npc 17761 has been researched along with bradykinin in 5 studies
Studies (npc 17761) | Trials (npc 17761) | Recent Studies (post-2010) (npc 17761) | Studies (bradykinin) | Trials (bradykinin) | Recent Studies (post-2010) (bradykinin) |
---|---|---|---|---|---|
5 | 0 | 0 | 14,195 | 355 | 1,520 |
Protein | Taxonomy | npc 17761 (IC50) | bradykinin (IC50) |
---|---|---|---|
B2 bradykinin receptor | Homo sapiens (human) | 0.0018 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Amrani, Y; Da Silva, A; Landry, Y; Trifilieff, A | 1 |
Abraham, WM; Burch, R; Forteza, R; Lauredo, IT | 1 |
Amrani, Y; Gies, JP; Landry, Y; Trifilieff, A | 1 |
Kyle, DJ; Lowe, VC; Noronha-Blob, L; Otterbein, L | 1 |
Cabrini, DA; Calixto, JB; Kyle, DJ | 1 |
5 other study(ies) available for npc 17761 and bradykinin
Article | Year |
---|---|
Involvement of B2 receptors in the bradykinin-induced relaxation of guinea-pig isolated trachea.
Topics: Animals; Bradykinin; Dose-Response Relationship, Drug; Guinea Pigs; Male; Melitten; Receptors, Adrenergic, beta-2; Relaxation; Thiorphan; Trachea | 1995 |
Extracellular metabolites of Pseudomonas aeruginosa produce bronchoconstriction by different mechanisms.
Topics: Administration, Inhalation; Aerosols; Airway Resistance; Animals; Atropine; Bradykinin; Bradykinin Receptor Antagonists; Bronchial Diseases; Bronchoalveolar Lavage Fluid; Chlorpheniramine; Constriction, Pathologic; Drug Evaluation, Preclinical; Endotoxins; Female; Inflammation; Kinins; Nedocromil; Phenazines; Premedication; Pseudomonas aeruginosa; Pyocyanine; Sheep | 1994 |
Comparative action of new highly potent bradykinin receptor antagonists in the guinea-pig trachea.
Topics: Animals; Binding, Competitive; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Kinins; Muscle Contraction; Muscle, Smooth; Oligopeptides; Receptors, Bradykinin; Trachea | 1993 |
Additive effects of a bradykinin antagonist, NPC 17761, and a leumedin, NPC 15669, on survival in animal models of sepsis.
Topics: Amino Acid Sequence; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Bradykinin Receptor Antagonists; Disease Models, Animal; Drug Synergism; Endotoxins; Leucine; Male; Mice; Molecular Sequence Data; Peritonitis; Rats; Rats, Sprague-Dawley; Shock, Septic; Survival Rate | 1993 |
A pharmacological analysis of receptor subtypes and the mechanisms mediating the biphasic response induced by kinins in the rat stomach fundus in vitro.
Topics: Animals; Bradykinin; Calcium; Gastric Fundus; In Vitro Techniques; Lipopolysaccharides; Male; Rats; Rats, Wistar; Receptors, Bradykinin | 1996 |