nitrendipine and isradipine

nitrendipine has been researched along with isradipine in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-199023 (33.33)18.7374
1990's35 (50.72)18.2507
2000's6 (8.70)29.6817
2010's5 (7.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dietel, M; Höllt, V; Kouba, M; Vogt, G1
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Einzinger, U; Hoda, JC; Huber, IG; Koschak, A; Obermair, GJ; Sartori, SB; Sinnegger-Brauns, MJ; Striessnig, J; Wild, C1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Reimão, JQ; Scotti, MT; Tempone, AG1
Sun, H1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Blanck, TJ; Fiskum, G; Hoehner, PJ; Rosenthal, RE; Roy, R1
Babcock, DF; Corron, ME; Florman, HM; Kim, TD1
Mason, RP; Moisey, DM; Shajenko, L1
Bladen, C; Dunn, SM1
Chou, MY; Shibuya, T; Watanabe, Y1
Little, HJ; Littleton, JM; Whittington, MA1
Battaini, F; Bergamaschi, S; Govoni, S; Meucci, O; Parenti, M; Schettini, G; Trabucchi, M1
Lepor, H; Rosenthal, E; Shapiro, E1
de Pascual, R; Gandía, L; García, AG; López, MG; Michelena, P1
Fujimoto, M; Mihara, S1
Butterworth, AR; Dolin, SJ; Little, HJ; Patch, TL; Siarey, RJ; Whittington, MA1
Murphy, BJ; Tuana, BS1
Pinchuk, GV; Pinchuk, LN; Rudenko, AE; Tkachenko, YV1
Rampe, D; Schilling, WP; Zaher, MC1
Böhm, M; Erdmann, E; Schwinger, RH1
Bristow, MR; Minobe, W; Rasmussen, RP1
Barradas, J; Gerbeau, C1
Hosey, MM; McMahon, KK; Ptasienski, J1
Benavides, J; Bertrand, P; Burgevin, MC; Doble, A; Ferris, O; Gueremy, C; Le Fur, G; Menager, J; Uzan, A; Vaucher, N1
Carpenter, CL; Greenberg, DA; Messing, RO1
Hosey, MM; Maan, AC; Ptasienski, J1
Brown, AM; Brush, K; Hamilton, SL; Schwartz, A; Yatani, A1
Brown, AM; Hamilton, SL; Hawkes, MJ; Kunze, DL1
DeRoth, L; Godfraind, T; Wibo, M1
Brown, AM; Kunze, DL; Yatani, A1
Askanas, V; Desnuelle, C; Engel, WK1
Massieu, L; Tapia, R1
Dunn, SM2
Callens, F; Charlemagne, D; Mayoux, E; Swynghedauw, B1
Aonuma, S; Fujisue, T; Ichida, S; Masada, A; Matsuda, N; Oda, Y1
Dodd, PR; Gundlach, AL; Harper, CG; Johnston, GA; Kril, JJ1
Ehrhardt, JD; Quennedey, MC; Rouot, B; Schwartz, J; Welsch, M1
Ferry, DR; Glossmann, H; Goll, A; Linn, T1
Leysen, JE; Pauwels, PJ; Van Assouw, HP1
Schilling, WP1
Navarro, J1
Oswald, RE; Weiland, GA1
Lee, HR; Roeske, WR; Yamamura, HI1
Ferry, DR; Glossmann, H; Goll, A1
Artalejo, CR; Cillero, FJ; de Casa-Juana, MF; de Pascual, R; García, AG; González-Morales, MA; López, MG; Priego, J; Sunkel, C; Villarroya, M1
Cross, AJ; Green, AR; Little, HJ; Misra, A; Watson, WP1
Kamp, TJ; Marbán, E; Pérez-García, MT1
Corbett, AM; Kramer, JW1
Akimoto, T; Ichida, S; Kishino, H; Matsuda, N; Nakazaki, S; Wada, T1
Fetkovska, N; Jakubovska, Z; Oravcova, J; Tison, P; Ulicna, L2
Ganunis, TF; Helfaer, MA; Hoehner, PJ; Kirsch, JR; Murphy, MT; Traystman, RJ1
Baraldi, M; Brandoli, C; di Bella, M; Parenti, C; Tait, A; Truzzi, C; Veneri, C; Zanoli, P1
Buxton, BF; Casley, D; Dauer, R; Gallicchio, M; Johnston, CI; Liu, JJ; Wojta, J1
Blanck, TJ; Fiskum, G; Fox, LG; Hoehner, PJ; Hurt, KJ; Rosenthal, RE; Werling, LL1
Burger, KJ; Lohmann, FW; Welzel, D1
Latifpour, J; Weiss, RM; Yoshida, M1
Fetkovska, N; Jakubovska, Z; Oravcova, J; Tison, P; Trnovec, T; Ulicna, L1
Ader, JL; Durand, D; Lloveras, JJ; Rostaing, L; Suc, JM; Tack, I; Tran-Van, T1
Gilar, M; Tesarová, E; Uhrová, M1
Brauns, T; Glossmann, H; Haugland, RP; Kimball, SD; Prinz, H; Striessnig, J1
Babcock, DF; Hille, B; Wennemuth, G; Westenbroek, RE; Xu, T1
Beydemir, S; Söyüt, H; Türkeş, C1

