norfloxacin and chloramphenicol

norfloxacin has been researched along with chloramphenicol in 116 studies

Research

Studies (116)

TimeframeStudies, this research(%)All Research%
pre-19907 (6.03)18.7374
1990's14 (12.07)18.2507
2000's31 (26.72)29.6817
2010's59 (50.86)24.3611
2020's5 (4.31)2.80

Authors

AuthorsStudies
Apiwattanakul, N; Endou, H; Jariyawat, S; Kanai, Y; Sekine, T; Sophasan, S; Takeda, M1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Drlica, K; Hussain, S; Malik, M1
Arpin, C; Ba, BB; Caignard, DH; Forfar-Bares, I; Grellet, J; Guillon, J; Jarry, C; Moreau, S; Quentin, C; Vidaillac, C1
Levy, SB; Nicoloff, H; Perreten, V1
Akamatsu, M; Fujikawa, M; Nakao, K; Shimizu, R1
Courvalin, P; Galimand, M; Périchon, B1
Al-Momani, W; Antunes, NT; Assunção, P; Ayling, RD; Mercier, P; Poveda, JB; Rosales, RS; Tavío, MM1
Beceiro, A; Bou, G; Canle, D; Fernández, A; Lasa, I; Latasa, C; Mallo, S; Molina, F; Pérez, A; Pérez, S; Poza, M; Tomás, Mdel M; Villanueva, R1
Ackerley, DF; Andersen, GL; Benoit, MR; Brodie, EL; Dixon, L; Hu, P; Keyhan, M; Lynch, SV; Matin, A1
Chen, T; Khalil, H; Riffon, R; Wang, R; Wang, Z1
Bammert, GF; Banitt, LS; Barbachyn, MR; Boyle, TP; Bundy, GL; Dolak, LA; Ford, CW; Graber, DR; Hamel, JC; Han, F; Harris, DW; Hromockyj, AE; Hurd, AR; Kamilar, GM; Marotti, KR; Martin, GE; Miller, AA; Mott, JE; Munzner, JB; Palmer, JR; Ruble, JC; Seest, EP; Skepner, JE; Sweeney, MT; Zhong, WZ; Zurenko, GE1
Long, F; Rouquette-Loughlin, C; Shafer, WM; Yu, EW1
Cattoir, V; Nordmann, P; Poirel, L1
Bailey, AM; Paulsen, IT; Piddock, LJ1
Chevalier, J; Davin-Regli, A; Dupont, M; Lavigne, JP; Pagès, JM; Sotto, A; Tran, QT1
Wang, X; Zhao, X1
Hiramatsu, K; Kikuchi, K; Ohtsuka, M; Ono, Y; Sasaki, T; Shimizu, K; Takahashi, N1
Hamamoto, H; Kurokawa, K; Lee, BL; Maki, H; Matsuo, M; Murakami, K; Nishida, S; Sekimizu, K; Yamane, N1
Espinal, P; Gibert, I; Marti, S; Martínez, P; Roca, I; Vila, J1
Gaillard, JL; Jackson, M; McDonnell, G; Niederweis, M; Skovierová, H; Svetlíková, Z1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Brasme, L; De Champs, C; Duval, V; Forte, D; Guillard, T; Madoux, J; Maiga, A; Maiga, I; Vernet-Garnier, V1
Hashida, Y; Konaka, R; Kourai, H; Maseda, H; Shirai, A1
Gebreyes, WA; Rajamohan, G; Srinivasan, VB1
Courvalin, P; Coyne, S; Guigon, G; Périchon, B1
Fàbrega, A; Martin, RG; Rosner, JL; Tavio, MM; Vila, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Hakanen, AJ; Huovinen, P; Kotilainen, P; Lehtopolku, M; Nakari, UM; Siitonen, A1
Alibert-Franco, S; Bolla, JM; Kuete, V; Ngadjui, BT; Ngameni, B; Pagès, JM; Tangmouo, JG1
Gan, LL; Zhang, FF; Zhou, CH1
Levy, SB; Ruiz, C1
Avdeef, A; Tam, KY1
Mima, T; Schweizer, HP1
Fang, B; Rao, XC; Zhou, CH1
Bohnert, JA; Karamian, B; Nikaido, H1
Chen, S; Chen, Z; Deng, Y; Huang, X; Liu, JH; Liu, Y; Sun, Y; Tian, W; Wu, C; Zeng, Z; Zhao, J1
Gadakh, AV; Karale, BK; Pandit, C; Rindhe, SS1
Gotoh, N; Hayashi, N; Okuda, J; Wakahara, Y1
Mali, MD; Patel, MM; Patel, SK1
Akamatsu, M1
Makawana, JA; Mungra, DC; Patel, MP; Patel, RG1
Akhaja, TN; Raval, JP1
Anderson, KC; Kellogg, GE; Sarkar, A1
Barad, HA; Gupta, VK; Kant, R; Pansuriya, BR; Parmar, NJ; Teraiya, SB1
Barad, HA; Gupta, VK; Kant, R; Pansuriya, BR; Parmar, NJ1
Patel, MP; Patel, RG; Shah, NM1
Bonifácio, VD; Gawande, MB; Mhaske, GR; Shelke, SN1
Damu, GL; Geng, RX; Zhang, L; Zhang, SL; Zhou, CH1
Chang, JJ; Damu, GL; Fang, B; Geng, RX; Zhang, SL; Zhou, CH; Zhou, XD1
Parmar, BD; Parmar, NJ; Patel, RA; Talpada, NP1
Kathrotiya, HG; Patel, MP1
Cui, SF; Damu, GL; Geng, RX; Peng, XM; Ren, Y; Zhang, SL; Zhou, CH1
Kanawade, SB; Rajani, DP; Toche, RB1
Cai, GX; Damu, GL; Zhang, HZ; Zhou, CH1
Jardosh, HH; Patel, MP1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Geng, RX; Peng, XM; Rasheed, S; Yan, CY; Yin, BT; Zhang, SL; Zhou, CH1
Kishore, B; Lv, JS; Peng, XM; Zhou, CH1
Kalaria, PN; Raval, DK; Satasia, SP1
Karad, SC; Purohit, VB; Raval, DK1
Karad, SC; Purohit, VB; Raval, DK; Thakkar, VR; Thakor, P1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Addla, D; Cui, SF; Zhou, CH1
Avula, SR; Jeyakkumar, P; Zhang, L; Zhou, CH1
Addla, D; Avula, SR; Cheng, Y; Gao, WW; Lin, JM; Tangadanchu, VKR; Zhang, L; Zhou, CH1
Kamani, RD; Karad, SC; Purohit, VB; Raval, DK; Ray, A; Thakkar, SS; Thakkar, VR; Thakor, P; Thummar, RP; Vaghasiya, BK1
Cheng, Y; Geng, RX; Gopala, L; Jeyakkumar, P; Liu, HB; Peng, XM; Zhou, CH1
Gan, LL; Gopala, L; He, SC; Peng, YJ; Tangadanchu, VKR; Zhang, HJ; Zhang, HZ; Zhou, CH1
Doshi, H; Ray, A; Thakkar, SS; Thakor, P1
Doshi, H; Ray, A; Thakkar, SS; Thakkar, VR; Thakor, P1
Bheemanaboina, RRY; Kannekanti, VK; Li, ZZ; Maddili, SK; Tangadanchu, VKR; Tuniki, B; Zhou, CH1
Bai, L; Deng, J; Feng, L; Lv, Z; Wang, Y; Xu, Z; Zhang, F; Zhao, S1
Bukharov, SV; Burilov, AR; Gibadullina, EM; Pazilova, NB; Pudovik, MA; Sapunova, AS; Starodubtseva, RR; Sudakov, IA; Voloshina, AD; Vyshtakalyuk, AB1
Zhang, B1
Ba, Y; Hou, X; Wang, S; Xu, Z; Yang, H; Zhang, J1
Gao, F; Huang, G; Xiao, J1
Beteck, RM; Jesumoroti, OJ; Legoabe, LJ; Patel, OPS1
Daraji, DG; Jayanthi, S; Patel, HD; Pithawala, EA; Rajani, DP; Rajani, SD1
Hannan, A1
Hancock, RE; Young, M1
Cook, T; Miller, IM; Vogel, R; Wittreich, JM1
Fukuda, H; Hashimoto, H; Hirai, K; Iyobe, S; Jakics, EB1
Agarwal, S; Guleria, JS; Madhu, SV; Talwar, V1
Avisar, R; Hundart, O; Lerner, N; Savir, H; Vender, T; Yasur, Y1
Cohen, SP; Hooper, DC; Levy, SB; McMurry, LM; Wolfson, JS1
Zeiler, HJ1
Martin, E; Nauciel, C1
Hackbarth, CJ; Sande, MA; Shibl, AM1
Bonanni, M; Iegri, F; Lorenzi, A; Mascellino, MT1
Drusano, GL; Morris, JG; Tenney, JH1
Li, XZ; Livermore, DM; Nikaido, H1
Mortimer, PG; Piddock, LJ1
Li, XZ; Nikaido, H; Poole, K1
Gotoh, N; Li, XZ; Neshat, S; Nishino, T; Poole, K; Tsujimoto, H; Wada, A; Yamagishi, J; Yamasaki, T; Zhao, Q1
Ishiguro, EE; Rodionov, DG1
Courvalin, P; Lynch, C; Nikaido, H1
Deguchi, K; Ishihara, R; Ishii, Y; Nakazawa, A; Suzuki, Y1
Araj, GF; Zouain, MG1
Bal, AM; Ghadage, DP1
Chan, CM; Li, L; Tan, DT; Theng, JT1
Tabata, M; Takata, T; Tsuruoka, T; Watabe, H1
Biswas, A; Kumar, AA; Ramakrishnan, MA; Shivachandra, SB; Singh, VP; Srivastava, SK1
Bassily, S; El Masry, NA; Haberberger, RL; Mikhail, I; Woody, JN; Yassa, M; Zakaria, S1
Gerkowicz, M; Gruszecka-Gerkowicz, R; Kosior-Jarecka, E; Pietraś-Trzpiel, M1
Li, XD; Liu, YC; Xu, WH; Zhang, G; Zou, SC1
Adam, E; Baitiche, M; Chevalier, J; Mahamoud, A; Pagès, JM1
Chen, CP; Chen, TL; Fan, NW; Lee, SM; Lin, PY1
Chu, LM; Pan, M1
Ahn, J; Ding, T; Jo, A; Kim, J; Lee, HY1
Akutagawa, M; Emoto, T; Harada, Y; Hou, Y; Kinouchi, Y; Mawatari, K; Nakahashi, M; Shimohata, T; Takahashi, A; Tsunedomi, A; Uebanso, T1
Abdenaceur, H; Beltifa, A; Ben Mansour, H; Ghorbel, A; Mehri, I; Reyns, T; Sire, O; Van Loco, J; Zouiten, A1
Al-Ajmi, D; Banu, S; Rahman, S1
Abebe, N; Ahmed, M; Awol, N; Bsrat, A; Gugsa, G; Hagos, Y; Tsegaye, Y1
Fang, C; Huang, Q; Liu, C; Shao, C; Wang, H; Wang, S; Xu, H1

