Page last updated: 2024-09-02

npc 12626 and selfotel

npc 12626 has been researched along with selfotel in 10 studies

Compound Research Comparison

Studies
(npc 12626)
Trials
(npc 12626)
Recent Studies (post-2010)
(npc 12626)
Studies
(selfotel)
Trials
(selfotel)
Recent Studies (post-2010) (selfotel)
5500250910

Protein Interaction Comparison

ProteinTaxonomynpc 12626 (IC50)selfotel (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.3428
Glutamate receptor 1Homo sapiens (human)0.967
Glutamate receptor 2Homo sapiens (human)0.967
Glutamate receptor 3Homo sapiens (human)0.967
Glutamate receptor 4Homo sapiens (human)0.967
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.362
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.3428
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.3428
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.3428
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.3428
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.3428

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Heikkila, RE; Riordan, DE; Sonsalla, PK1
Liljequist, S1
Abreu, M; Ferkany, J; French, ED; Levenson, S1
Mansbach, RS1
Ferkany, JW; Kaplita, PV1
Brandsgaard, RR; Clissold, DB; Ferkany, JW; Hamilton, GS; Hartman, TL; Willetts, J1
Balster, RL; Bobelis, DJ1
Beart, PM; Cheung, NS; Dutton, R; O'Callaghan, D; Ryan, MC; Wong, MG1
Boon, F; Cain, DP; Saucier, D1
Kirsch, JR; Koehler, RC; Miyabe, M; Nishikawa, T; Traystman, RJ1

Other Studies

10 other study(ies) available for npc 12626 and selfotel

ArticleYear
Competitive and noncompetitive antagonists at N-methyl-D-aspartate receptors protect against methamphetamine-induced dopaminergic damage in mice.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Amino Acids; Animals; Corpus Striatum; Dizocilpine Maleate; Male; Methamphetamine; Mice; N-Methylaspartate; Pipecolic Acids; Piperidines; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; Tyrosine 3-Monooxygenase

1991
Genetic differences in the effects of competitive and non-competitive NMDA receptor antagonists on locomotor activity in mice.
    Psychopharmacology, 1991, Volume: 104, Issue:1

    Topics: Amino Acids; Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Motor Activity; Phencyclidine; Pipecolic Acids; Receptors, N-Methyl-D-Aspartate; Species Specificity

1991
Effects of competitive N-methyl-D-aspartate antagonists on midbrain dopamine neurons: an electrophysiological and behavioral comparison to phencyclidine.
    Neuropharmacology, 1991, Volume: 30, Issue:10

    Topics: Amino Acids; Amphetamine; Animals; Behavior, Animal; Dopamine; Electrophysiology; Limbic System; Male; Mesencephalon; Motor Activity; N-Methylaspartate; Neurons; Nucleus Accumbens; Oxidopamine; Phencyclidine; Pipecolic Acids; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1991
Effects of NMDA receptor ligands on sensorimotor gating in the rat.
    European journal of pharmacology, 1991, Sep-04, Volume: 202, Issue:1

    Topics: Acoustic Stimulation; Amino Acids; Animals; Dizocilpine Maleate; Ligands; Male; N-Methylaspartate; Pipecolic Acids; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Reflex; Reflex, Startle

1991
Evidence for direct interactions between the NMDA and glycine recognition sites in brain.
    European journal of pharmacology, 1990, Mar-13, Volume: 188, Issue:2-3

    Topics: Amino Acids; Animals; Brain Chemistry; In Vitro Techniques; Kynurenic Acid; Male; Pipecolic Acids; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Serine

1990
Behavioral pharmacology of NPC 17742, a competitive N-methyl-D-aspartate (NMDA) antagonist.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Behavior, Animal; Binding, Competitive; Dose-Response Relationship, Drug; Isoquinolines; Male; Mice; Pipecolic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1993
Pharmacological specificity of the discriminative stimulus properties of 2-amino-4,5-(1,2-cyclohexyl)-7-phosphono-heptanoic acid (NPC 12626), a competitive N-methyl-D-aspartate receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Amino Acids; Animals; Binding, Competitive; Conditioning, Operant; Diazepam; Discrimination Learning; Generalization, Stimulus; Male; Phencyclidine; Pipecolic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1993
Structure-activity relationships of competitive NMDA receptor antagonists.
    European journal of pharmacology, 1996, Oct-10, Volume: 313, Issue:1-2

    Topics: Amino Acids; Animals; Binding, Competitive; Biphenyl Compounds; Cells, Cultured; Cerebral Cortex; Excitatory Amino Acid Antagonists; Isoquinolines; Mice; Models, Molecular; Neurons; Pipecolic Acids; Propionates; Radioligand Assay; Receptors, N-Methyl-D-Aspartate; Stereoisomerism; Structure-Activity Relationship

1996
Testing hypotheses of spatial learning: the role of NMDA receptors and NMDA-mediated long-term potentiation.
    Behavioural brain research, 1997, Volume: 84, Issue:1-2

    Topics: Amino Acids; Animals; Behavior, Animal; Discrimination Learning; Electrophysiology; Excitatory Amino Acid Antagonists; Learning; Long-Term Potentiation; Male; Maze Learning; N-Methylaspartate; Pipecolic Acids; Rats; Receptors, N-Methyl-D-Aspartate; Space Perception

1997
Comparative analysis of brain protection by N-methyl-D-aspartate receptor antagonists after transient focal ischemia in cats.
    Critical care medicine, 1997, Volume: 25, Issue:6

    Topics: Amino Acids; Animals; Brain; Brain Damage, Chronic; Cats; Cerebrovascular Circulation; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Ischemic Attack, Transient; Male; Neuroprotective Agents; Pipecolic Acids; Prospective Studies; Receptors, N-Methyl-D-Aspartate

1997