Trials

5 trial(s) available for nitrendipine and isradipine

ArticleYear
Effects of dihydropyridines and their combination with aspirin on blood pressure and circadian platelet activity in patients with essential hypertension.
    American journal of hypertension, 1994, Volume: 7, Issue:7 Pt 2

    Topics: Adult; Aspirin; Blood Platelets; Blood Pressure; Circadian Rhythm; Dihydropyridines; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Isradipine; Male; Middle Aged; Nitrendipine

1994
Treatment of hypertension with dihydropyridine calcium antagonists and aspirin.
    Blood pressure. Supplement, 1994, Volume: 1

    Topics: Adult; Aspirin; Blood Platelets; Blood Pressure; Calcium Channel Blockers; Circadian Rhythm; Dihydropyridines; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Isradipine; Male; Middle Aged; Nitrendipine

1994
[Circadian antihypertensive action and tolerability of a sustained-release form of isradipine in an intra-individual comparison with nitrendipine].
    Arzneimittel-Forschung, 1993, Volume: 43, Issue:5

    Topics: Adolescent; Adult; Aged; Blood Pressure; Calcium Channel Blockers; Circadian Rhythm; Delayed-Action Preparations; Double-Blind Method; Female; Humans; Hypertension; Isradipine; Male; Middle Aged; Nitrendipine

1993
Treatment of hypertension with calcium antagonists and aspirin. Effects on 24-h platelet activity.
    American journal of hypertension, 1993, Volume: 6, Issue:3 Pt 2

    Topics: Adult; Aspirin; Circadian Rhythm; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Isradipine; Male; Middle Aged; Nitrendipine; Platelet Aggregation; Treatment Outcome

1993
Renal functional reserve in calcium channel blocker-treated hypertensive recipients of kidney transplant.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 1995, Volume: 10 Suppl 6

    Topics: Adult; Amino Acids; Calcium Channel Blockers; Cyclosporine; Female; Glomerular Filtration Rate; Humans; Hypertension, Renal; Isradipine; Kidney Transplantation; Male; Middle Aged; Nifedipine; Nitrendipine; Renal Plasma Flow; Retrospective Studies

1995

Other Studies

64 other study(ies) available for nitrendipine and isradipine

ArticleYear
Stereoisomers of calcium antagonists which differ markedly in their potencies as calcium blockers are equally effective in modulating drug transport by P-glycoprotein.
    Biochemical pharmacology, 1992, Jun-23, Volume: 43, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Biological Transport; Calcium Channel Blockers; Cell Line; Dihydropyridines; Drug Resistance; Haplorhini; Immunoblotting; Membrane Glycoproteins; Mice; RNA, Messenger; Stereoisomerism; Verapamil; Vinblastine

1992
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Expression and 1,4-dihydropyridine-binding properties of brain L-type calcium channel isoforms.
    Molecular pharmacology, 2009, Volume: 75, Issue:2

    Topics: Amino Acid Motifs; Animals; Brain; Calcium Channels, L-Type; Dihydropyridines; Female; Gene Expression; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Protein Isoforms

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Anti-leishmanial and anti-trypanosomal activities of 1,4-dihydropyridines: In vitro evaluation and structure-activity relationship study.
    Bioorganic & medicinal chemistry, 2010, Nov-15, Volume: 18, Issue:22

    Topics: Animals; Antiprotozoal Agents; Cell Line; Cricetinae; Dihydropyridines; Erythrocytes; Leishmania; Macaca mulatta; Mice; Parasitic Sensitivity Tests; Quantitative Structure-Activity Relationship; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma cruzi

2010
Capture hydrolysis signals in the microsomal stability assay: molecular mechanisms of the alkyl ester drug and prodrug metabolism.
    Bioorganic & medicinal chemistry letters, 2012, Jan-15, Volume: 22, Issue:2