Reviews

6 review(s) available for norfloxacin and chloramphenicol

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Benzofuran derivatives and their anti-tubercular, anti-bacterial activities.
    European journal of medicinal chemistry, 2019, Jan-15, Volume: 162

    Topics: Anti-Bacterial Agents; Antitubercular Agents; Benzofurans; Humans; Structure-Activity Relationship

2019
Comprehensive review on the anti-bacterial activity of 1,2,3-triazole hybrids.
    European journal of medicinal chemistry, 2019, Apr-15, Volume: 168

    Topics: Anti-Bacterial Agents; Bacteria; Bacterial Infections; Dose-Response Relationship, Drug; Humans; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Triazoles

2019
Nitroimidazole-containing compounds and their antibacterial and antitubercular activities.
    European journal of medicinal chemistry, 2019, Oct-01, Volume: 179

    Topics: Anti-Bacterial Agents; Bacterial Infections; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Molecular Structure; Nitroimidazoles

2019
Current scenario of tetrazole hybrids for antibacterial activity.
    European journal of medicinal chemistry, 2019, Dec-15, Volume: 184

    Topics: Anti-Bacterial Agents; Bacteria; Dose-Response Relationship, Drug; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Tetrazoles

2019
Metronidazole-conjugates: A comprehensive review of recent developments towards synthesis and medicinal perspective.
    European journal of medicinal chemistry, 2021, Jan-15, Volume: 210

    Topics: Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Antiprotozoal Agents; Drug Development; Humans; Hypoglycemic Agents; Metronidazole

2021

Trials

2 trial(s) available for norfloxacin and chloramphenicol

ArticleYear
The safety and efficacy of topical norfloxacin compared with chloramphenicol for the treatment of external ocular bacterial infections. The Norfloxacin-Chloramphenicol Ophthalmic Study Group.
    Eye (London, England), 1992, Volume: 6 ( Pt 1)

    Topics: Acute Disease; Adolescent; Adult; Aged; Aged, 80 and over; Blepharitis; Child; Child, Preschool; Chloramphenicol; Conjunctivitis, Bacterial; Double-Blind Method; Female; Humans; Male; Middle Aged; Norfloxacin

1992
[Changes in bacterial flora of conjunctival sac in patients prophylacticaly treated with antibiotic before cataract operation].
    Klinika oczna, 2005, Volume: 107, Issue:10-12

    Topics: Antibiotic Prophylaxis; Cataract; Cataract Extraction; Chloramphenicol; Conjunctiva; Conjunctivitis, Bacterial; Female; Gentamicins; Humans; Male; Norfloxacin; Ofloxacin

2005

Other Studies

108 other study(ies) available for norfloxacin and chloramphenicol

ArticleYear
The interaction and transport of beta-lactam antibiotics with the cloned rat renal organic anion transporter 1.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:2

    Topics: Animals; Anion Transport Proteins; Anti-Bacterial Agents; Biological Transport; Carrier Proteins; Cell Survival; Cephaloridine; Cephalosporins; In Vitro Techniques; Kidney; Kinetics; Oocytes; p-Aminohippuric Acid; Penicillin G; Rats; Recombinant Proteins; Xenopus laevis

1999
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Effect of anaerobic growth on quinolone lethality with Escherichia coli.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:1

    Topics: Aerobiosis; Anaerobiosis; Anti-Infective Agents; Chloramphenicol; Ciprofloxacin; DNA Fragmentation; DNA Gyrase; DNA, Bacterial; DnaB Helicases; Dose-Response Relationship, Drug; Drug Resistance, Bacterial; Escherichia coli; Microbial Sensitivity Tests; Models, Biological; Molecular Structure; Nalidixic Acid; Quinolones

2007
Synthesis of omeprazole analogues and evaluation of these as potential inhibitors of the multidrug efflux pump NorA of Staphylococcus aureus.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:3

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Culture Media; Drug Resistance, Multiple, Bacterial; Enzyme Inhibitors; Indicators and Reagents; Kinetics; Microbial Sensitivity Tests; Multidrug Resistance-Associated Proteins; Norfloxacin; Omeprazole; Staphylococcus aureus; Structure-Activity Relationship

2007
Increased genome instability in Escherichia coli lon mutants: relation to emergence of multiple-antibiotic-resistant (Mar) mutants caused by insertion sequence elements and large tandem genomic amplifications.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:4

