nordazepam and diazepam

nordazepam has been researched along with diazepam in 379 studies

Research

Studies (379)

TimeframeStudies, this research(%)All Research%
pre-1990240 (63.32)18.7374
1990's69 (18.21)18.2507
2000's31 (8.18)29.6817
2010's30 (7.92)24.3611
2020's9 (2.37)2.80

Authors

AuthorsStudies
Collins, RJ; Gall, M; Kamdar, BV1
Blair, T; Webb, GA1
Aoyama, T; Ichikawa, H; Suzuki, Y1
Blanton, CD; Fatmi, AA; Iturrian, WB; Vaidya, NA1
Lukovits, I1
Babbini, M; Barbaro, AM; Bartoletti, M; Biagi, GL; Borea, PA; Gaiardi, M; Guerra, MC1
Lopata, A; Lukovits, I1
Johnston, GA; Maddalena, DJ1
Karplus, M; So, SS1
Ghuloum, AM; Jain, AN; Sage, CR1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Topliss, JG; Yoshida, F1
Ertl, P; Rohde, B; Selzer, P1
Artursson, P; Luthman, K; Norinder, U; Stenberg, P1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Caron, G; Ermondi, G1
Fitos, I; Mády, G; Simonyi, M; Visy, J; Zsila, F1
Du-Cuny, L; Huwyler, J; Kansy, M; Wiese, M1
Lombardo, F; Obach, RS; Waters, NJ1
Campillo, NE; Guerra, A; Páez, JA1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC1
Clarke, CH; Ferres, HM; Nicholson, AN; Stone, BM1
Golovenko, NIa; Zin'kovskii, VG1
Erkkola, R; Kangas, L; Kanto, J; Piiroinen, O1
Andreoli, V; Maffei, F; Montanaro, N; Morandini, G1
Pape, BE; Ribick, MA1
de Angelis, L; Traversa, U; Vertua, R1
Bertler, A; Lindgren, S; Malmgren, H; Post, C1
Dorrity, F; Linnoila, M1
Greenblatt, DJ2
Greenblatt, DJ; Shader, RI1
Linnoila, M; Viukari, M1
Allen, MD; Georgotas, A; Greenblatt, DJ; Harmatz, JS; Shader, RI1
Airoldi, L; Lanzoni, J; Marcucci, F; Mussini, E1
Baird, ES; Hailey, DM1
Allen, MD; Bodem, G; Greenblatt, DJ; Harmatz, JS; Ochs, HR; Shader, RI1
de Angelis, L; File, SE1
Baars, AM; Hekster, YA; O'Reilly, WJ; van der Kleijn, E; Vree, TB1
Georgotas, A; Greenblatt, DJ; Harmatz, JS; Shader, RI1
't Hart, BJ; de Gier, JJ1
Bugge, A1
Fresia, P; Govoni, S; Spano, PF; Trabucchi, M1
Das, S; Datta, SC; Dey, S; Guin, AK; Sengupta, D1
Kangas, L; Korttila, K1
Antonin, KH; Bieck, PR; Brügel, H; Klotz, U1
Cesco, G; Fabbruci, I; Giannico, S; Montanaro, N; Scaggiante, L1
Lader, M1
Rutherford, DM1
Clarke, CH; Nicholson, AN2
Klotz, U2
Khoo, KC; Posmanter, HN; Puglisi, CV; Weinfeld, RE1
Airoldi, L; Facchinetti, T; Garattini, S; Marcucci, F; Mussini, E1
Cano, JP; Reynier, JP; Rispe, R; Viala, A1
Steyn, JM; van der Merew, PJ1
Kabra, PM; Marton, LJ; Stevens, GL1
Brodie, RR; Chasseaud, LF; Taylor, T1
Perchalski, RJ; Wilder, BJ1
Cleary, W; Eng, L; McMillan, S; Missen, AW1
Okoko, A; Rutherford, DM; Tyrer, PJ1
Haataja, M; Hurme, P; Kanto, J; Sellman, R1
Ishihama, H; Kimata, H1
Ishihama, H; Kimata, H; Matsumoto, S1
Allen, MD; Greenblatt, DJ; Orsulak, PJ; Shader, RI; Woo, E1
Sun, SR1
Babbini, M; Bartoletti, M; Gaiardi, M1
Helmsing, PJ; van der Woude, J; van Eupen, OM1
Bredesen, JE; Langslet, A; Lunde, PK; Meberg, A2
Konishi, M1
Klotz, U; Müller-Seydlitz, P1
Dhar, AK; Kutt, H1
Cohen, ME; Duffner, PK; Jusko, WJ; MacKichan, JJ1
Bartenbach, D; Carrigan, PJ1
Kanto, J; Mäenpää, M; Mäntylä, R; Sellman, R; Valovirta, E1
Schwertner, HA; Shimek, EL; Wallace, JE1
Miller, F; Nulsen, J1
Aderjan, R; Schmidt, G1
Delaney, M; Dixon, R; Earley, J; Glover, W1
Sellers, EM; Wong, GB1
Cook, L; Grodsky, FS; Sepinwall, J1
Allen, MD; Greenblatt, DJ; MacLaughlin, DS; Sahder, RI; Weinberger, DR1
Brooks, MA; Dixon, R; Hackman, MR; Moore, JD; Postma, E; Schwartz, MA; Spector, S1
Antonin, KH; Bieck, PR; Klotz, U1
Alberti, GG; De Maio, D; Franciosi, P; Gomeni, R; Scieghi, G; Tognoni, G1
Hanifl, E; Rosenmund, H; Wad, N1
Beischlag, TV; Inaba, T; Kalow, W; Mahon, WA1
Constant, H; Duthel, JM; Miachon, S; Rochet, T; Vallon, JJ1
Guentert, TW; Stebler, T2
Chiba, K; Ishizaki, T; Jang, IJ; Kusaka, M; Shin, JG; Shin, SG; Sohn, DR1
Bruce, I; Hooper, WD; Reilly, PE1
de la Rey, N; Hundt, HK; Luus, HG; Meyer, BH; Müller, FO; Röthig, HJ1
Basile, AS; Harrison, PM; Hughes, RD; Jones, EA; Murata, Y; Pannell, L; Skolnick, P; Williams, R1
Dickey, KM; Martin, WR; Sloan, JW; Wala, E1
Martin, WR; Sloan, JW; Wala, EP2
Corcoran, KD; Lukey, BJ; Solana, RP1
Anthenelli, RM; Blunt, B; Monteiro, MG; Schuckit, MA1
Hooper, WD; Mason, SR; Reilly, PE; Thompson, DA1
Benazzi, F1
Hole, K; Rosland, JH1
Wong, PT1
Andersson, T; Cederberg, C; Edvardsson, G; Heggelund, A; Lundborg, P1
Dusci, LJ; Good, SM; Hall, RW; Ilett, KF1
Caccia, S; Conti, I; Tridico, RV1
Heikkinen, H; Heinälä, P; Piepponen, T1
Eckardt, MJ; Granger, A; Lane, E; Linnoila, M; Lister, R; Moss, H; Stapleton, JM1
Andersson, T; Andrén, K; Cederberg, C; Edvardsson, G; Heggelund, A; Lundborg, P1
Camsonne, R1
Bertilsson, L; Henthorn, TK; Sanz, E; Säwe, J; Tybring, G; Villén, T1
Klotz, U; Unseld, E1
Kubo, H; Miura, H; Nishida, A; Nishikawa, T; Ohtani, H; Sudo, Y; Sunaoshi, W1
Fischer, C; Klotz, U; Krishna, DR; Unseld, E1
Chenery, RJ; Lockwood, GF; Seddon, T1
Corrie, JE; Dowie, LJ; Fraser, R; Gray, CE; Holloway, CD; Kenyon, CJ1
Friedman, H; Greenblatt, DJ; Harmatz, JS; Locniskar, A; Shader, RI1
D'Eramo, C; Iacovelli, W; Salvadori, A; Stocchetti, N1
Iwaya, N; Miyoshi, K; Morita, Y1
Appel, M; Bron, HN; Hooymans, PM; Janknegt, R1
Benetello, P; Bertin, I; Colombo, G; Furlanut, M1
Fassbender, CP; Hönack, D; Löscher, W1
D'Eramo, C; Maestri, D; Tirelli, F2
Klockowski, PM; Levy, G3
Bertolissi, M; de Angelis, L; Della Loggia, R; Nardini, G; Traversa, U; Vertua, R1
Bergert, RJ; Deutsch, DG; Soo, VA1
Spealman, RD2
Greenblatt, DJ; Harmatz, JS; Locniskar, A; Shader, RI; Zinny, MA1
Bareggi, SR; Leva, S; Lorini, M; Nielsen, NP; Pirola, R; Zecca, L1
Greenblatt, DJ; Locniskar, A; Ochs, HR; Weinbrenner, J1
Bertolotti, G; Galdangelo, F; Mazzuero, G; Tavazzi, L; Zotti, AM1
Barone, D; Garattini, S; Gobbi, M; Mennini, T1
D'Eramo, C; Follini, L; Stocchetti, N; Taverna, A; Zennaro, F1
Dammann, HG; Gottlieb, W; Keohane, PP; Klotz, U1
Badian, M; Hundt, HK; Joubert, AL; Luus, HG; Meyer, BH; Müller, FO1
Bareggi, SR; Leva, S; Pirola, R; Smirne, S; Truci, G; Zecca, L1
Bareggi, SR; Leva, S; Pirola, R; Smirne, S; Truci, G1
Boxenbaum, HG; Divoll, MK; Greenblatt, DJ; Harmatz, JS; Shader, RI; Soong, MH1
Corbo, M; Struzziero, E; Zeppa, G1
Cafaggi, G; Ciotola, G; Ciritella, P; Di Gregorio, AM; Scafuro, M1
Maurer, R; Möhler, H; Ranalder, U; Schmidt, K; Vetter, W; Wildmann, J1
De Blas, AL; Fales, HM; Friedrich, P; Sangameswaran, L1
Laufen, H; Leitold, M; Räder, K; Yeates, RA1
Abernethy, DR; Friedman, H; Greenblatt, DJ; Shader, RI1
Hasselstrøm, L; Ostergård, D; Ravnborg, M1
Gwee, MC; Lee, HS; Wong, PT; Yoong, YL1
Brase, DA; Dewey, WL; Glennon, RA; Young, R1
Cowen, PJ; Franklin, M; Fraser, S; Gosden, B; Murdock, P; Nutt, DJ1
Gumulka, SW; Janicki, PK; Jedrzejowska, H; Pisarski, W; Rewekant, M1
Cone, EJ; Darwin, WD; Gorodetzky, CW; Griffiths, RR; Preston, KL1
Bonanzinga, M; De Domenico, P; Di Perri, R; Gallitto, G; Musolino, R; Sacchi, C; Troilo, G1
Ecobichon, DJ; Ungar, W1
Chan, M; Ko, W; Kumana, CR; Lauder, IJ; Lin, HJ1
Dolan, S; Lau, CE; Tang, M1
Alazia, M; Cano, JP; Crevat-Pisano, P; Drouet, C; Francois, G; Lacarelle, B1
Kanto, J; Scheinin, M1
Hole, K; Hunskaar, S; Rosland, JH1
Bareggi, SR; Ferrario, P; Pirola, R; Zecca, L1
Boisse, NR; Guarino, JJ; Samoriski, GM1
Igarashi, T; Kitagawa, H; Ohmori, S; Okiyama, M; Ueno, K1
Bergstrom, RF; Bosomworth, JC; Lemberger, L; Rowe, H; Tenbarge, JB1
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E1
Beightol, LA; Farthing, D; Karnes, HT; Serafin, RJ1
Imamura, T; Kimura, K; Kudo, K; Nagata, T; Noda, M1
García Ruiz, A; Gómez Luque, A; Martos Crespo, F; Sánchez de la Cuesta, F1
Brown, C; File, SE; Greenblatt, DJ; Martin, IL1
Clarke, P; Ewen, JM; Stevenson, IH; Swift, CG1
Moroji, T; Motomura, H; Noguchi, T; Sekiguchi, R; Tada, K1
Berwish, NJ; Bond, WS; Swift, B1
Löscher, W; Schwark, WS1
Gugler, R; Jensen, JC1
Martin, WR; McNicholas, LF; Pruitt, TA1
Lee, HS; Low, PS; Quak, SH; Ti, TY; Wong, HB1
Ellinwood, EH; Heatherly, D; Nikaido, A1
Davenport, R; Haidukewych, D; Rodin, EA1
Meeles, MT; Thys, CP; Tjaden, UR; van der Kaay, M1
Paradiso, L; Rapisarda, V1
Dudkiewicz, J; Misterek, K1
Vozeh, S1
El-Hazmi, MA1
Ballabio, M; Caccia, S; Carli, M; Garattini, S; Samanin, R1
Burrows, GD; Fulton, A; Maguire, KP; Norman, TR1
Ciraulo, DA; Divoll, M; Georgotas, A; Greenblatt, DJ; Harmatz, JS; Shader, RI1
Ciraulo, DA; Greenblatt, DJ; Harmatz, JS; Shader, RI1
Dorow, RG; Schneider, HH; Seidler, J1
Caccia, S; Cotecchia, S; Garattini, S; Mennini, T1
Greenblatt, DJ; Knüchel, M; Locniskar, A; Ochs, HR; Steinhaus, E1
Nicholson, AN1
Kostowski, W; Lipińska, T; Puciłowski, O; Płaźnik, A; Trzaskowska, E1
Löscher, W1
Henderson, JG1
Hashimoto, S; Mizobuchi, M; Momose, T; Sakurai, E; Takahashi, S; Yamamoto, K1
Cocchi, R; Macci, F; Passanisi, S1
Colin, P; Lelorier, J; Sirois, G1
Coffey, B; Greenblatt, DJ; Shader, RI1
Greenblatt, DJ; Kaschell, HJ; Ochs, HR; Rauh, HW1
Betts, T; Crowe, A; Hawksworth, G; Knight, R; Nyemitei-Addo, I; Parry, K; Parsons, A; Petrie, JC; Raffle, A1
Käferstein, H; Norpoth, T; Staak, M; Sticht, G1
Allison, S; Greenblatt, DJ; Harmatz, JS; Locniskar, A; Pary, RJ; Shader, RI1
Arcidiacono, G; Cappelli, N; Cuoci, L; Fornaro, P; Guarneri, M; Moggi, G; Pacifici, GM; Placidi, GF1
Greenblatt, DJ; Locniskar, A; Ochs, HR; Verburg-Ochs, B1
Itoh, N; Mimaki, T; Ono, J; Tagawa, T; Tanaka, J; Terada, H; Yabuuchi, H1
Dawling, S; Flanagan, RJ; Moreton, K; Riley, P; Treasaden, I; Tyrer, P1
Agrawal, KK; Gupta, A; Tayal, G; Tekur, U1
Greenblatt, DJ; Martyn, JA; Quinby, WC1
Eckardt, B; Greenblatt, DJ; Harmatz, JS; Ochs, HR; Shader, RI1
Abernethy, DR; Divoll, M; Greenblatt, DJ; Ochs, HR; Shader, RI1
Brendle, A; Erwin, CW; Linnoila, M; Simpson, D1
Ochs, HR2
de Gier, JJ; t Hart, BJ; Wilting, J1
Kuhnz, W; Nau, H1
Greenblatt, DJ; Locniskar, A; Shader, RI1
Ballabio, M; Caccia, S; Garattini, S; Guiso, G; Reginato, R1
Colburn, WA; Jack, ML1
Colburn, WA; Wills, RJ1
Kuhnz, W; Luck, W; Nau, H1
Colburn, WA; Cotler, S; Gustafson, JH1
Abernethy, DR; Greenblatt, DJ; Harmatz, JS; Morse, DS; Shader, RI1
Case, WG; Dixon, R; Downing, RW; Fridman, R; Rickels, K1
Ghoneim, MM; Hinrichs, JV; Mewaldt, SP1
Kuhnz, W; Luck, W; Nau, H; Wegener, S1
Booij, LH; Crul, JF; Driessen, JJ; van Egmond, J; Vree, TB1
Greenblatt, DJ; Ochs, HR; Verburg-Ochs, B1
Busto, U; Harrison, M; Kaplan, HL; Naranjo, CA; Sellers, EM1
Cuoci, L; Pacifici, GM; Placidi, GF1
Rickels, K; Winokur, A1
Frey, HH; Philippin, HP; Scheuler, W1
McCurdy, HH; Rhodes, PJ; Rhodes, RS1
Aranko, K; Aranko, S; Mattila, MJ; Seppälä, T1
Bjornsson, TD; Kitchell, BB; Linnoila, M; Routledge, PA; Shand, DG; Skinner, T1
Abel, JG; Giles, HG; Naranjo, CA; Sellers, EM1
Klotz, U; Reimann, I3
Hallstrom, C; Lader, MH1
Kolenda, KD1
Allen, MD; Greenblatt, DJ; Harmatz, JS; Shader, RI1
Müller, FO; Steyn, JM1
Coffman, WB; McFarland, SA; Meyer, EA; Mumford, R; Wynn, RL1
Dietrichson, P; Lossius, R; Lunde, PK1
Dextraze, PG; Diamond, I; Foreman, JM; Griffiths, WC1
Greenblatt, DJ; Lloyd, BL; Ochs, HR1
Friel, PN; Graaff, PR; Opheim, KE; Raisys, VA; Wilensky, AJ1
Harris, SC; Shimek, EL; Wallace, JE1
Elsass, P; Hansen, T; Hendel, J; Hvidberg, EF; Møller, IW; Sørensen, KH1
Elsass, P; Gymoese, E; Hansen, T; Hendel, J; Hvidberg, EF; Rathje, J1
Nel, P; Walters, L1
Stenchever, MA; Williamson, RA1
Allen, MD; Greenblatt, DJ; Harmatz, JS; Laughren, TP; Shader, RI1
Abernethy, DR; Greenblatt, DJ1
Divoll, M; Greenblatt, DJ; Lacasse, Y; Shader, RI1
Britt, RH; Conley, FK; Hollister, LE; Shuer, L1
Bittencourt, PR; Richens, A; Smith, AT; Wade, P1
Cazzullo, CL; Scarone, S; Strambi, LF1
Dumont, CH; Rangno, RE; Sitar, DS1
Dhillon, S; Richens, A2
Divoll, M; Greenblatt, DJ1
Bowden, CL; Fisher, JG1
Gustafson, JH; Holazo, AA; Kaplan, SA; Khoo, KC; Weinfeld, RE; Weissman, L1
Dixon, R1
Greenblatt, DJ; Lauven, PM; Ochs, HR; Rommelsheim, K; Stoeckel, H1
Fornaro, P; Gomeni, R; Pacifici, GM; Placidi, GF1
Abernethy, DR; Divoll, M; Greenblatt, DJ; Shader, RI1
Bosatra, A; Poli, P; Vertua, R1
Frey, HH; Löscher, W1
Battey, YW; Greenblatt, DJ; Laughren, TP1
Bondiolotti, GP; Carruba, MO; Corli, O; Galva, MD; Picotti, GB1
Aoyagi, N; Ejima, A; Kaniwa, N; Koibuchi, M; Nishida, Y; Ogata, H; Ogawa, Y; Shibazaki, T; Shimamoto, T; Uda, Y; Yashiki, T1
Richter, K; Scherber, A1
Greenblatt, DJ; Rickels, K; Schatz, NJ; Snyder, PJ; Winokur, A1
Yang, SK1
Chiba, K; Chiba, T; Hirano, T; Horii, H; Ishizaki, T; Kato, Y1
Jing, X; Sloan, JW; Wala, EP2
Caraco, Y; Tateishi, T; Wood, AJ1
Chiba, K; Hayashi, M; Horai, Y; Ishizaki, T; Koyama, E; Manabe, K; Tomono, Y; Toyoki, T; Yamato, C; Yasuda, S1
Conjeevaram, HS; Kaminsky-Russ, K; Mullen, KD1
Ambre, J; de Wit, H; Dudish, S1
Desor, D; Humbert, AC; Koziel, V; Nehlig, A; Schroeder, H1
Capra, C; Casella, G; Costagli, V; Ramella, G; Sogni, A1
Barel, S; Bialer, M; Cipolla, G; Gatti, G; Gips, M; Perucca, E; Soback, S; Spina, E1
Andersson, T; Birkett, DJ; Miners, JO; Veronese, ME1
Aantaa, R; Himberg, JJ; Kanto, J; Katila, A; Kirvelä, O1
Basile, AS; Gu, ZQ; Harrison, PM; Hughes, RD; Jones, EA; McKinney, A; Pannell, L; Williams, R1
Ihara, N; Kokufu, T; Nosaka, K; Ohta, T; Sugioka, N1
Kamali, F1
Pang, KS; St-Pierre, MV1
Alcorn, J; Papich, MG1
Lu, Y; Pan, B; Wang, D1
Franke, M; Kingston, HM; Winek, CL1
Chaba, P; Dziklińska, A; Kur, E; Matsumoto, H; Skalski, M; Stencka, K; Szelenberger, W; Wasilewski, D; Woźny, E1
Sloan, JW; Wala, EP1
Jindrová, O; Lamka, J1
Berry, D; Fernandes, C; File, SE1
Baldinelli, L; Consolati, E; Cordioli, G; Galzigna, L; Luisetto, F; Manani, G1
Garretty, DJ; Hay, AW; Raistrick, D; Wolff, K1
Dressler, C; Franke, KP; Herzig, M; Nagel, U1
Baris, BA; Gardner, MJ; Preskorn, SH; Wilner, KD1
Bolognesi, R; Conti, M; Manca, C; Tsialtas, D; Vasini, P1
Court, MH; Greenblatt, DJ; Norman, WM1
Camaris, C; Little, D1
Gunaratna, C; Kissinger, PT1
Camara, P; Davidson, D; Fitz, E; Rosen, S; Swift, R1
Ardizzone, G; Arrigo, A; Avallone, R; Baraldi, M; Centanaro, M; Corsi, L; Farina, F; Kleinschnitz, M; Schreier, P; Venturini, I; Zeneroli, ML1
Brown, S; Patsalos, PN; Shorvon, SD; Tong, X; Walker, MC1
Gelboin, HV; Gonzalez, FJ; Korzekwa, KR; Shou, M; Yang, SK; Yang, TJ1
Ali, HM; Azzam, RM; Notarianni, LJ1
Hemmersbach, P; Ragnar Norli, H; Rasmussen, KE; Reubsaet, KJ1
Baillie, TA; Dai, R; Ettore, MW; Mei, Q; Rushmore, TH; Shou, M1
He, N; Huang, SL; Ou-Yang, DS; Qin, XP; Wang, W; Wang, YJ; Xie, HG; Xu, ZH; Zhou, HH1
Kristensen, PA; Moller, JT; Rasmussen, H; Rasmussen, LS; Steentoft, A1
Atta-Politou, J; Dona, A; Koutselinis, A; Parissi-Poulou, M1
Schmoldt, A; Schulz, M; Stein, S1
Krogh, M; Rasmussen, KE; Ugland, HG1
Arditti, J; Bourdon, JH; de Haro, L; Hayek-Lanthois, M; Iliadis, A; Valli, M1
Mørland, J; Olsen, KM; Skuterud, B; Smith-Kielland, A1
Contel, N; Grossman, S; Liu, Z; Ren, S; Rose, A; Short, J; Unger, S1
Bell, RR; Crookham, SB; Dunn, WA; Grates, KM; Reiber, TM1
Bergman, J; Knebel, N; Munzar, P; Paronis, C; Redhi, G; Tober, C; Yasar, S; Zschiesche, M1
Djeridane, Y; Touitou, Y1
Andersson, TB; Bredberg, E; Eriksson, UG; Eriksson-Lepkowska, M; Frison, L; Johansson, S; Larsson, M; Thuresson, A1
Holmgren, P; Jones, AW1
Jones, AW; Larsson, H1
Holmgren, A; Holmgren, P; Jones, AW1
Atta-Politou, J; Panderi, I; Valavani, P1
Musteata, FM; Musteata, ML; Pawliszyn, J1
Grubwieser, P; Libiseller, K; Pavlic, M; Rabl, W; Schubert, H1
Bouchonnet, S; Kinani, S; Milan, N; Ricordel, I1
Bertilsson, L; Laine, K; Neuvonen, PJ; Olkkola, KT; Saari, TI1
Barroso, M; Gallardo, E; Margalho, C; Monsanto, P; Vieira, DN1
Lehmann, C; Wannarka, GL1
Acikgöz, A; Bader, A; Giri, S; Karim, N; Schmidt-Heck, W1
Cole, B; Fishbain, DA; Gao, J; Lewis, JE; Rosomoff, RS1
Iannello, C; Mandrioli, R; Matrisciano, F; Mercolini, L; Nicoletti, F; Raggi, MA1
Abe, K; Kobayashi, N; Nakamura, K; Nishiya, Y; Okazaki, O; Okudaira, N1
Chronister, CW; Goldberger, BA; Merves, ML1
Acikgöz, A; Bader, A; Giri, S; Maringka, M; Nieber, K1
Mariani, CL; Musulin, SE; Papich, MG1
Bowron, P; Fu, S; Lewis, J; Molnar, A; Wang, H1
KuKanich, B; Nauss, JL1
Andrews, P; Lamson, MJ; Mesa, M; Pellock, J; Sitki-Green, D; Wannarka, GL1
Holmgren, A; Jones, AW1
Roth, T; Verster, JC1
Cox, S; Martin, T; Moyers, TD; Probst, CW; Thomas, WB1
Charabidze, D; Delabarde, T; Keyser, C; Ludes, B; Tracqui, A1
Burch, HJ; Clarke, EJ; Hubbard, AM; Scott-Ham, M1
Breborowicz, GH; Florek, E; Krzyscin, M; Kulza, M; Lechowicz, E; Markwitz, W; Mazela, J; Merritt, TA; Miechowicz, I; Piekoszewski, W; Senczuk-Przybylowska, M1
Liang, C; Ni, C; Rao, Y; Wang, R; Wang, X; Xiong, L; Zhang, Y1
Atayee, RS; Best, BM; Luk, S; Ma, JD1
Bertol, E; Boscolo Berto, R; Favretto, D; Mannaioni, G; Mari, F; Vaiano, F1
Bankstahl, M; Gramer, M; Hausknecht, M; Klein, S; Löscher, W1
Li, J; Liu, H; Wu, L; Zhang, J1
Aboul-Enein, HY; Adib, N; Talebpour, Z; Torabizadeh, M1
Darwish, WS; Hayami, A; Ikenaka, Y; Ishizuka, M; Kawai, YK; Mizukawa, H; Nakayama, SM; Watanabe, KP1
Jia, J; Jiang, F; Johansen, SS; Linnet, K; Rao, Y; Wang, X; Zhang, Y1
Castro, A; Costa, P; Franco, JM; Melo, P; Quintas, MJ; Tarelho, S; Teixeira, HM1
Boxho, P; Charlier, C; Denooz, R; Dubois, N; Lemaire, E; Schmidt, C1
Du, P; Gao, T; Hou, L; Li, J; Li, X; Wang, C; Xu, Z; Yang, J; Zhang, H1
Bugelli, V; Campobasso, CP; Chericoni, S; Fornaro, S; Giusiani, M; Papi, L; Stefanelli, F; Vanin, S1
Barclay, VKH; Johansson, IM; Pettersson, CE; Tyrefors, NL1
Concheiro, M; Cooper, G; Mei, V; Pardi, J1
Andresen-Streichert, H; Froch-Cortis, J; Lehmann, S; Mercer-Chalmers-Bender, K; Rothschild, MA; Sczyslo, A; Thevis, M1
Cui, GF; He, Y; Ren, XX; Wang, LL; Wei, ZW; Yun, KM1
Falcon, M; Fernadez-Lopez, L; Luna, A; Mancini, R; Pellegrini, M; Rotolo, M1
Ballardini, M; Carelli, C; Freni, F; Moretti, M; Morini, L; Vignali, C1
Broussou, D; Düe, M; Lagershausen, H; Lallemand, E; Machnik, M; Meuly, A; Roques, BB; Röttgen, H; Schenk, I; Thevis, M; Toutain, PL1
Diogo, HP; Ramos, JJM1
Burkat, PM1
Frankenfeld, F; Jacobs, CM; Meyer, MR; Wagmann, L1
Adhikari, S; Barron, LP; Bhatnagar, A; Bowes, DA; Coronado-Apodaca, KG; Driver, EM; Halden, RU; Kumar, R; Martínez-Ruiz, M; McCall, KL; Melchor-Martínez, EM; Ng, KT; Oyervides-Muñoz, MA; Parra-Saldivar, R; Piper, BJ; Smith, T; Sosa-Hernandez, JE1

