H; Yan, T; Zhou, X1
Artinian, L; Estes, S; Rehder, V1
Chuang, VTG; Ikeda, M; Ikeda, T; Ishida, T; Ishima, Y; Kinoshita, R; Maruyama, T; Otagiri, M; Watanabe, H1
Krutsenko, Y; Lezgyieva, K; Martin, E; Sharina, I1

Other Studies

30 other study(ies) available for ns 2028 and oxadiazoles

ArticleYear
Characterization of NS 2028 as a specific inhibitor of soluble guanylyl cyclase.
    British journal of pharmacology, 1998, Volume: 123, Issue:2

    Topics: Animals; Cattle; Cells, Cultured; Cerebellum; Cyclic GMP; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Guinea Pigs; Heme; Humans; In Vitro Techniques; Kinetics; Male; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Oxadiazoles; Oxazines; Rabbits; Solubility; Spectrophotometry; Structure-Activity Relationship; Swine; Umbilical Veins

1998
Rapid and delayed p42/p44 mitogen-activated protein kinase activation by nitric oxide: the role of cyclic GMP and tyrosine phosphatase inhibition.
    Journal of immunology (Baltimore, Md. : 1950), 1998, Nov-01, Volume: 161, Issue:9

    Topics: Acetylcysteine; Animals; Biphenyl Compounds; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Cyclic GMP; Enzyme Activation; Free Radical Scavengers; Glomerular Mesangium; Glutathione; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Molsidomine; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitroso Compounds; Onium Compounds; Oxadiazoles; Oxazines; Phosphorylation; Protein Processing, Post-Translational; Protein Tyrosine Phosphatases; Rats; S-Nitrosoglutathione; Second Messenger Systems

1998
Isometric contraction induces the Ca2+-independent activation of the endothelial nitric oxide synthase.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Feb-02, Volume: 96, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Aorta, Thoracic; Benzoquinones; Calcium; Calmodulin; Cells, Cultured; Cyclic GMP; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Female; Genistein; Hydroquinones; Imidazoles; In Vitro Techniques; Indoles; Isometric Contraction; Lactams, Macrocyclic; Male; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroarginine; Oxadiazoles; Oxazines; Quinones; Rabbits; Rifabutin; Staurosporine

1999
Vascular smooth muscle contraction is an independent regulator of endothelial nitric oxide production.
    Scandinavian cardiovascular journal : SCJ, 1999, Volume: 33, Issue:2

    Topics: Animals; Endothelium, Vascular; Enzyme Inhibitors; Male; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Oxazines; Rats; Rats, Wistar; Vasomotor System

1999
Nitroglycerin-mediated vasorelaxation is modulated by endothelial calcium-activated potassium channels.
    Cardiovascular research, 1999, Aug-15, Volume: 43, Issue:3

    Topics: Animals; Calcium; Coronary Vessels; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Ion Channel Gating; Male; Nitroglycerin; Oxadiazoles; Oxazines; Peptides; Perfusion; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Regional Blood Flow; Regression Analysis; Swine; Vasodilator Agents

1999
Accumulation of HIF-1alpha under the influence of nitric oxide.
    Blood, 2001, Feb-15, Volume: 97, Issue:4

    Topics: Animals; Benzoates; Cell Hypoxia; Cell Line; Cobalt; Coculture Techniques; Deferoxamine; DNA-Binding Proteins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Glutathione; Guanylate Cyclase; Hydrazines; Hypoxia-Inducible Factor 1; Hypoxia-Inducible Factor 1, alpha Subunit; Imidazoles; Inflammation; Kidney Tubules, Proximal; Macrophage Activation; Macrophages; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitrogen Oxides; Nitroso Compounds; Nuclear Proteins; Oxadiazoles; Oxazines; S-Nitrosoglutathione; Spermine; Swine; Transcription Factors

2001
Both serotonin and a nitric-oxide donor cause chloride secretion in rat colonocytes by stimulating cGMP.
    Surgery, 2001, Volume: 130, Issue:2

    Topics: Animals; Chlorides; Colon; Cyclic GMP; Enzyme Inhibitors; Guanylate Cyclase; Male; Nitric Oxide Donors; Oxadiazoles; Oxazines; Polyamines; Rats; Rats, Sprague-Dawley; Serotonin

2001
Comparative vasodilation of peroxynitrite and 3-morpholinosydnonimine.
    Life sciences, 2001, Oct-05, Volume: 69, Issue:20