    Topics: Anti-Bacterial Agents; DNA Transposable Elements; DNA-Binding Proteins; DNA, Bacterial; Drug Resistance, Multiple, Bacterial; Escherichia coli; Escherichia coli Proteins; Gene Amplification; Genome, Bacterial; Genomic Instability; Multidrug Resistance-Associated Proteins; Mutation; Protease La

2007
QSAR study on permeability of hydrophobic compounds with artificial membranes.
    Bioorganic & medicinal chemistry, 2007, Jun-01, Volume: 15, Issue:11

    Topics: Biological Transport; Caco-2 Cells; Drug Evaluation, Preclinical; Humans; Hydrophobic and Hydrophilic Interactions; Membranes, Artificial; Permeability; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship

2007
Transferable resistance to aminoglycosides by methylation of G1405 in 16S rRNA and to hydrophilic fluoroquinolones by QepA-mediated efflux in Escherichia coli.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:7

    Topics: Amino Acid Motifs; Amino Acid Sequence; Aminoglycosides; Anti-Bacterial Agents; Anti-Infective Agents; Conjugation, Genetic; Conserved Sequence; DNA, Bacterial; Drug Resistance, Multiple, Bacterial; Enterobacteriaceae; Escherichia coli; Escherichia coli Proteins; Fluoroquinolones; Genes, rRNA; Methylation; Methyltransferases; Microbial Sensitivity Tests; Molecular Sequence Data; Norfloxacin; Plasmids; Sequence Analysis, DNA; Sequence Homology, Amino Acid

2007
In vitro susceptibilities of Mycoplasma putrefaciens field isolates.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:9

    Topics: Anti-Bacterial Agents; France; Humans; Jordan; Lincomycin; Macrolides; Microbial Sensitivity Tests; Mycoplasma; Mycoplasma Infections; Tetracycline Resistance

2007
Cloning, nucleotide sequencing, and analysis of the AcrAB-TolC efflux pump of Enterobacter cloacae and determination of its involvement in antibiotic resistance in a clinical isolate.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:9

    Topics: Bacterial Proteins; Base Sequence; beta-Lactamases; Carrier Proteins; Cloning, Molecular; DNA, Bacterial; Drug Resistance, Bacterial; Enterobacter cloacae; Enterobacteriaceae Infections; Genes, MDR; Genetic Vectors; Humans; Microbial Sensitivity Tests; Molecular Sequence Data; Plasmids; Porins

2007
Role of the rapA gene in controlling antibiotic resistance of Escherichia coli biofilms.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:10

    Topics: Anti-Bacterial Agents; beta-Lactamases; Biofilms; Blotting, Western; DNA Primers; Drug Resistance, Bacterial; Escherichia coli K12; Gene Deletion; Genes, Bacterial; Genetic Complementation Test; Genetic Vectors; Penicillin G; Penicillin-Binding Proteins; Plasmids; Polysaccharides

2007
Synergy between polyethylenimine and different families of antibiotics against a resistant clinical isolate of Pseudomonas aeruginosa.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:5

    Topics: Aminoglycosides; Anti-Bacterial Agents; Carbenicillin; Ceftazidime; Ciprofloxacin; Drug Resistance, Bacterial; Drug Synergism; Humans; Microbial Sensitivity Tests; Novobiocin; Ofloxacin; Piperacillin; Polyethyleneimine; Pseudomonas aeruginosa; Pseudomonas Infections; Rifampin; Ticarcillin; Tobramycin

2008
Discovery and characterization of QPT-1, the progenitor of a new class of bacterial topoisomerase inhibitors.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Area Under Curve; Bacteria; Bacterial Infections; Bacterial Proteins; Cell Line; Cell Proliferation; Metabolic Clearance Rate; Mice; Microbial Sensitivity Tests; Molecular Structure; Staphylococcus aureus; Stereoisomerism; Topoisomerase II Inhibitors

2008
Functional cloning and characterization of the multidrug efflux pumps NorM from Neisseria gonorrhoeae and YdhE from Escherichia coli.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:9

    Topics: Anti-Bacterial Agents; Antiporters; ATP-Binding Cassette Transporters; Bacterial Proteins; Cloning, Molecular; Drug Resistance, Bacterial; Escherichia coli; Escherichia coli Proteins; Ethidium; Fluorescence Polarization; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Norfloxacin

2008
Plasmid-mediated quinolone resistance pump QepA2 in an Escherichia coli isolate from France.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:10

    Topics: Aged; Base Sequence; DNA Primers; DNA, Bacterial; Drug Resistance, Bacterial; Escherichia coli; Escherichia coli Infections; Escherichia coli Proteins; Female; Fluoroquinolones; France; Genes, Bacterial; Humans; Models, Genetic; Molecular Sequence Data; Plasmids

2008
RamA confers multidrug resistance in Salmonella enterica via increased expression of acrB, which is inhibited by chlorpromazine.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:10

    Topics: Anti-Bacterial Agents; Antipsychotic Agents; Bacterial Proteins; Base Sequence; Chlorpromazine; DNA Primers; DNA, Bacterial; Drug Resistance, Multiple, Bacterial; Drug Synergism; Ethidium; Gene Expression; Genes, Bacterial; Humans; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Mutation; Oligonucleotide Array Sequence Analysis; Phenothiazines; Salmonella typhimurium; Trans-Activators

2008
Occurrence of efflux mechanism and cephalosporinase variant in a population of Enterobacter aerogenes and Klebsiella pneumoniae isolates producing extended-spectrum beta-lactamases.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:4

    Topics: Bacterial Proteins; beta-Lactamases; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cefepime; Cephalosporinase; Cephalosporins; Drug Resistance, Bacterial; Enterobacter aerogenes; Humans; Klebsiella pneumoniae; Microbial Sensitivity Tests

2009
Contribution of oxidative damage to antimicrobial lethality.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:4

    Topics: 2,2'-Dipyridyl; Anti-Bacterial Agents; Bacterial Proteins; Catalase; Escherichia coli; Escherichia coli Proteins; Hydroxyl Radical; Microbial Sensitivity Tests; Norfloxacin; Oxidative Stress; Superoxide Dismutase; Thiourea

2009
Emergence of quinolone-resistant Bordetella pertussis in Japan.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:7

    Topics: Anti-Bacterial Agents; Bordetella pertussis; Child; DNA Gyrase; Fluoroquinolones; Humans; Japan; Microbial Sensitivity Tests; Mutation; Nalidixic Acid; Quinolones

2009
Evaluation of target specificity of antibacterial agents using Staphylococcus aureus ddlA mutants and D-cycloserine in a silkworm infection model.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:9

    Topics: Animals; Anti-Bacterial Agents; Bombyx; Cephalosporins; Chloramphenicol; Cycloserine; Inhibitory Concentration 50; Larva; Microbial Sensitivity Tests; Staphylococcus aureus; Tetracycline; Vancomycin

2009
CraA, a major facilitator superfamily efflux pump associated with chloramphenicol resistance in Acinetobacter baumannii.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:9

    Topics: Acinetobacter baumannii; Aminoglycosides; Anti-Bacterial Agents; Bacterial Proteins; Chloramphenicol Resistance; Drug Resistance, Multiple, Bacterial; Imipenem; Microbial Sensitivity Tests; Polymerase Chain Reaction; Quinolones; Tetracyclines

2009
Role of porins in the susceptibility of Mycobacterium smegmatis and Mycobacterium chelonae to aldehyde-based disinfectants and drugs.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:9

    Topics: Antitubercular Agents; Disinfectants; Drug Resistance, Bacterial; Glutaral; Microbial Sensitivity Tests; Molecular Sequence Data; Mutation; Mycobacterium chelonae; Mycobacterium smegmatis; o-Phthalaldehyde; Porins

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
High prevalence of CTX-M-type beta-lactamases among clinical isolates of Enterobacteriaceae in Bamako, Mali.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:11

