Page last updated: 2024-09-03

nnc 711 and gamma-aminobutyric acid

nnc 711 has been researched along with gamma-aminobutyric acid in 71 studies

Compound Research Comparison

Studies
(nnc 711)
Trials
(nnc 711)
Recent Studies (post-2010)
(nnc 711)
Studies
(gamma-aminobutyric acid)
Trials
(gamma-aminobutyric acid)
Recent Studies (post-2010) (gamma-aminobutyric acid)
11202140,2151,4239,631

Protein Interaction Comparison

ProteinTaxonomynnc 711 (IC50)gamma-aminobutyric acid (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0292
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0332
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0323
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.152
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0333
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.2623
Sodium- and chloride-dependent taurine transporterHomo sapiens (human)354
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)2.51
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)6.349
Sodium- and chloride-dependent GABA transporter 2Mus musculus (house mouse)7.0795
Sodium- and chloride-dependent GABA transporter 3Mus musculus (house mouse)8.1283
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent betaine transporterHomo sapiens (human)6.4082
Sodium- and chloride-dependent GABA transporter 3Homo sapiens (human)3.9953
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0333
GABA theta subunitRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0292

Research

Studies (71)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's21 (29.58)18.2507
2000's35 (49.30)29.6817
2010's14 (19.72)24.3611
2020's1 (1.41)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Andersen, KE; Frederiksen, K; Knutsen, LJ; Nielsen, EB; Suzdak, PD; Sørensen, PO1
Marsden, CA; Martin, KF; Rowley, HL1
Carvalho, AP; Carvalho, CM; Duarte, CB; Ferreira, IL; Santos, PF1
Carvalho, AL; Carvalho, AP; Duarte, CB; Ferreira, IL1
Agostinho, P; Carvalho, AP; Duarte, CB; Oliveira, CR1
Agostinho, P; Carvalho, AP; Caseiro, P; Duarte, CB; Oliveira, CR1
Alfonso, M; Carvalho, AP; Duarte, CB; Duran, R; Ferreira, IL1
Carvalho, AP; Duarte, CB; Ferreira, IL; Oliveira, CR; Santos, PF1
Carvalho, AP; Carvalho, CM; Duarte, CB; Ferreira, IL1
Feuerstein, TJ; Hüring, H; Landwehrmeyer, GB; Lücking, CH; van Velthoven, V1
Chen, DZ; Katsura, M; Kuriyama, K; Narihara, H; Ohkuma, S1
Johnson, KM; Lonart, G; Wang, J1
Bowery, NG; Richards, DA1
Nicklas, WJ; Zeevalk, GD1
Gaspary, HL; Richerson, GB; Wang, W1
Hanania, T; Johnson, KM1
Blythin, DJ; Kerr, DI; Marino, V; Ong, J; Parker, DA1
Bowery, NG; Davies, CC; Sutch, RJ1
Davies, JA; Shakesby, A1
Delaney, AJ; Sah, P1
Banks, MI; Pearce, RA; White, JA1
Brodie, JD; Dewey, SL; Gerasimov, MR; Lennon, IC; Schiffer, WK; Taylor, SJ1
Jones, MV; Overstreet, LS; Westbrook, GL1
Bernard, LP; Nicklas, WJ; Stokes, AH; Zeevalk, GD1
Mac, M; Nałecz, KA; Nałecz, MJ; Sacher, A; Wawrzeńczyk, A1
Overstreet, LS; Westbrook, GL1
Johnson, SW; Shen, KZ1
Ichinose, T; Lukasiewicz, PD1
Manzino, L; Sonsalla, PK; Zeevalk, GD1
Yang, CY1
Peng, W; Simantov, R1
Duan, SH; Fei, J; Guo, LH; Hu, JH; Jiang, J; Ma, YH; Mei, ZT; Yang, N; Zhou, XG1
Fei, J; Guo, LH; Hu, JH; Jiang, J; Ma, YH; Mei, ZT; Yang, N; Zhang, XY; Zhou, XG1
Houser, CR; Mody, I; Peng, Z; Wei, W; Zhang, N1
Himmelreich, NH; Linetska, MV; Storchak, LG; Tarasenko, AS1
Fei, J; Guo, LH; Hu, JH; Ma, YH; Mei, ZT; Yang, N; Zhang, MH1
Flade, A; Hanitzsch, R; Küppers, L1
Höfner, G; Wanner, KT1
Huttu, K; Kaila, K; Sipilä, S; Voipio, J1
Cherubini, E; Marchionni, I; Petrini, EM; Sieghart, W; Zacchi, P1
Ananthalakshmi, KV; Edafiogho, IO; Kombian, SB1
Hablitz, JJ; Keros, S1
Cherubini, E; Conti, F; Fattorini, G; Safiulina, VF1
Glykys, J; Mody, I1
de Groat, WC; Fink, DJ; Liu, J; Mata, M; Peng, XM; Tai, C1
Ben-Ari, Y; Chiron, C; Gozlan, H; Quilichini, PP1
Kubin, L; Volgin, DV1
Marino, V; Nassery, K; Parker, DA1
Cherubini, E; Marchionni, I; Omrani, A1
De Mello, FG; De Mello, MC; De Melo Reis, RA; De Sampaio Schitine, C; Kubrusly, RC; Yamasaki, EN1
Bowery, NG; Smith, CG; Whitehead, KJ1
Brawek, B; Feuerstein, TJ; Löffler, M; Weyerbrock, A1
Gonzalez-Burgos, G; Lewis, DA; Povysheva, NV; Rotaru, DC; Zaitsev, AV1
Fujiwara, A; Kamei, C; Takechi, K; Watanabe, Y1
Hardy-Yamada, M; Ishizeki, J; Kubo, K; Nishikawa, K; Saito, S; Yanagawa, Y1
Dvorzhak, A; Kirischuk, S; Kirmse, K; Myakhar, O; Unichenko, P1
Angulo, MC; Audinat, E; Butt, AM; Maldonado, PP; Vélez-Fort, M1
Chen, CC; Cheng, SJ; Lin, CC; Lu, HC; Min, MY; Wang, HY; Wu, Y; Yang, HW1
Feuerstein, TJ; Freiman, TM; Kammerer, M; Rassner, MP1
Acheson, SK; Fleming, RL; Moore, SD; Swartzwelder, HS; Wilson, WA1
Bagley, EE; Chefer, VI; Chieng, BC; Christie, MJ; Hacker, J; Mallet, C; McNally, GP; Perroud, J; Shippenberg, TS1
Kirischuk, S; Myakhar, O; Unichenko, P1
Calaza, KC; Guimarães-Souza, EM1
Dai, XY; Hao, YJ; Li, YX; Liu, HY; Sun, T; Wang, HY; Yu, JQ1
Broberg, BV; Dalby, NO; Kjaerby, C; Kristiansen, U1
Antkowiak, B; Hawellek, DJ; Hentschke, H; Razik, DS1
Baraban, SC; Looke-Stewart, E; Sebe, JY1
Borisova, T; Dudarenko, M; Himmelreich, N; Krupko, O; Pozdnyakova, N; Yatsenko, L1
Friauf, E; Stephan, J1
Gao, S; Guo, Y; Li, R; Liu, J; Lyu, S; Ma, B; Tang, G; Wang, Y; Yang, J; Zhang, L1