    Topics: Carboxylic Acids; Cytochrome P-450 Enzyme System; Esters; Humans; Hydrolysis; Microsomes; Models, Molecular; Molecular Structure; Prodrugs; Quantum Theory; Signal Transduction

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Alteration of voltage-dependent calcium channels in canine brain during global ischemia and reperfusion.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1992, Volume: 12, Issue:3

    Topics: Animals; Binding Sites; Brain Ischemia; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Dihydropyridines; Dogs; Female; Isradipine; Nitrendipine; Reperfusion; Synaptosomes

1992
Activation of voltage-dependent calcium channels of mammalian sperm is required for zona pellucida-induced acrosomal exocytosis.
    Developmental biology, 1992, Volume: 152, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acrosome; Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels; Cattle; Dihydropyridines; Exocytosis; Isradipine; Male; Mice; Nitrendipine; Sheep; Spermatozoa; Zona Pellucida

1992
Cholesterol alters the binding of Ca2+ channel blockers to the membrane lipid bilayer.
    Molecular pharmacology, 1992, Volume: 41, Issue:2

    Topics: Amlodipine; Animals; Calcium Channel Blockers; Cattle; Cell Membrane; Cholesterol; Dihydropyridines; Diltiazem; Electrons; Isradipine; Lipid Bilayers; Myocardium; Nifedipine; Nimodipine; Nitrendipine; Phosphatidylcholines; Rabbits; Verapamil

1992
Kinetics of binding of dihydropyridine calcium channel ligands to skeletal muscle membranes: evidence for low-affinity sites and for the involvement of G proteins.
    Biochemistry, 1991, Jun-11, Volume: 30, Issue:23

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Isradipine; Kinetics; Ligands; Membrane Proteins; Microsomes; Muscles; Nitrendipine; Oxadiazoles; Rabbits; Receptors, Nicotinic; Stereoisomerism; Thionucleotides

1991
Neuropsychopharmacological studies of a Ca2+ channel blocker on the modulation of brain Ca2+ mobilization of spontaneously hypertensive rats under mild stress.
    Neuroscience research, 1991, Volume: 12, Issue:2

    Topics: Acoustic Stimulation; Animals; Binding Sites; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Diazepam; Dihydropyridines; Hippocampus; Isoindoles; Isradipine; Kinetics; Male; Motor Activity; Nitrendipine; Organ Specificity; Piperazines; Pyrimidines; Rats; Rats, Inbred SHR; Reference Values; Stress, Psychological; Synaptosomes

1991
Effects of dihydropyridine calcium channel antagonists in ethanol withdrawal; doses required, stereospecificity and actions of Bay K 8644.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Ethanol; Isradipine; Male; Mice; Nimodipine; Nitrendipine; Oxadiazoles; Stereoisomerism; Substance Withdrawal Syndrome; Time Factors

1990
Modulation of dihydropyridine-sensitive calcium channels: a role for G proteins.
    European neurology, 1990, Volume: 30 Suppl 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Dihydropyridines; GTP-Binding Proteins; Guanosine Triphosphate; Isradipine; Neurons; Nitrendipine; Oxadiazoles; Rats; Tumor Cells, Cultured

1990
Characterization of 1,4, dihydropyridine calcium channel binding sites in the human prostate.
    The Journal of urology, 1990, Volume: 144, Issue:6

    Topics: Binding Sites; Calcium Channel Blockers; Calcium Channels; Humans; In Vitro Techniques; Isradipine; Male; Nitrendipine; Oxadiazoles; Prostate; Prostatic Hyperplasia; Receptors, Nicotinic

1990
Different sensitivities to dihydropyridines of catecholamine release from cat and ox adrenals.
    Neuroreport, 1990, Volume: 1, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Catecholamines; Cats; Cattle; Dihydropyridines; In Vitro Techniques; Isradipine; Male; Nitrendipine; Perfusion; Species Specificity

1990
Effect of S-312, a new calcium channel blocker, on the 1,4-dihydropyridine binding sites in porcine basilar blood vessels and rat aortic smooth muscle cells.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:3

    Topics: Animals; Aorta; Basilar Artery; Binding Sites; Calcium; Calcium Channel Blockers; Cells, Cultured; Dihydropyridines; Isradipine; Muscle, Smooth, Vascular; Nicardipine; Nitrendipine; Oxadiazoles; Rats; Swine