Reviews

10 review(s) available for nordazepam and diazepam

ArticleYear
Neural networks applied to quantitative structure-activity relationship analysis.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Animals; Azirines; Benzodiazepines; Carbazilquinone; Nerve Net; Nervous System; Regression Analysis; Structure-Activity Relationship

1990
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea

2020
[Clinical pharmacokinetics of diazepam and its biologically active metabolites (author's transl)].
    Klinische Wochenschrift, 1978, Sep-15, Volume: 56, Issue:18

    Topics: Biotransformation; Diazepam; Half-Life; Humans; Kinetics; Models, Biological; Nordazepam; Oxazepam

1978
Benzodiazepines: are they of natural origin?
    Pharmaceutical research, 1989, Volume: 6, Issue:1

    Topics: Animals; Benzodiazepines; Diazepam; Nordazepam

1989
[Current intravenous anesthetics].
    Polski tygodnik lekarski (Warsaw, Poland : 1960), 1980, Volume: 35, Issue:43

    Topics: Anesthesia, Intravenous; Anesthetics; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Etomidate; Flunitrazepam; Imidazoles; Injections, Intravenous; Lorazepam; Medazepam; Midazolam; Nordazepam

1980
Benzodiazepine kinetics: implications for therapeutics and pharmacogeriatrics.
    Drug metabolism reviews, 1983, Volume: 14, Issue:2

    Topics: Adolescent; Adult; Age Factors; Aged; Benzodiazepines; Biotransformation; Child; Diazepam; Flurazepam; Half-Life; Humans; Kinetics; Middle Aged; Nordazepam; Oxidation-Reduction

1983
[Benzodiazepines: significance of kinetics for therapy].
    Klinische Wochenschrift, 1983, Mar-01, Volume: 61, Issue:5

    Topics: Age Factors; Aged; Benzodiazepines; Diazepam; Humans; Kinetics; Metabolic Clearance Rate; Nordazepam; Sex Factors; Triazolam

1983
[Drug catabolism and its significance for pharmacotherapy].
    Medizinische Klinik, 1980, Mar-28, Volume: 75, Issue:7

    Topics: Biotransformation; Cytochrome P-450 Enzyme System; Diazepam; Digitoxin; Digoxin; Drug Interactions; Drug Therapy; Drug Therapy, Combination; Enzyme Induction; Ethanol; Kidney; Kidney Diseases; Liver; Liver Diseases; Nordazepam; Receptors, Drug

1980
Studies of "endogenous" benzodiazepine in human hepatic encephalopathy.
    Alcohol and alcoholism (Oxford, Oxfordshire). Supplement, 1993, Volume: 2

    Topics: Animals; Benzodiazepines; Diazepam; Hepatic Encephalopathy; Humans; Models, Biological; Nordazepam

1993
Blood drug concentrations of benzodiazepines correlate poorly with actual driving impairment.
    Sleep medicine reviews, 2013, Volume: 17, Issue:2

    Topics: Anti-Anxiety Agents; Automobile Driving; Diazepam; GABA-A Receptor Agonists; Humans; Nordazepam; Psychomotor Performance

2013

Trials

65 trial(s) available for nordazepam and diazepam

ArticleYear
Effect of N-desmethyldiazepam (nordiazepam) and a precursor, potassium clorazepate, on sleep in man.
    British journal of clinical pharmacology, 1976, Volume: 3, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Humans; Male; Nordazepam; Sleep; Sleep Stages; Time Factors

1976
Double-blind cross-over clinical comparison of two 2'-chloro benzodiazepines: 7-chloro-5-(2-chlorophenyl)-1,3-dihydro-2H-1,4-benzodiazepin-2-one (chlordesmethyldiazepam) versus 7-chloro-5-(o-chlorophenyl)-1,3-dihydro-3-hydroxy-2H-1,4-benzodiazepin-2-one (
    Arzneimittel-Forschung, 1977, Volume: 27, Issue:2

    Topics: Adult; Aged; Anti-Anxiety Agents; Anxiety Disorders; Brief Psychiatric Rating Scale; Clinical Trials as Topic; Diazepam; Drug Evaluation; Female; Humans; Lorazepam; Middle Aged; Nordazepam; Psychiatric Status Rating Scales

1977
Impaired absorption of desmethyldiazepam from clorazepate by magnesium aluminum hydroxide.
    Clinical pharmacology and therapeutics, 1978, Volume: 24, Issue:3

    Topics: Adult; Aged; Aluminum Hydroxide; Anti-Anxiety Agents; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Drug Combinations; Female; Humans; Hypnotics and Sedatives; Intestinal Absorption; Kinetics; Magnesium; Magnesium Hydroxide; Male; Middle Aged; Nordazepam; Time Factors

1978
Disposition of diazepam and its major metabolite desmethyldiazepam in patients with liver disease.
    Clinical pharmacology and therapeutics, 1977, Volume: 21, Issue:4

    Topics: Adult; Biological Availability; Biotransformation; Clinical Trials as Topic; Diazepam; Half-Life; Hepatitis; Humans; Liver; Liver Cirrhosis; Liver Diseases; Middle Aged; Nordazepam

1977
Single-blind evaluation of hypnotic activity of chlordesmethyldiazepam in No-placebo-reactor medical patients.
    Arzneimittel-Forschung, 1977, Volume: 27, Issue:1

    Topics: Clinical Trials as Topic; Diazepam; Drug Evaluation; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Nordazepam; Placebos; Sleep Initiation and Maintenance Disorders

1977
Activity of N-desmethyldiazepam (nordiazepam) [proceedings].
    British journal of clinical pharmacology, 1977, Volume: 4, Issue:5

    Topics: Adult; Diazepam; Humans; Male; Motor Skills; Nordazepam

1977
Immediate and residual effects in man of the metabolites of diazepam.
    British journal of clinical pharmacology, 1978, Volume: 6, Issue:4

    Topics: Adult; Choice Behavior; Diazepam; Humans; Male; Motor Skills; Nordazepam; Oxazepam; Placebos; Reaction Time; Temazepam; Time Factors

1978
Plasma concentration of diazepam and N-desmethyldiazepam in children after a single rectal or intramuscular dose of diazepam.
    European journal of clinical pharmacology, 1978, Dec-01, Volume: 14, Issue:4

    Topics: Child; Child, Preschool; Clinical Trials as Topic; Diazepam; Humans; Hypnotics and Sedatives; Injections, Intramuscular; Nordazepam; Rectum; Suppositories; Time Factors

1978
Effect of a cocktail on diazepam absorption.
    Psychopharmacology, 1978, Apr-28, Volume: 57, Issue:2

    Topics: Adult; Alcoholic Beverages; Diazepam; Ethanol; Female; Humans; Intestinal Absorption; Kinetics; Male; Nordazepam

1978
Pharmacokinetics of N-demethyldiazepam in patients suffering from insomnia and treated with nortriptyline.
    British journal of clinical pharmacology, 1975, Volume: 2, Issue:3

    Topics: Adult; Aged; Clinical Trials as Topic; Diazepam; Drug Evaluation; Drug Therapy, Combination; Half-Life; Humans; Male; Middle Aged; Nordazepam; Nortriptyline; Placebos; Sleep Initiation and Maintenance Disorders

1975
The effects of felodipine on the pharmacokinetics of diazepam.
    International journal of clinical pharmacology, therapy, and toxicology, 1992, Volume: 30, Issue:4

    Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Felodipine; Humans; Male; Nordazepam

1992
Amnestic effects of intravenous diazepam in healthy young men.
    The American journal of drug and alcohol abuse, 1991, Volume: 17, Issue:2

    Topics: Adolescent; Adult; Diazepam; Dose-Response Relationship, Drug; Humans; Infusions, Intravenous; Male; Memory, Short-Term; Mental Recall; Nordazepam; Retention, Psychology; Verbal Learning

1991
Effect of omeprazole treatment on diazepam plasma levels in slow versus normal rapid metabolizers of omeprazole.
    Clinical pharmacology and therapeutics, 1990, Volume: 47, Issue:1

    Topics: Adult; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Drug Interactions; Humans; Male; Metabolic Clearance Rate; Nordazepam; Omeprazole; Random Allocation

1990
Effects of single doses of alprazolam and diazepam, alone and in combination with ethanol, on psychomotor and cognitive performance and on autonomic nervous system reactivity in healthy volunteers.
    European journal of clinical pharmacology, 1990, Volume: 39, Issue:1

    Topics: Adult; Affect; Alprazolam; Anxiety; Autonomic Nervous System; Cognition; Diazepam; Drug Interactions; Ethanol; Female; Humans; Nordazepam; Norepinephrine; Psychomotor Performance

1990
Effect of omeprazole and cimetidine on plasma diazepam levels.
    European journal of clinical pharmacology, 1990, Volume: 39, Issue:1

    Topics: Adult; Cimetidine; Diazepam; Double-Blind Method; Drug Interactions; Half-Life; Humans; Male; Nordazepam; Omeprazole

1990
Double-blind placebo cross-over study of long-acting (chlordesmethyldiazepam) versus short-acting (lorazepam) benzodiazepines in generalized anxiety disorders.
    International journal of clinical pharmacology research, 1989, Volume: 9, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Diazepam; Double-Blind Method; Female; Humans; Lorazepam; Male; Middle Aged; Nordazepam; Psychiatric Status Rating Scales

1989
[Chlordesmethyldiazepam and prolactinemia during surgical stress].
    Acta bio-medica de L'Ateneo parmense : organo della Societa di medicina e scienze naturali di Parma, 1989, Volume: 60, Issue:5-6

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Male; Middle Aged; Nordazepam; Preanesthetic Medication; Prolactin; Stress, Physiological; Surgery, Plastic; Surgical Procedures, Operative; Thiopental

1989
Influence of propranolol coadministration or cigarette smoking on the kinetics of desmethyldiazepam following intravenous clorazepate.
    Klinische Wochenschrift, 1986, Dec-01, Volume: 64, Issue:23

    Topics: Adult; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Drug Interactions; Female; Humans; Infusions, Intravenous; Kinetics; Male; Metabolic Clearance Rate; Nordazepam; Propranolol; Smoking

1986
Effects of propranolol, atenolol, and chlordesmethyldiazepam on response to mental stress in patients with recent myocardial infarction.
    Clinical cardiology, 1987, Volume: 10, Issue:6

    Topics: Adult; Aged; Anti-Anxiety Agents; Atenolol; Benzodiazepines; Diazepam; Electrocardiography; Hemodynamics; Humans; Male; Middle Aged; Myocardial Infarction; Nordazepam; Propranolol; Psychophysiology; Stress, Psychological

1987
Nocturnal doses of ranitidine and nizatidine do not affect the disposition of diazepam.
    Journal of clinical pharmacology, 1987, Volume: 27, Issue:3

    Topics: Adult; Diazepam; Drug Interactions; Histamine H2 Antagonists; Humans; Male; Nizatidine; Nordazepam; Ranitidine; Thiazoles

1987
Effects of HOE 760 (histamine H2-receptor antagonist) on diazepam pharmacokinetics.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1988, Apr-02, Volume: 73, Issue:7

    Topics: Adult; Clinical Trials as Topic; Diazepam; Double-Blind Method; Half-Life; Histamine H2 Antagonists; Humans; Male; Nordazepam; Piperidines; Time Factors

1988
Pharmacokinetics and bioavailability of intravenous and oral chlordesmethyldiazepam in humans.
    European journal of clinical pharmacology, 1988, Volume: 34, Issue:1

    Topics: Absorption; Administration, Oral; Adult; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Biological Availability; Diazepam; Half-Life; Humans; Injections, Intravenous; Male; Nordazepam; Random Allocation; Tablets; Time Factors

1988
[Effects of chlordemethyldiazepam on blood cortisol during surgical stress].
    Acta bio-medica de L'Ateneo parmense : organo della Societa di medicina e scienze naturali di Parma, 1988, Volume: 59, Issue:5-6