Reviews

2 review(s) available for nnc 711 and gamma-aminobutyric acid

ArticleYear
Glutamate receptor modulation of [3H]GABA release and intracellular calcium in chick retina cells.
    Annals of the New York Academy of Sciences, 1995, May-10, Volume: 757

    Topics: Animals; Calcium; Calcium Channels; Chick Embryo; gamma-Aminobutyric Acid; Glutamates; Ion Channel Gating; Membrane Potentials; Nicotinic Acids; Nipecotic Acids; Nitrendipine; omega-Conotoxin GVIA; Oximes; Peptides; Potassium; Receptors, Glutamate; Retina

1995
Reactive oxygen species on GABA release.
    Annals of the New York Academy of Sciences, 1994, Nov-17, Volume: 738

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Ascorbic Acid; Calcium; Calcium Channel Blockers; Cells, Cultured; Chickens; Dizocilpine Maleate; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Iron; Nicotinic Acids; Nipecotic Acids; Nitrendipine; omega-Conotoxin GVIA; Oximes; Peptides; Reactive Oxygen Species; Retina

1994

Other Studies

69 other study(ies) available for nnc 711 and gamma-aminobutyric acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization.
    European journal of pharmacology, 1992, Dec-02, Volume: 224, Issue:2-3

    Topics: Animals; Anticonvulsants; Astrocytes; Behavior, Animal; Brain; Carbolines; Cells, Cultured; Convulsants; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Neurons; Nicotinic Acids; Nipecotic Acids; Oximes; Pentylenetetrazole; Rats; Seizures; Synaptosomes; Tiagabine

1992
Decreased GABA release following tonic-clonic seizures is associated with an increase in extracellular glutamate in rat hippocampus in vivo.
    Neuroscience, 1995, Volume: 68, Issue:2

    Topics: Amino Acids; Animals; Anticonvulsants; Bicuculline; Calcium; Electroshock; Epilepsy, Tonic-Clonic; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Male; Microdialysis; Nickel; Nicotinic Acids; Nipecotic Acids; Oximes; Rats; Synaptic Transmission

1995
Release of [3H]GABA evoked by glutamate receptor agonists in cultured chick retina cells: effect of Ca2+.
    Brain research, 1994, Nov-21, Volume: 664, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium; Cells, Cultured; Chick Embryo; Dizocilpine Maleate; Excitatory Amino Acid Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kainic Acid; N-Methylaspartate; Nicotinic Acids; Nipecotic Acids; Oximes; Quisqualic Acid; Retina; Tritium