    Topics: beta-Lactamases; Drug Resistance, Bacterial; Enterobacteriaceae; Humans; Random Amplified Polymorphic DNA Technique

2009
Mutational upregulation of a resistance-nodulation-cell division-type multidrug efflux pump, SdeAB, upon exposure to a biocide, cetylpyridinium chloride, and antibiotic resistance in Serratia marcescens.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:12

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Cetylpyridinium; Disinfectants; Drug Resistance, Multiple, Bacterial; Membrane Proteins; Mutation; Norfloxacin; Quaternary Ammonium Compounds; Serratia marcescens

2009
Role of AbeS, a novel efflux pump of the SMR family of transporters, in resistance to antimicrobial agents in Acinetobacter baumannii.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:12

    Topics: Acinetobacter baumannii; Amino Acid Sequence; Anti-Bacterial Agents; Bacterial Proteins; Drug Resistance, Multiple, Bacterial; Escherichia coli; Membrane Transport Proteins; Microbial Sensitivity Tests; Molecular Sequence Data; Sequence Homology, Amino Acid

2009
Screening and quantification of the expression of antibiotic resistance genes in Acinetobacter baumannii with a microarray.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:1

    Topics: Acinetobacter baumannii; Anti-Bacterial Agents; DNA, Bacterial; DNA, Complementary; Drug Resistance, Bacterial; Drug Resistance, Multiple, Bacterial; Genes, MDR; Metals, Heavy; Microbial Sensitivity Tests; Mutation; Oligonucleotide Array Sequence Analysis; Reproducibility of Results; Reverse Transcriptase Polymerase Chain Reaction; RNA, Bacterial

2010
Constitutive SoxS expression in a fluoroquinolone-resistant strain with a truncated SoxR protein and identification of a new member of the marA-soxS-rob regulon, mdtG.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:3

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Base Sequence; Drug Resistance, Bacterial; Escherichia coli; Escherichia coli Proteins; Fluoroquinolones; Gene Expression Regulation, Bacterial; Humans; Microbial Sensitivity Tests; Molecular Sequence Data; Oligonucleotide Array Sequence Analysis; Promoter Regions, Genetic; Regulon; Sequence Analysis, DNA; Trans-Activators; Transcription Factors

2010
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Antimicrobial susceptibilities of multidrug-resistant Campylobacter jejuni and C. coli strains: in vitro activities of 20 antimicrobial agents.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:3

    Topics: Anti-Bacterial Agents; Campylobacter coli; Campylobacter Infections; Campylobacter jejuni; Carbapenems; Drug Resistance, Multiple, Bacterial; Erythromycin; Feces; Finland; Humans; Macrolides; Microbial Sensitivity Tests; Minocycline; Tigecycline

2010
Efflux pumps are involved in the defense of Gram-negative bacteria against the natural products isobavachalcone and diospyrone.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:5

    Topics: Bacterial Proteins; Carrier Proteins; Chalcones; Diospyros; Drug Discovery; Drug Resistance, Bacterial; Drug Resistance, Multiple; Enterobacter aerogenes; Enterobacter cloacae; Escherichia coli; Gram-Negative Bacteria; Klebsiella pneumoniae; Membrane Transport Proteins; Plant Proteins; Pseudomonas aeruginosa

2010
Synthesis, antibacterial and antifungal activities of some carbazole derivatives.
    Bioorganic & medicinal chemistry letters, 2010, Mar-15, Volume: 20, Issue:6

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aspergillus fumigatus; Bacteria; Candida albicans; Carbazoles; Microbial Sensitivity Tests

2010
Many chromosomal genes modulate MarA-mediated multidrug resistance in Escherichia coli.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:5

    Topics: Anti-Bacterial Agents; Bacterial Outer Membrane Proteins; Chromosomes, Bacterial; Colicins; Cyclic AMP Receptor Protein; DNA-Binding Proteins; Drug Resistance, Bacterial; Drug Resistance, Multiple; Escherichia coli; Escherichia coli Proteins; Fimbriae Proteins; Gene Expression Regulation, Bacterial; Lipoproteins; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Mutagenesis; Polynucleotide Adenylyltransferase

2010
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
The BpeAB-OprB efflux pump of Burkholderia pseudomallei 1026b does not play a role in quorum sensing, virulence factor production, or extrusion of aminoglycosides but is a broad-spectrum drug efflux system.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:8

    Topics: Aminoglycosides; Anti-Bacterial Agents; Bacterial Outer Membrane Proteins; Burkholderia pseudomallei; Culture Media; Drug Resistance, Multiple, Bacterial; Humans; Membrane Transport Proteins; Microbial Sensitivity Tests; Mutation; Periplasmic Proteins; Quorum Sensing; Singapore; Virulence Factors

2010
Synthesis and biological activities of novel amine-derived bis-azoles as potential antibacterial and antifungal agents.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:9

    Topics: Amines; Anti-Bacterial Agents; Antifungal Agents; Azoles; Bacteria; Fungi; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Structure-Activity Relationship

2010
Optimized Nile Red efflux assay of AcrAB-TolC multidrug efflux system shows competition between substrates.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:9

    Topics: Anti-Bacterial Agents; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Chlortetracycline; Dipeptides; Doxorubicin; Doxycycline; Drug Resistance, Multiple, Bacterial; Escherichia coli; Escherichia coli Proteins; Minocycline; Onium Compounds; Organophosphorus Compounds; Tetracycline

2010
Prevalence and dissemination of oqxAB in Escherichia coli isolates from animals, farmworkers, and the environment.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:10

    Topics: Animals; Anti-Bacterial Agents; Drug Resistance, Multiple, Bacterial; Electrophoresis, Gel, Pulsed-Field; Escherichia coli; Escherichia coli Proteins; Humans; Microbial Sensitivity Tests; Molecular Sequence Data; Plasmids; Quinolones

2010
Synthesis and antimicrobial activity of novel fluorine containing 4-(substituted-2-hydroxybenzoyl)-1H-pyrazoles and pyrazolyl benzo[d]oxazoles.
    Bioorganic & medicinal chemistry letters, 2010, Sep-15, Volume: 20, Issue:18

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Bacillus subtilis; Bacteria; Bacterial Infections; Candida albicans; Candidiasis; Escherichia coli; Fluorine; Humans; Microbial Sensitivity Tests; Oxazoles; Pseudomonas aeruginosa; Pyrazoles; Staphylococcus aureus; Structure-Activity Relationship

2010
Reduced expression of the vca0421 gene of Vibrio cholerae O1 results in innate resistance to ciprofloxacin.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:11

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Ciprofloxacin; Fluoroquinolones; Quinolones; Reverse Transcriptase Polymerase Chain Reaction; Vibrio cholerae O1

2010
Bernthsen synthesis, antimicrobial activities and cytotoxicity of acridine derivatives.
    Bioorganic & medicinal chemistry letters, 2010, Nov-01, Volume: 20, Issue:21

    Topics: Acridines; Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Antineoplastic Agents; Aspergillus niger; Bacteria; Gram-Negative Bacteria; Gram-Positive Bacteria; Indicators and Reagents; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Spectrophotometry, Infrared

2010
Importance of physicochemical properties for the design of new pesticides.
    Journal of agricultural and food chemistry, 2011, Apr-13, Volume: 59, Issue:7

    Topics: Anabasine; Animals; Biological Availability; Cell Membrane Permeability; Chemical Phenomena; Drug Design; Humans; Imidazoles; Insecticides; Neonicotinoids; Nitro Compounds; Pesticides; Quantitative Structure-Activity Relationship; Receptors, Nicotinic

2011
Microwave assisted synthesis and antimicrobial evaluation of new fused pyran derivatives bearing 2-morpholinoquinoline nucleus.
    Bioorganic & medicinal chemistry letters, 2011, Oct-15, Volume: 21, Issue:20

