Page last updated: 2024-09-02

npc 12626 and phencyclidine

npc 12626 has been researched along with phencyclidine in 15 studies

Compound Research Comparison

Studies
(npc 12626)
Trials
(npc 12626)
Recent Studies (post-2010)
(npc 12626)
Studies
(phencyclidine)
Trials
(phencyclidine)
Recent Studies (post-2010) (phencyclidine)
550028,2943877,796

Protein Interaction Comparison

ProteinTaxonomynpc 12626 (IC50)phencyclidine (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.1299
Lysosomal Pro-X carboxypeptidaseHomo sapiens (human)0.091
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.1299
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.1299
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.1299
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.5563
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.205
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)1.2589
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.1299
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.1299
Sigma non-opioid intracellular receptor 1Rattus norvegicus (Norway rat)0.53
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.1299

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's11 (73.33)18.2507
2000's3 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balster, RL; Compton, AD; Porter, JH; Wiley, JL1
Balster, RL; Bobelis, DJ; Grech, DM1
Clissold, DB; Ferkany, JW; Pontecorvo, MJ; White, MF1
Liljequist, S1
Abreu, M; Ferkany, J; French, ED; Levenson, S1
Balster, RL; Jortani, SA; Mansbach, RS; Willetts, J1
Tortella, FC; Witkin, JM1
Balster, RL; Bobelis, DJ; Willetts, J1
Balster, RL; Bobelis, DJ1
Balster, RL; Cristello, AF; Wiley, JL1
Edwards, MA; Kantak, KM; O'Connor, TP1
Balster, RL; Jones, HE; Nicholson, KL1
Balster, RL; Nicholson, KL2
Balster, RL; Wiley, JL1

Other Studies

15 other study(ies) available for npc 12626 and phencyclidine

ArticleYear
Antipunishment effects of acute and repeated administration of phencyclidine and NPC 12626 in rats.
    Life sciences, 1992, Volume: 50, Issue:20

    Topics: Amino Acids; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Male; Phencyclidine; Punishment; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1992
Drug discrimination analysis of ethanol as an N-methyl-D-aspartate receptor antagonist.
    European journal of pharmacology, 1992, Nov-03, Volume: 222, Issue:1

    Topics: Amino Acids; Animals; Binding, Competitive; Discrimination Learning; Discrimination, Psychological; Ethanol; Male; Phencyclidine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1992
N-methyl-D-aspartate antagonists and working memory performance: comparison with the effects of scopolamine, propranolol, diazepam, and phenylisopropyladenosine.
    Behavioral neuroscience, 1991, Volume: 105, Issue:4

    Topics: Amino Acids; Animals; Appetitive Behavior; Brain; Diazepam; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Mental Recall; Phencyclidine; Phenylisopropyladenosine; Piperazines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic; Retention, Psychology; Scopolamine

1991
Genetic differences in the effects of competitive and non-competitive NMDA receptor antagonists on locomotor activity in mice.
    Psychopharmacology, 1991, Volume: 104, Issue:1

    Topics: Amino Acids; Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Motor Activity; Phencyclidine; Pipecolic Acids; Receptors, N-Methyl-D-Aspartate; Species Specificity

1991
Effects of competitive N-methyl-D-aspartate antagonists on midbrain dopamine neurons: an electrophysiological and behavioral comparison to phencyclidine.
    Neuropharmacology, 1991, Volume: 30, Issue:10

    Topics: Amino Acids; Amphetamine; Animals; Behavior, Animal; Dopamine; Electrophysiology; Limbic System; Male; Mesencephalon; Motor Activity; N-Methylaspartate; Neurons; Nucleus Accumbens; Oxidopamine; Phencyclidine; Pipecolic Acids; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1991
NMDA antagonists: lack of antipunishment effect in squirrel monkeys.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:4

    Topics: Amino Acids; Animals; Conditioning, Operant; Isoflurophate; Male; Midazolam; N-Methylaspartate; Pentobarbital; Phencyclidine; Piperazines; Punishment; Receptors, N-Methyl-D-Aspartate; Reinforcement Schedule; Saimiri

1991
Modulators of N-methyl-D-aspartate protect against diazepam- or phenobarbital-resistant cocaine convulsions.
    Life sciences, 1991, Volume: 48, Issue:11

    Topics: Amino Acids; Animals; Anticonvulsants; Cocaine; Diazepam; Dizocilpine Maleate; Male; Mice; Phencyclidine; Phenobarbital; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Time Factors

1991
Drug discrimination based on the competitive N-methyl-D-aspartate antagonist, NPC 12626.
    Psychopharmacology, 1989, Volume: 99, Issue:4

    Topics: Amino Acids; Animals; Aspartic Acid; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; N-Methylaspartate; Pentobarbital; Phencyclidine; Rats; Rats, Inbred Strains

1989
Pharmacological specificity of the discriminative stimulus properties of 2-amino-4,5-(1,2-cyclohexyl)-7-phosphono-heptanoic acid (NPC 12626), a competitive N-methyl-D-aspartate receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Amino Acids; Animals; Binding, Competitive; Conditioning, Operant; Diazepam; Discrimination Learning; Generalization, Stimulus; Male; Phencyclidine; Pipecolic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1993
Effects of site-selective NMDA receptor antagonists in an elevated plus-maze model of anxiety in mice.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Amino Acids; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phencyclidine; Punishment; Quinoxalines; Rats; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1995
Modulation of the discriminative stimulus and rate-altering effects of cocaine by competitive and noncompetitive N-methyl-D-aspartate antagonists.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 59, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Binding, Competitive; Cocaine; Discrimination Learning; Dizocilpine Maleate; Dopamine Uptake Inhibitors; Drug Interactions; Excitatory Amino Acid Antagonists; Magnesium Chloride; Male; Phencyclidine; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Reinforcement Schedule

1998
Evaluation of the reinforcing and discriminative stimulus effects of the N-methyl-D-aspartate competitive antagonist NPC 17742 in rhesus monkeys.
    Behavioural pharmacology, 1997, Volume: 8, Issue:5

    Topics: Amino Acids; Animals; Binding, Competitive; Discrimination, Psychological; Excitatory Amino Acid Antagonists; Female; Macaca mulatta; Male; N-Methylaspartate; Phencyclidine; Reinforcement, Psychology; Self Administration

1997
Evaluation of the discriminative stimulus effects of the low-affinity N-methyl-D-aspartate channel blockers AR-R 13950AA and AR-R 16283AA in rats and rhesus monkeys.
    Behavioural pharmacology, 2002, Volume: 13, Issue:7

    Topics: Acetamides; Amino Acids; Animals; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Food; Macaca mulatta; Male; Phencyclidine; Pyrazines; Rats; Receptors, N-Methyl-D-Aspartate; Reinforcement Schedule

2002
Effects of modulators of N-methyl-D-aspartate receptor-mediated neurotransmission on diazepam discrimination in rats.
    Life sciences, 2004, May-28, Volume: 75, Issue:2

    Topics: Amino Acids; Animals; Biguanides; Binding Sites; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Male; N-Methylaspartate; Pentobarbital; Phencyclidine; Piperazines; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Riluzole

2004
The discriminative stimulus effects of N-methyl-D-aspartate glycine-site ligands in NMDA antagonist-trained rats.
    Psychopharmacology, 2009, Volume: 203, Issue:2

    Topics: Amino Acids; Animals; Behavior, Animal; Binding Sites; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Male; Phencyclidine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

2009