1994
Effect of oxidative stress on the release of [3H]GABA in cultured chick retina cells.
    Brain research, 1994, Aug-29, Volume: 655, Issue:1-2

    Topics: Animals; Ascorbic Acid; Aspartic Acid; Cells, Cultured; Chick Embryo; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Iron; Lipid Peroxidation; Nicotinic Acids; Nipecotic Acids; Oxidative Stress; Oximes; Potassium; Receptors, Glutamate; Retina

1994
Domoic acid induced release of [3H]GABA in cultured chick retina cells.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Cells, Cultured; Chick Embryo; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Neurotoxins; Nicotinic Acids; Nipecotic Acids; Oximes; Quinoxalines; Retina

1994
Glutamate increases the [Ca2+]i but stimulates Ca(2+)-independent release of [3H]GABA in cultured chick retina cells.
    Brain research, 1993, May-14, Volume: 611, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Chick Embryo; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Nicotinic Acids; Nipecotic Acids; Nitrendipine; omega-Conotoxin GVIA; Oximes; Peptides; Retina; Veratridine

1993
Relation of exocytotic release of gamma-aminobutyric acid to Ca2+ entry through Ca2+ channels or by reversal of the Na+/Ca2+ exchanger in synaptosomes.
    Pflugers Archiv : European journal of physiology, 1993, Volume: 423, Issue:3-4

    Topics: Animals; Calcium; Calcium Channels; Carrier Proteins; Cerebral Cortex; Egtazic Acid; Exocytosis; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Nicotinic Acids; Nipecotic Acids; Organic Anion Transporters; Oximes; Potassium Chloride; Rats; Rats, Sprague-Dawley; Sodium-Calcium Exchanger; Synaptosomes

1993
5-HT1D-like receptors inhibit the release of endogenously formed [3H]GABA in human, but not in rabbit, neocortex.
    Neuroscience letters, 1996, May-17, Volume: 209, Issue:3

    Topics: 3-Mercaptopropionic Acid; Adult; Animals; Cerebral Cortex; Electric Stimulation; Female; GABA Agents; GABA Antagonists; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Male; Middle Aged; Nicotinic Acids; Nipecotic Acids; Oximes; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Sumatriptan; Tetrodotoxin

1996
Nitric oxide-evoked [3H] gamma-aminobutyric acid release is mediated by two distinct release mechanisms.
    Brain research. Molecular brain research, 1996, Volume: 36, Issue:1

    Topics: Animals; Biological Transport; Calcium; Cells, Cultured; Cerebral Cortex; gamma-Aminobutyric Acid; Mice; Neurons; Nipecotic Acids; Nitric Oxide; Nitroprusside; Oximes; Penicillamine; Proline; S-Nitroso-N-Acetylpenicillamine; Sodium; Tritium

1996
Glutamate receptor activation induces carrier mediated release of endogenous GABA from rat striatal slices.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:1-2

    Topics: Animals; Calcium; Carrier Proteins; Electric Stimulation; Excitatory Amino Acid Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Neostriatum; Neurotransmitter Agents; Nipecotic Acids; Oximes; Potassium; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate

1996
Comparative effects of the GABA uptake inhibitors, tiagabine and NNC-711, on extracellular GABA levels in the rat ventrolateral thalamus.
    Neurochemical research, 1996, Volume: 21, Issue:2

    Topics: Analysis of Variance; Animals; Anticonvulsants; Basal Metabolism; Drug Evaluation, Preclinical; Epilepsy; gamma-Aminobutyric Acid; Male; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Rats; Rats, Wistar; Thalamus; Tiagabine

1996
Activity at the GABA transporter contributes to acute cellular swelling produced by metabolic impairment in retina.
    Vision research, 1997, Volume: 37, Issue:24

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Carrier Proteins; Chick Embryo; Culture Techniques; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glycolysis; Iodoacetates; Ischemia; Isoxazoles; Membrane Proteins; Membrane Transport Proteins; Muscimol; Nipecotic Acids; Organic Anion Transporters; Oximes; Proline; Retina

1997
Carrier-mediated GABA release activates GABA receptors on hippocampal neurons.
    Journal of neurophysiology, 1998, Volume: 80, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Carrier Proteins; Cells, Cultured; Fetus; GABA Agents; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Neurons; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Picrotoxin; Potassium; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sodium; Tetrodotoxin

1998
Regulation of neurotransmitter release by endogenous nitric oxide in striatal slices.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Acetylcholine; Animals; Carbon Radioisotopes; Corpus Striatum; Enzyme Inhibitors; Excitatory Amino Acid Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; N-Methylaspartate; Neurotransmitter Agents; Nipecotic Acids; Nitric Oxide; Nitroarginine; Oximes; Rats; Rats, Sprague-Dawley; Tritium