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Clinical Trials as Topic; Diazepam; Humans; Hydrocortisone; Male; Middle Aged; Nordazepam; Preanesthetic Medication; Random Allocation; Stress, Physiological; Surgical Procedures, Operative

1988
Premedication with oral and rectal diazepam.
    Acta anaesthesiologica Scandinavica, 1986, Volume: 30, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Aged; Anesthesia, General; Anxiety; Diazepam; Double-Blind Method; Drug Evaluation; Humans; Kinetics; Middle Aged; Nordazepam; Preanesthetic Medication; Random Allocation; Rectum; Time Factors

1986
Diazepam and methadone blood levels following concurrent administration of diazepam and methadone.
    Drug and alcohol dependence, 1986, Volume: 18, Issue:2

    Topics: Adult; Chromatography, Thin Layer; Diazepam; Drug Interactions; Humans; Immunoenzyme Techniques; Kinetics; Male; Meiosis; Methadone; Nordazepam

1986
Diazepam: prediction of pharmacodynamics from pharmacokinetics.
    Psychopharmacology, 1984, Volume: 83, Issue:3

    Topics: Adult; Diazepam; Humans; Kinetics; Male; Nordazepam; Receptors, Cell Surface; Receptors, GABA-A

1984
Steady-state plasma desmethyldiazepam during long-term clorazepate use: effects of antacids.
    Clinical pharmacology and therapeutics, 1982, Volume: 31, Issue:2

    Topics: Adult; Aluminum Hydroxide; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Drug Combinations; Drug Interactions; Female; Gastric Acid; Humans; Magnesium; Magnesium Hydroxide; Male; Nordazepam; Time Factors

1982
A radioreceptor assay to study the affinity of benzodiazepines and their receptor binding activity in human plasma including their active metabolites.
    British journal of clinical pharmacology, 1982, Volume: 13, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Biotransformation; Blood Proteins; Diazepam; Female; Humans; Lorazepam; Male; Nitrazepam; Nordazepam; Protein Binding; Radioligand Assay; Receptors, Drug; Receptors, GABA-A

1982
Desmethyldiazepam kinetics after intravenous, intramuscular, and oral administration of clorazepate dipotassium.
    Klinische Wochenschrift, 1982, Apr-15, Volume: 60, Issue:8

    Topics: Administration, Oral; Adult; Aged; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Female; Half-Life; Humans; Injections, Intramuscular; Injections, Intravenous; Kinetics; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam

1982
Value of a single night-time dose of potassium clorazepate in anxiety: a controlled trial comparison with diazepam.
    Scottish medical journal, 1982, Volume: 27, Issue:4

    Topics: Adolescent; Adult; Anti-Anxiety Agents; Anxiety; Blood Pressure; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Nordazepam; Patient Compliance; Psychological Tests

1982
Diazepam/beta-adrenoceptor antagonist interactions.
    British journal of clinical pharmacology, 1984, Volume: 17 Suppl 1

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Animals; Atenolol; Diazepam; Drug Interactions; Emotions; Humans; In Vitro Techniques; Kinetics; Male; Metoprolol; Microsomes, Liver; Nordazepam; Propranolol; Psychomotor Performance; Rats; Rats, Inbred Strains; Reaction Time; Visual Acuity

1984
Plasma concentrations and clinical effects after single oral doses of prazepam, clorazepate, and diazepam.
    The Journal of clinical psychiatry, 1984, Volume: 45, Issue:10

    Topics: Administration, Oral; Adult; Anti-Anxiety Agents; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Double-Blind Method; Emotions; Female; Humans; Intestinal Absorption; Kinetics; Male; Nordazepam; Prazepam; Sleep

1984
Psychomotor effects of diazepam in anxious patients and healthy volunteers.
    Journal of clinical psychopharmacology, 1983, Volume: 3, Issue:2

    Topics: Adult; Anxiety Disorders; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Male; Nordazepam; Personality Inventory; Psychiatric Status Rating Scales; Psychomotor Performance

1983
Clinical importance of the interaction of diazepam and cimetidine.
    The New England journal of medicine, 1984, Jun-21, Volume: 310, Issue:25

    Topics: Adult; Anxiety; Cimetidine; Clinical Trials as Topic; Diazepam; Double-Blind Method; Drug Interactions; Drug Therapy, Combination; Female; Half-Life; Humans; Male; Middle Aged; Nordazepam; Psychomotor Performance; Reaction Time; Sleep Wake Disorders

1984
Dose-response analysis of the behavioral effects of diazepam: II. Psychomotor performance, cognition and mood.
    Psychopharmacology, 1984, Volume: 82, Issue:4

    Topics: Adolescent; Adult; Circadian Rhythm; Cognition; Diazepam; Dose-Response Relationship, Drug; Emotions; Half-Life; Humans; Nordazepam; Posture; Psychomotor Performance

1984
Withdrawal responses to abrupt discontinuation of desmethyldiazepam.
    The American journal of psychiatry, 1984, Volume: 141, Issue:11

    Topics: Acute Disease; Adult; Anxiety Disorders; Clinical Trials as Topic; Depression; Diazepam; Feeding and Eating Disorders; Female; Half-Life; Humans; Nausea; Nordazepam; Placebos; Psychiatric Status Rating Scales; Sleep Wake Disorders; Substance Withdrawal Syndrome

1984
Anxiety and sedation during a stressful situation after single dose of diazepam versus N-desmethyldiazepam--a controlled trial.
    Psychopharmacology, 1980, Volume: 70, Issue:3

    Topics: Adult; Anxiety; Breast Neoplasms; Diazepam; Double-Blind Method; Drug Evaluation; Emotions; Female; Humans; Hypnotics and Sedatives; Middle Aged; Nordazepam

1980
Kinetics and neuropsychologic effects of IV diazepam in the presence and absence of its active N-desmethyl metabolite in humans.
    Psychopharmacology, 1980, Volume: 70, Issue:3

    Topics: Adolescent; Adult; Anxiety; Diazepam; Electroencephalography; Emotions; Female; Humans; Injections, Intravenous; Kinetics; Male; Nordazepam; Reaction Time

1980
The relationship between peak velocity of saccadic eye movements and serum benzodiazepine concentration.
    British journal of clinical pharmacology, 1981, Volume: 12, Issue:4

    Topics: Adult; Benzodiazepines; Diazepam; Double-Blind Method; Eye Movements; Flurazepam; Humans; Male; Nitrazepam; Nordazepam; Reticular Formation; Saccades; Temazepam

1981
Effects of two dosages of chlordesmethyldiazepam on mnestic-information processes in normal subjects.
    Clinical therapeutics, 1981, Volume: 4, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Male; Memory; Mental Recall; Nordazepam; Random Allocation

1981
Clearance of diazepam can be impaired by its major metabolite desmethyldiazepam.
    European journal of clinical pharmacology, 1981, Volume: 21, Issue:2

    Topics: Adult; Diazepam; Humans; Metabolic Clearance Rate; Nordazepam

1981
Relationship of diazepam serum level to antianxiety effects.
    Journal of clinical psychopharmacology, 1982, Volume: 2, Issue:2

    Topics: Adult; Anxiety Disorders; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Personality Inventory

1982
Effects of oral chlordemethyldiazepam on plasma adrenaline and noradrenaline and cardiovascular reactivity in preoperative patients.
    European journal of clinical pharmacology, 1982, Volume: 23, Issue:5

    Topics: Abortion, Induced; Adolescent; Adult; Anti-Anxiety Agents; Benzodiazepines; Blood Pressure; Diazepam; Epinephrine; Female; Heart Rate; Hemodynamics; Humans; Nordazepam; Norepinephrine; Plethysmography; Pregnancy; Preoperative Care

1982
Withdrawal reaction from long-term, low-dosage administration of diazepam. A double-blind, placebo-controlled case study.
    Archives of general psychiatry, 1980, Volume: 37, Issue:1

    Topics: Adult; Anxiety; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Male; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1980
Interethnic difference in omeprazole's inhibition of diazepam metabolism.
    Clinical pharmacology and therapeutics, 1995, Volume: 58, Issue:1

    Topics: Adult; Asian People; China; Cross-Over Studies; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Debrisoquin; Diazepam; Double-Blind Method; Drug Interactions; Ethnicity; Humans; Male; Mephenytoin; Nordazepam; Omeprazole; Tennessee; White People

1995
Comparison of the interaction potential of a new proton pump inhibitor, E3810, versus omeprazole with diazepam in extensive and poor metabolizers of S-mephenytoin 4'-hydroxylation.
    Clinical pharmacology and therapeutics, 1995, Volume: 58, Issue:2

    Topics: 2-Pyridinylmethylsulfinylbenzimidazoles; Analysis of Variance; Aryl Hydrocarbon Hydroxylases; Benzimidazoles; Cross-Over Studies; Cytochrome P-450 CYP2C19; Cytochrome P-450 Enzyme System; Diazepam; Drug Interactions; Half-Life; Humans; Hydroxylation; Male; Mephenytoin; Mixed Function Oxygenases; Nordazepam; Omeprazole; Proton Pump Inhibitors; Rabeprazole; Reference Values; Single-Blind Method

1995
Subjective and behavioral effects of diazepam depend on its rate of onset.
    Psychopharmacology, 1993, Volume: 112, Issue:2-3

    Topics: Adult; Affect; Alcohol Drinking; Behavior; Breath Tests; Cognition; Diazepam; Double-Blind Method; Euphoria; Humans; Male; Nordazepam; Psychomotor Performance; Sleep

1993
[Preanesthesia in elderly patients undergoing subarachnoid anesthesia: chlordesmethyldiazepam versus diazepam].
    Minerva anestesiologica, 1994, Volume: 60, Issue:4

    Topics: Aged; Anesthesia, Spinal; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Female; Humans; Male; Nordazepam; Preanesthetic Medication

1994
Inhibition of diazepam metabolism by fluvoxamine: a pharmacokinetic study in normal volunteers.
    Clinical pharmacology and therapeutics, 1994, Volume: 56, Issue:5

    Topics: Adult; Biotransformation; Diazepam; Female; Fluvoxamine; Humans; Male; Nordazepam

1994
Metabolic and subjective responses to oral diazepam and midazolam.
    European journal of anaesthesiology, 1994, Volume: 11, Issue:5

    Topics: Administration, Oral; Adult; Arousal; Calorimetry, Indirect; Carbon Dioxide; Cognition; Diazepam; Double-Blind Method; Energy Metabolism; Humans; Hypnotics and Sedatives; Male; Memory; Midazolam; Monitoring, Physiologic; Nordazepam; Oxygen Consumption; Placebos

1994
Absorption of diazepam after its rectal administration in dogs.
    American journal of veterinary research, 1995, Volume: 56, Issue:12

    Topics: Absorption; Administration, Rectal; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cross-Over Studies; Diazepam; Dogs; Dose-Response Relationship, Drug; Fluorescence Polarization Immunoassay; Injections, Intravenous; Male; Nordazepam; Oxazepam; Time Factors

1995
[Determination of diazepam concentration in maternal and fetal serum after intravenous administration during active phase of labor and its effects on neonates].
    Zhonghua fu chan ke za zhi, 1995, Volume: 30, Issue:12

    Topics: Adult; Apgar Score; Asphyxia Neonatorum; Diazepam; Female; Fetal Blood; Humans; Infant, Newborn; Injections, Intravenous; Labor Onset; Nordazepam; Pregnancy

1995
Premedication with chlordemethyldiazepam and anxiolytic effect of diazepeam in implantology.
    Anesthesia progress, 1995, Volume: 42, Issue:3-4

    Topics: Adult; Anesthesia, Dental; Anti-Anxiety Agents; Benzodiazepines; Chi-Square Distribution; Dental Anxiety; Dental Implantation; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Preanesthetic Medication

1995
Effect of sertraline on the pharmacokinetics and protein binding of diazepam in healthy volunteers.
    Clinical pharmacokinetics, 1997, Volume: 32 Suppl 1

    Topics: 1-Naphthylamine; Adolescent; Adult; Anti-Anxiety Agents; Antidepressive Agents; Aryl Hydrocarbon Hydroxylases; Blood Proteins; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Diazepam; Double-Blind Method; Drug Interactions; Humans; Male; Mixed Function Oxygenases; Nordazepam; Protein Binding; Selective Serotonin Reuptake Inhibitors; Sertraline

1997
Naltrexone effects on diazepam intoxication and pharmacokinetics in humans.
    Psychopharmacology, 1998, Volume: 135, Issue:3

    Topics: Adult; Affect; Aged; Anti-Anxiety Agents; Central Nervous System Depressants; Diazepam; Ethanol; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Neuropsychological Tests; Nordazepam; Psychomotor Performance

1998
Benzodiazepines and postoperative cognitive dysfunction in the elderly. ISPOCD Group. International Study of Postoperative Cognitive Dysfunction.
    British journal of anaesthesia, 1999, Volume: 83, Issue:4

    Topics: Abdomen; Age Factors; Aged; Aged, 80 and over; Anesthesia, General; Anti-Anxiety Agents; Cognition Disorders; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Postoperative Complications; Psychometrics; Regression Analysis

1999
A modified simple and rapid reversed phase liquid chromatographic method for quantification of diazepam and nordiazepam in plasma.
    Journal of pharmaceutical and biomedical analysis, 1999, Volume: 20, Issue:1-2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Calibration; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Middle Aged; Nordazepam; Reference Standards; Reproducibility of Results; Solvents

1999
Urinary excretion of diazepam metabolites in healthy volunteers and drug users.
    Scandinavian journal of clinical and laboratory investigation, 2001, Volume: 61, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Chromatography, Gas; Chromatography, High Pressure Liquid; Creatinine; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Substance Abuse Detection; Substance-Related Disorders; Temazepam

2001
Ximelagatran, an oral direct thrombin inhibitor, has a low potential for cytochrome P450-mediated drug-drug interactions.
    Clinical pharmacokinetics, 2003, Volume: 42, Issue:8

    Topics: Administration, Oral; Adult; Aged; Amidines; Anticoagulants; Area Under Curve; Azetidines; Benzylamines; Cross-Over Studies; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diazepam; Diclofenac; Drug Interactions; Glycine; Humans; In Vitro Techniques; Infusions, Intravenous; Microsomes, Liver; Middle Aged; Nifedipine; Nordazepam; Prodrugs; Thrombin

2003
Distribution of diazepam and nordiazepam between plasma and whole blood and the influence of hematocrit.
    Therapeutic drug monitoring, 2004, Volume: 26, Issue:4

    Topics: Adult; Body Water; Chromatography, Gas; Diazepam; Erythrocytes; Female; Hematocrit; Humans; In Vitro Techniques; Male; Middle Aged; Nordazepam; Plasma; Sex Factors

2004
Voriconazole and fluconazole increase the exposure to oral diazepam.
    European journal of clinical pharmacology, 2007, Volume: 63, Issue:10

    Topics: Administration, Oral; Adult; Antifungal Agents; Area Under Curve; Aryl Hydrocarbon Hydroxylases; Biotransformation; Cognition; Cross-Over Studies; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diazepam; Drug Interactions; Enzyme Inhibitors; Female; Fluconazole; Genotype; Half-Life; Humans; Hypnotics and Sedatives; Male; Mixed Function Oxygenases; Nordazepam; Pyrimidines; Triazoles; Voriconazole; Wakefulness

2007
Bioavailability and dose proportionality of intramuscular diazepam administered by autoinjector.
    Journal of clinical pharmacology, 2008, Volume: 48, Issue:4

    Topics: Adult; Anticonvulsants; Area Under Curve; Biotransformation; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Half-Life; Humans; Injections, Intramuscular; Male; Nordazepam; Therapeutic Equivalency

2008
Diazepam pharmacokinetics after nasal drop and atomized nasal administration in dogs.
    Journal of veterinary pharmacology and therapeutics, 2011, Volume: 34, Issue:1

    Topics: Administration, Intranasal; Animals; Anticonvulsants; Diazepam; Dogs; Dosage Forms; Drug Administration Routes; Female; Half-Life; Male; Nordazepam; Oxazepam

2011
Pharmacokinetics of diazepam administered intramuscularly by autoinjector versus rectal gel in healthy subjects: a phase I, randomized, open-label, single-dose, crossover, single-centre study.
    Clinical drug investigation, 2011, Volume: 31, Issue:8

    Topics: Administration, Rectal; Adult; Anticonvulsants; Area Under Curve; Cross-Over Studies; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Injections, Intramuscular; Male; Nordazepam; Young Adult

2011
Evaluation of plasma diazepam and nordiazepam concentrations following administration of diazepam intravenously or via suppository per rectum in dogs.
    American journal of veterinary research, 2013, Volume: 74, Issue:4

    Topics: Administration, Rectal; Animals; Anticonvulsants; Area Under Curve; Cross-Over Studies; Diazepam; Dogs; Female; Half-Life; Injections, Intravenous; Male; Nordazepam; Suppositories

2013

Other Studies

304 other study(ies) available for nordazepam and diazepam

ArticleYear
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles

1978
Electronic factors in the structure-activity relationship of some 1,4-benzodiazepin-2-ones.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:9

    Topics: Benzodiazepinones; Electrochemistry; Structure-Activity Relationship

1977
Synthesis of previously inaccessible quinazolines and 1,4-benzodiazepines as potential anticonvulsants.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:6

    Topics: Animals; Anticonvulsants; Benzodiazepines; Mice; Pentylenetetrazole; Quinazolines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
Quantitative structure-activity relationships employing independent quantum chemical indices.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:8

    Topics: Amines; Benzodiazepines; Benzylamines; Mathematics; Quantum Theory; Structure-Activity Relationship; Tetracyclines

1983
Rm values and structure-activity relationship of benzodiazepines.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:2

    Topics: Animals; Benzodiazepines; Chromatography, Thin Layer; Conflict, Psychological; Exploratory Behavior; Models, Biological; Rats; Solubility; Structure-Activity Relationship

1980
Decomposition of pharmacological activity indices into mutually independent components using principal component analysis.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:4

    Topics: Animals; Anti-Infective Agents; Benzodiazepines; Hydroxyquinolines; Mathematics; Pharmacology; Rifamycins; Seizures; Statistics as Topic; Structure-Activity Relationship

1980
Prediction of receptor properties and binding affinity of ligands to benzodiazepine/GABAA receptors using artificial neural networks.
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Binding Sites; Ligands; Neural Networks, Computer; Predictive Value of Tests; Receptors, GABA-A; Structure-Activity Relationship

1995
Genetic neural networks for quantitative structure-activity relationships: improvements and application of benzodiazepine affinity for benzodiazepine/GABAA receptors.
    Journal of medicinal chemistry, 1996, Dec-20, Volume: 39, Issue:26

    Topics: Algorithms; Benzodiazepines; Models, Genetic; Nerve Net; Protein Binding; Receptors, GABA-A; Structure-Activity Relationship

1996
Molecular hashkeys: a novel method for molecular characterization and its application for predicting important pharmaceutical properties of molecules.
    Journal of medicinal chemistry, 1999, May-20, Volume: 42, Issue:10

    Topics: Drug Design; Intestinal Absorption; Models, Molecular; Pharmaceutical Preparations; Structure-Activity Relationship

1999
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Fast calculation of molecular polar surface area as a sum of fragment-based contributions and its application to the prediction of drug transport properties.
    Journal of medicinal chemistry, 2000, Oct-05, Volume: 43, Issue:20

    Topics: Biological Availability; Biological Transport; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Reproducibility of Results

2000
Experimental and computational screening models for the prediction of intestinal drug absorption.
    Journal of medicinal chemistry, 2001, Jun-07, Volume: 44, Issue:12

    Topics: Biological Transport; Carbon Radioisotopes; Cell Line; Cell Membrane; Cell Membrane Permeability; Ciprofloxacin; Computational Biology; Drug Design; Foscarnet; Humans; Hydrogen Bonding; Intestinal Absorption; Intestinal Mucosa; Lactulose; Mannitol; Models, Biological; Raffinose; Surface Properties; Tritium; Verapamil

2001
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Conformation selectivity in the binding of diazepam and analogues to alpha1-acid glycoprotein.
    Bioorganic & medicinal chemistry, 2007, Jul-15, Volume: 15, Issue:14

    Topics: Circular Dichroism; Diazepam; Genetic Variation; Humans; Molecular Conformation; Orosomucoid; Protein Binding; Serum Albumin