    Topics: Adenine; Animals; Benzoates; Cattle; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Enzyme Inhibitors; Female; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Mammary Arteries; Molsidomine; Muscle Relaxation; Muscle, Smooth, Vascular; Oxadiazoles; Oxazines; Oxidants; Peroxynitrous Acid; Vasodilation; Vasodilator Agents

2001
Facilitatory role of NO in neural norepinephrine release in the rat kidney.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 282, Issue:5

    Topics: Animals; Benzoates; Cyclic GMP; Electric Stimulation; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Indazoles; Kidney; Male; Nervous System; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroarginine; Norepinephrine; Oxadiazoles; Oxazines; Perfusion; Pressure; Rats; Rats, Wistar

2002
Post-transcriptional regulation of soluble guanylyl cyclase expression in rat aorta.
    The Journal of biological chemistry, 2003, Jan-24, Volume: 278, Issue:4

    Topics: 3' Untranslated Regions; Animals; Antigens, Surface; Aorta; Base Sequence; Blotting, Northern; Blotting, Western; Cell Nucleus; Cells, Cultured; Dactinomycin; Down-Regulation; ELAV Proteins; ELAV-Like Protein 1; Enzyme Activators; Guanylate Cyclase; Indazoles; Male; Molecular Sequence Data; Muscle, Smooth; Nucleic Acid Synthesis Inhibitors; Oxadiazoles; Oxazines; Poly A; Protein Binding; Protein Structure, Tertiary; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; RNA; RNA Processing, Post-Transcriptional; RNA-Binding Proteins; RNA, Messenger; RNA, Small Interfering; Soluble Guanylyl Cyclase; Time Factors; Transcription, Genetic; Transfection

2003
Guanylyl cyclase inhibitors NS2028 and ODQ and protein kinase G (PKG) inhibitor KT5823 trigger apoptotic DNA fragmentation in immortalized uterine epithelial cells: anti-apoptotic effects of basal cGMP/PKG.
    Molecular human reproduction, 2003, Volume: 9, Issue:12

    Topics: Animals; Apoptosis; Carbazoles; Cell Line, Transformed; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; DNA; DNA Fragmentation; Enzyme Inhibitors; Epithelial Cells; Female; Guanylate Cyclase; Indoles; Oxadiazoles; Oxazines; Quinoxalines; Signal Transduction; Uterus

2003
Insulin induces the release of vasodilator compounds from platelets by a nitric oxide-G kinase-VAMP-3-dependent pathway.
    The Journal of experimental medicine, 2004, Feb-02, Volume: 199, Issue:3

    Topics: Adenosine; Adenosine Triphosphate; Blood Platelets; Carbazoles; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Humans; In Vitro Techniques; Indoles; Insulin; Nitric Oxide; Oxadiazoles; Oxazines; Protein Kinase Inhibitors; Serotonin; Vasodilation

2004
Nitric oxide inhibits gastric acid secretion by increasing intraparietal cell levels of cGMP in isolated human gastric glands.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 289, Issue:6

    Topics: Adult; Cyclic GMP; Dibutyryl Cyclic GMP; Gastric Acid; Guanylate Cyclase; Histamine; Histamine Antagonists; Humans; Male; Nitric Oxide; Oxadiazoles; Oxazines; Parietal Cells, Gastric; S-Nitroso-N-Acetylpenicillamine

2005
Up-regulation of microglial CD11b expression by nitric oxide.
    The Journal of biological chemistry, 2006, May-26, Volume: 281, Issue:21

    Topics: Animals; CD11b Antigen; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Gene Expression Regulation; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Microglia; Neurodegenerative Diseases; Nitric Oxide; Oxadiazoles; Oxazines; Up-Regulation

2006
NO mobilizes intracellular Zn2+ via cGMP/PKG signaling pathway and prevents mitochondrial oxidant damage in cardiomyocytes.
    Cardiovascular research, 2007, Jul-15, Volume: 75, Issue:2

    Topics: Animals; Cells, Cultured; Chlorides; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Flavonoids; Guanylate Cyclase; Membrane Potential, Mitochondrial; Microscopy, Confocal; Mitochondria, Heart; Mitogen-Activated Protein Kinase Kinases; Myocytes, Cardiac; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Oxazines; Oxidation-Reduction; Penicillamine; Phosphorylation; Quinoxalines; Rats; Signal Transduction; Zinc; Zinc Compounds