1998
Antagonism of GABA(B) receptors by morpholino-2-acetic acid derivatives Sch 54679 and Sch 51324 in rat brain.
    European journal of pharmacology, 1999, Mar-12, Volume: 369, Issue:1

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Morpholines; Neocortex; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Tritium

1999
GABA release and uptake measured in crude synaptosomes from Genetic Absence Epilepsy Rats from Strasbourg (GAERS).
    Neurochemistry international, 1999, Volume: 34, Issue:5

    Topics: Aminooxyacetic Acid; Animals; Autoradiography; beta-Alanine; Cerebral Cortex; Epilepsy; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Nipecotic Acids; Oximes; Rats; Rats, Mutant Strains; Synaptosomes; Thalamus; Tiagabine; Tritium

1999
Blockade of GABA uptake potentiates GABA-induced depolarizations in adult mouse cortical slices.
    Neuroscience letters, 1999, May-14, Volume: 266, Issue:3

    Topics: Animals; Bicuculline; Carrier Proteins; Cerebral Cortex; Drug Synergism; Female; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Nerve Tissue Proteins; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Oximes

1999
GABA receptors inhibited by benzodiazepines mediate fast inhibitory transmission in the central amygdala.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Nov-15, Volume: 19, Issue:22

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Bicuculline; Evoked Potentials; Flurazepam; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Neurons; Nipecotic Acids; Nitrazepam; Oximes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Strychnine; Synaptic Transmission

1999
Interactions between distinct GABA(A) circuits in hippocampus.
    Neuron, 2000, Volume: 25, Issue:2

    Topics: Animals; Computer Simulation; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Membrane Potentials; Models, Neurological; Neural Inhibition; Neural Pathways; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Pyramidal Cells; Rats; Receptors, GABA-A; Theta Rhythm

2000
gamma-aminobutyric acid mimetic drugs differentially inhibit the dopaminergic response to cocaine.
    European journal of pharmacology, 2000, Apr-28, Volume: 395, Issue:2

    Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Molecular Mimicry; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sodium Chloride

2000
Slow desensitization regulates the availability of synaptic GABA(A) receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Nov-01, Volume: 20, Issue:21

    Topics: Animals; Biological Transport; Carrier Proteins; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Ion Channel Gating; Membrane Proteins; Membrane Transport Proteins; Neural Inhibition; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

2000
Attenuation of malonate toxicity in primary mesencephalic cultures using the GABA transport blocker, NO-711.
    Journal of neuroscience research, 2001, Apr-01, Volume: 64, Issue:1

    Topics: Animals; Cells, Cultured; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Malonates; Mesencephalon; Muscimol; Neurons; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species

2001
Transport of L-carnitine in isolated cerebral cortex neurons.
    European journal of biochemistry, 2001, Volume: 268, Issue:7

    Topics: Animals; beta-Alanine; Betaine; Binding, Competitive; Biological Transport, Active; Carnitine; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Neurons; Nipecotic Acids; Oocytes; Organic Anion Transporters; Organic Cation Transport Proteins; Oximes; Rats; Rats, Wistar; Solute Carrier Family 22 Member 5; Taurine; Xenopus laevis

2001
Paradoxical reduction of synaptic inhibition by vigabatrin.
    Journal of neurophysiology, 2001, Volume: 86, Issue:2

    Topics: 4-Aminobutyrate Transaminase; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Presynaptic; Synaptic Transmission; Tetrodotoxin; Vigabatrin

2001
Potentiation of GABA(A) receptor agonists by GABA uptake inhibitors in the rat ventral midbrain.
    European journal of pharmacology, 2001, Sep-28, Volume: 428, Issue:1

    Topics: Animals; Carrier Proteins; Drug Synergism; Electrophysiology; GABA Agonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Mesencephalon; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sodium; Suprachiasmatic Nucleus

2001
GABA transporters regulate inhibition in the retina by limiting GABA(C) receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Apr-15, Volume: 22, Issue:8

    Topics: Animals; Carrier Proteins; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Kainic Acid; Membrane Proteins; Membrane Transport Proteins; Neural Inhibition; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Photic Stimulation; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Stimulation, Chemical; Synaptic Transmission; Urodela; Vision, Ocular

2002
Protection of malonate-induced GABA but not dopamine loss by GABA transporter blockade in rat striatum.
    Experimental neurology, 2002, Volume: 176, Issue:1

    Topics: Animals; Carrier Proteins; Catheterization; Corpus Striatum; Dopamine; Drug Administration Routes; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Malonates; Membrane Proteins; Membrane Transport Proteins; Neuroprotective Agents; Nipecotic Acids; Organic Anion Transporters; Oximes; Rats; Rats, Sprague-Dawley

2002
gamma-aminobutyric acid transporter-mediated current from bipolar cells in tiger salamander retinal slices.
    Vision research, 1998, Volume: 38, Issue:17