2007
Computational aqueous solubility prediction for drug-like compounds in congeneric series.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Benzodiazepines; Computer Simulation; Crystallography, X-Ray; Databases, Factual; Least-Squares Analysis; Models, Chemical; Organic Chemicals; Pharmaceutical Preparations; Principal Component Analysis; Solubility; Sulfonamides; Water

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
[Analysis of the structure of the components of the convulsive action of corazole following administration of sulazepam and its metabolites to mice].
    Biulleten' eksperimental'noi biologii i meditsiny, 1976, Volume: 82, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred CBA; Nordazepam; Oxazepam; Pentylenetetrazole; Seizures; Time Factors

1976
Feto-maternal concentrations of diazepam and W-demethyldiazepam after intra-amniotic diazepam injection.
    International journal of gynaecology and obstetrics: the official organ of the International Federation of Gynaecology and Obstetrics, 1976, Volume: 14, Issue:3

    Topics: Adolescent; Adult; Amniotic Fluid; Brain Chemistry; Diazepam; Female; Fetal Blood; Humans; Injections; Injections, Intramuscular; Kinetics; Liver; Maternal-Fetal Exchange; Nordazepam; Oxazepam; Pregnancy

1976
Analysis of medazepam, diazepam, and metabolites in plasma by gas-liquid chromatography with electrolytic conductivity detection.
    Journal of chromatography, 1977, Jun-01, Volume: 136, Issue:1

    Topics: Anti-Anxiety Agents; Chromatography, Gas; Chromatography, Liquid; Diazepam; Electric Conductivity; Medazepam; Microchemistry; Nordazepam

1977
On the hypnogenic and anticonvulsant activities of demethyldiazepam and chlordemethyldiazepam: time-effect relations.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:8

    Topics: Animals; Anticonvulsants; Chlorprothixene; Diazepam; Female; Hexobarbital; Hypnotics and Sedatives; Mice; Nordazepam; Pentylenetetrazole; Time Factors

1977
Pharmacokinetics of N-desmethyldiazepam in healthy volunteers after single daily doses of dipotassium chlorazepate.
    Psychopharmacology, 1977, Jul-18, Volume: 53, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Body Weight; Clorazepate Dipotassium; Diazepam; Drug Interactions; Female; Half-Life; Humans; Kinetics; Male; Nordazepam

1977
Rapid gas chromatographic assay of serum diazepam, N-desmethyldiazepam, and N-desalkylflurazepam.
    Acta pharmacologica et toxicologica, 1977, Volume: 41, Issue:5

    Topics: Anti-Anxiety Agents; Chromatography, Gas; Diazepam; Flurazepam; Humans; Nordazepam; Time Factors

1977
Determination of desmethyldiazepam in plasma by electron-capture GLC: application to pharmacokinetic studies of clorazepate.
    Journal of pharmaceutical sciences, 1978, Volume: 67, Issue:3

    Topics: Anti-Anxiety Agents; Chromatography, Gas; Clorazepate Dipotassium; Diazepam; Female; Humans; Kinetics; Nordazepam; Time Factors

1978
Pharmacokinetic understanding of antianxiety drug therapy.
    Southern medical journal, 1978, Volume: 71 Suppl 2

    Topics: Adult; Anti-Anxiety Agents; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Dose-Response Relationship, Drug; Humans; Nordazepam; Oxazepam; Prazepam

1978
Serum medazepam, diazepam, and N-desmethyldiazepam levels after single and multiple oral doses of medazepam.
    Annals of clinical research, 1977, Volume: 9, Issue:5

    Topics: Administration, Oral; Adolescent; Adult; Anti-Anxiety Agents; Chemical Phenomena; Chemistry; Diazepam; Humans; Intellectual Disability; Male; Medazepam; Nordazepam

1977
Gas chromatographic determination of chlorodesmethyldiazepam and lorazepam in rats and mice.
    Journal of chromatography, 1979, Jan-11, Volume: 168, Issue:1

    Topics: Adipose Tissue; Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Chromatography, Gas; Diazepam; Kinetics; Lorazepam; Male; Mass Spectrometry; Methods; Mice; Nordazepam; Rats

1979
Plasma concentrations of medazepam and its metabolites after oral administration.
    British journal of anaesthesia, 1979, Volume: 51, Issue:6

    Topics: Administration, Oral; Adult; Anti-Anxiety Agents; Diazepam; Humans; Male; Medazepam; Nordazepam; Time Factors

1979
Effect of age and Billroth gastrectomy on absorption of desmethyldiazepam from clorazepate.
    Clinical pharmacology and therapeutics, 1979, Volume: 26, Issue:4

    Topics: Adult; Age Factors; Aged; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Female; Gastrectomy; Humans; Intestinal Absorption; Male; Middle Aged; Nordazepam

1979
Acute and chronic effects of three benzodiazepines in the social interaction anxiety test in mice.
    Psychopharmacology, 1979, Aug-08, Volume: 64, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Humans; Interpersonal Relations; Lighting; Male; Mice; Nordazepam; Time Factors

1979
Simultaneous determination of diazepam and its metabolies N-desmethyldiazepam, oxydiazepam and oxazepam in plasma and urine of man and dog by means of high-performance liquid chromatography.
    Journal of chromatography, 1979, Apr-11, Volume: 162, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Humans; Nordazepam; Oxazepam; Species Specificity; Temazepam

1979
Self-rated sedation and plasma concentrations of desmethyldiazepam following single doses of clorazepate.
    Psychopharmacology, 1979, Volume: 66, Issue:3

    Topics: Adult; Aged; Anti-Anxiety Agents; Biotransformation; Clorazepate Dipotassium; Diazepam; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Nordazepam

1979
Sensitive gas chromatographic method for the determination of diazepam and N-desmethyldiazepam in plasma.
    Journal of chromatography, 1979, Jul-21, Volume: 163, Issue:3

    Topics: Chromatography, Gas; Diazepam; Humans; Nordazepam

1979
Quantitative high-performance liquid chromatography of diazepam and N-desmethyldiazepam in blood.
    Journal of chromatography, 1976, Nov-17, Volume: 128, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Forensic Medicine; Methods; Microchemistry; Nordazepam; Silicon Dioxide

1976
Effect of desmethyldiazepam and chlordesmethyldiazepam on 3',5'-cyclic guanosine monophosphate levels in rat cerebellum.
    Psychopharmacology, 1976, Nov-24, Volume: 50, Issue:3

    Topics: Age Factors; Animals; Animals, Newborn; Cerebellum; Cyclic AMP; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Male; Nordazepam; Rats

1976
In vitro effects of diazepam, desmethyldiazepam & nitrazepam on ATPase activity of human fetal brain.
    Indian journal of experimental biology, 1979, Volume: 17, Issue:9

    Topics: Adenosine Triphosphatases; Brain; Calcium-Transporting ATPases; Cell-Free System; Diazepam; Humans; Microsomes; Nitrazepam; Nordazepam; Sodium-Potassium-Exchanging ATPase; Synaptosomes

1979
Unchanged protein binding and the increase of serum diazepam levels after food intake.
    Acta pharmacologica et toxicologica, 1977, Volume: 40, Issue:2

    Topics: Adult; Diazepam; Dietary Carbohydrates; Dietary Fats; Eating; Fatty Acids, Nonesterified; Humans; Injections, Intravenous; Male; Nordazepam; Protein Binding; Time Factors

1977
Allergy to diazepam.
    British medical journal, 1977, Apr-16, Volume: 1, Issue:6067

    Topics: Cross Reactions; Diazepam; Humans; Nordazepam

1977
Rapid micro-method for the measurement of diazepam and desmethyldiazepam in blood plasma by gas-liquid chromatography.
    Journal of chromatography, 1977, Jul-21, Volume: 137, Issue:2

    Topics: Chromatography, Gas; Chromatography, Liquid; Diazepam; Humans; Methods; Microchemistry; Nordazepam; Solvents

1977
[Important factors determining human distribution and elimination of diazepam].
    Fortschritte der Medizin, 1977, Aug-25, Volume: 95, Issue:32

    Topics: Animals; Biological Availability; Diazepam; Dogs; Guinea Pigs; Humans; Liver; Nordazepam; Protein Binding; Rabbits; Rats

1977
Rapid determination of diazepam and nordiazepam in plasma by electron capture gas--liquid chromatography. Application in clinical pharmacokinetic studies.
    Journal of chromatography, 1977, Nov-01, Volume: 143, Issue:6

    Topics: Autoanalysis; Chromatography, Gas; Chromatography, Liquid; Diazepam; Humans; Nordazepam

1977
Hydroxylation of three benzodiazepines in vitro.
    Journal of pharmaceutical sciences, 1977, Volume: 66, Issue:10

    Topics: Animals; Biotransformation; Diazepam; Hydroxylation; In Vitro Techniques; Kinetics; Male; Microsomes, Liver; Nordazepam; Rats

1977
Determination of N-desmethyldiazepam in plasma by gas chromatography with an internal standard.
    Journal of chromatography, 1978, Jan-11, Volume: 147

    Topics: Chromatography, Gas; Diazepam; Dose-Response Relationship, Drug; Humans; Nordazepam

1978
Thin-layer chromatographic method for determination of diazepam and its major metabolite, N-desmethyldiazepam, in human serum.
    Journal of chromatography, 1978, Feb-01, Volume: 148, Issue:2

    Topics: Chromatography, Thin Layer; Diazepam; Humans; Nordazepam

1978
High-pressure liquid chromatographic analysis of diazepam, oxazepam and N-desmethyldiazepam in human blood.
    Journal of chromatography, 1978, Mar-21, Volume: 150, Issue:2

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam

1978
High-performance liquid chromatographic determination of benzodiazepines in human plasma.
    Journal of chromatography, 1978, Mar-21, Volume: 150, Issue:2

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam

1978
Determination of benzodiazepine anticonvulsants in plasma by high-performance liquid chromatography.
    Analytical chemistry, 1978, Volume: 50, Issue:4

    Topics: Benzodiazepinones; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Humans; Nordazepam; Spectrophotometry, Ultraviolet

1978
Diazepam, alcohol and drivers.
    The New Zealand medical journal, 1978, Apr-26, Volume: 87, Issue:610

    Topics: Accidents, Traffic; Automobile Driving; Diazepam; Ethanol; Humans; Legislation as Topic; New Zealand; Nordazepam; Wounds and Injuries

1978
Plasma concentrations of diazepam and desmethyldiazepam during chronic diazepam therapy.
    British journal of clinical pharmacology, 1978, Volume: 6, Issue:1

    Topics: Adult; Age Factors; Aged; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Sex Factors; Time Factors

1978
Plasma and urine concentrations of diazepam and its metabolites in children, adults and in diazepam-intoxicated patients.
    International journal of clinical pharmacology and biopharmacy, 1978, Volume: 16, Issue:6

    Topics: Adult; Aging; Biotransformation; Child; Creatinine; Diazepam; Female; Humans; Infant; Infant, Newborn; Kinetics; Male; Nordazepam; Oxazepam

1978
[Binding of prazepam, desalkylprazepam and diazepam to human serum albumin (author's transl)].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 1978, Volume: 98, Issue:6

    Topics: Diazepam; Humans; Nordazepam; Prazepam; Protein Binding; Serum Albumin

1978
[Studies on metabolism of prazepam. II. Metabolism of prazepam, diazepam and desalkylprazepam by rat liver microsomes (author's transl)].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 1978, Volume: 98, Issue:6

    Topics: Animals; Diazepam; In Vitro Techniques; Microsomes, Liver; Nordazepam; Prazepam; Rats

1978
Rapid recovery from massive diazepam overdose.
    JAMA, 1978, Oct-20, Volume: 240, Issue:17

    Topics: Adult; Biotransformation; Diazepam; Female; Half-Life; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Remission, Spontaneous; Suicide, Attempted; Temazepam; Time Factors

1978
Simultaneous gas-chromatographic analysis for diazepam and its major metabolite, desmethyldiazepam, with use of double internal standardization.
    Clinical chemistry, 1978, Volume: 24, Issue:10

    Topics: Adult; Benzodiazepinones; Chromatography, Gas; Diazepam; Female; Humans; Nordazepam; Reference Standards

1978
Fluorescence--TLC densitometric determination of diazepam and other 1,4-benzodiazepines in serum.
    Journal of pharmaceutical sciences, 1978, Volume: 67, Issue:10

    Topics: Benzodiazepines; Chromatography, Thin Layer; Densitometry; Diazepam; Humans; Methods; Nordazepam; Oxazepam; Spectrometry, Fluorescence

1978
Influence of the 2'-chloro substitution on central activity of desmethyldiazepam.
    Pharmacology, 1978, Volume: 17, Issue:3

    Topics: Animals; Avoidance Learning; Behavior, Animal; Choice Behavior; Diazepam; Electroencephalography; Male; Motor Activity; Nordazepam; Rats; Structure-Activity Relationship

1978
A micromethod for simultaneous estimation of blood levels of some commonly used antiepileptic drugs.
    Clinica chimica acta; international journal of clinical chemistry, 1978, Oct-16, Volume: 89, Issue:2

    Topics: Anticonvulsants; Carbamazepine; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Humans; Microchemistry; Nordazepam; Phenobarbital; Phenytoin

1978
Plasma concentrations of diazepam and N-desmethyldiazepam in newborn infants after intravenous, intramuscular, rectal and oral administration.
    Acta paediatrica Scandinavica, 1978, Volume: 67, Issue:6

    Topics: Administration, Oral; Diazepam; Female; Humans; Infant, Newborn; Infant, Newborn, Diseases; Injections, Intramuscular; Injections, Intravenous; Nordazepam; Pregnancy; Rectum; Seizures; Time Factors

1978
Dose-dependent pharmacokinetics of 7-chloro-1,3-dihydro-5-(2'-chlorophenyl)-2H-1,4-benzodiazepin-2-one in dogs.
    Journal of pharmaceutical sciences, 1978, Volume: 67, Issue:12

    Topics: Animals; Diazepam; Dogs; Dose-Response Relationship, Drug; Kinetics; Male; Models, Biological; Nordazepam

1978
Altered elimination of desmethyldiazepam in the elderly.
    British journal of clinical pharmacology, 1979, Volume: 7, Issue:1

    Topics: Adult; Aged; Aging; Diazepam; Half-Life; Humans; Liver; Nordazepam; Time Factors

1979
Monitoring diazepam and desmethyldiazepam concentrations in plasma by gas-liquid chromatography, with use of a nitrogen-sensitive detector.
    Clinical chemistry, 1979, Volume: 25, Issue:1

    Topics: Chromatography, Gas; Diazepam; Epilepsy; Humans; Microchemistry; Nitrogen; Nordazepam

1979
Liquid-chromatographic assay of diazepam and its major metabolites in plasma.
    Clinical chemistry, 1979, Volume: 25, Issue:6

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam

1979
Elimination half-life of nordiazepam.
    Southern medical journal, 1979, Volume: 72, Issue:6

    Topics: Diazepam; Half-Life; Humans; Kinetics; Nordazepam

1979
Effect of age on the pharmacokinetics of diazepam given in conjunction with spinal anesthesia.
    Anesthesiology, 1979, Volume: 51, Issue:2

    Topics: Adult; Age Factors; Aged; Anesthesia, Spinal; Body Water; Diazepam; Humans; Kinetics; Middle Aged; Nordazepam; Oxazepam; Temazepam

1979
Analysis for diazepam and nordiazepam by electron-capture gas chromatography and by liquid chromatography.
    Clinical chemistry, 1979, Volume: 25, Issue:7

    Topics: Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Humans; Methods; Nordazepam

1979
Single case study. Diazepam (Valium) detoxification.
    The Journal of nervous and mental disease, 1979, Volume: 167, Issue:10

    Topics: Adult; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Metabolic Clearance Rate; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1979
[A screening radioimmunoassay for 1,4-benzodiazepines in human blood, serum, and urine using anti-oxazepam-hemisuccinate-antibodies (author's transl)].
    Zeitschrift fur Rechtsmedizin. Journal of legal medicine, 1979, Volume: 83, Issue:3

    Topics: Benzodiazepines; Chromatography, Gas; Chromatography, Thin Layer; Diazepam; Humans; Nordazepam; Oxazepam; Radioimmunoassay; Succinates

1979
Desmethyldiazepam: a specific radioimmunoassay.
    Journal of pharmaceutical sciences, 1979, Volume: 68, Issue:11

    Topics: Antibody Specificity; Diazepam; Humans; Methods; Nordazepam; Radioimmunoassay

1979
Intravascular factors affecting diazepam binding to human serum albumin.
    Biochemical pharmacology, 1979, Nov-15, Volume: 28, Issue:22

    Topics: Binding, Competitive; Dialysis; Diazepam; Fatty Acids; Humans; Nordazepam; Oleic Acids; Oxazepam; Palmitic Acids; Protein Binding; Serum Albumin

1979
Conflict behavior in the squirrel monkey: effects of chlordiazepoxide, diazepam and N-desmethyldiazepam.
    The Journal of pharmacology and experimental therapeutics, 1978, Volume: 204, Issue:1

    Topics: Animals; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Haplorhini; Male; Nordazepam; Reinforcement Schedule; Saimiri; Time Factors

1978
N-desmethyldiazepam: a new metabolite of chlordiazepoxide in man.
    Clinical pharmacology and therapeutics, 1976, Volume: 20, Issue:4

    Topics: Animals; Chlordiazepoxide; Chromatography, Gas; Diazepam; Humans; Nordazepam; Rabbits; Radioimmunoassay; Time Factors

1976
Pharmacokinetics and plasma binding of diazepam in man, dog, rabbit, guinea pig and rat.
    The Journal of pharmacology and experimental therapeutics, 1976, Volume: 199, Issue:1

    Topics: Adult; Animals; Blood Proteins; Body Surface Area; Diazepam; Dogs; Guinea Pigs; Half-Life; Humans; Kinetics; Male; Nordazepam; Protein Binding; Rabbits; Rats; Species Specificity; Swine

1976
A simplified quantitative method for the simultaneous determination of diazepam and its metabolites in serum by thin-layer chromatography.
    Journal of chromatography, 1976, Nov-17, Volume: 128, Issue:1

    Topics: Absorption; Chromatography, Thin Layer; Diazepam; Hot Temperature; Methods; Nordazepam

1976
Diazepam metabolism by rat and human liver in vitro: inhibition by mephenytoin.
    Xenobiotica; the fate of foreign compounds in biological systems, 1992, Volume: 22, Issue:5

    Topics: Animals; Chromatography, Gas; Diazepam; Humans; Hydroxylation; In Vitro Techniques; Kinetics; Liver; Male; Mephenytoin; Methylation; Nordazepam; Polymorphism, Genetic; Rats; Temazepam

1992
Quantitation by gas chromatography with selected-ion monitoring mass spectrometry of "natural" diazepam, N-desmethyldiazepam and oxazepam in normal human serum.
    Journal of chromatography, 1992, Aug-07, Volume: 579, Issue:1

    Topics: Adult; Analysis of Variance; Diazepam; Female; Gas Chromatography-Mass Spectrometry; Humans; Male; Nordazepam; Oxazepam

1992
Studies on the excretion of diazepam and nordazepam into milk for the prediction of milk-to-plasma drug concentration ratios.
    Pharmaceutical research, 1992, Volume: 9, Issue:10

    Topics: Animals; Diazepam; Diffusion; Fats; Female; Infusions, Intravenous; Jugular Veins; Milk, Human; Models, Biological; Nordazepam; Pregnancy; Protein Binding; Rabbits

1992
Incidence of S-mephenytoin hydroxylation deficiency in a Korean population and the interphenotypic differences in diazepam pharmacokinetics.
    Clinical pharmacology and therapeutics, 1992, Volume: 52, Issue:2

    Topics: Adult; Asian People; Creatinine; Diazepam; Female; Humans; Hydroxylation; Korea; Male; Mephenytoin; Mixed Function Oxygenases; Nordazepam; Phenotype; Polymorphism, Genetic

1992
Comparative metabolism of clinically important precursors of N-desmethyldiazepam using phenobarbitone-pretreated rat liver microsomes.
    Biochemical pharmacology, 1992, Mar-17, Volume: 43, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Diazepam; Hydroxylation; Male; Methylation; Microsomes, Liver; Nordazepam; Phenobarbital; Prazepam; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1992
Elevated brain concentrations of 1,4-benzodiazepines in fulminant hepatic failure.
    The New England journal of medicine, 1991, Aug-15, Volume: 325, Issue:7

