Page last updated: 2024-09-04

norcisapride and metoclopramide

norcisapride has been researched along with metoclopramide in 1 studies

Compound Research Comparison

Studies
(norcisapride)
Trials
(norcisapride)
Recent Studies (post-2010)
(norcisapride)
Studies
(metoclopramide)
Trials
(metoclopramide)
Recent Studies (post-2010) (metoclopramide)
8305,0441,216623

Protein Interaction Comparison

ProteinTaxonomynorcisapride (IC50)metoclopramide (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.383
MyeloperoxidaseHomo sapiens (human)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)2.721
Cytochrome P450 2D6Homo sapiens (human)0.8
D(2) dopamine receptorHomo sapiens (human)0.127
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.8
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 2AHomo sapiens (human)3.675
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.383
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)7.8
D(3) dopamine receptorHomo sapiens (human)0.2
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.88
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.63
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.8
D(2) dopamine receptorRattus norvegicus (Norway rat)0.6237
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.88

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barberich, TJ; Hewitt, MC; Shao, L; Wang, F1

Other Studies

1 other study(ies) available for norcisapride and metoclopramide

ArticleYear
mu-Opioid/5-HT4 dual pharmacologically active agents-efforts towards an effective opioid analgesic with less GI and respiratory side effects (Part I).
    Bioorganic & medicinal chemistry letters, 2009, Oct-01, Volume: 19, Issue:19

    Topics: Analgesics, Opioid; Cisapride; Gastrointestinal Transit; Humans; Metoclopramide; Receptors, Opioid, mu; Receptors, Serotonin, 5-HT4; Respiratory System; Serotonin 5-HT4 Receptor Agonists; Stereoisomerism; Tramadol

2009