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Candida albicans; Fungi; Gram-Negative Bacteria; Gram-Negative Bacterial Infections; Gram-Positive Bacteria; Gram-Positive Bacterial Infections; Humans; Microbial Sensitivity Tests; Microwaves; Mycoses; Pyrans; Quinolines

2011
1,3-Dihydro-2H-indol-2-ones derivatives: design, synthesis, in vitro antibacterial, antifungal and antitubercular study.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:11

    Topics: Antifungal Agents; Antitubercular Agents; Chemistry Techniques, Synthetic; Drug Design; Fungi; Indoles; Microbial Sensitivity Tests; Mycobacterium tuberculosis

2011
Computational analysis of structure-based interactions and ligand properties can predict efflux effects on antibiotics.
    European journal of medicinal chemistry, 2012, Volume: 52

    Topics: Anti-Bacterial Agents; beta-Lactams; Computational Biology; Drug Resistance, Bacterial; Hydrophobic and Hydrophilic Interactions; Ligands; Membrane Transport Proteins; Microbial Sensitivity Tests; Models, Molecular; Protein Binding; Protein Conformation; Quantitative Structure-Activity Relationship; Regression Analysis; Thermodynamics

2012
An efficient one-pot synthesis, structure, antimicrobial and antioxidant investigations of some novel quinolyldibenzo[b,e][1,4]diazepinones.
    Bioorganic & medicinal chemistry letters, 2012, Jun-01, Volume: 22, Issue:11

    Topics: Anti-Infective Agents; Antioxidants; Azepines; Crystallography, X-Ray; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Conformation; Quinolines

2012
An improved microwave assisted one-pot synthesis, and biological investigations of some novel aryldiazenyl chromeno fused pyrrolidines.
    Bioorganic & medicinal chemistry letters, 2012, Jun-15, Volume: 22, Issue:12

    Topics: Antifungal Agents; Antitubercular Agents; Aspergillus fumigatus; Azo Compounds; Benzopyrans; Candida albicans; Crystallography, X-Ray; Gram-Negative Bacteria; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Microwaves; Molecular Structure; Mycobacterium tuberculosis; Pyrrolidines; Stereoisomerism; Thiosemicarbazones

2012
New N-arylamino biquinoline derivatives: synthesis, antimicrobial, antituberculosis, and antimalarial evaluation.
    European journal of medicinal chemistry, 2012, Volume: 54

    Topics: Antimalarials; Antitubercular Agents; Chemistry Techniques, Synthetic; Electrons; Fungi; Hydrophobic and Hydrophilic Interactions; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Plasmodium falciparum; Quinolines

2012
Green synthesis and anti-infective activities of fluorinated pyrazoline derivatives.
    Bioorganic & medicinal chemistry letters, 2012, Sep-01, Volume: 22, Issue:17

    Topics: Anti-Infective Agents; Antitubercular Agents; Bacteria; Bacterial Infections; Fungi; Green Chemistry Technology; Halogenation; Humans; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Mycoses; Pyrazoles; Tuberculosis

2012
Synthesis and biological evaluation of novel benzimidazole derivatives and their binding behavior with bovine serum albumin.
    European journal of medicinal chemistry, 2012, Volume: 55

    Topics: Animals; Anti-Infective Agents; Bacteria; Benzimidazoles; Cattle; Chemistry Techniques, Synthetic; Fungi; Microbial Sensitivity Tests; Serum Albumin, Bovine; Thermodynamics

2012
Novel berberine triazoles: synthesis, antimicrobial evaluation and competitive interactions with metal ions to human serum albumin.
    Bioorganic & medicinal chemistry letters, 2013, Feb-15, Volume: 23, Issue:4

    Topics: Anti-Bacterial Agents; Antifungal Agents; Berberine; Binding, Competitive; Cations; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Metals; Microbial Sensitivity Tests; Serum Albumin; Triazoles

2013
An efficient domino reaction in ionic liquid: synthesis and biological evaluation of some pyrano- and thiopyrano-fused heterocycles.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Aldehydes; Anti-Bacterial Agents; Coumarins; Gram-Negative Bacteria; Gram-Positive Bacteria; Heterocyclic Compounds; Ionic Liquids; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Pyrans; Pyrazolones; Quinolines; Structure-Activity Relationship

2013
Synthesis and identification of β-aryloxyquinoline based diversely fluorine substituted N-aryl quinolone derivatives as a new class of antimicrobial, antituberculosis and antioxidant agents.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Anti-Infective Agents; Antioxidants; Antitubercular Agents; Artemia; Aspergillus fumigatus; Candida albicans; Dose-Response Relationship, Drug; Fluorine; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Models, Chemical; Molecular Structure; Mycobacterium tuberculosis; Ovum; Quinolines; Structure-Activity Relationship

2013
Synthesis and biological evaluation of a class of quinolone triazoles as potential antimicrobial agents and their interactions with calf thymus DNA.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Anti-Infective Agents; Bacteria; Cattle; DNA; DNA Replication; Drug Evaluation, Preclinical; Fungi; Intercalating Agents; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Quinolones; Spectrophotometry, Ultraviolet; Triazoles

2013
Synthetic tactics of new class of 4-aminothieno[2,3-d]pyrimidine-6-carbonitrile derivatives acting as antimicrobial agents.
    European journal of medicinal chemistry, 2013, Volume: 64

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzoxazines; Dose-Response Relationship, Drug; Fungi; Microbial Sensitivity Tests; Molecular Structure; Piperidines; Structure-Activity Relationship

2013
Design, synthesis and antimicrobial evaluation of novel benzimidazole type of Fluconazole analogues and their synergistic effects with Chloromycin, Norfloxacin and Fluconazole.
    European journal of medicinal chemistry, 2013, Volume: 64

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzimidazoles; Dose-Response Relationship, Drug; Drug Design; Drug Synergism; Fluconazole; Fungi; Microbial Sensitivity Tests; Norfloxacin; Structure-Activity Relationship

2013
Design and synthesis of biquinolone-isoniazid hybrids as a new class of antitubercular and antimicrobial agents.
    European journal of medicinal chemistry, 2013, Volume: 65

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Antitubercular Agents; Artemia; Bacteria; Dose-Response Relationship, Drug; Drug Design; Fungi; Isoniazid; Microbial Sensitivity Tests; Molecular Structure; Motor Activity; Quinolones; Structure-Activity Relationship; Tuberculosis

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Synthesis and biological evaluation of α-triazolyl chalcones as a new type of potential antimicrobial agents and their interaction with calf thymus DNA and human serum albumin.
    European journal of medicinal chemistry, 2014, Volume: 71

    Topics: Animals; Anti-Infective Agents; Bacteria; Bacterial Infections; Cattle; Chalcones; DNA; Fungi; Humans; Microbial Sensitivity Tests; Mycoses; Serum Albumin; Triazoles

2014
1,2,3-Triazole-derived naphthalimides as a novel type of potential antimicrobial agents: synthesis, antimicrobial activity, interaction with calf thymus DNA and human serum albumin.
    Bioorganic & medicinal chemistry letters, 2014, Jan-01, Volume: 24, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Bacteria; Cattle; DNA; DNA Replication; Dose-Response Relationship, Drug; Humans; Microbial Sensitivity Tests; Molecular Structure; Naphthalimides; Serum Albumin; Static Electricity; Structure-Activity Relationship; Triazoles

2014
Synthesis, characterization and pharmacological screening of some novel 5-imidazopyrazole incorporated polyhydroquinoline derivatives.
    European journal of medicinal chemistry, 2014, May-06, Volume: 78

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antimalarials; Bacteria; Dose-Response Relationship, Drug; Fungi; Microbial Sensitivity Tests; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymers; Pyrazoles; Quinolines; Structure-Activity Relationship

2014
Design, synthesis and characterization of fluoro substituted novel pyrazolylpyrazolines scaffold and their pharmacological screening.
    European journal of medicinal chemistry, 2014, Sep-12, Volume: 84