    Topics: Adult; Aged; Benzodiazepines; Brain Chemistry; Chromatography; Diazepam; Flumazenil; Frontal Lobe; gamma-Aminobutyric Acid; Hepatic Encephalopathy; Humans; Mass Spectrometry; Middle Aged; Nordazepam; Receptors, GABA-A; Synaptic Transmission

1991
Chronic administration of and dependence on halazepam, diazepam, and nordiazepam in the dog.
    Drug and alcohol dependence, 1991, Volume: 28, Issue:3

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Dogs; Dose-Response Relationship, Drug; Flumazenil; Neurologic Examination; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Distribution of diazepam, nordiazepam, and oxazepam between brain extraneuronal space, brain tissue, plasma, and cerebrospinal fluid in diazepam and nordiazepam dependent dogs.
    Psychopharmacology, 1991, Volume: 105, Issue:4

    Topics: Animals; Brain; Diazepam; Dogs; Extracellular Space; Female; Nordazepam; Oxazepam; Substance-Related Disorders

1991
Pharmacokinetics of diazepam intramuscularly administered to rhesus monkeys.
    Journal of pharmaceutical sciences, 1991, Volume: 80, Issue:10

    Topics: Animals; Anticonvulsants; Blood Proteins; Diazepam; Hematocrit; Injections, Intramuscular; Macaca mulatta; Male; Nordazepam; Protein Binding; Seizures; Soman

1991
Determination of diazepam and nordazepam in milk and plasma in the presence of oxazepam and temazepam.
    Journal of chromatography, 1991, Mar-08, Volume: 564, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Flurazepam; Humans; Hydrogen-Ion Concentration; Milk, Human; Nordazepam; Oxazepam; Temazepam

1991
Cytochrome P450IIIA enzymes in rat liver microsomes: involvement in C3-hydroxylation of diazepam and nordazepam but not N-dealkylation of diazepam and temazepam.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Cytochrome P-450 Enzyme System; Diazepam; Female; Hydroxylation; Kinetics; Male; Microsomes, Liver; Nordazepam; Oxidoreductases, N-Demethylating; Phenobarbital; Rats; Rats, Inbred Strains; Sex Factors; Species Specificity; Substrate Specificity; Temazepam

1990
Depressive stupor treated with intramuscular chlordesmethyldiazepam.
    Canadian journal of psychiatry. Revue canadienne de psychiatrie, 1990, Volume: 35, Issue:3

    Topics: Anti-Anxiety Agents; Arousal; Benzodiazepines; Depressive Disorder; Diazepam; Female; Humans; Injections, Intramuscular; Middle Aged; Nordazepam

1990
Benzodiazepine-induced antagonism of opioid antinociception may be abolished by spinalization or blockade of the benzodiazepine receptor.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Analgesics; Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Male; Mice; Midazolam; Morphine; Narcotics; Nordazepam; Psychomotor Performance; Reaction Time; Receptors, GABA-A; Receptors, Opioid; Skin Temperature; Spinal Cord

1990
Characterization by saturation studies of the in vivo binding of [3H]flunitrazepam in mouse brain.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:2

    Topics: Animals; Brain; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Flunitrazepam; Kinetics; Mice; Nordazepam; Oxazepam

1991
Excretion of diazepam and its metabolites in human milk during withdrawal from combination high dose diazepam and oxazepam.
    British journal of clinical pharmacology, 1990, Volume: 29, Issue:1

    Topics: Adult; Diazepam; Drug Combinations; Female; Humans; Infant; Milk, Human; Nordazepam; Oxazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam

1990
Effect of chronic oral delorazepam on in vitro and in vivo hepatic drug-metabolizing enzyme activities in the rat.
    Research communications in chemical pathology and pharmacology, 1990, Volume: 67, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cytochrome P-450 Enzyme System; Diazepam; Enzyme Induction; In Vitro Techniques; Liver; Male; Mixed Function Oxygenases; Nordazepam; Phenobarbital; Rats; Rats, Inbred Strains

1990
Diazepam loading in alcohol withdrawal: clinical pharmacokinetics.
    International journal of clinical pharmacology, therapy, and toxicology, 1990, Volume: 28, Issue:5

    Topics: Administration, Oral; Adult; Diazepam; Ethanol; Half-Life; Humans; Male; Middle Aged; Nordazepam; Substance Withdrawal Syndrome; Time Factors

1990
Endogenous benzodiazepines in brain: right or wrong?
    Trends in neurosciences, 1988, Volume: 11, Issue:3

    Topics: Benzodiazepines; Brain; Diazepam; Female; Humans; Male; Nordazepam

1988
Importance of genetic factors in the regulation of diazepam metabolism: relationship to S-mephenytoin, but not debrisoquin, hydroxylation phenotype.
    Clinical pharmacology and therapeutics, 1989, Volume: 45, Issue:4

    Topics: Adult; Benzodiazepines; Debrisoquin; Diazepam; Female; Humans; Hydantoins; Isoquinolines; Male; Mephenytoin; Mixed Function Oxygenases; Nordazepam; Phenotype; Smoking

1989
Radioreceptor assay of clonazepam and diazepam in blood for therapeutic drug monitoring.
    Therapeutic drug monitoring, 1989, Volume: 11, Issue:4

    Topics: Adolescent; Animals; Child; Child, Preschool; Chromatography, Gas; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Flunitrazepam; Humans; Male; Nordazepam; Radioligand Assay; Rats

1989
Detection of desmethyldiazepam and diazepam in brain of different species and plants.
    Biochemical pharmacology, 1989, Aug-01, Volume: 38, Issue:15

    Topics: Animals; Benzodiazepines; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Nordazepam; Plants; Radioligand Assay; Species Specificity

1989
In vitro drug metabolism and pharmacokinetics of diazepam in cynomolgus monkey hepatocytes during culture for six days.
    Biochemical pharmacology, 1989, Aug-15, Volume: 38, Issue:16

    Topics: Animals; Cells, Cultured; Cytochrome P-450 Enzyme System; Diazepam; Liver; Macaca fascicularis; Male; Models, Biological; Nordazepam; Oxazepam; Oxygenases; Temazepam; Time Factors

1989
Effect of the benzodiazepines diazepam, des-N-methyldiazepam and midazolam on corticosteroid biosynthesis in bovine adrenocortical cells in vitro; location of site of action.
    Journal of steroid biochemistry, 1989, Volume: 33, Issue:2

    Topics: Adrenal Cortex; Aldosterone; Animals; Benzodiazepines; Cattle; Diazepam; Hydrocortisone; In Vitro Techniques; Midazolam; Nordazepam

1989
A large-sample study of diazepam pharmacokinetics.
    Therapeutic drug monitoring, 1989, Volume: 11, Issue:6

    Topics: Adolescent; Adult; Body Weight; Chromatography, Gas; Diazepam; Half-Life; Humans; Male; Nordazepam

1989
[Control of the side effects of ketamine: chlordemethyldiazepam vs diazepam in pre-anesthesia].
    Minerva anestesiologica, 1989, Volume: 55, Issue:10

    Topics: Adolescent; Adult; Age Factors; Anti-Anxiety Agents; Benzodiazepines; Blood Pressure; Child; Child, Preschool; Diazepam; Drug Evaluation; Female; Heart Rate; Humans; Infant; Infant, Newborn; Ketamine; Male; Nordazepam; Preanesthetic Medication

1989
Determination of pharmacodynamics of diazepam by quantitative pharmaco-EEG.
    The Japanese journal of psychiatry and neurology, 1989, Volume: 43, Issue:4

    Topics: Adult; Computer Systems; Diazepam; Dose-Response Relationship, Drug; Electroencephalography; Evoked Potentials; Humans; Infusions, Intravenous; Male; Nordazepam; Reaction Time; Signal Processing, Computer-Assisted

1989
Efficacy of flumazenil in COPD patient with therapeutic diazepam levels.
    Lancet (London, England), 1989, Feb-18, Volume: 1, Issue:8634

    Topics: Aged; Diazepam; Drug Evaluation; Flumazenil; Humans; Lung Diseases, Obstructive; Male; Nordazepam

1989
Physical dependence on diazepam in the dog: precipitation of different abstinence syndromes by the benzodiazepine receptor antagonists Ro 15-1788 and ZK 93426.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1989
Kinetics of drug action in disease states. XXV. Effect of experimental hypovolemia on the pharmacodynamics and pharmacokinetics of desmethyldiazepam.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:2

    Topics: Animals; Cerebral Cortex; Diazepam; Kinetics; Male; Nordazepam; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Reflex; Shock

1988
Effects of caffeine and chlor-desmethyldiazepam on fighting behavior of mice with different reactivity baselines.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:2

    Topics: Aggression; Animals; Anti-Anxiety Agents; Benzodiazepines; Caffeine; Dextroamphetamine; Diazepam; Electroshock; Male; Mice; Nordazepam; Pentylenetetrazole; Seizures

1985
Screening and quantification of hypnotic sedatives in serum by capillary gas chromatography with a nitrogen-phosphorus detector, and confirmation by capillary gas chromatography-mass spectrometry.
    Clinical chemistry, 1986, Volume: 32, Issue:2

    Topics: Amobarbital; Barbiturates; Chromatography, Gas; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Hypnotics and Sedatives; Nordazepam; Pentobarbital; Secobarbital; Toxicology

1986
Disruption of schedule-controlled behavior by Ro 15-1788 one day after acute treatment with benzodiazepines.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Conditioning, Operant; Convulsants; Diazepam; Flumazenil; Male; Nordazepam; Reinforcement Schedule; Saimiri

1986
Interaction of diazepam with famotidine and cimetidine, two H2-receptor antagonists.
    Journal of clinical pharmacology, 1986, Volume: 26, Issue:4

    Topics: Adult; Biotransformation; Cimetidine; Diazepam; Drug Interactions; Famotidine; Half-Life; Histamine H2 Antagonists; Humans; Infusions, Parenteral; Kinetics; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam; Thiazoles

1986
Age-related multiple-dose pharmacokinetics and anxiolytic effects of delorazepam (chlordesmethyldiazepam).
    International journal of clinical pharmacology research, 1986, Volume: 6, Issue:4

    Topics: Adult; Aged; Aging; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Diazepam; Female; Humans; Kinetics; Male; Middle Aged; Nordazepam

1986
Diazepam and desmethyldiazepam differ in their affinities and efficacies at 'central' and 'peripheral' benzodiazepine receptors.
    The Journal of pharmacy and pharmacology, 1987, Volume: 39, Issue:5

    Topics: Adrenal Glands; Animals; Benzodiazepines; Brain; Cerebellum; Cerebral Cortex; Diazepam; In Vitro Techniques; Male; Nordazepam; Rats; Receptors, GABA-A

1987
[Chlordesmethyldiazepam as an anesthesia-inducing agent: time of loss of consciousness. Statistical analysis in man].
    Acta bio-medica de L'Ateneo parmense : organo della Societa di medicina e scienze naturali di Parma, 1987, Volume: 58, Issue:1-2

    Topics: Adult; Aged; Anesthesia, Intravenous; Anesthetics; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Middle Aged; Nordazepam; Preanesthetic Medication; Time Factors; Unconsciousness

1987
Effect of food on absorption of chlordemethyldiazepam.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Food; Half-Life; Humans; Intestinal Absorption; Male; Nordazepam

1988
Desmethyldiazepam pharmacokinetics: studies following intravenous and oral desmethyldiazepam, oral clorazepate, and intravenous diazepam.
    Journal of clinical pharmacology, 1988, Volume: 28, Issue:9

    Topics: Administration, Oral; Adult; Aged; Anti-Anxiety Agents; Biological Availability; Clorazepate Dipotassium; Diazepam; Female; Half-Life; Humans; Injections, Intravenous; Male; Middle Aged; Nordazepam

1988
[A ketamine-chlordemethyldiazepam combination in celioscopy].
    Minerva ginecologica, 1988, Volume: 40, Issue:12

    Topics: Adolescent; Adult; Aged; Anesthesia, General; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Combinations; Drug Evaluation; Female; Humans; Ketamine; Laparoscopy; Middle Aged; Nordazepam

1988
[Use of a chlordemethyldiazepam-fentanyl combination in invasive neuroradiologic examinations].
    Minerva anestesiologica, 1988, Volume: 54, Issue:9

    Topics: Adolescent; Adult; Aged; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Evaluation; Drug Therapy, Combination; Female; Fentanyl; Humans; Male; Middle Aged; Neuroradiography; Nordazepam; Premedication

1988
Kinetics of drug action in disease states. XXIV. Pharmacodynamics of diazepam and its active metabolites in rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Female; Nordazepam; Oxazepam; Rats; Rats, Inbred Lew; Reflex; Temazepam

1988
Discriminative-stimulus effects of midazolam in squirrel monkeys: comparison with other drugs and antagonism by Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Azabicyclo Compounds; Barbital; Benzodiazepines; Benzodiazepinones; Buspirone; Caffeine; Chlordiazepoxide; Cinanserin; Clozapine; Conditioning, Operant; Cyproheptadine; Diazepam; Diphenhydramine; Discrimination Learning; Electroshock; Flumazenil; Male; Midazolam; Muscimol; Nordazepam; Pentobarbital; Piperazines; Pyridazines; Pyrimidines; Saimiri; Tripelennamine

1985
Diazepam and N-desmethyldiazepam are found in rat brain and adrenal and may be of plant origin.
    Journal of neural transmission, 1987, Volume: 70, Issue:3-4

    Topics: Adrenal Glands; Animals; Brain Chemistry; Cerebellum; Cerebral Cortex; Diazepam; Male; Nordazepam; Pituitary Gland; Rats; Specific Pathogen-Free Organisms; Tissue Extracts; Triticum

1987
Purification of a benzodiazepine from bovine brain and detection of benzodiazepine-like immunoreactivity in human brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:23

    Topics: Animals; Antibodies, Monoclonal; Benzodiazepines; Brain Chemistry; Cattle; Chromatography, High Pressure Liquid; Diazepam; Humans; Immunologic Techniques; Mass Spectrometry; Nordazepam; Receptors, GABA-A; Spectrum Analysis

1986
Preliminary study of the pharmacokinetics of desmethyldiazepam administered as drops or tablets.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:1

    Topics: Adult; Diazepam; Female; Humans; Kinetics; Male; Nordazepam; Sex Factors; Solutions; Tablets; Time Factors

1986
The pharmacokinetics of diazepam and desmethyldiazepam in rat brain and plasma.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Blood Proteins; Brain; Diazepam; Half-Life; Male; Nordazepam; Protein Binding; Rats; Time Factors

1986
Acute tolerance to diazepam in mice: pharmacokinetic considerations.
    Clinical and experimental pharmacology & physiology, 1986, Volume: 13, Issue:2

    Topics: Animals; Brain Chemistry; Cycloheximide; Diazepam; Drug Tolerance; Kinetics; Male; Mice; Microsomes, Liver; Nordazepam

1986
Potencies of diazepam metabolites in rats trained to discriminate diazepam.
    Life sciences, 1986, Jul-07, Volume: 39, Issue:1

    Topics: Animals; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Nordazepam; Oxazepam; Rats; Rats, Inbred Strains; Temazepam

1986
The effect of diazepam on indices of 5-HT function in man.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:5

    Topics: Adult; Blood Platelets; Diazepam; Humans; Hypnotics and Sedatives; Imipramine; Male; Nordazepam; Prolactin; Serotonin; Time Factors; Tryptophan

1986
Serum concentrations of diazepam and its metabolite desmethyldiazepam in epileptic patients after chronic diazepam treatment.
    Acta neurologica, 1986, Volume: 8, Issue:4

    Topics: Adult; Aged; Diazepam; Epilepsy; Humans; Middle Aged; Nordazepam

1986
[Epilepsy induced by penicillin in rabbits: comparative study of the anticonvulsant effects of diazepam and chlordesmethyldiazepam].
    Bollettino chimico farmaceutico, 1986, Volume: 125, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Epilepsy; Male; Nordazepam; Penicillins; Rabbits

1986
Diazepam metabolism in the guinea pig materno-fetal model: effects of cigarette smoke.
    Drug and chemical toxicology, 1986, Volume: 9, Issue:3-4

    Topics: Animals; Biotransformation; Dealkylation; Diazepam; Female; Guinea Pigs; Maternal-Fetal Exchange; Microsomes, Liver; Nordazepam; Pregnancy; Smoking

1986
Differences in diazepam pharmacokinetics in Chinese and white Caucasians--relation to body lipid stores.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:2

    Topics: Adult; Asian People; Diazepam; Humans; Kinetics; Lipids; Male; Nordazepam; White People

1987
Microsample determination of diazepam and its three metabolites in serum by reversed-phase high-performance liquid chromatography.
    Journal of chromatography, 1987, Apr-24, Volume: 416, Issue:1

    Topics: Animals; Biotransformation; Chlordiazepoxide; Chromatography, High Pressure Liquid; Diazepam; Hydrogen-Ion Concentration; Indicators and Reagents; Nordazepam; Rats; Spectrophotometry, Ultraviolet; Temazepam

1987
Validation of a radioreceptor assay technique for monitoring pharmacological active material during intensive diazepam tetanus therapy.
    International journal of clinical pharmacology, therapy, and toxicology, 1987, Volume: 25, Issue:7

    Topics: Biotransformation; Chromatography, Gas; Cimetidine; Diazepam; Humans; Kinetics; Middle Aged; Nordazepam; Oxazepam; Radioligand Assay; Tetanus

1987
Placental and blood-CSF transfer of orally administered diazepam in the same person.
    Pharmacology & toxicology, 1987, Volume: 61, Issue:1

    Topics: Adult; Biotransformation; Diazepam; Female; Fetal Blood; Humans; Maternal-Fetal Exchange; Nordazepam; Oxazepam; Pregnancy

1987
The effect of diazepam on nociception in mice.
    Pharmacology & toxicology, 1987, Volume: 61, Issue:2

    Topics: Analgesics; Animals; Diazepam; Male; Mice; Nordazepam; Pain Measurement; Psychomotor Performance

1987
Analysis of chlorodesmethyldiazepam and its metabolites in plasma and urine.
    Journal of chromatography, 1987, Sep-25, Volume: 420, Issue:2

    Topics: Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Glucuronates; Humans; Lorazepam; Nordazepam; Oxazepam

1987
Simultaneous determination of diazepam and its active metabolites in rat serum, brain and cerebrospinal fluid by high-performance liquid chromatography.
    Journal of chromatography, 1987, Nov-27, Volume: 422

    Topics: Animals; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Female; Nordazepam; Oxazepam; Postural Balance; Rats; Rats, Inbred Strains; Temazepam

1987
Apparent lesser physical dependence potential of nor-diazepam compared to diazepam in the rat.
    NIDA research monograph, 1987, Volume: 76

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Male; Nordazepam; Rats; Rats, Inbred Strains; Substance-Related Disorders

1987
Imipramine treatment alters the pharmacokinetics and pharmacodynamics of diazepam.
    Journal of pharmaceutical sciences, 1987, Volume: 76, Issue:12

    Topics: Animals; Blood Proteins; Brain Chemistry; Diazepam; Drug Interactions; Imipramine; Liver; Male; Nordazepam; Oxazepam; Pentylenetetrazole; Protein Binding; Rats; Rats, Inbred Strains; Temazepam

1987
The effect of fluoxetine on the pharmacokinetics and psychomotor responses of diazepam.
    Clinical pharmacology and therapeutics, 1988, Volume: 43, Issue:4

    Topics: Adult; Diazepam; Drug Interactions; Fluoxetine; Humans; Male; Middle Aged; Nordazepam; Propylamines; Psychomotor Performance

1988
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Improved method for the determination of diazepam and N-desmethyldiazepam in plasma using capillary gas chromatography and nitrogen-phosphorus detection.
    Journal of chromatography, 1988, Feb-26, Volume: 424, Issue:2

    Topics: Chromatography, Gas; Diazepam; Humans; Nitrogen; Nordazepam; Phosphorus; Solvents

1988
Sensitive determination of diazepam and N-desmethyldiazepam in human material using capillary gas chromatography-mass spectrometry.
    Journal of chromatography, 1988, Oct-14, Volume: 431, Issue:2

    Topics: Aged; Aged, 80 and over; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Indicators and Reagents; Male; Muscles; Nordazepam