    Topics: Animals; Carrier Proteins; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ion Channels; Membrane Proteins; Membrane Transport Proteins; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Picrotoxin; Retina; Sodium; Urodela

1998
Altered gene expression in frontal cortex and midbrain of 3,4-methylenedioxymethamphetamine (MDMA) treated mice: differential regulation of GABA transporter subtypes.
    Journal of neuroscience research, 2003, Apr-15, Volume: 72, Issue:2

    Topics: Animals; Carrier Proteins; Cloning, Molecular; Frontal Lobe; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Male; Membrane Proteins; Membrane Transport Proteins; Mesencephalon; Mice; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Nerve Tissue Proteins; Nipecotic Acids; Organic Anion Transporters; Oximes; Protein Isoforms; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Tiagabine

2003
Hyperalgesic effects of gamma-aminobutyric acid transporter I in mice.
    Journal of neuroscience research, 2003, Aug-15, Volume: 73, Issue:4

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Brain; Carrier Proteins; Dose-Response Relationship, Drug; Drug Tolerance; Formaldehyde; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Hyperalgesia; Male; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Transgenic; Morphine; Nipecotic Acids; Organic Anion Transporters; Oximes; Pain Measurement; Reaction Time; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spinal Cord; Substance-Related Disorders; Synaptosomes; Time Factors

2003
Decrease of morphine-induced reward effects and withdrawal symptoms in mice overexpressing gamma-aminobutyric acid transporter I.
    Journal of neuroscience research, 2003, Nov-15, Volume: 74, Issue:4

    Topics: Adaptation, Physiological; Animals; Brain; Carrier Proteins; Conditioning, Psychological; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Transgenic; Morphine Dependence; Naloxone; Narcotic Antagonists; Nipecotic Acids; Organic Anion Transporters; Oximes; Receptors, Opioid, mu; Reinforcement, Psychology; Substance Withdrawal Syndrome

2003
Perisynaptic localization of delta subunit-containing GABA(A) receptors and their activation by GABA spillover in the mouse dentate gyrus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Nov-19, Volume: 23, Issue:33

    Topics: Animals; Carrier Proteins; Dendrites; Dentate Gyrus; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Immunohistochemistry; In Vitro Techniques; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Nipecotic Acids; Organic Anion Transporters; Oximes; Patch-Clamp Techniques; Protein Subunits; Receptors, GABA-A; Synapses; Temperature; Zinc

2003
Involvement of membrane GABA transporter in alpha-latrotoxin-stimulated [3H]GABA release.
    Neurochemistry international, 2004, Volume: 44, Issue:5

    Topics: Algorithms; Animals; Calcium; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Carrier Proteins; Cell Membrane; Enzyme Inhibitors; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ionophores; Macrolides; Male; Membrane Proteins; Membrane Transport Proteins; Nipecotic Acids; Organic Anion Transporters; Oximes; Rats; Rats, Wistar; Spider Venoms; Stimulation, Chemical; Synaptic Transmission; Synaptosomes

2004
Up-regulation of gamma-aminobutyric acid transporter I mediates ethanol sensitivity in mice.
    Neuroscience, 2004, Volume: 123, Issue:4

    Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Carrier Proteins; Central Nervous System Depressants; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Enzyme Inhibitors; Ethanol; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Kinetics; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Transgenic; Motor Activity; Nipecotic Acids; Organic Anion Transporters; Oximes; Reaction Time; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sleep; Survival; Synaptosomes; Time Factors; Tritium; Up-Regulation

2004
The effect of GABA and the GABA-uptake-blocker NO-711 on the b-wave of the ERG and the responses of horizontal cells to light.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 2004, Volume: 242, Issue:9

    Topics: Animals; Electroretinography; Enzyme Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Light; Neuroglia; Nipecotic Acids; Oximes; Photic Stimulation; Rabbits; Retina; Vigabatrin

2004
Evaluation of GABA uptake in subcellular fractions of bovine frontal cortex and brainstem.
    Neuroscience letters, 2004, Jun-24, Volume: 364, Issue:1

    Topics: Animals; Blotting, Western; Brain Stem; Carrier Proteins; Cattle; Frontal Lobe; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Inhibitory Concentration 50; Kidney; Membrane Proteins; Membrane Transport Proteins; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Sodium; Subcellular Fractions

2004
GABA uptake via GABA transporter-1 modulates GABAergic transmission in the immature hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jun-30, Volume: 24, Issue:26

    Topics: Animals; Animals, Newborn; Bicuculline; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Membrane Transport Proteins; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Synaptic Transmission; Tetrodotoxin

2004
Clustering of extrasynaptic GABA(A) receptors modulates tonic inhibition in cultured hippocampal neurons.
    The Journal of biological chemistry, 2004, Oct-29, Volume: 279, Issue:44