2007
Nitric oxide mediates lymphatic vessel activation via soluble guanylate cyclase alpha1beta1-impact on inflammation.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2008, Volume: 22, Issue:2

    Topics: Cell Movement; Cell Proliferation; Cells, Cultured; Cyclic GMP; Edema; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Guanylate Cyclase; Humans; Immunity, Cellular; Inflammation; Lymphatic Vessels; Nitric Oxide; Nitric Oxide Synthase Type III; Oxadiazoles; Oxazines; Receptors, Cytoplasmic and Nuclear; S-Nitroso-N-Acetylpenicillamine; Soluble Guanylyl Cyclase

2008
cGMP-independent anti-tumour actions of the inhibitor of soluble guanylyl cyclase, ODQ, in prostate cancer cell lines.
    British journal of pharmacology, 2008, Volume: 155, Issue:6

    Topics: Antineoplastic Agents; Caspase 3; Cell Death; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cyclic GMP; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; Humans; Male; Nitroprusside; Oxadiazoles; Oxazines; Prostatic Neoplasms; RNA Interference; Solubility

2008
Effects of carbon monoxide on trout and lamprey vessels.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2009, Volume: 296, Issue:1

    Topics: Animals; Aorta; Branchial Region; Carbon Monoxide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Heme Oxygenase (Decyclizing); Hydrogen Sulfide; Muscle, Smooth, Vascular; Myography; Nitric Oxide; Nitroprusside; Norepinephrine; Oncorhynchus mykiss; Organometallic Compounds; Oxadiazoles; Oxazines; Petromyzon; Polarography; Potassium Channel Blockers; Potassium Chloride; Protoporphyrins; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2009
The soluble guanylyl cyclase inhibitor NS-2028 reduces vascular endothelial growth factor-induced angiogenesis and permeability.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2010, Volume: 298, Issue:3

    Topics: Animals; Aorta; Capillary Permeability; Cell Division; Cell Movement; Cells, Cultured; Cornea; Drug Interactions; Endothelial Cells; Enzyme Inhibitors; Fibroblast Growth Factor 2; Guanylate Cyclase; Humans; Neovascularization, Physiologic; Oxadiazoles; Oxazines; p38 Mitogen-Activated Protein Kinases; Rabbits; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Umbilical Veins; Vascular Endothelial Growth Factor A; Vasodilation

2010
Endothelium-derived nitric oxide inhibits the relaxation of the porcine coronary artery to natriuretic peptides by desensitizing big conductance calcium-activated potassium channels of vascular smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 334, Issue:1

    Topics: Animals; Coronary Vessels; Cyclic GMP; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Ion Channel Gating; Large-Conductance Calcium-Activated Potassium Channels; Muscle, Smooth, Vascular; Natriuretic Peptides; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Oxazines; Patch-Clamp Techniques; Peptides; Swine; Vasodilation

2010
Methodological proof of immunochemistry for specific identification of 8-nitroguanosine 3',5'-cyclic monophosphate formed in glia cells.
    Nitric oxide : biology and chemistry, 2011, Aug-01, Volume: 25, Issue:2

    Topics: Animals; Antibodies, Monoclonal, Murine-Derived; Blotting, Western; Cells, Cultured; Chromatography, Liquid; Cyclic GMP; Cytokines; Cytoprotection; Epitopes; Guanylate Cyclase; Immunohistochemistry; Lipopolysaccharides; Neuroglia; Nitric Oxide Synthase Type II; Nitrites; omega-N-Methylarginine; Oxadiazoles; Oxazines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase

2011
The soluble guanylyl cyclase activator YC-1 increases intracellular cGMP and cAMP via independent mechanisms in INS-1E cells.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 338, Issue:3

    Topics: Animals; Blotting, Western; Cell Line; Cyclic AMP; Cyclic GMP; Enzyme Activators; Enzyme Inhibitors; Glucose; Guanylate Cyclase; Indazoles; Insulin-Secreting Cells; Mitogen-Activated Protein Kinases; Morpholines; Oxadiazoles; Oxazines; Phosphoric Diester Hydrolases; Pyrimidines; Quinoxalines; Rats; Transcription, Genetic

2011
Fluorescence dequenching makes haem-free soluble guanylate cyclase detectable in living cells.
    PloS one, 2011, Volume: 6, Issue:8

