Page last updated: 2024-09-03

nnc 711 and nipecotic acid

nnc 711 has been researched along with nipecotic acid in 12 studies

Compound Research Comparison

Studies
(nnc 711)
Trials
(nnc 711)
Recent Studies (post-2010)
(nnc 711)
Studies
(nipecotic acid)
Trials
(nipecotic acid)
Recent Studies (post-2010) (nipecotic acid)
112021308043

Protein Interaction Comparison

ProteinTaxonomynnc 711 (IC50)nipecotic acid (IC50)
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.3367
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)8.1516

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (25.00)18.2507
2000's8 (66.67)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Chapman, AG; Meldrum, BS; Parvez, NS; Smith, SE1
Chen, DZ; Katsura, M; Kuriyama, K; Narihara, H; Ohkuma, S1
Nicklas, WJ; Zeevalk, GD1
Bernard, LP; Nicklas, WJ; Stokes, AH; Zeevalk, GD1
Mac, M; Nałecz, KA; Nałecz, MJ; Sacher, A; Wawrzeńczyk, A1
Himmelreich, NH; Linetska, MV; Storchak, LG; Tarasenko, AS1
Hablitz, JJ; Keros, S1
Kreil, A; Richter, A1
Marino, V; Nassery, K; Parker, DA1
De Mello, FG; De Mello, MC; De Melo Reis, RA; De Sampaio Schitine, C; Kubrusly, RC; Yamasaki, EN1
Allen, CN; Cravetchi, O; Moldavan, M1

Other Studies

12 other study(ies) available for nnc 711 and nipecotic acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
The gamma-aminobutyric acid uptake inhibitor, tiagabine, is anticonvulsant in two animal models of reflex epilepsy.
    European journal of pharmacology, 1995, Feb-06, Volume: 273, Issue:3

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Behavior, Animal; Carbamazepine; Epilepsy; Female; GABA Agents; Male; Motor Activity; Myoclonus; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Oximes; Papio; Photic Stimulation; Proline; Rats; Rats, Inbred Strains; Tiagabine

1995
Nitric oxide-evoked [3H] gamma-aminobutyric acid release is mediated by two distinct release mechanisms.
    Brain research. Molecular brain research, 1996, Volume: 36, Issue:1

    Topics: Animals; Biological Transport; Calcium; Cells, Cultured; Cerebral Cortex; gamma-Aminobutyric Acid; Mice; Neurons; Nipecotic Acids; Nitric Oxide; Nitroprusside; Oximes; Penicillamine; Proline; S-Nitroso-N-Acetylpenicillamine; Sodium; Tritium

1996
Activity at the GABA transporter contributes to acute cellular swelling produced by metabolic impairment in retina.
    Vision research, 1997, Volume: 37, Issue:24

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Carrier Proteins; Chick Embryo; Culture Techniques; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glycolysis; Iodoacetates; Ischemia; Isoxazoles; Membrane Proteins; Membrane Transport Proteins; Muscimol; Nipecotic Acids; Organic Anion Transporters; Oximes; Proline; Retina

1997
Attenuation of malonate toxicity in primary mesencephalic cultures using the GABA transport blocker, NO-711.
    Journal of neuroscience research, 2001, Apr-01, Volume: 64, Issue:1

    Topics: Animals; Cells, Cultured; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Malonates; Mesencephalon; Muscimol; Neurons; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species

2001
Transport of L-carnitine in isolated cerebral cortex neurons.
    European journal of biochemistry, 2001, Volume: 268, Issue:7

    Topics: Animals; beta-Alanine; Betaine; Binding, Competitive; Biological Transport, Active; Carnitine; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Neurons; Nipecotic Acids; Oocytes; Organic Anion Transporters; Organic Cation Transport Proteins; Oximes; Rats; Rats, Wistar; Solute Carrier Family 22 Member 5; Taurine; Xenopus laevis

2001
Involvement of membrane GABA transporter in alpha-latrotoxin-stimulated [3H]GABA release.
    Neurochemistry international, 2004, Volume: 44, Issue:5

    Topics: Algorithms; Animals; Calcium; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Carrier Proteins; Cell Membrane; Enzyme Inhibitors; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ionophores; Macrolides; Male; Membrane Proteins; Membrane Transport Proteins; Nipecotic Acids; Organic Anion Transporters; Oximes; Rats; Rats, Wistar; Spider Venoms; Stimulation, Chemical; Synaptic Transmission; Synaptosomes

2004
Subtype-specific GABA transporter antagonists synergistically modulate phasic and tonic GABAA conductances in rat neocortex.
    Journal of neurophysiology, 2005, Volume: 94, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Animals, Newborn; Anisoles; Bicuculline; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Synergism; Electric Stimulation; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Membrane Transport Modulators; Membrane Transport Proteins; Models, Neurological; Muscimol; Neocortex; Neural Inhibition; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors

2005
Antidystonic efficacy of gamma-aminobutyric acid uptake inhibitors in the dtsz mutant.
    European journal of pharmacology, 2005, Oct-03, Volume: 521, Issue:1-3

    Topics: Animals; Cricetinae; Disease Progression; Dose-Response Relationship, Drug; Dystonia; Female; GABA Antagonists; Injections, Intraperitoneal; Male; Mutation; Nipecotic Acids; Oximes; Random Allocation; Severity of Illness Index; Tiagabine; Time Factors; Treatment Outcome

2005
Uptake and release of [(3)H]GABA in human dental pulp.
    Archives of oral biology, 2007, Volume: 52, Issue:7

    Topics: Adult; Autoreceptors; Baclofen; Dental Pulp; Electric Stimulation; Female; GABA Agents; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Male; Morpholines; Nipecotic Acids; Oximes; Radiopharmaceuticals; Receptors, GABA; Time Factors; Tritium

2007
GABA uptake by purified avian Müller glia cells in culture.
    Neurotoxicity research, 2007, Volume: 12, Issue:2

    Topics: Analysis of Variance; Animals; Biological Transport; Cells, Cultured; Chick Embryo; Chlorides; Coculture Techniques; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Neuroglia; Neurons; Nipecotic Acids; Oximes; Retina; Sodium; Temperature; Tritium

2007
GABA transporters regulate tonic and synaptic GABA
    Journal of neurophysiology, 2017, 12-01, Volume: 118, Issue:6

    Topics: Animals; Anisoles; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; Male; Neurons; Nipecotic Acids; Oximes; Period Circadian Proteins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Suprachiasmatic Nucleus; Synaptic Potentials

2017