    Topics: Animals; Cells, Cultured; Flurazepam; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Nipecotic Acids; Nocodazole; Oximes; Protein Subunits; Rats; Receptors, GABA-A; Tetrodotoxin

2004
Anticonvulsant enaminones depress excitatory synaptic transmission in the rat brain by enhancing extracellular GABA levels.
    British journal of pharmacology, 2005, Volume: 145, Issue:7

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Brain; Cyclohexanes; Cyclohexanones; Cyclohexylamines; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; N-Methylaspartate; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Nucleus Accumbens; Oximes; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Synaptic Transmission

2005
Subtype-specific GABA transporter antagonists synergistically modulate phasic and tonic GABAA conductances in rat neocortex.
    Journal of neurophysiology, 2005, Volume: 94, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Animals, Newborn; Anisoles; Bicuculline; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Synergism; Electric Stimulation; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Membrane Transport Modulators; Membrane Transport Proteins; Models, Neurological; Muscimol; Neocortex; Neural Inhibition; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors

2005
GABAergic signaling at mossy fiber synapses in neonatal rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-11, Volume: 26, Issue:2

    Topics: Action Potentials; Aminobutyrates; Animals; Animals, Newborn; Bicuculline; Cation Transport Proteins; Dentate Gyrus; Electric Stimulation; Excitatory Amino Acid Agonists; Flurazepam; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Glutamic Acid; Interneurons; Mossy Fibers, Hippocampal; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Propanolamines; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Reaction Time; Receptors, AMPA; Receptors, GABA-A; Synaptic Transmission; Vesicular Glutamate Transport Protein 1

2006
Hippocampal network hyperactivity after selective reduction of tonic inhibition in GABA A receptor alpha5 subunit-deficient mice.
    Journal of neurophysiology, 2006, Volume: 95, Issue:5

    Topics: Analysis of Variance; Animals; Animals, Newborn; Bicuculline; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscimol; Nerve Net; Neural Inhibition; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Pyramidal Cells; Receptors, GABA-A

2006
Release of GABA from sensory neurons transduced with a GAD67-expressing vector occurs by non-vesicular mechanisms.
    Brain research, 2006, Feb-16, Volume: 1073-1074

    Topics: Analysis of Variance; Animals; Cells, Cultured; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Glutamate Decarboxylase; Glutamic Acid; Glutamine; Isoenzymes; Neurons, Afferent; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Simplexvirus; Spinal Nerves; Transfection; Tubulin

2006
Stiripentol, a putative antiepileptic drug, enhances the duration of opening of GABA-A receptor channels.
    Epilepsia, 2006, Volume: 47, Issue:4

    Topics: Animals; Animals, Newborn; Anticonvulsants; Chloride Channels; Dioxolanes; Disease Models, Animal; Drug Interactions; Epilepsy; Excitatory Postsynaptic Potentials; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Neural Inhibition; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Pentobarbital; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission

2006
Regionally selective effects of GABA on hypothalamic GABAA receptor mRNA in vitro.
    Biochemical and biophysical research communications, 2007, Feb-16, Volume: 353, Issue:3

    Topics: Animals; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypothalamus; Isoenzymes; Male; Muscimol; Nipecotic Acids; Oximes; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Tetrodotoxin

2007
Uptake and release of [(3)H]GABA in human dental pulp.
    Archives of oral biology, 2007, Volume: 52, Issue:7

    Topics: Adult; Autoreceptors; Baclofen; Dental Pulp; Electric Stimulation; Female; GABA Agents; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Male; Morpholines; Nipecotic Acids; Oximes; Radiopharmaceuticals; Receptors, GABA; Time Factors; Tritium

2007
In the developing rat hippocampus a tonic GABAA-mediated conductance selectively enhances the glutamatergic drive of principal cells.
    The Journal of physiology, 2007, Jun-01, Volume: 581, Issue:Pt 2

    Topics: Animals; Animals, Newborn; Electric Stimulation; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamine; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Neuronal Plasticity; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Picrotoxin; Pyramidal Cells; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission; Time Factors

2007
GABA uptake by purified avian Müller glia cells in culture.
    Neurotoxicity research, 2007, Volume: 12, Issue:2

    Topics: Analysis of Variance; Animals; Biological Transport; Cells, Cultured; Chick Embryo; Chlorides; Coculture Techniques; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Neuroglia; Neurons; Nipecotic Acids; Oximes; Retina; Sodium; Temperature; Tritium

2007
GABA transporter type 1 (GAT-1) uptake inhibition reduces stimulated aspartate and glutamate release in the dorsal spinal cord in vivo via different GABAergic mechanisms.
    Neuropharmacology, 2007, Volume: 53, Issue:8

    Topics: Analysis of Variance; Animals; Aspartic Acid; Bicuculline; Dose-Response Relationship, Drug; Drug Combinations; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Morpholines; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Potassium Chloride; Rats; Rats, Wistar; Spinal Cord