1991
Chronic dihydropyridine treatment can reverse the behavioural consequences of and prevent adaptations to, chronic ethanol treatment.
    British journal of pharmacology, 1991, Volume: 103, Issue:3

    Topics: Adaptation, Psychological; Administration, Inhalation; Animals; Behavior, Animal; Bicuculline; Brain; Calcium Channel Blockers; Dihydropyridines; Dose-Response Relationship, Drug; Ethanol; Isradipine; Male; Mice; Mice, Inbred C57BL; Nimodipine; Nitrendipine; Seizures; Substance Withdrawal Syndrome

1991
Calcium ions inhibit the allosteric interaction between the dihydropyridine and phenylalkylamine binding site on the voltage-gated calcium channel in heart sarcolemma but not in skeletal muscle transverse tubules.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:11

    Topics: Allosteric Regulation; Aniline Compounds; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Heart; In Vitro Techniques; Isradipine; Kinetics; Muscles; Myocardium; Nitrendipine; Oxadiazoles; Rabbits; Receptors, Nicotinic; Sarcolemma; Verapamil

1990
Calcium channel ligand binding to intact, concanavalin A and cyclic AMP-treated cells of the immune system.
    Immunology letters, 1990, Volume: 26, Issue:3

    Topics: Animals; Bucladesine; Calcium Channels; Concanavalin A; Isradipine; Leukocytes, Mononuclear; Lymphocyte Activation; Mice; Mice, Inbred CBA; Nitrendipine; Oxadiazoles; Spleen; Verapamil

1990
Effect of inorganic calcium channel blockers on dihydropyridine binding to cardiac sarcolemma.
    Molecular pharmacology, 1990, Volume: 37, Issue:1

    Topics: Animals; Cadmium; Calcimycin; Calcium; Calcium Channel Blockers; Dihydropyridines; Dogs; In Vitro Techniques; Isradipine; Lanthanum; Myocardium; Nitrendipine; Ouabain; Oxadiazoles; Quinuclidinyl Benzilate; Sarcolemma

1990
Different negative inotropic activity of Ca2(+)-antagonists in human myocardial tissue.
    Klinische Wochenschrift, 1990, Aug-17, Volume: 68, Issue:16

    Topics: Calcium Channel Blockers; Depression, Chemical; Diltiazem; Heart Atria; Heart Failure; Heart Transplantation; Humans; Isradipine; Myocardial Contraction; Nifedipine; Nitrendipine; Papillary Muscles; Pyridines; Verapamil

1990
Calcium antagonist binding sites in failing and nonfailing human ventricular myocardium.
    Biochemical pharmacology, 1990, Feb-15, Volume: 39, Issue:4

    Topics: Calcium Channel Blockers; Calcium Channels; Cardiomyopathy, Dilated; Cell Membrane; Humans; Iodocyanopindolol; Isradipine; Kinetics; Myocardium; Nitrendipine; Oxadiazoles; Pindolol; Receptors, Adrenergic, beta; Receptors, Nicotinic

1990
A radioreceptor assay for determination of nicardipine in human serum using 3H(+)PN 200-110 as radioligand.
    Journal of immunoassay, 1990, Volume: 11, Issue:3

    Topics: Animals; Binding, Competitive; Calcium Channels; Humans; In Vitro Techniques; Isradipine; Kinetics; Male; Nicardipine; Nitrendipine; Oxadiazoles; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Reproducibility of Results; Stereoisomerism; Tritium

1990
High and low affinity states of the dihydropyridine and phenylalkylamine receptors on the cardiac calcium channel and their interconversion by divalent cations.
    Biochemical and biophysical research communications, 1985, Jun-28, Volume: 129, Issue:3

    Topics: Animals; Calcium; Cations, Divalent; Chickens; Dihydropyridines; Heart; Ion Channels; Isradipine; Magnesium; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Pyridines; Receptors, Drug; Verapamil

1985
Dihydropyridine and peripheral type benzodiazepine binding sites: subcellular distribution and molecular size determination.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Fractionation; Dogs; Ion Channels; Isoquinolines; Isradipine; Male; Molecular Weight; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Nicotinic; Sarcolemma; Sarcoplasmic Reticulum; Verapamil

1985
Depolarization-dependent binding of the calcium channel antagonist, (+)-[3H]PN200-110, to intact cultured PC12 cells.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Cells, Cultured; Isradipine; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Onium Compounds; Organophosphorus Compounds; Oxadiazoles; Potassium; Pyridines; Tritium