1988
[Effect of sodium valproate on brain levels of diazepam and N-desmethyldiazepam in the rat].
    Archivos de farmacologia y toxicologia, 1985, Volume: 11, Issue:1

    Topics: Animals; Brain Chemistry; Diazepam; Male; Nordazepam; Rats; Rats, Inbred Strains; Valproic Acid

1985
Long-lasting anticonvulsant effects of diazepam in different mouse strains: correlations with brain concentrations and receptor occupancy.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Anticonvulsants; Brain Chemistry; Diazepam; Mice; Mice, Inbred C3H; Nordazepam; Oxazepam; Pentylenetetrazole; Seizures; Species Specificity; Time Factors

1985
Responsiveness to oral diazepam in the elderly: relationship to total and free plasma concentrations.
    British journal of clinical pharmacology, 1985, Volume: 20, Issue:2

    Topics: Adult; Aged; Aging; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Hypnotics and Sedatives; Male; Nordazepam; Posture; Protein Binding; Psychomotor Performance

1985
Liquid-chromatographic assay of diazepam and its major metabolites in serum, and application to pharmacokinetic study of high doses of diazepam in schizophrenics.
    Clinical chemistry, 1985, Volume: 31, Issue:10

    Topics: Administration, Oral; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Kinetics; Nordazepam; Oxazepam; Schizophrenia; Temazepam

1985
Severe withdrawal syndrome after substitution of a short-acting benzodiazepine for a long-acting benzodiazepine.
    Drug intelligence & clinical pharmacy, 1985, Volume: 19, Issue:10

    Topics: Diazepam; Female; Half-Life; Humans; Middle Aged; Nordazepam; Oxazepam; Substance Withdrawal Syndrome

1985
Development of tolerance to the anticonvulsant effect of diazepam in amygdala-kindled rats.
    Experimental neurology, 1985, Volume: 90, Issue:2

    Topics: Amygdala; Animals; Anticonvulsants; Diazepam; Drug Tolerance; Electric Stimulation; Female; Kindling, Neurologic; Kinetics; Nordazepam; Rats; Rats, Inbred Strains; Time Factors

1985
Omeprazole inhibits oxidative drug metabolism. Studies with diazepam and phenytoin in vivo and 7-ethoxycoumarin in vitro.
    Gastroenterology, 1985, Volume: 89, Issue:6

    Topics: Adult; Benzimidazoles; Coumarins; Diazepam; Drug Interactions; Humans; In Vitro Techniques; Kinetics; Male; Microsomes, Liver; Nordazepam; Omeprazole; Oxidation-Reduction; Phenytoin

1985
N-desmethyldiazepam physical dependence in dogs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Analysis of Variance; Animals; Body Weight; Diazepam; Dogs; Drinking; Energy Intake; Female; Lorazepam; Muscle Spasticity; Nordazepam; Oxazepam; Paresthesia; Substance Withdrawal Syndrome; Temazepam; Time Factors

1985
Plasma concentrations of diazepam and N-desmethyldiazepam in Asian children after an intravenous or rectal dose of diazepam.
    The Journal of the Singapore Paediatric Society, 1985, Volume: 27, Issue:3-4

    Topics: Child; Child, Preschool; Diazepam; Female; Humans; Injections, Intravenous; Male; Nordazepam; Rectum

1985
Monitoring clorazepate dipotassium as desmethyldiazepam in plasma by electron-capture gas--liquid chromatography.
    Clinical chemistry, 1980, Volume: 26, Issue:1

    Topics: Anti-Anxiety Agents; Chromatography, Gas; Clorazepate Dipotassium; Diazepam; Dose-Response Relationship, Drug; Humans; Nordazepam

1980
Determination of some benzodiazepines and metabolites in serum, urine and saliva by high-performance liquid chromatography.
    Journal of chromatography, 1980, Feb-08, Volume: 181, Issue:2

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Humans; Mathematics; Nordazepam; Oxazepam; Saliva; Temazepam

1980
The psychosedative effect of chlordesmethyldiazepam on anxiety states in neurotic and psychotic inpatients.
    Clinical therapeutics, 1980, Volume: 3, Issue:3

    Topics: Adolescent; Adult; Aged; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Diazepam; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Neurotic Disorders; Nordazepam; Psychiatric Status Rating Scales; Psychotic Disorders; Reaction Time

1980
[Pharmacokinetic of benzodiazepines in old age].
    Schweizerische medizinische Wochenschrift, 1981, Nov-21, Volume: 111, Issue:47

    Topics: Adult; Aged; Aging; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Half-Life; Humans; Lorazepam; Metabolic Clearance Rate; Middle Aged; Nitrazepam; Nordazepam; Oxazepam

1981
Aspects of the interaction of thyroxine and its binding serum proteins with 1,4-benzodiazepine tranquillizers.
    Biochemical medicine, 1981, Volume: 26, Issue:2

    Topics: Anti-Anxiety Agents; Autoradiography; Binding, Competitive; Chlordiazepoxide; Diazepam; Electrophoresis, Polyacrylamide Gel; Humans; Male; Nordazepam; Oxazepam; Temazepam; Thyroxine; Thyroxine-Binding Proteins

1981
Studies on some pharmacological activities of 7-nitro-2-amino-5-phenyl-3H-1,5-benzodiazepine (CP 1414 S) in the rat. A comparison with diazepam.
    Arzneimittel-Forschung, 1981, Volume: 31, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Brain Chemistry; Conflict, Psychological; Diazepam; Female; Kinetics; Motor Activity; Nordazepam; Pentylenetetrazole; Rats; Rats, Inbred Strains

1981
Pharmacokinetics of N-desmethyldiazepam after a single oral dose of clorazepate: the effect of smoking.
    European journal of clinical pharmacology, 1981, Volume: 21, Issue:3

    Topics: Administration, Oral; Adult; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Humans; Kinetics; Male; Nordazepam; Smoking

1981
Effect of age and sex on disposition of desmethyldiazepam formed from its precursor clorazepate.
    Psychopharmacology, 1981, Volume: 75, Issue:2

    Topics: Adult; Age Factors; Aged; Anti-Anxiety Agents; Biotransformation; Clorazepate Dipotassium; Diazepam; Female; Humans; Liver; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam; Sex Factors

1981
Does ethyl-beta-carboline-3-carboxylate interact with mouse brain benzodiazepine receptors in vivo?
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:6

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Diazepam; Indoles; Mice; Nordazepam; Receptors, Drug; Receptors, GABA-A

1982
[Anxiolytics in man: studies on sleep and performance (author's transl)].
    L'Encephale, 1982, Volume: 8, Issue:2

    Topics: Anti-Anxiety Agents; Anxiety Disorders; Arousal; Attention; Benzodiazepines; Benzodiazepinones; Clobazam; Clorazepate Dipotassium; Diazepam; Dose-Response Relationship, Drug; Humans; Motor Skills; Nordazepam; Sleep Stages; Visual Perception

1982
Some behavioral effects of chlorodesmethyldiazepam and lorazepam.
    Polish journal of pharmacology and pharmacy, 1981, Volume: 33, Issue:6

    Topics: Acoustic Stimulation; Aggression; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Diazepam; Humans; Lorazepam; Male; Mice; Nordazepam; Rats; Seizures

1981
Rapid gas chromatographic measurement of diazepam and its metabolites desmethyldiazepam, oxazepam, and 3-hydroxydiazepam (temazepam) in small samples of plasma.
    Therapeutic drug monitoring, 1982, Volume: 4, Issue:3

    Topics: Anti-Anxiety Agents; Biotransformation; Chromatography, Gas; Diazepam; Humans; Nordazepam; Oxazepam; Temazepam

1982
Determination of peptidoaminobenzophenone (2-o-chlorobenzoyl-4-chloro-N-methyl-N'-glycylglycinanilide) and its metabolites in human plasma by glass capillary gas chromatography negative ion chemical ionization mass spectrometry--1.
    Biomedical mass spectrometry, 1982, Volume: 9, Issue:12

    Topics: Anti-Anxiety Agents; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Glycine; Humans; Lorazepam; Nordazepam

1982
Does chlordesmethyldiazepam have a specific anti-erotic effect? Report on five observations.
    Acta psychiatrica Belgica, 1982, Volume: 82, Issue:6

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Therapy, Combination; Female; Humans; Libido; Male; Middle Aged; Neurotic Disorders; Nordazepam

1982
High-performance liquid chromatography determination of dipotassium clorazepate and its major metabolite nordiazepam in plasma.
    Journal of chromatography, 1983, Apr-08, Volume: 273, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Clorazepate Dipotassium; Diazepam; Dogs; Half-Life; Humans; Kinetics; Nordazepam

1983
Pharmacokinetics of benzodiazepines and psychostimulants in children.
    Journal of clinical psychopharmacology, 1983, Volume: 3, Issue:4

    Topics: Adolescent; Adult; Anti-Anxiety Agents; Attention Deficit Disorder with Hyperactivity; Biotransformation; Child; Child Development; Child, Preschool; Diazepam; Epilepsy; Female; Half-Life; Humans; Infant; Infant, Newborn; Kinetics; Male; Methylphenidate; Nordazepam

1983
Clorazepate dipotassium and diazepam in renal insufficiency: serum concentrations and protein binding of diazepam and desmethyldiazepam.
    Nephron, 1984, Volume: 37, Issue:2

    Topics: Adult; Aged; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Kidney Failure, Chronic; Kinetics; Male; Middle Aged; Nordazepam; Protein Binding

1984
[Pharmacokinetics and metabolite pattern of tetrazepam and chlordesmethyldiazepam].
    Beitrage zur gerichtlichen Medizin, 1984, Volume: 42

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Biotransformation; Diazepam; Humans; Kinetics; Male; Nordazepam

1984
Placental transfer of pinazepam and its metabolite N-desmethyldiazepam in women at term.
    European journal of clinical pharmacology, 1984, Volume: 27, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Diazepam; Female; Humans; Labor, Obstetric; Maternal-Fetal Exchange; Milk, Human; Nordazepam; Placenta; Pregnancy

1984
Comparative single-dose kinetics of oxazolam, prazepam, and clorazepate: three precursors of desmethyldiazepam.
    Journal of clinical pharmacology, 1984, Volume: 24, Issue:10

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Clorazepate Dipotassium; Diazepam; Female; Humans; Kinetics; Male; Molecular Weight; Nordazepam; Prazepam

1984
Antiepileptic effect and serum levels of clorazepate on children with refractory seizures.
    Brain & development, 1984, Volume: 6, Issue:6

    Topics: Adolescent; Adult; Anti-Anxiety Agents; Anticonvulsants; Child; Child, Preschool; Clorazepate Dipotassium; Diazepam; Drug Therapy, Combination; Epilepsies, Myoclonic; Epilepsies, Partial; Epilepsy; Epilepsy, Absence; Humans; Infant; Nordazepam; Spasms, Infantile

1984
Value of serum diazepam and nordiazepam measurements in anxious patients.
    Journal of affective disorders, 1984, Volume: 7, Issue:1

    Topics: Adult; Aged; Anxiety Disorders; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Nordazepam; Patient Compliance; Time Factors

1984
Blood concentrations of diazepam and its metabolites in children and neonates with tetanus.
    The Journal of pediatrics, 1983, Volume: 102, Issue:1

    Topics: Child; Diazepam; Female; Humans; Infant, Newborn; Infant, Newborn, Diseases; Male; Nordazepam; Oxazepam; Tetanus

1983
Diazepam kinetics in patients with severe burns.
    Anesthesia and analgesia, 1983, Volume: 62, Issue:3

    Topics: Adult; Aged; Burns; Diazepam; Female; Half-Life; Humans; Kinetics; Male; Middle Aged; Nordazepam

1983
Repeated diazepam dosing in cirrhotic patients: cumulation and sedation.
    Clinical pharmacology and therapeutics, 1983, Volume: 33, Issue:4

    Topics: Adult; Diazepam; Half-Life; Humans; Hypnotics and Sedatives; Kinetics; Liver Cirrhosis; Male; Middle Aged; Nordazepam

1983
The role of buffer composition during equilibrium dialysis in determining concentrations of free diazepam in serum.
    Methods and findings in experimental and clinical pharmacology, 1983, Volume: 5, Issue:1

    Topics: Buffers; Dialysis; Diazepam; Humans; Male; Nordazepam; Protein Binding

1983
Differences in in vitro binding of diazepam and N-desmethyldiazepam to maternal and fetal plasma proteins at birth: relation to free fatty acid concentration and other parameters.
    Clinical pharmacology and therapeutics, 1983, Volume: 34, Issue:2

    Topics: Adolescent; Adult; Blood Proteins; Diazepam; Fatty Acids, Nonesterified; Female; Fetal Blood; Humans; Infant, Newborn; Labor, Obstetric; Middle Aged; Nordazepam; Pregnancy; Protein Binding

1983
Halazepam as a precursor of desmethyldiazepam: quantitation by electron-capture gas-liquid chromatography.
    Psychopharmacology, 1983, Volume: 80, Issue:2

    Topics: Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chromatography, Gas; Diazepam; Humans; Kinetics; Nordazepam

1983
Metabolic and pharmacological studies with N-methyl-N'-methyl-2'-allyl-2-benzoyl-4-chloro-glycinanilide (F 1797).
    Arzneimittel-Forschung, 1983, Volume: 33, Issue:7

    Topics: Anilides; Animals; Anticonvulsants; Brain Chemistry; Diazepam; Male; Nordazepam; Pentylenetetrazole; Rats; Rats, Inbred Strains

1983
Pharmacokinetic model for diazepam and its major metabolite desmethyldiazepam following diazepam administration.
    Journal of pharmaceutical sciences, 1983, Volume: 72, Issue:11

    Topics: Adult; Clorazepate Dipotassium; Diazepam; Humans; Kinetics; Male; Models, Biological; Nordazepam

1983
Multiple-dose pharmacokinetics of diazepam following once-daily administration of a controlled-release capsule.
    Therapeutic drug monitoring, 1983, Volume: 5, Issue:4

    Topics: Adult; Biological Availability; Delayed-Action Preparations; Diazepam; Female; Half-Life; Humans; Kinetics; Male; Middle Aged; Nordazepam

1983
Decreased serum protein binding of diazepam and its major metabolite in the neonate during the first postnatal week relate to increased free fatty acid levels.
    British journal of clinical pharmacology, 1984, Volume: 17, Issue:1

    Topics: Adult; Bilirubin; Blood Proteins; Diazepam; Fatty Acids, Nonesterified; Female; Fetal Blood; Humans; Infant, Newborn; Nordazepam; Pregnancy; Protein Binding; Serum Albumin

1984
Pharmacokinetics of diazepam and nordiazepam in the cat.
    Journal of pharmaceutical sciences, 1984, Volume: 73, Issue:3

    Topics: Animals; Cats; Diazepam; Female; Injections, Intravenous; Kinetics; Liver Circulation; Nordazepam; Time Factors

1984
Diazepam and desmethyldiazepam plasma concentrations in chronic anxious outpatients.
    Pharmacopsychiatry, 1984, Volume: 17, Issue:2

    Topics: Adult; Anxiety Disorders; Chronic Disease; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam

1984
Serum protein binding of diazepam, desmethyldiazepam, furosemide, indomethacin, warfarin, and phenobarbital in human fetus, mother, and newborn infant.
    Pediatric pharmacology (New York, N.Y.), 1983, Volume: 3, Issue:3-4

    Topics: Blood Proteins; Diazepam; Fatty Acids, Nonesterified; Female; Fetal Blood; Furosemide; Humans; Indomethacin; Infant, Newborn; Maternal-Fetal Exchange; Nordazepam; Phenobarbital; Pregnancy; Protein Binding; Warfarin

1983
In vitro interaction of diazepam and oxazepam with pancuronium and suxamethonium.
    British journal of anaesthesia, 1984, Volume: 56, Issue:10

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Muscle Contraction; Neuromuscular Junction; Nordazepam; Oxazepam; Pancuronium; Rats; Rats, Inbred Strains; Succinylcholine; Temazepam

1984
Propranolol interactions with diazepam, lorazepam, and alprazolam.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:4

    Topics: Adolescent; Adult; Alprazolam; Benzodiazepines; Biotransformation; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Female; Humans; Injections, Intravenous; Kinetics; Lorazepam; Male; Nordazepam; Propranolol

1984
Diazepam tapering in detoxification for high-dose benzodiazepine abuse.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:4

    Topics: Adult; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Humans; Inactivation, Metabolic; Kinetics; Male; Mental Status Schedule; Middle Aged; Nordazepam; Prospective Studies; Substance-Related Disorders

1984
Subcellular distribution of pinazepam and its metabolite N-desmethyldiazepam in rat liver.
    General pharmacology, 1984, Volume: 15, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cell Nucleus; Cytosol; Diazepam; Liver; Male; Microsomes, Liver; Nordazepam; Rats; Rats, Inbred Strains; Subcellular Fractions

1984
Development of tolerance to the anticonvulsant effect of diazepam in dogs.
    European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2

    Topics: Animals; Anticonvulsants; Diazepam; Dogs; Drug Tolerance; Electrocardiography; Electroencephalography; Female; Male; Nordazepam; Pentylenetetrazole; Seizures; Time Factors

1984
Elimination kinetics and symptomatology of diazepam withdrawal in abusers.
    Journal of toxicology. Clinical toxicology, 1984, Volume: 22, Issue:4

    Topics: Diazepam; Half-Life; Humans; Kinetics; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
The contribution of the active metabolites to the tolerance developing to diazepam in man: relationship to bioassayed serum benzodiazepine levels.
    Medical biology, 1984, Volume: 62, Issue:5

    Topics: Adult; Benzodiazepines; Biological Assay; Diazepam; Double-Blind Method; Drug Tolerance; Female; Humans; Male; Nordazepam; Oxazepam; Psychomotor Performance

1984
Diazepam and N-desmethyldiazepam redistribution after heparin.
    Clinical pharmacology and therapeutics, 1980, Volume: 27, Issue:4

    Topics: Adult; Biotransformation; Blood Proteins; Diazepam; Drug Interactions; Heparin; Humans; Male; Nordazepam; Protein Binding

1980
Diurnal variations in plasma diazepam concentrations associated with reciprocal changes in free fraction.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:3

    Topics: Adolescent; Adult; Circadian Rhythm; Diazepam; Female; Food; Humans; Injections, Intravenous; Male; Nordazepam; Time Factors

1980
Delayed clearance of diazepam due to cimetidine.
    The New England journal of medicine, 1980, May-01, Volume: 302, Issue:18

    Topics: Adult; Antipyrine; Cimetidine; Diazepam; Drug Interactions; Drug Synergism; Female; Guanidines; Half-Life; Humans; Kinetics; Male; Nordazepam

1980
Diazepam and N-desmethyldiazepam concentrations in saliva, plasma and CSF.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:4

    Topics: Adult; Diazepam; Female; Humans; Hydrogen-Ion Concentration; Male; Nordazepam; Protein Binding; Saliva; Time Factors

1980
Desmethyldiazepam kinetics in the elderly after oral prazepam.
    Clinical pharmacology and therapeutics, 1980, Volume: 28, Issue:2

    Topics: Adult; Age Factors; Aged; Blood Proteins; Diazepam; Female; Half-Life; Humans; Kinetics; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam; Prazepam; Protein Binding; Regression Analysis; Sex Factors; Smoking

1980
Comparative effects of two commercially available blood collection tubes on plasma concentrations of drugs.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1980, Jan-26, Volume: 57, Issue:4

    Topics: Acebutolol; Blood Specimen Collection; Carbamazepine; Diazepam; Digoxin; Ethosuximide; Humans; Nordazepam; Penbutolol; Pharmaceutical Preparations; Propranolol; Quinidine; Salicylates; Time Factors; Valproic Acid; Warfarin

1980
Structure activity relationships of selected benzodiazepines as anticonvulsants to local anesthetics.
    Pharmacology and therapeutics in dentistry, 1980, Volume: 5, Issue:1-2

    Topics: Anesthetics, Local; Animals; Anticonvulsants; Benzodiazepines; Diazepam; Lidocaine; Male; Mepivacaine; Mice; Nitrazepam; Nordazepam; Oxazepam; Prilocaine; Seizures; Structure-Activity Relationship; Temazepam

1980
Effect of diazepam and desmethyldiazepam in spasticity and rigidity. A quantitative study of reflexes and plasma concentrations.
    Acta neurologica Scandinavica, 1980, Volume: 61, Issue:6