2007
Effects of gabapentin and pregabalin on K+-evoked 3H-GABA and 3H-glutamate release from human neocortical synaptosomes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2009, Volume: 379, Issue:4

    Topics: Adolescent; Adult; Aged; Amines; Amino Acids, Cyclic; Anticonvulsants; Aspartic Acid; Calcium Channel Blockers; Child; Child, Preschool; Cyclohexanecarboxylic Acids; Exocytosis; Female; Gabapentin; gamma-Aminobutyric Acid; Glutamic Acid; Humans; Infant; Isoleucine; Male; Middle Aged; Neocortex; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Potassium; Pregabalin; Synaptosomes; Tacrolimus; Young Adult

2009
GABA transporter GAT1 prevents spillover at proximal and distal GABA synapses onto primate prefrontal cortex neurons.
    Journal of neurophysiology, 2009, Volume: 101, Issue:2

    Topics: Animals; Electric Stimulation; Female; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Macaca fascicularis; Macaca mulatta; Male; Models, Neurological; Neurons; Nipecotic Acids; Organophosphorus Compounds; Oximes; Patch-Clamp Techniques; Prefrontal Cortex; Pyridazines; Synapses

2009
Participation of GABA-ergic system in epileptogenic activity induced by teicoplanin in mice.
    Epilepsy research, 2009, Volume: 84, Issue:2-3

    Topics: Animals; Anti-Bacterial Agents; Bicuculline; Brain; Disease Models, Animal; Dizocilpine Maleate; Electric Stimulation; Electroencephalography; Epilepsy; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Nipecotic Acids; Oximes; Phosphinic Acids; Pyridines; Teicoplanin

2009
Thermal hyperalgesia via supraspinal mechanisms in mice lacking glutamate decarboxylase 65.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:1

    Topics: Animals; Behavior, Animal; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hot Temperature; Hyperalgesia; Inhibitory Postsynaptic Potentials; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Nipecotic Acids; Oximes; Pain Measurement; Patch-Clamp Techniques; Spinal Cord

2009
Estimation of ambient GABA levels in layer I of the mouse neonatal cortex in brain slices.
    The Journal of physiology, 2010, Jul-01, Volume: 588, Issue:Pt 13

    Topics: 3-Mercaptopropionic Acid; Animals; Anisoles; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neocortex; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Quinoxalines; Receptors, GABA-B

2010
Postnatal switch from synaptic to extrasynaptic transmission between interneurons and NG2 cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, May-19, Volume: 30, Issue:20

    Topics: Age Factors; Animals; Animals, Newborn; Biophysics; Calcium; Cell Line, Transformed; Cerebral Cortex; Electric Conductivity; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Luminescent Proteins; Lysine; Mice; Mice, Transgenic; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oligodendroglia; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Pyridazines; Pyridines; Quinoxalines; Statistics, Nonparametric; Stem Cells; Synapses; Synaptic Transmission

2010
GABAB receptor-mediated tonic inhibition of noradrenergic A7 neurons in the rat.
    Journal of neurophysiology, 2011, Volume: 105, Issue:6

    Topics: Analysis of Variance; Animals; Anisoles; Baclofen; Barium; Bee Venoms; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation; In Vitro Techniques; Lysine; Male; Morpholines; Neural Inhibition; Neurons; Nipecotic Acids; Norepinephrine; Organophosphorus Compounds; Oximes; Patch-Clamp Techniques; Pons; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; RNA, Messenger

2011
Effects of antiepileptic drugs on GABA release from rat and human neocortical synaptosomes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 384, Issue:1

    Topics: Adolescent; Adult; Aged; Amines; Animals; Anticonvulsants; Calcium; Carbamazepine; Child; Child, Preschool; Cyclohexanecarboxylic Acids; Female; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Infant; Lamotrigine; Levetiracetam; Male; Middle Aged; Neocortex; Nipecotic Acids; Oximes; Phenytoin; Piracetam; Potassium; Pregabalin; Rats; Rats, Wistar; Synaptosomes; Tetanus Toxin; Tetrodotoxin; Triazines; Valproic Acid; Veratridine; Young Adult

2011
GABA transport modulates the ethanol sensitivity of tonic inhibition in the rat dentate gyrus.
    Alcohol (Fayetteville, N.Y.), 2011, Volume: 45, Issue:6

    Topics: Aging; Animals; Dentate Gyrus; Ethanol; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Hippocampus; Neurons; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2011
Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors.
    Nature neuroscience, 2011, Oct-30, Volume: 14, Issue:12

    Topics: Analysis of Variance; Animals; Disease Models, Animal; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Microdialysis; Morphine; Naloxone; Narcotic Antagonists; Nipecotic Acids; Oximes; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Time Factors

2011
Intracellular Na+ concentration influences short-term plasticity of glutamate transporter-mediated currents in neocortical astrocytes.
    Glia, 2012, Volume: 60, Issue:4