    Topics: Amino Acid Motifs; Amino Acid Sequence; Animals; Benzoates; CHO Cells; Cricetinae; Cricetulus; Cyclic GMP; Cysteine; Enzyme Activation; Enzyme Activators; Fluorescence; Fluorescent Dyes; Guanylate Cyclase; Heme; Humans; Molecular Sequence Data; Mutation; Nitric Oxide; Oxadiazoles; Oxazines; Oxidation-Reduction; Protein Engineering; Receptors, Cytoplasmic and Nuclear; Rotenone; Signal Transduction; Soluble Guanylyl Cyclase; Spectrometry, Fluorescence

2011
The inotropic effects of ammonia on isolated perfused rat hearts and the mechanisms involved.
    The Journal of experimental biology, 2011, Dec-01, Volume: 214, Issue:Pt 23

    Topics: Adenosine Triphosphatases; Ammonia; Ammonium Chloride; Animals; Cardiotonic Agents; Creatine Kinase; Cyclic GMP; Guanylate Cyclase; Heart; Heart Ventricles; Hydrogen-Ion Concentration; In Vitro Techniques; KATP Channels; L-Lactate Dehydrogenase; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Oxazines; Perfusion; Pressure; Rats; Signal Transduction; Small-Conductance Calcium-Activated Potassium Channels; Sodium Hydroxide; Solubility

2011
Portal pressure regulation following Kupffer cell activation: control of prostaglandin production by heme oxygenases.
    Digestion, 2013, Volume: 87, Issue:2

    Topics: Animals; Carbon Monoxide; Enzyme Inhibitors; Guanylate Cyclase; Heme Oxygenase (Decyclizing); Kupffer Cells; Liver; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxadiazoles; Oxazines; Portal Pressure; Prostaglandins; Protoporphyrins; Rats; Rats, Sprague-Dawley

2013
Lack of effect of ODQ does not exclude cGMP signalling via NO-sensitive guanylyl cyclase.
    British journal of pharmacology, 2013, Volume: 170, Issue:2

    Topics: Adult; Animals; Aorta; Cyclic GMP; Female; Guanylate Cyclase; HEK293 Cells; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Oxazines; Signal Transduction

2013
The role of cGMP in ocular growth and the development of form-deprivation myopia in guinea pigs.
    Investigative ophthalmology & visual science, 2013, Dec-03, Volume: 54, Issue:13

    Topics: Animals; Collagen; Conjunctiva; Cyclic GMP; Disease Progression; Eye; Guanylate Cyclase; Guinea Pigs; Injections; Myopia; Oxadiazoles; Oxazines; Radioimmunoassay; Retina; Sclera; Sensory Deprivation

2013
Modulation of growth cone filopodial length by carbon monoxide.
    Developmental neurobiology, 2017, Volume: 77, Issue:6

    Topics: Action Potentials; Animals; Calcium; Carbazoles; Carbon Monoxide; Enzyme Inhibitors; Ganglia, Invertebrate; Growth Cones; Heme Oxygenase-1; Neurons; Nitric Oxide; Organometallic Compounds; Oxadiazoles; Oxazines; Patch-Clamp Techniques; Pseudopodia; Quinoxalines; Signal Transduction; Snails; Time Factors

2017
Apoptosis induction of poly-S-nitrosated human serum albumin in resistant solid tumor under hypoxia can be restored by phosphodiesterase 5 inhibition.
    Nitric oxide : biology and chemistry, 2017, Sep-30, Volume: 69

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Apoptosis; Caspase 3; Cell Line, Tumor; Colonic Neoplasms; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 5; Drug Resistance, Neoplasm; Drug Synergism; Drugs, Chinese Herbal; Humans; Hypoxia; Male; Mice, Inbred BALB C; Nitroso Compounds; Oxadiazoles; Oxazines; Phosphodiesterase 5 Inhibitors; Plant Extracts; Reactive Oxygen Species; Serum Albumin, Human; Soluble Guanylyl Cyclase; Vardenafil Dihydrochloride

2017
Higher susceptibility to heme oxidation and lower protein stability of the rare α
    Biochemical pharmacology, 2021, Volume: 186

    Topics: Animals; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Genetic Variation; Heme; Humans; Moyamoya Disease; Oxadiazoles; Oxazines; Oxidation-Reduction; Protein Stability; Protein Structure, Secondary; Sf9 Cells; Soluble Guanylyl Cyclase

2021