    Topics: Adult; Diazepam; Female; Humans; Injections, Intravenous; Male; Middle Aged; Muscle Rigidity; Muscle Spasticity; Muscle Tonus; Nordazepam; Reflex

1980
Simultaneous assay of diazepam, chlordiazepoxide, N-desmethyldiazepam, N-desmethylchloridazepoxide, and demoxepam in serum by high performance, liquid chromatography.
    Clinical biochemistry, 1980, Volume: 13, Issue:3

    Topics: Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chromatography, High Pressure Liquid; Diazepam; Humans; Methods; Nordazepam

1980
Entry of diazepam and its major matabolite into cerebrospinal fluid.
    Psychopharmacology, 1980, Volume: 70, Issue:1

    Topics: Animals; Blood Proteins; Diazepam; Dogs; Nordazepam; Protein Binding

1980
High-performance liquid chromatographic and gas-liquid chromatographic determination of diazepam and nordiazepam in plasma.
    Journal of chromatography, 1980, Oct-10, Volume: 183, Issue:4

    Topics: Adult; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Humans; Male; Nordazepam; Status Epilepticus

1980
Evaluation of an enzyme immunoassay for determining diazepam and nordiazepam in serum and urine.
    Clinical chemistry, 1980, Volume: 26, Issue:13

    Topics: Chromatography, High Pressure Liquid; Depression; Diazepam; Evaluation Studies as Topic; Humans; Immunoenzyme Techniques; Nordazepam

1980
Pharmacological requirements of patients during alcohol withdrawal.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1981, Jan-24, Volume: 59, Issue:4

    Topics: Alcoholism; Diazepam; Ethanol; Humans; Nordazepam

1981
The effect of diazepam on rates of fertilization in the CF-1 mouse.
    American journal of obstetrics and gynecology, 1981, Jan-15, Volume: 139, Issue:2

    Topics: Animals; Chorionic Gonadotropin; Chromatin; Copulation; Diazepam; Female; Fertilization; Meiosis; Mice; Mice, Inbred Strains; Nordazepam; Ovum; Superovulation

1981
Influence of cimetidine on the pharmacokinetics of desmethyldiazepam and oxazepam.
    European journal of clinical pharmacology, 1980, Volume: 18, Issue:6

    Topics: Adult; Cimetidine; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; Guanidines; Humans; Kinetics; Liver; Male; Nordazepam; Oxazepam

1980
Plasma diazepam and desmethyldiazepam concentrations during long-term diazepam therapy.
    British journal of clinical pharmacology, 1981, Volume: 11, Issue:1

    Topics: Adult; Aged; Diazepam; Humans; Male; Middle Aged; Nordazepam; Time Factors

1981
Effects of desmethyldiazepam on diazepam kinetics: a study of effects of a metabolite on parent drug disposition.
    Clinical pharmacology and therapeutics, 1981, Volume: 29, Issue:6

    Topics: Adult; Diazepam; Female; Humans; Kinetics; Male; Nordazepam

1981
Benzodiazepine overdosage: plasma concentrations and clinical outcome.
    Psychopharmacology, 1981, Volume: 73, Issue:4

    Topics: Adolescent; Adult; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Female; Humans; Male; Middle Aged; Nordazepam

1981
[Plasma levels following high diazepam doses in intensive-care medicine (author's transl)].
    Anasthesie, Intensivtherapie, Notfallmedizin, 1981, Volume: 16, Issue:3

    Topics: Adult; Critical Care; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam

1981
Long-term use of diazepam.
    JAMA, 1981, Oct-02, Volume: 246, Issue:14

    Topics: Adult; Aged; Diazepam; Female; Humans; Kinetics; Male; Middle Aged; Muscle Cramp; Nordazepam; Pain; Substance-Related Disorders; Time Factors

1981
Effect of ethanol ingestion on outcome of drug overdose.
    Critical care medicine, 1982, Volume: 10, Issue:3

    Topics: Adolescent; Adult; Aged; Antidepressive Agents, Tricyclic; Barbiturates; Benzodiazepines; Coma; Diazepam; Drug Interactions; Ethanol; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Nordazepam; Phenothiazines; Poisoning; Salicylates; Suicide, Attempted

1982
Valproic acid and diazepam interaction in vivo.
    British journal of clinical pharmacology, 1982, Volume: 13, Issue:4

    Topics: Adult; Blood Proteins; Diazepam; Drug Interactions; Humans; Kinetics; Male; Nordazepam; Protein Binding; Valproic Acid

1982
Binding of diazepam and desmethyldiazepam to plasma protein: concentration-dependence and interactions.
    Psychopharmacology, 1981, Volume: 75, Issue:4

    Topics: Binding, Competitive; Blood Proteins; Dialysis; Diazepam; Humans; In Vitro Techniques; Nordazepam; Protein Binding

1981
Pharmacokinetics of diazepam in epileptic patients and normal volunteers following intravenous administration.
    British journal of clinical pharmacology, 1981, Volume: 12, Issue:6

    Topics: Adult; Diazepam; Epilepsy; Half-Life; Humans; Injections, Intravenous; Male; Nordazepam

1981
Clinical bioavailability evaluation of a controlled release formulation of diazepam.
    Journal of pharmacokinetics and biopharmaceutics, 1981, Volume: 9, Issue:6

    Topics: Adult; Biological Availability; Biopharmaceutics; Delayed-Action Preparations; Diazepam; Humans; Nordazepam; Time Factors

1981
Radioimmunoassay of benzodiazepines.
    Methods in enzymology, 1982, Volume: 84

    Topics: Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Flurazepam; Humans; Microchemistry; Nitrazepam; Nordazepam; Oxazepam; Radioimmunoassay

1982
Kinetics of high-dose i.v. diazepam.
    British journal of anaesthesia, 1982, Volume: 54, Issue:8

    Topics: Adult; Critical Care; Diazepam; Half-Life; Humans; Injections, Intravenous; Kinetics; Male; Middle Aged; Nordazepam

1982
Pinazepam: a precursor of N-desmethyldiazepam.
    European journal of clinical pharmacology, 1982, Volume: 22, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Diazepam; Half-Life; Humans; Kinetics; Male; Nordazepam

1982
Prolongation of drug half-life due to obesity: studies of desmethyldiazepam (clorazepate).
    Journal of pharmaceutical sciences, 1982, Volume: 71, Issue:8

    Topics: Adult; Aged; Body Weight; Clorazepate Dipotassium; Diazepam; Female; Half-Life; Humans; Male; Middle Aged; Nordazepam; Obesity

1982
Sensitivity of auditory lateralization and temporal order tests to benzodiazepines.
    Audiology : official organ of the International Society of Audiology, 1982, Volume: 21, Issue:5

    Topics: Adult; Anti-Anxiety Agents; Auditory Pathways; Benzodiazepines; Diazepam; Ear; Functional Laterality; Hearing Tests; Humans; Loudness Perception; Middle Aged; Nordazepam; Sound Localization; Time Factors

1982
Anticonvulsant potency of unmetabolized diazepam.
    Pharmacology, 1982, Volume: 25, Issue:3

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Male; Mice; Nordazepam; Oxazepam; Pentylenetetrazole; Time Factors

1982
Chronic diazepam treatment in psychiatric outpatients.
    The Journal of clinical psychiatry, 1982, Volume: 43, Issue:11

    Topics: Adult; Aged; Ambulatory Care; Anxiety Disorders; Chronic Disease; Diazepam; Humans; Male; Middle Aged; Nordazepam; Psychiatric Status Rating Scales

1982
Correlation of the bioavailability of diazepam from uncoated tablets in beagle dogs with its dissolution rate and bioavailability in humans.
    International journal of clinical pharmacology, therapy, and toxicology, 1982, Volume: 20, Issue:12

    Topics: Animals; Biological Availability; Body Weight; Diazepam; Dogs; Humans; Hydrogen-Ion Concentration; Nordazepam; Solubility; Species Specificity; Tablets

1982
[The distribution of drugs between plasma, brain and cerebrospinal fluid in the human].
    Sammlung zwangloser Abhandlungen aus dem Gebiete der Psychiatrie und Neurologie, 1982, Volume: 50

    Topics: Blood-Brain Barrier; Brain; Brain Neoplasms; Carbamazepine; Diazepam; Humans; Lithium; Nordazepam; Phenobarbital; Phenytoin; Primidone; Protein Binding; Psychotropic Drugs; Serum Albumin; Sulfamerazine

1982
Acid-base equilibria of 1,4-benzodiazepine 4-oxides by spectrophotometry.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:5

    Topics: Chemical Phenomena; Chemistry, Physical; Chlordiazepoxide; Diazepam; Hydrogen-Ion Concentration; Indicators and Reagents; Kinetics; Nordazepam; Spectrophotometry, Ultraviolet

1995
Development and preliminary application of high-performance liquid chromatographic assay of urinary metabolites of diazepam in humans.
    Journal of chromatography. B, Biomedical applications, 1995, Jun-09, Volume: 668, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Reproducibility of Results; Temazepam

1995
Flunitrazepam and nordiazepam slowly released from silastic capsules induce physical dependence in rat.
    Drug and alcohol dependence, 1995, Volume: 39, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antidotes; Biological Availability; Delayed-Action Preparations; Diazepam; Drug Implants; Female; Flumazenil; Flunitrazepam; Nordazepam; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

1995
Behavioral and metabolic consequences of neonatal exposure to diazepam in rat pups.
    Experimental neurology, 1995, Volume: 131, Issue:1

    Topics: Animals; Animals, Newborn; Behavior, Animal; Brain; Diazepam; Glucose; Locomotion; Nordazepam; Postural Balance; Posture; Rats

1995
Diazepam metabolism by human liver microsomes is mediated by both S-mephenytoin hydroxylase and CYP3A isoforms.
    British journal of clinical pharmacology, 1994, Volume: 38, Issue:2

    Topics: Aryl Hydrocarbon Hydroxylases; Benzoflavones; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP2E1; Cytochrome P-450 Enzyme System; Diazepam; Humans; In Vitro Techniques; Isoenzymes; Mephenytoin; Microsomes, Liver; Mixed Function Oxygenases; Nordazepam; Temazepam

1994
Relationship between plasma benzodiazepine receptor ligand concentrations and severity of hepatic encephalopathy.
    Hepatology (Baltimore, Md.), 1994, Volume: 19, Issue:1

    Topics: Adult; Benzodiazepines; Diazepam; Female; Gas Chromatography-Mass Spectrometry; Hepatic Encephalopathy; Humans; Ligands; Male; Nordazepam; Prognosis; Receptors, GABA-A

1994
Inhibitory effect of diltiazem on diazepam metabolism in the mouse hepatic microsomes.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:3

    Topics: Animals; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diazepam; Diltiazem; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Microsomes, Liver; Nordazepam; Oxidoreductases, N-Demethylating

1993
Determination of plasma diazepam and desmethyldiazepam by solid-phase extraction and reversed-phase high-performance liquid chromatography.
    Journal of pharmaceutical and biomedical analysis, 1993, Volume: 11, Issue:7

    Topics: Calibration; Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Reference Standards; Spectrophotometry, Ultraviolet

1993
Pharmacokinetics of nordiazepam in physical dependence and precipitated abstinence in dogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Administration, Oral; Animals; Blood Proteins; Diazepam; Dogs; Female; Flumazenil; Hydrolysis; Injections, Intravenous; Nordazepam; Oxazepam; Protein Binding; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Kinetics of sequential metabolism. II. Formation and metabolism of nordiazepam and oxazepam from diazepam in the perfused murine liver.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: Animals; Diazepam; Kinetics; Male; Mice; Microsomes, Liver; Nordazepam; Oxazepam; Perfusion

1993
Extraction of selected drugs from serum using microwave irradiation.
    Forensic science international, 1996, Jul-31, Volume: 81, Issue:1

    Topics: Analgesics; Blood Chemical Analysis; Chromatography, Gas; Dextropropoxyphene; Diazepam; Humans; Lidocaine; Methadone; Microwaves; Narcotics; Nordazepam; Retrospective Studies

1996
Assessment of diazepam loading dose therapy of delirium tremens.
    Alcohol and alcoholism (Oxford, Oxfordshire), 1996, Volume: 31, Issue:3

    Topics: Adult; Alcohol Withdrawal Delirium; Anti-Anxiety Agents; Diazepam; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Humans; Male; Middle Aged; Neurologic Examination; Nordazepam; Psychoses, Alcoholic; Treatment Outcome

1996
Flumazenil, diazepam, nordiazepam and oxazepam interactions on plasma protein binding.
    Pharmacological research, 1995, Volume: 32, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Blood Proteins; Diazepam; Dogs; Drug Interactions; Flumazenil; In Vitro Techniques; Nordazepam; Oxazepam; Protein Binding

1995
Lymphatic bioavailability of diazepam and desmethyldiazepam in the rat.
    Physiological research, 1996, Volume: 45, Issue:1

    Topics: Animals; Biological Availability; Chemical Phenomena; Chemistry, Physical; Chromatography, Gas; Diazepam; Duodenum; GABA Modulators; Infusions, Intravenous; Injections; Injections, Intravenous; Lipid Metabolism; Lymph; Lymphatic System; Nordazepam; Rats

1996
Evidence against oppositional and pharmacokinetic mechanisms of tolerance to diazepam's sedative effects.
    Brain research, 1996, Sep-23, Volume: 734, Issue:1-2

    Topics: Animals; Diazepam; Drug Tolerance; Hypnotics and Sedatives; Male; Motor Activity; Nordazepam; Osmolar Concentration; Rats; Rats, Inbred Strains; Time Factors

1996
Benzodiazepine misuse by drug addicts.
    Annals of clinical biochemistry, 1997, Volume: 34 ( Pt 1)

    Topics: Alcoholism; Benzodiazepines; Chromatography, High Pressure Liquid; Diazepam; Humans; Narcotics; Nitrazepam; Nordazepam; Substance-Related Disorders; Temazepam

1997
[Benzodiazepines in geriatrics--a case report on prolonged action].
    Anaesthesiologie und Reanimation, 1996, Volume: 21, Issue:5

    Topics: Aged; Anti-Anxiety Agents; Dementia; Diazepam; Diverticulitis, Colonic; Drug Therapy, Combination; Emergencies; Female; Humans; Intestinal Perforation; Metabolic Clearance Rate; Nordazepam; Postoperative Complications

1996
Abnormal ventricular repolarization mimicking myocardial infarction after heterocyclic antidepressant overdose.
    The American journal of cardiology, 1997, Jan-15, Volume: 79, Issue:2

    Topics: Adult; Amitriptyline; Anti-Anxiety Agents; Antidepressive Agents; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Benzodiazepines; Bundle-Branch Block; Diagnosis, Differential; Diazepam; Electrocardiography; Female; Heart Ventricles; Humans; Hypnotics and Sedatives; Long QT Syndrome; Maprotiline; Myocardial Infarction; Nordazepam; Perphenazine; Triazolam

1997
Age-related changes in the pharmacokinetic disposition of diazepam in foals.
    American journal of veterinary research, 1997, Volume: 58, Issue:8

    Topics: Adjuvants, Anesthesia; Aging; Animals; Diazepam; Female; Half-Life; Horses; Male; Metabolic Clearance Rate; Nordazepam

1997
A fatality due to moclobemide.
    Journal of forensic sciences, 1997, Volume: 42, Issue:5

    Topics: Antidepressive Agents; Benzamides; Diazepam; Fatal Outcome; Female; Flumazenil; Humans; Liver; Middle Aged; Moclobemide; Nordazepam; Trifluoperazine

1997
Application of microdialysis to study the in vitro metabolism of drugs in liver microsomes.
    Journal of pharmaceutical and biomedical analysis, 1997, Volume: 16, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anti-Arrhythmia Agents; Anti-Inflammatory Agents, Non-Steroidal; Chromatography, High Pressure Liquid; Diazepam; Ibuprofen; Kinetics; Microdialysis; Microsomes, Liver; Nordazepam; Rats; Salicylates; Salicylic Acid; Temazepam

1997
Benzodiazepine-like compounds in the plasma of patients with fulminant hepatic failure.
    Scandinavian journal of gastroenterology, 1998, Volume: 33, Issue:3

    Topics: Adult; Benzodiazepines; Chromatography, High Pressure Liquid; Diazepam; Female; Hepatic Encephalopathy; Humans; Liver Failure; Male; Mass Spectrometry; Middle Aged; Nordazepam; Radioligand Assay

1998
Comparison of single- and repeated-dose pharmacokinetics of diazepam.
    Epilepsia, 1998, Volume: 39, Issue:3

    Topics: Animals; Chromatography, High Pressure Liquid; Clinical Protocols; Diazepam; Dose-Response Relationship, Drug; Humans; Injections, Intraperitoneal; Male; Nordazepam; Rats; Rats, Sprague-Dawley; Status Epilepticus

1998
Role of cDNA-expressed human cytochromes P450 in the metabolism of diazepam.
    Biochemical pharmacology, 1998, Mar-15, Volume: 55, Issue:6

    Topics: Cytochrome P-450 Enzyme System; Diazepam; DNA, Complementary; Gene Expression Regulation, Enzymologic; Humans; Isoenzymes; Kinetics; Linear Models; Microsomes, Liver; Nordazepam; Temazepam

1998
The effect of chronic benzodiazepines exposure on body weight in rats.
    Pharmacological research, 1998, Volume: 37, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; GABA Modulators; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Sex Factors; Time Factors; Weight Gain

1998
Rapid and simple chromatographic method for the determination of diazepam and its major metabolites in human plasma and urine.
    Journal of chromatography. B, Biomedical sciences and applications, 1998, Apr-24, Volume: 708, Issue:1-2

    Topics: Calibration; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Temazepam

1998
Determination of benzodiazepines in human urine and plasma with solvent modified solid phase micro extraction and gas chromatography; rationalisation of method development using experimental design strategies.
    Journal of pharmaceutical and biomedical analysis, 1998, Volume: 18, Issue:4-5

    Topics: Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Flunitrazepam; Humans; Hydrogen-Ion Concentration; Models, Chemical; Nordazepam; Oxazepam; Research Design

1998
Sigmoidal kinetic model for two co-operative substrate-binding sites in a cytochrome P450 3A4 active site: an example of the metabolism of diazepam and its derivatives.
    The Biochemical journal, 1999, Jun-15, Volume: 340 ( Pt 3)

    Topics: Adult; Allosteric Regulation; Allosteric Site; Antibodies, Monoclonal; Catalysis; Cell Line; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Kinetics; Male; Microsomes, Liver; Middle Aged; Mixed Function Oxygenases; Models, Chemical; Nordazepam; Oxidation-Reduction; Temazepam

1999
Effect of the gene dosage of CgammaP2C19 on diazepam metabolism in Chinese subjects.
    Clinical pharmacology and therapeutics, 1999, Volume: 66, Issue:6

    Topics: Adult; Anti-Anxiety Agents; Area Under Curve; Aryl Hydrocarbon Hydroxylases; Asian People; China; Cytochrome P-450 CYP2C19; Cytochrome P-450 Enzyme System; Diazepam; Gene Dosage; Half-Life; Heterozygote; Homozygote; Humans; Male; Mixed Function Oxygenases; Nordazepam; Phenotype; Reference Values

1999
Fatal intoxication with melperone.
    Forensic science international, 2000, Sep-11, Volume: 113, Issue:1-3

    Topics: Adult; Anti-Anxiety Agents; Antimanic Agents; Antipsychotic Agents; Autopsy; Butyrophenones; Carbamazepine; Cause of Death; Diazepam; Drug Synergism; Fatal Outcome; Female; Homicide; Humans; Nordazepam; Substance Abuse Detection; Suicide

2000
Liquid-phase microextraction as a sample preparation technique prior to capillary gas chromatographic-determination of benzodiazepines in biological matrices.
    Journal of chromatography. B, Biomedical sciences and applications, 2000, Nov-10, Volume: 749, Issue:1

    Topics: Chromatography, Gas; Diazepam; Humans; Nordazepam; Reproducibility of Results; Sensitivity and Specificity

2000
Diazepam poisoning with one-month monitoring of diazepam and nordiazepam blood levels.
    Veterinary and human toxicology, 2001, Volume: 43, Issue:3

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Humans; Male; Middle Aged; Nordazepam; Poisoning; Suicide, Attempted; Treatment Outcome