    Topics: Action Potentials; Amino Acid Transport System X-AG; Animals; Animals, Newborn; Anisoles; Aspartic Acid; Astrocytes; Benzofurans; Biophysics; Cadmium Chloride; Calcium Channel Blockers; Electric Stimulation; Ethers, Cyclic; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Intracellular Fluid; Mice; Mice, Inbred C57BL; Neocortex; Neuronal Plasticity; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Rhodamines; Sodium; Sodium Channel Blockers; Synaptic Transmission; Tetrodotoxin

2012
Selective activation of group III metabotropic glutamate receptor subtypes produces different patterns of γ-aminobutyric acid immunoreactivity and glutamate release in the retina.
    Journal of neuroscience research, 2012, Volume: 90, Issue:12

    Topics: Amacrine Cells; Anilides; Animals; Benzhydryl Compounds; Calcium; Chickens; Cyclohexanecarboxylic Acids; Dizocilpine Maleate; GABA Plasma Membrane Transport Proteins; GABAergic Neurons; gamma-Aminobutyric Acid; Glutamic Acid; Nipecotic Acids; Oximes; Phosphoserine; Quinoxalines; Receptors, Metabotropic Glutamate

2012
Effects of oxymatrine on the neuropathic pain induced by chronic constriction injury in mice.
    CNS neuroscience & therapeutics, 2012, Volume: 18, Issue:12

    Topics: Alkaloids; Animals; Chronic Disease; Constriction; Disease Models, Animal; Dose-Response Relationship, Drug; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Male; Mice; Mice, Inbred ICR; Muscimol; Neuralgia; Neuroprotective Agents; Nipecotic Acids; Oximes; Pain Measurement; Pain Threshold; Quinolizines; Receptors, GABA-A; Spinal Cord

2012
Impaired GABAergic inhibition in the prefrontal cortex of early postnatal phencyclidine (PCP)-treated rats.
    Cerebral cortex (New York, N.Y. : 1991), 2014, Volume: 24, Issue:9

    Topics: Animals; Animals, Newborn; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Interneurons; Miniature Postsynaptic Potentials; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phencyclidine; Prefrontal Cortex; Pyramidal Cells; Pyridazines; Rats, Inbred ACI; Receptors, GABA-A; Tissue Culture Techniques

2014
Impairment of GABA transporter GAT-1 terminates cortical recurrent network activity via enhanced phasic inhibition.
    Frontiers in neural circuits, 2013, Volume: 7

    Topics: Action Potentials; Animals; Anisoles; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Male; Neocortex; Nerve Net; Neural Inhibition; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Rats

2013
GABAB receptors in maintenance of neocortical circuit function.
    Experimental neurology, 2014, Volume: 261

    Topics: Animals; Animals, Newborn; Calbindin 2; DNA-Binding Proteins; Embryo, Mammalian; gamma-Aminobutyric Acid; Green Fluorescent Proteins; In Vitro Techniques; Mice; Mice, Inbred BALB C; Mice, Transgenic; Neocortex; Nerve Net; Neuropeptide Y; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Piperidines; Pyrimidines; Receptors, GABA-B; Stem Cell Transplantation; Synaptic Potentials; Transcription Factors

2014
Perinatal hypoxia: different effects of the inhibitors of GABA transporters GAT1 and GAT3 on the initial velocity of [3H]GABA uptake by cortical, hippocampal, and thalamic nerve terminals.
    Croatian medical journal, 2014, Jun-01, Volume: 55, Issue:3

    Topics: Animals; Animals, Newborn; beta-Alanine; Cerebral Cortex; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Hypoxia; Male; Nipecotic Acids; Oximes; Rats; Rats, Wistar; Synaptosomes; Thalamus

2014
Functional analysis of the inhibitory neurotransmitter transporters GlyT1, GAT-1, and GAT-3 in astrocytes of the lateral superior olive.
    Glia, 2014, Volume: 62, Issue:12

    Topics: Action Potentials; Animals; Animals, Newborn; Anisoles; Astrocytes; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glycine; Glycine Plasma Membrane Transport Proteins; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neural Inhibition; Nipecotic Acids; Olivary Nucleus; Oximes; Patch-Clamp Techniques; Sarcosine; Synaptic Transmission

2014
Blockade of GABA transporter-1 and GABA transporter-3 in the lateral habenula improves depressive-like behaviors in a rat model of Parkinson's disease.
    Neuropharmacology, 2020, 12-15, Volume: 181

    Topics: Animals; Anisoles; Behavior, Animal; Depression; Dopamine; Dose-Response Relationship, Drug; Electrophysiological Phenomena; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Habenula; Hydroxydopamines; Male; Nipecotic Acids; Oximes; Parkinson Disease, Secondary; Rats; Rats, Sprague-Dawley; Swimming

2020