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antimalarials; Bacteria; Dose-Response Relationship, Drug; Drug Design; Fungi; Microbial Sensitivity Tests; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrazoles; Structure-Activity Relationship

2014
Novel morpholinoquinoline nucleus clubbed with pyrazoline scaffolds: Synthesis, antibacterial, antitubercular and antimalarial activities.
    European journal of medicinal chemistry, 2016, Apr-13, Volume: 112

    Topics: Anti-Infective Agents; Antimalarials; Antitubercular Agents; Bacteria; Bacterial Infections; Fungi; Humans; Malaria, Falciparum; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Mycoses; Plasmodium falciparum; Pyrazoles; Quinolines; Structure-Activity Relationship; Tuberculosis

2016
Novel 3-Aminothiazolquinolones: Design, Synthesis, Bioactive Evaluation, SARs, and Preliminary Antibacterial Mechanism.
    Journal of medicinal chemistry, 2016, 05-26, Volume: 59, Issue:10

    Topics: Animals; Anti-Bacterial Agents; Cell Line; Cell Proliferation; Cell Survival; DNA Gyrase; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; PC12 Cells; Quinolones; Rats; Structure-Activity Relationship; Thiazoles

2016
Design, synthesis and biological evaluation of berberine-benzimidazole hybrids as new type of potentially DNA-targeting antimicrobial agents.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: Animals; Anti-Infective Agents; Bacteria; Benzimidazoles; Berberine; Cattle; Cell Membrane Permeability; Chemistry Techniques, Synthetic; DNA; Drug Design; Fungi; Humans; Microbial Sensitivity Tests; Molecular Docking Simulation; Protein Conformation; Serum Albumin; Water

2016
Multi-targeting exploration of new 2-aminothiazolyl quinolones: Synthesis, antimicrobial evaluation, interaction with DNA, combination with topoisomerase IV and penetrability into cells.
    European journal of medicinal chemistry, 2016, Nov-29, Volume: 124

    Topics: Animals; Anti-Infective Agents; Biological Transport; Cattle; Cell Line; Cell Membrane Permeability; Chemistry Techniques, Synthetic; DNA; DNA Replication; DNA Topoisomerase IV; Drug Design; Kinetics; Mice; Microbial Sensitivity Tests; Molecular Docking Simulation; Permeability; Quinolones

2016
Synthesis and biological screening of novel 2-morpholinoquinoline nucleus clubbed with 1,2,4-oxadiazole motifs.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Anti-Infective Agents; Bacteria; Bacterial Proteins; Catalytic Domain; Chemistry Techniques, Synthetic; Drug Evaluation, Preclinical; Fungi; Microbial Sensitivity Tests; Molecular Docking Simulation; Oxadiazoles; Quinolines; Structure-Activity Relationship

2017
Novel benzimidazolyl tetrahydroprotoberberines: Design, synthesis, antimicrobial evaluation and multi-targeting exploration.
    Bioorganic & medicinal chemistry letters, 2017, 04-15, Volume: 27, Issue:8

    Topics: Animals; Anti-Infective Agents; Bacteria; Bacterial Infections; Benzimidazoles; Berberine Alkaloids; Cattle; DNA; Fungi; Humans; Microbial Sensitivity Tests; Molecular Docking Simulation; Mycoses

2017
Design, synthesis and antimicrobial evaluation of novel benzimidazole-incorporated sulfonamide analogues.
    European journal of medicinal chemistry, 2017, Aug-18, Volume: 136

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Benzimidazoles; Cattle; DNA; Dose-Response Relationship, Drug; Drug Design; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Molecular Structure; Serum Albumin; Structure-Activity Relationship; Sulfonamides

2017
1,2,4-Triazole and 1,3,4-oxadiazole analogues: Synthesis, MO studies, in silico molecular docking studies, antimalarial as DHFR inhibitor and antimicrobial activities.
    Bioorganic & medicinal chemistry, 2017, 08-01, Volume: 25, Issue:15

    Topics: Anti-Infective Agents; Antimalarials; Folic Acid Antagonists; Molecular Docking Simulation; Oxadiazoles; Spectrum Analysis; Triazoles

2017
Benzothiazole analogues: Synthesis, characterization, MO calculations with PM6 and DFT, in silico studies and in vitro antimalarial as DHFR inhibitors and antimicrobial activities.
    Bioorganic & medicinal chemistry, 2017, 10-15, Volume: 25, Issue:20

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antimalarials; Benzothiazoles; Cell Survival; Computer Simulation; Dose-Response Relationship, Drug; Folic Acid Antagonists; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Plasmodium falciparum; Quantum Theory; Schizosaccharomyces; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2017
Azoalkyl ether imidazo[2,1-b]benzothiazoles as potentially antimicrobial agents with novel structural skeleton.
    Bioorganic & medicinal chemistry letters, 2018, 08-01, Volume: 28, Issue:14

    Topics: Anti-Bacterial Agents; Antifungal Agents; Benzothiazoles; Dose-Response Relationship, Drug; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Quantum Theory; Structure-Activity Relationship

2018
Design, synthesis, and biological activity of novel ammonium salts containing sterically hindered phenolic fragment and phosphoryl group.
    MedChemComm, 2018, Dec-01, Volume: 9, Issue:12

    Topics:

2018
Structure based design, synthesis, and biological evaluation of imidazole derivatives targeting dihydropteroate synthase enzyme.
    Bioorganic & medicinal chemistry letters, 2021, 03-15, Volume: 36

    Topics: Anti-Bacterial Agents; Dihydropteroate Synthase; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Imidazoles; Ligands; Microbial Sensitivity Tests; Molecular Structure; Staphylococcus aureus; Structure-Activity Relationship; Vancomycin-Resistant Enterococci

2021
Comparative in vitro activity of enoxacin and other fluoroquinolones against multi-resistant strains of Salmonella typhi.
    Current medical research and opinion, 1992, Volume: 12, Issue:9

    Topics: Ampicillin; Anti-Infective Agents; Chloramphenicol; Drug Resistance, Microbial; Enoxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Norfloxacin; Pefloxacin; Quinolones; Salmonella typhi; Species Specificity; Trimethoprim, Sulfamethoxazole Drug Combination; Typhoid Fever

1992
Fluoroquinolone supersusceptibility mediated by outer membrane protein OprH overexpression in Pseudomonas aeruginosa: evidence for involvement of a nonporin pathway.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:11

    Topics: Anti-Infective Agents; Bacterial Outer Membrane Proteins; Cell Membrane; Chloramphenicol; Ciprofloxacin; Drug Resistance, Microbial; Fleroxacin; Gene Expression; Norfloxacin; Porins; Pseudomonas aeruginosa

1992
Occurrence of the nfxB type mutation in clinical isolates of Pseudomonas aeruginosa.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:11

    Topics: Carbenicillin; Chloramphenicol; Drug Resistance, Microbial; Genes, Bacterial; Gentamicins; Imipenem; Microbial Sensitivity Tests; Mutation; Norfloxacin; Phenotype; Plasmids; Pseudomonas aeruginosa; Transformation, Bacterial

1992
The problem of emerging chloramphenicol resistance in typhoid fever--a preliminary report.
    The Journal of the Association of Physicians of India, 1991, Volume: 39, Issue:6

    Topics: Chloramphenicol; Chloramphenicol Resistance; Disease Outbreaks; Humans; India; Microbial Sensitivity Tests; Norfloxacin; Salmonella typhi; Typhoid Fever

1991
Norfloxacin ophthalmic versus chloramphenicol in bacterial conjunctivitis and blepharoconjunctivitis.
    DICP : the annals of pharmacotherapy, 1990, Volume: 24, Issue:6