2001
The simultaneous determination of diazepam and its three metabolites in dog plasma by high-performance liquid chromatography with mass spectroscopy detection.
    Journal of pharmaceutical and biomedical analysis, 2001, Volume: 26, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Mass Spectrometry; Nordazepam; Oxazepam; Reproducibility of Results; Temazepam

2001
A contemporaneous finding of fenproporex in a polydrug suicide.
    Journal of analytical toxicology, 2001, Volume: 25, Issue:7

    Topics: Adult; Amphetamines; Anti-Allergic Agents; Anticonvulsants; Appetite Depressants; Autopsy; Diazepam; Diphenhydramine; Drug Overdose; Female; Humans; Hydroxybutyrates; Nordazepam; Stomach; Suicide

2001
Evaluation of the novel antiepileptic drug, AWD 131-138, for benzodiazepine-like discriminative stimulus and reinforcing effects in squirrel monkeys.
    European journal of pharmacology, 2003, Apr-04, Volume: 465, Issue:3

    Topics: Animals; Anticonvulsants; Behavior, Animal; Chromatography, High Pressure Liquid; Cocaine; Diazepam; Discrimination Learning; GABA Modulators; GABA-A Receptor Agonists; Imidazoles; Injections, Intramuscular; Injections, Intravenous; Male; Midazolam; Nordazepam; Reinforcement, Psychology; Saimiri; Self Administration

2003
Effects of diazepam and its metabolites on nocturnal melatonin secretion in the rat pineal and Harderian glands. A comparative in vivo and in vitro study.
    Chronobiology international, 2003, Volume: 20, Issue:2

    Topics: Animals; Circadian Rhythm; Diazepam; Harderian Gland; In Vitro Techniques; Male; Melatonin; Nordazepam; Oxazepam; Perfusion; Pineal Gland; Rats; Rats, Wistar; Temazepam

2003
Coexistence and concentrations of ethanol and diazepam in postmortem blood specimens: risk for enhanced toxicity?
    Journal of forensic sciences, 2003, Volume: 48, Issue:6

    Topics: Central Nervous System Depressants; Chromatography, Gas; Diazepam; Drug Interactions; Ethanol; Forensic Medicine; GABA Modulators; Humans; Nordazepam; Risk Factors

2003
High concentrations of diazepam and nordiazepam in blood of impaired drivers: association with age, gender and spectrum of other drugs present.
    Forensic science international, 2004, Nov-10, Volume: 146, Issue:1

    Topics: Adolescent; Adult; Age Distribution; Amphetamine; Anti-Anxiety Agents; Automobile Driving; Central Nervous System Depressants; Central Nervous System Stimulants; Databases as Topic; Diazepam; Dronabinol; Ethanol; Female; Forensic Medicine; Gas Chromatography-Mass Spectrometry; Hallucinogens; Humans; Hypnotics and Sedatives; Male; Middle Aged; Morphine; Narcotics; Nordazepam; Sex Distribution; Substance Abuse Detection; Substance-Related Disorders; Sweden

2004
Development and validation of a liquid chromatographic/electrospray ionization mass spectrometric method for the quantitation of prazepam and its main metabolites in human plasma.
    Journal of mass spectrometry : JMS, 2005, Volume: 40, Issue:4

    Topics: Calibration; Chromatography, Liquid; Diazepam; Humans; Molecular Structure; Nordazepam; Oxazepam; Prazepam; Reference Standards; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization

2005
Fast in vivo microextraction: a new tool for clinical analysis.
    Clinical chemistry, 2006, Volume: 52, Issue:4

    Topics: Animals; Biocompatible Materials; Blood Chemical Analysis; Blood Specimen Collection; Calibration; Chemistry Techniques, Analytical; Chromatography, Liquid; Diazepam; Dogs; Mass Spectrometry; Nordazepam; Oxazepam; Polyethylene Glycols; Polymers; Pyrroles; Silicon Dioxide

2006
Medicolegal aspects of tetrazepam metabolism.
    International journal of legal medicine, 2007, Volume: 121, Issue:3

    Topics: Adult; Benzodiazepines; Diazepam; Female; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Half-Life; Humans; Male; Molecular Structure; Muscle Relaxants, Central; Nordazepam

2007
A sensitive and selective method for the detection of diazepam and its main metabolites in urine by gas chromatography-tandem mass spectrometry.
    Journal of chromatography. A, 2007, Feb-02, Volume: 1141, Issue:1

    Topics: Benzodiazepinones; Diazepam; Gas Chromatography-Mass Spectrometry; Nordazepam; Oxazepam; Reproducibility of Results; Tandem Mass Spectrometry; Time Factors

2007
Massive intoxication involving unusual high concentration of amitriptyline.
    Human & experimental toxicology, 2007, Volume: 26, Issue:8

    Topics: Adult; Amitriptyline; Antidepressive Agents, Tricyclic; Depression; Diazepam; Female; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Nordazepam; Nortriptyline; Spectrometry, Mass, Electrospray Ionization; Suicide

2007
Two compartment model of diazepam biotransformation in an organotypical culture of primary human hepatocytes.
    Toxicology and applied pharmacology, 2009, Jan-15, Volume: 234, Issue:2

    Topics: Anti-Inflammatory Agents; Antithyroid Agents; Biotransformation; Cell Separation; Chlorodiphenyl (54% Chlorine); Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Dexamethasone; Diazepam; Enzyme Induction; Hepatocytes; Humans; Hypnotics and Sedatives; Models, Biological; Models, Statistical; Nordazepam; Organ Culture Techniques; Oxazepam; Phenobarbital; Temazepam

2009
Alleged breaches of "standards of medical care" in a patient overdose death possibly related to chronic opioid analgesic therapy, application of the controlled substances model guidelines: case report.
    Pain medicine (Malden, Mass.), 2009, Volume: 10, Issue:3

    Topics: Adult; Analgesics, Opioid; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Diazepam; Doxepin; Drug Overdose; Female; Heroin Dependence; Humans; Hydrocodone; Malpractice; Methadone; Nordazepam; Pain; Pain Measurement; Practice Guidelines as Topic; Shoulder; Shoulder Injuries; Temazepam

2009
Simultaneous analysis of diazepam and its metabolites in rat plasma and brain tissue by HPLC-UV and SPE.
    Talanta, 2009, Nov-15, Volume: 80, Issue:1

    Topics: Animals; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Nordazepam; Oxazepam; Rats; Reproducibility of Results; Solid Phase Extraction; Spectrophotometry, Ultraviolet; Temazepam

2009
Effects of organic solvents on the time-dependent inhibition of CYP3A4 by diazepam.
    Xenobiotica; the fate of foreign compounds in biological systems, 2010, Volume: 40, Issue:1

    Topics: Acetonitriles; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Diazepam; Dimethyl Sulfoxide; GABA Modulators; Humans; Kinetics; Methanol; Microsomes, Liver; Nordazepam; Solvents; Temazepam

2010
Quantitation of benzodiazepines in blood and urine using gas chromatography-mass spectrometry (GC-MS).
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Lorazepam; Nordazepam; Oxazepam; Solid Phase Extraction; Triazolam

2010
Biotransformation of diazepam in a clinically relevant flat membrane bioreactor model using primary porcine hepatocytes.
    Fundamental & clinical pharmacology, 2011, Volume: 25, Issue:3

    Topics: Adult; Animals; Bioreactors; Biotransformation; Cells, Cultured; Culture Media; Culture Media, Serum-Free; Diazepam; Female; Hepatocytes; Humans; Inactivation, Metabolic; Liver, Artificial; Male; Nordazepam; Oxazepam; Swine; Temazepam; Young Adult

2011
Reduction of temazepam to diazepam and lorazepam to delorazepam during enzymatic hydrolysis.
    Analytical and bioanalytical chemistry, 2011, Volume: 400, Issue:1

    Topics: Benzodiazepines; Chromatography, Liquid; Diazepam; Glucuronidase; Humans; Hydrolysis; Lorazepam; Mass Spectrometry; Nordazepam; Reference Standards; Temazepam

2011
Pharmacokinetics of the cytochrome P-450 substrates phenytoin, theophylline, and diazepam in healthy Greyhound dogs.
    Journal of veterinary pharmacology and therapeutics, 2012, Volume: 35, Issue:3

    Topics: Animals; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Diazepam; Dogs; Female; Fluorescence Polarization Immunoassay; Gas Chromatography-Mass Spectrometry; Injections, Intravenous; Male; Nordazepam; Oxazepam; Phenytoin; Theophylline

2012
Concentrations of diazepam and nordiazepam in 1,000 blood samples from apprehended drivers--therapeutic use or abuse of anxiolytics?
    Journal of pharmacy practice, 2013, Volume: 26, Issue:3

    Topics: Automobile Driving; Chromatography, Gas; Databases, Factual; Diazepam; Forensic Toxicology; Humans; Limit of Detection; Nordazepam; Prescription Drug Misuse; Substance Abuse Detection

2013
The potential of forensic analysis on human bones found in riverine environment.
    Forensic science international, 2013, May-10, Volume: 228, Issue:1-3

    Topics: Adult; Animals; Bone and Bones; Diatoms; Diazepam; DNA Fingerprinting; Feeding Behavior; Forensic Anthropology; Forensic Toxicology; Humans; Hypnotics and Sedatives; Male; Muscidae; Nordazepam; Postmortem Changes; Pupa; Rivers; Young Adult

2013
Concentrations of drugs determined in blood samples collected from suspected drugged drivers in England and Wales.
    Journal of forensic and legal medicine, 2013, Volume: 20, Issue:4

    Topics: Adolescent; Adult; Amphetamine; Automobile Driving; Central Nervous System Depressants; Chromatography, Liquid; Cocaine; Diazepam; England; Ethanol; Female; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Ketamine; Male; Methadone; Methamphetamine; N-Methyl-3,4-methylenedioxyamphetamine; Narcotics; Nordazepam; Sodium Oxybate; Substance Abuse Detection; Substance-Related Disorders; Wales; Young Adult

2013
Diazepam and its metabolites in the mothers' and newborns' hair as a biomarker of prenatal exposure.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2013, Volume: 64, Issue:4

    Topics: Biomarkers; Chromatography, Liquid; Diazepam; Female; Hair; Humans; Infant, Newborn; Maternal-Fetal Exchange; Mothers; Nordazepam; Pregnancy; Pregnancy Trimesters; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry

2013
Direct determination of diazepam and its glucuronide metabolites in human whole blood by μElution solid-phase extraction and liquid chromatography-tandem mass spectrometry.
    Forensic science international, 2013, Dec-10, Volume: 233, Issue:1-3

    Topics: Chromatography, Liquid; Diazepam; Forensic Toxicology; Humans; Hypnotics and Sedatives; Limit of Detection; Nordazepam; Oxazepam; Reproducibility of Results; Solid Phase Extraction; Tandem Mass Spectrometry; Temazepam

2013
Urinary diazepam metabolite distribution in a chronic pain population.
    Journal of analytical toxicology, 2014, Volume: 38, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Chromatography, High Pressure Liquid; Chronic Pain; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Diazepam; Drug Interactions; Esomeprazole; Female; Fluoxetine; Humans; Male; Methadone; Nordazepam; Oxazepam; Retrospective Studies; Specimen Handling; Temazepam

2014
A mixed MDPV and benzodiazepine intoxication in a chronic drug abuser: determination of MDPV metabolites by LC-HRMS and discussion of the case.
    Forensic science international, 2014, Volume: 243

    Topics: Adult; Alprazolam; Benzodiazepines; Benzodioxoles; Chlordiazepoxide; Chromatography, Liquid; Diazepam; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nordazepam; Oxazepam; Psychotropic Drugs; Pyrrolidines; Substance-Related Disorders; Synthetic Cathinone; Temazepam

2014
Low doses of ethanol markedly potentiate the anti-seizure effect of diazepam in a mouse model of difficult-to-treat focal seizures.
    Epilepsy research, 2014, Volume: 108, Issue:10

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Disease Models, Animal; Drug Compounding; Drug Synergism; Electroencephalography; Epilepsy, Temporal Lobe; Ethanol; Female; Kainic Acid; Mice; Nordazepam; Oxazepam; Seizures; Solvents; Temazepam; Water

2014
A comparative study of primary secondary amino (PSA) and multi-walled carbon nanotubes (MWCNTs) as QuEChERS absorbents for the rapid determination of diazepam and its major metabolites in fish samples by high-performance liquid chromatography-electrospray
    Journal of the science of food and agriculture, 2016, Jan-30, Volume: 96, Issue:2

    Topics: Adsorption; Animals; Chromatography, High Pressure Liquid; Diazepam; Fishes; Food Contamination; Nanotubes, Carbon; Nordazepam; Oxazepam; Seafood; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Temazepam

2016
Preparation of a novel sorptive stir bar based on vinylpyrrolidone-ethylene glycol dimethacrylate monolithic polymer for the simultaneous extraction of diazepam and nordazepam from human plasma.
    Journal of separation science, 2016, Volume: 39, Issue:7

    Topics: Adsorption; Chromatography, High Pressure Liquid; Diazepam; Humans; Methacrylates; Nordazepam; Polymerization; Pyrrolidinones; Surface Properties

2016
Characterization of equine cytochrome P450: role of CYP3A in the metabolism of diazepam.
    Journal of veterinary pharmacology and therapeutics, 2016, Volume: 39, Issue:5

    Topics: Animals; Chlorocebus aethiops; COS Cells; Cytochrome P-450 CYP3A; Diazepam; Horses; Hypnotics and Sedatives; Male; Microsomes, Liver; Nordazepam; Oxazepam; Phylogeny; Protein Isoforms; Rats; Rats, Sprague-Dawley; Species Specificity; Temazepam

2016
Deposition of diazepam and its metabolites in hair following a single dose of diazepam.
    International journal of legal medicine, 2017, Volume: 131, Issue:1

    Topics: Adult; Asian People; Chromatography, Liquid; Diazepam; Female; Hair; Healthy Volunteers; Humans; Hypnotics and Sedatives; Male; Nordazepam; Oxazepam; Tandem Mass Spectrometry; Temazepam; Young Adult

2017
Pentobarbital in the context of possible suicides: Analysis of a Case.
    Forensic science international, 2017, Volume: 274

    Topics: Adult; Central Nervous System Depressants; Diazepam; Ethanol; Gastrointestinal Contents; Humans; Male; Nordazepam; Oxazepam; Pentobarbital; Suicide; Temazepam

2017
Site-, Technique-, and Time-Related Aspects of the Postmortem Redistribution of Diazepam, Methadone, Morphine, and their Metabolites: Interest of Popliteal Vein Blood Sampling.
    Journal of forensic sciences, 2017, Volume: 62, Issue:6

    Topics: Adult; Blood Specimen Collection; Chromatography, Liquid; Diazepam; Female; Femoral Vein; Forensic Toxicology; Humans; Male; Methadone; Middle Aged; Morphine; Morphine Derivatives; Nordazepam; Oxazepam; Popliteal Vein; Postmortem Changes; Subclavian Vein; Young Adult

2017
Occurrence of diazepam and its metabolites in wastewater and surface waters in Beijing.
    Environmental science and pollution research international, 2017, Volume: 24, Issue:18

    Topics: Beijing; Cities; Diazepam; Nordazepam; Wastewater; Water Pollutants, Chemical

2017
Entomotoxicology in burnt bodies: a case of maternal filicide-suicide by fire.
    International journal of legal medicine, 2017, Volume: 131, Issue:5

    Topics: Adult; Animals; Automobiles; Burns; Carbon Monoxide Poisoning; Carboxyhemoglobin; Child; Child, Preschool; Diazepam; Diptera; Feeding Behavior; Female; Fires; Gasoline; Homicide; Humans; Hypnotics and Sedatives; Kidney; Larva; Liver; Male; Nordazepam; Oxazepam; Postmortem Changes; Suicide

2017
Acidic transformation of nordiazepam can affect recovery estimate during trace analysis of diazepam and nordiazepam in environmental water samples by liquid chromatography-tandem mass spectrometry.
    Analytical and bioanalytical chemistry, 2019, Volume: 411, Issue:17

    Topics: Acids; Chromatography, Liquid; Diazepam; Hydrogen-Ion Concentration; Limit of Detection; Nordazepam; Solid Phase Extraction; Tandem Mass Spectrometry; Water Pollutants, Chemical

2019
Validation of an LC-MS/MS Method for the Quantification of 13 Designer Benzodiazepines in Blood.
    Journal of analytical toxicology, 2019, Oct-17, Volume: 43, Issue:9

    Topics: Benzodiazepines; Chromatography, Liquid; Diazepam; Humans; Nordazepam; Substance Abuse Detection; Tandem Mass Spectrometry

2019
Organ distribution of diclazepam, pyrazolam and 3-fluorophenmetrazine.
    Forensic science international, 2019, Volume: 303

    Topics: Adult; Benzodiazepines; Bile; Body Fluids; Brain Chemistry; Designer Drugs; Diazepam; Forensic Toxicology; Gastrointestinal Contents; Humans; Kidney; Liver; Lorazepam; Lung; Male; Nordazepam; Pericardial Fluid; Phenmetrazine; Postmortem Changes; Psoas Muscles; Tandem Mass Spectrometry

2019
An Experimental Pharmacokinetics Study of Diazepam and Its Metabolites in Oral Fluid of Chinese Population.
    Journal of analytical toxicology, 2020, May-18, Volume: 44, Issue:4

    Topics: Adult; Chromatography, High Pressure Liquid; Diazepam; Healthy Volunteers; Humans; Nordazepam; Saliva; Solid Phase Extraction

2020
Postmortem Analysis of Benzodiazepines in Human Bone by Gas Chromatography-Mass Spectrometry.
    Journal of analytical toxicology, 2021, Jan-21, Volume: 44, Issue:9

    Topics: Alprazolam; Autopsy; Benzodiazepines; Chromatography, Liquid; Clonazepam; Diazepam; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Liquid-Liquid Extraction; Lorazepam; Nordazepam; Oxazepam; Tandem Mass Spectrometry

2021
A case report on fatal intoxication by tapentadol: Study of distribution and metabolism.
    Forensic science international, 2021, Volume: 324

    Topics: Adult; Analgesics, Opioid; Benzodiazepines; Bile; Chromatography, Liquid; Diazepam; Dibenzothiazepines; Gas Chromatography-Mass Spectrometry; Gastrointestinal Contents; Hair; Humans; Male; Nordazepam; Prisoners; Tapentadol; Tranquilizing Agents; Valproic Acid

2021
Kinetic disposition of diazepam and its metabolites after intravenous administration of diazepam in the horse: Relevance for doping control.
    Journal of veterinary pharmacology and therapeutics, 2021, Volume: 44, Issue:5

    Topics: Administration, Intravenous; Animals; Chromatography, Liquid; Diazepam; Doping in Sports; Horses; Nordazepam

2021
TSDC and DSC Investigation on the Molecular Mobility in the Amorphous Solid State and in the Glass Transformation Region of Two Benzodiazepine Derivatives: Diazepam and Nordazepam.
    Journal of pharmaceutical sciences, 2022, Volume: 111, Issue:8

    Topics: Anti-Anxiety Agents; Calorimetry, Differential Scanning; Diazepam; Glass; Hypnotics and Sedatives; Nordazepam

2022
Physiologically Based Pharmacokinetic and Pharmacodynamic Modeling of Diazepam: Unbound Interstitial Brain Concentrations Correspond to Clinical End Points.
    Journal of clinical pharmacology, 2022, Volume: 62, Issue:10

    Topics: Benzodiazepines; Brain; Diazepam; gamma-Aminobutyric Acid; Humans; Nordazepam

2022
Clinical Toxicological Follow-Up Analysis of a Suicide Attempt Using Chloroquine.
    Journal of analytical toxicology, 2023, Jan-24, Volume: 46, Issue:9

    Topics: Chloroquine; Diazepam; Follow-Up Studies; Humans; Nordazepam; Suicide, Attempted

2023
Occurrence of Z-drugs, benzodiazepines, and ketamine in wastewater in the United States and Mexico during the Covid-19 pandemic.
    The Science of the total environment, 2023, Jan-20, Volume: 857, Issue:Pt 2

    Topics: Alprazolam; Benzodiazepines; Clonazepam; COVID-19; Diazepam; Humans; Ketamine; Lorazepam; Mexico; Nordazepam; Pandemics; Tandem Mass Spectrometry; Temazepam; United States; Wastewater; Zolpidem

2023