Page last updated: 2024-09-03

nnc 711 and sr 95531

nnc 711 has been researched along with sr 95531 in 9 studies

Compound Research Comparison

Studies
(nnc 711)
Trials
(nnc 711)
Recent Studies (post-2010)
(nnc 711)
Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010) (sr 95531)
1120216100209

Protein Interaction Comparison

ProteinTaxonomynnc 711 (IC50)sr 95531 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.24
GABA theta subunitRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.24

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's6 (66.67)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Delaney, AJ; Sah, P1
Overstreet, LS; Westbrook, GL1
Mody, I; Nusser, Z1
Kubin, L; Volgin, DV1
Cherubini, E; Marchionni, I; Omrani, A1
Dvorzhak, A; Grantyn, R; Kirischuk, S; Kirmse, K1
Gonzalez-Burgos, G; Lewis, DA; Povysheva, NV; Rotaru, DC; Zaitsev, AV1
Angulo, MC; Audinat, E; Butt, AM; Maldonado, PP; VĂ©lez-Fort, M1
Broberg, BV; Dalby, NO; Kjaerby, C; Kristiansen, U1

Other Studies

9 other study(ies) available for nnc 711 and sr 95531

ArticleYear
GABA receptors inhibited by benzodiazepines mediate fast inhibitory transmission in the central amygdala.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Nov-15, Volume: 19, Issue:22

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Bicuculline; Evoked Potentials; Flurazepam; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Neurons; Nipecotic Acids; Nitrazepam; Oximes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Strychnine; Synaptic Transmission

1999
Paradoxical reduction of synaptic inhibition by vigabatrin.
    Journal of neurophysiology, 2001, Volume: 86, Issue:2

    Topics: 4-Aminobutyrate Transaminase; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Presynaptic; Synaptic Transmission; Tetrodotoxin; Vigabatrin

2001
Selective modulation of tonic and phasic inhibitions in dentate gyrus granule cells.
    Journal of neurophysiology, 2002, Volume: 87, Issue:5

    Topics: Animals; Dentate Gyrus; GABA Agonists; GABA Antagonists; Neural Inhibition; Neurons; Nipecotic Acids; Organ Culture Techniques; Oximes; Pyridazines; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Zolpidem

2002
Regionally selective effects of GABA on hypothalamic GABAA receptor mRNA in vitro.
    Biochemical and biophysical research communications, 2007, Feb-16, Volume: 353, Issue:3

    Topics: Animals; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypothalamus; Isoenzymes; Male; Muscimol; Nipecotic Acids; Oximes; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Tetrodotoxin

2007
In the developing rat hippocampus a tonic GABAA-mediated conductance selectively enhances the glutamatergic drive of principal cells.
    The Journal of physiology, 2007, Jun-01, Volume: 581, Issue:Pt 2

    Topics: Animals; Animals, Newborn; Electric Stimulation; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamine; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Neuronal Plasticity; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Picrotoxin; Pyramidal Cells; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission; Time Factors

2007
GABA transporter 1 tunes GABAergic synaptic transmission at output neurons of the mouse neostriatum.
    The Journal of physiology, 2008, Dec-01, Volume: 586, Issue:23

    Topics: Action Potentials; Animals; Animals, Newborn; Baclofen; Bicuculline; Electric Impedance; Electric Stimulation; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Neostriatum; Neurons; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Pyridazines; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Tetrodotoxin

2008
GABA transporter GAT1 prevents spillover at proximal and distal GABA synapses onto primate prefrontal cortex neurons.
    Journal of neurophysiology, 2009, Volume: 101, Issue:2

    Topics: Animals; Electric Stimulation; Female; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Macaca fascicularis; Macaca mulatta; Male; Models, Neurological; Neurons; Nipecotic Acids; Organophosphorus Compounds; Oximes; Patch-Clamp Techniques; Prefrontal Cortex; Pyridazines; Synapses

2009
Postnatal switch from synaptic to extrasynaptic transmission between interneurons and NG2 cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, May-19, Volume: 30, Issue:20

    Topics: Age Factors; Animals; Animals, Newborn; Biophysics; Calcium; Cell Line, Transformed; Cerebral Cortex; Electric Conductivity; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Luminescent Proteins; Lysine; Mice; Mice, Transgenic; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oligodendroglia; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Pyridazines; Pyridines; Quinoxalines; Statistics, Nonparametric; Stem Cells; Synapses; Synaptic Transmission

2010
Impaired GABAergic inhibition in the prefrontal cortex of early postnatal phencyclidine (PCP)-treated rats.
    Cerebral cortex (New York, N.Y. : 1991), 2014, Volume: 24, Issue:9

    Topics: Animals; Animals, Newborn; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Interneurons; Miniature Postsynaptic Potentials; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phencyclidine; Prefrontal Cortex; Pyramidal Cells; Pyridazines; Rats, Inbred ACI; Receptors, GABA-A; Tissue Culture Techniques

2014