    Topics: Chloramphenicol; Conjunctivitis, Bacterial; Humans; Norfloxacin

1990
Cross-resistance to fluoroquinolones in multiple-antibiotic-resistant (Mar) Escherichia coli selected by tetracycline or chloramphenicol: decreased drug accumulation associated with membrane changes in addition to OmpF reduction.
    Antimicrobial agents and chemotherapy, 1989, Volume: 33, Issue:8

    Topics: Anti-Infective Agents; Bacterial Outer Membrane Proteins; Bacteriophages; Chloramphenicol; DNA, Bacterial; Drug Resistance, Microbial; Electrophoresis, Polyacrylamide Gel; Escherichia coli; Microbial Sensitivity Tests; Mutation; Norfloxacin; Tetracycline

1989
Evaluation of the in vitro bactericidal action of ciprofloxacin on cells of Escherichia coli in the logarithmic and stationary phases of growth.
    Antimicrobial agents and chemotherapy, 1985, Volume: 28, Issue:4

    Topics: Chloramphenicol; Ciprofloxacin; Drug Interactions; Escherichia coli; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Norfloxacin; Quinolines; Time Factors

1985
[Comparative efficacy of ampicillin, chloramphenicol, cefotaxime, ceftriaxone and pefloxacin in experimental Salmonella typhimurium infection].
    Pathologie-biologie, 1987, Volume: 35, Issue:9

    Topics: Ampicillin; Animals; Anti-Bacterial Agents; Cefotaxime; Ceftriaxone; Chloramphenicol; Female; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Norfloxacin; Pefloxacin; Salmonella Infections, Animal; Salmonella typhimurium

1987
Evaluation of pefloxacin in experimental Escherichia coli meningitis.
    Antimicrobial agents and chemotherapy, 1986, Volume: 29, Issue:3

    Topics: Animals; Anti-Infective Agents; Cefotaxime; Chloramphenicol; Escherichia coli Infections; Humans; Meningitis; Microbial Sensitivity Tests; Norfloxacin; Pefloxacin; Rabbits; Time Factors

1986
Antimicrobial activity of norfloxacin in enteric and urinary tract infections: combined effect of norfloxacin with aminoglycosides, tetracycline and chloramphenicol.
    Drugs under experimental and clinical research, 1986, Volume: 12, Issue:4

    Topics: Acinetobacter; Aminoglycosides; Anti-Bacterial Agents; Bacterial Infections; Chloramphenicol; Drug Combinations; Enterobacteriaceae; Gastrointestinal Diseases; Humans; Microbial Sensitivity Tests; Norfloxacin; Pipemidic Acid; Pseudomonas; Tetracycline; Urinary Tract Infections

1986
In vitro susceptibility of pathogenic Vibrio species to norfloxacin and six other antimicrobial agents.
    Antimicrobial agents and chemotherapy, 1985, Volume: 28, Issue:3

    Topics: Ampicillin; Chloramphenicol; Gentamicins; In Vitro Techniques; Microbial Sensitivity Tests; Nalidixic Acid; Norfloxacin; Sulfamethoxazole; Tetracycline; Trimethoprim; Vibrio

1985
Role of efflux pump(s) in intrinsic resistance of Pseudomonas aeruginosa: resistance to tetracycline, chloramphenicol, and norfloxacin.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:8

    Topics: Chloramphenicol; Chloramphenicol Resistance; Drug Resistance, Microbial; Membrane Proteins; Mutation; Norfloxacin; Pseudomonas aeruginosa; Tetracycline; Tetracycline Resistance

1994
The accumulation of five antibacterial agents in porin-deficient mutants of Escherichia coli.
    The Journal of antimicrobial chemotherapy, 1993, Volume: 32, Issue:2

    Topics: Anti-Infective Agents; Cefoxitin; Cephalosporins; Chloramphenicol; Escherichia coli; Microbial Sensitivity Tests; Mutation; Norfloxacin; Phenotype; Porins; Tetracycline

1993
Role of mexA-mexB-oprM in antibiotic efflux in Pseudomonas aeruginosa.
    Antimicrobial agents and chemotherapy, 1995, Volume: 39, Issue:9

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacterial Outer Membrane Proteins; Chloramphenicol; DNA Transposable Elements; Microbial Sensitivity Tests; Norfloxacin; Operon; Penicillin G; Penicillins; Pseudomonas aeruginosa; Tetracycline

1995
Overexpression of the mexC-mexD-oprJ efflux operon in nfxB-type multidrug-resistant strains of Pseudomonas aeruginosa.
    Molecular microbiology, 1996, Volume: 21, Issue:4

    Topics: Amino Acid Sequence; Anti-Bacterial Agents; Bacterial Outer Membrane Proteins; Bacterial Proteins; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Chloramphenicol; Cloning, Molecular; DNA-Binding Proteins; Drug Resistance, Microbial; Drug Resistance, Multiple; Gene Expression Regulation, Bacterial; Genes, Bacterial; Ionophores; Molecular Sequence Data; Norfloxacin; Operon; Point Mutation; Pseudomonas aeruginosa; Transcription Factors

1996
Dependence of peptidoglycan metabolism on phospholipid synthesis during growth of Escherichia coli.
    Microbiology (Reading, England), 1996, Volume: 142 ( Pt 10)

    Topics: Ampicillin; Ampicillin Resistance; Cerulenin; Chloramphenicol; Enzyme Inhibitors; Escherichia coli; Glycerol; Guanosine Tetraphosphate; Norfloxacin; Penicillins; Peptidoglycan; Phospholipids; Protein Synthesis Inhibitors; Topoisomerase II Inhibitors

1996
Active efflux of antimicrobial agents in wild-type strains of enterococci.
    Antimicrobial agents and chemotherapy, 1997, Volume: 41, Issue:4

    Topics: Anti-Bacterial Agents; Chloramphenicol; Enterococcus faecalis; Enterococcus faecium; Microbial Sensitivity Tests; Norfloxacin; Tetracycline

1997
[The drug susceptibility pattern of the presumed etiologic agents of infectious enteritis including verotoxin-producing Escherichia coli O-157].
    The Japanese journal of antibiotics, 1997, Volume: 50, Issue:10

    Topics: Aerobiosis; Ampicillin; Anaerobiosis; Anti-Bacterial Agents; Anti-Infective Agents; Campylobacter jejuni; Cefaclor; Cephalosporins; Chloramphenicol; Drug Resistance, Microbial; Enteritis; Escherichia coli O157; Fosfomycin; Humans; Microbial Sensitivity Tests; Minocycline; Norfloxacin; Penicillins; Salmonella; Tetracycline; Vibrio parahaemolyticus

1997
Antimicrobial resistance of Enterococci in Lebanon.
    International journal of antimicrobial agents, 2001, Volume: 17, Issue:3

    Topics: Aminoglycosides; Ampicillin; Anti-Bacterial Agents; Anti-Infective Agents; Chloramphenicol; Ciprofloxacin; Drug Resistance, Microbial; Enterococcus; Erythromycin; Gentamicins; Humans; Lebanon; Microbial Sensitivity Tests; Norfloxacin; Penicillins; Rifampin; Streptomycin; Teicoplanin; Tetracycline; Vancomycin

2001
Antibiotic susceptibility pattern of Salmonella worthington isolated from neonates--a retrospective study.
    Japanese journal of infectious diseases, 2002, Volume: 55, Issue:2

    Topics: Amikacin; Anti-Bacterial Agents; Anti-Infective Agents; Cefotaxime; Chloramphenicol; Ciprofloxacin; Drug Resistance, Multiple, Bacterial; Humans; Infant, Newborn; Infant, Newborn, Diseases; Meningitis; Norfloxacin; Penicillins; Prevalence; Retrospective Studies; Salmonella; Salmonella Infections; Sepsis; Time Factors

2002
Microsporidial keratoconjunctivitis in healthy individuals: a case series.
    Ophthalmology, 2003, Volume: 110, Issue:7

    Topics: Adolescent; Adult; Albendazole; Antiprotozoal Agents; Chloramphenicol; Cornea; Cyclohexanes; Drug Therapy, Combination; Eye Infections, Parasitic; Fatty Acids, Unsaturated; HIV Seronegativity; Humans; Keratoconjunctivitis; Male; Microsporidiosis; Norfloxacin; Retrospective Studies; Sesquiterpenes

2003
[Activity of fosfomycin against Escherichia coli O157:H7--morphological changes and production of Shiga toxins].
    The Japanese journal of antibiotics, 2003, Volume: 56, Issue:6

    Topics: Ampicillin; Anti-Bacterial Agents; Bacteriolysis; Cell Wall; Chloramphenicol; Dose-Response Relationship, Drug; Escherichia coli O157; Fosfomycin; Kanamycin; Norfloxacin; Shiga Toxins

2003
Antibiotic sensitivity patterns among Indian strains of avian Pasteurella multocida.
    Tropical animal health and production, 2004, Volume: 36, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Chloramphenicol; Doxycycline; Enrofloxacin; Fluoroquinolones; India; Lincomycin; Microbial Sensitivity Tests; Norfloxacin; Pasteurella Infections; Pasteurella multocida; Poultry; Poultry Diseases; Quinolones; Species Specificity; Sulfadiazine

2004
The use of quinolones in the treatment of acute bacterial diarrhea: a comparative therapeutic trial.
    Journal of chemotherapy (Florence, Italy), 1989, Volume: 1, Issue:4 Suppl

    Topics: Acute Disease; Adolescent; Anti-Infective Agents; Bacteria; Bacterial Infections; Chloramphenicol; Diarrhea; Feces; Female; Humans; Male; Norfloxacin; Quinolones; Randomized Controlled Trials as Topic; Tetracycline; Trimethoprim, Sulfamethoxazole Drug Combination

1989
Determination of selected antibiotics in the Victoria Harbour and the Pearl River, South China using high-performance liquid chromatography-electrospray ionization tandem mass spectrometry.
    Environmental pollution (Barking, Essex : 1987), 2007, Volume: 145, Issue:3

    Topics: Amoxicillin; Anti-Bacterial Agents; China; Chloramphenicol; Chromatography, High Pressure Liquid; Climate; Erythromycin; Hong Kong; Macrolides; Norfloxacin; Ofloxacin; Quinolones; Rivers; Seasons; Seawater; Spectrometry, Mass, Electrospray Ionization; Sulfanilamides; Time Factors; Waste Management; Water Pollutants, Chemical

2007
An alkylaminoquinazoline restores antibiotic activity in Gram-negative resistant isolates.
    Microbiology (Reading, England), 2011, Volume: 157, Issue:Pt 2

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Chloramphenicol; Drug Resistance, Multiple, Bacterial; Fluoroquinolones; Gram-Negative Bacteria; Membrane Transport Proteins; Microbial Sensitivity Tests; Nalidixic Acid; Norfloxacin; Quinazolines

2011
Treatment of microsporidial keratoconjunctivitis with repeated corneal swabbing.
    American journal of ophthalmology, 2012, Volume: 154, Issue:6

    Topics: Adult; Aged; Anti-Bacterial Agents; Chloramphenicol; Cornea; DNA, Bacterial; Drug Therapy, Combination; Eye Infections, Fungal; Female; Humans; Keratoconjunctivitis; Male; Microsporidia; Microsporidiosis; Middle Aged; Norfloxacin; Polymerase Chain Reaction; Retrospective Studies; RNA, Bacterial; RNA, Ribosomal, 16S; Surgical Sponges; Young Adult

2012
Phytotoxicity of veterinary antibiotics to seed germination and root elongation of crops.
    Ecotoxicology and environmental safety, 2016, Volume: 126

    Topics: Animals; Anti-Bacterial Agents; Chloramphenicol; Crops, Agricultural; Cucumis sativus; Daucus carota; Erythromycin; Germination; Lactuca; Norfloxacin; Plant Roots; Quantitative Structure-Activity Relationship; Seeds; Soil Pollutants; Solanum lycopersicum; Sulfamethazine; Tetracycline; Veterinary Drugs

2016
Assessment of altered binding specificity of bacteriophage for ciprofloxacin-induced antibiotic-resistant Salmonella Typhimurium.
    Archives of microbiology, 2016, Volume: 198, Issue:6

    Topics: Ampicillin; Anti-Bacterial Agents; Bacterial Proteins; Bacteriophages; beta-Lactamases; Binding Sites; Chloramphenicol; Ciprofloxacin; Drug Resistance, Multiple, Bacterial; Membrane Transport Proteins; Microbial Sensitivity Tests; Norfloxacin; Salmonella typhimurium; Tetracycline; Trans-Activators

2016
Combined treatment of UVA irradiation and antibiotics induces greater bactericidal effects on Vibrio parahaemolyticus.
    The journal of medical investigation : JMI, 2016, Volume: 63, Issue:1-2

    Topics: Ampicillin; Anti-Bacterial Agents; Chloramphenicol; Disinfection; Gentamicins; Humans; Norfloxacin; Ultraviolet Rays; Vibrio parahaemolyticus

2016
Designation of pathogenic resistant bacteria in the Sparusaurata sea collected in Tunisia coastlines: Correlation with high performance liquid chromatography-tandem mass spectrometry analysis of antibiotics.
    Microbial pathogenesis, 2017, Volume: 106

    Topics: Amoxicillin; Animals; Anti-Bacterial Agents; Aquaculture; Bacteria; Chloramphenicol; Chromatography, High Pressure Liquid; Colistin; DNA, Bacterial; Drug Resistance, Multiple, Bacterial; Fish Diseases; Fisheries; Food Contamination; Fusidic Acid; Microbial Sensitivity Tests; Norfloxacin; Sea Bream; Seafood; Seawater; Tandem Mass Spectrometry; Tunisia; Vibrio alginolyticus; Vibrio Infections; Vibrio parahaemolyticus; Water Pollutants, Chemical

2017
Occurrence, virulence genes, and antimicrobial profiles of Escherichia coli O157 isolated from ruminants slaughtered in Al Ain, United Arab Emirates.
    BMC microbiology, 2020, 07-16, Volume: 20, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Camelus; Cattle; Cefotaxime; Chloramphenicol; Ciprofloxacin; Escherichia coli Infections; Escherichia coli Proteins; Feces; Female; Food Microbiology; Goats; Male; Microbial Sensitivity Tests; Norfloxacin; Polymyxin B; Prevalence; Ruminants; Sheep; Shiga-Toxigenic Escherichia coli; United Arab Emirates; Virulence Factors

2020
Isolation, identification, and antimicrobial susceptibility pattern of Campylobacter jejuni and Campylobacter coli from cattle, goat, and chicken meats in Mekelle, Ethiopia.
    PloS one, 2021, Volume: 16, Issue:2

    Topics: Amoxicillin; Ampicillin; Animals; Anti-Bacterial Agents; Campylobacter coli; Campylobacter Infections; Campylobacter jejuni; Cattle; Chickens; Chloramphenicol; Cross-Sectional Studies; Drug Resistance, Multiple, Bacterial; Erythromycin; Ethiopia; Goats; Meat; Microbial Sensitivity Tests; Norfloxacin; Prevalence; Streptomycin; Sulfamethoxazole; Trimethoprim

2021
Simultaneous removal of norfloxacin and chloramphenicol using cold atmospheric plasma jet (CAPJ): Enhanced performance, synergistic effect, plasma-activated water (PAW) contribution, mechanism and toxicity evaluation.
    Journal of hazardous materials, 2023, 06-15, Volume: 452

    Topics: Anti-Bacterial Agents; Chloramphenicol; Humans; Norfloxacin; Plasma Gases; Reactive Nitrogen Species; Reactive Oxygen Species; Water

2023