1986
Influence of Mg++ on the effect of diltiazem to increase dihydropyridine binding to receptors on Ca++-channels in chick cardiac and skeletal muscle membranes.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Chickens; Diltiazem; Dose-Response Relationship, Drug; Ion Channels; Isradipine; Magnesium; Membranes; Muscles; Myocardium; Nitrendipine; Oxadiazoles; Receptors, Nicotinic

1986
A comparison between the binding and electrophysiological effects of dihydropyridines on cardiac membranes.
    Molecular pharmacology, 1987, Volume: 31, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Heart; Ion Channels; Isradipine; Kinetics; Membrane Potentials; Membranes; Myocardium; Nicotinic Acids; Nimodipine; Nitrendipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1987
Dihydropyridine binding and calcium channel function in clonal rat adrenal medullary tumor cells.
    Molecular pharmacology, 1987, Volume: 31, Issue:4

    Topics: Adrenal Gland Neoplasms; Animals; Calcium; Cell Membrane; Clone Cells; Electrophysiology; Ion Channels; Isradipine; Mathematics; Membrane Potentials; Nitrendipine; Oxadiazoles; Pheochromocytoma; Rats

1987
Pharmacologic relevance of dihydropyridine binding sites in membranes from rat aorta: kinetic and equilibrium studies.
    Circulation research, 1988, Volume: 62, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Binding, Competitive; Calcium; Calcium Channels; Ion Channels; Isradipine; Kinetics; Muscle, Smooth, Vascular; Nifedipine; Nisoldipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Stereoisomerism

1988
Effects of dihydropyridine calcium channel modulators on cardiac sodium channels.
    The American journal of physiology, 1988, Volume: 254, Issue:1 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Heart; Ion Channels; Isradipine; Myocardium; Nitrendipine; Oxadiazoles; Rats; Receptors, Nicotinic; Sodium; Stereoisomerism

1988
Dihydropyridine-sensitive Ca2+ channel in aneurally cultured human muscles. Relationship between high-affinity binding site and inhibition of calcium uptake.
    FEBS letters, 1988, Mar-28, Volume: 230, Issue:1-2

    Topics: Calcium; Calcium Channel Blockers; Calcium Radioisotopes; Cells, Cultured; Dihydropyridines; Electrophysiology; Humans; Ion Channels; Isradipine; Muscles; Nitrendipine; Oxadiazoles; Potassium

1988
Relationship of dihydropyridine binding sites with calcium-dependent neurotransmitter release in synaptosomes.
    Journal of neurochemistry, 1988, Volume: 51, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; gamma-Aminobutyric Acid; Ion Channels; Isradipine; Lanthanum; Male; Mice; Neurotransmitter Agents; Nifedipine; Nitrendipine; Oxadiazoles; Potassium; Receptors, Nicotinic; Ruthenium Red; Synaptosomes

1988
Multiple calcium channels in synaptosomes: voltage dependence of 1,4-dihydropyridine binding and effects on function.
    Biochemistry, 1988, Jul-12, Volume: 27, Issue:14

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dihydropyridines; Ion Channels; Isradipine; Kinetics; Male; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Spectrometry, Fluorescence; Synaptosomes; Verapamil

1988
Adaptational process of the cardiac Ca2+ channels to pressure overload: biochemical and physiological properties of the dihydropyridine receptors in normal and hypertrophied rat hearts.
    Journal of cardiovascular pharmacology, 1988, Volume: 12, Issue:4

    Topics: Adaptation, Physiological; Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Cardiomegaly; Heart; In Vitro Techniques; Isradipine; Kinetics; Male; Myocardium; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Sarcolemma

1988
Voltage-dependent calcium channels in skeletal muscle transverse tubules. Measurements of calcium efflux in membrane vesicles.
    The Journal of biological chemistry, 1989, Jul-05, Volume: 264, Issue:19

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzothiazoles; Calcium Channel Blockers; Calcium Channels; Calcium Radioisotopes; Carbocyanines; Cell Membrane; Dihydropyridines; Edetic Acid; Fluorescent Dyes; Isradipine; Lanthanum; Membrane Potentials; Muscles; Nitrendipine; Oxadiazoles; Potassium; Rabbits; Verapamil

1989
Characteristics of specific bindings of nitrendipine and PN200-110 to various crude membranes: induction of irreversible bindings by UV irradiation.
    Journal of biochemistry, 1989, Volume: 105, Issue:5

    Topics: Animals; Calcium Channel Blockers; Female; In Vitro Techniques; Isradipine; Male; Membranes; Muscle, Smooth; Muscles; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Spectrophotometry, Ultraviolet; Time Factors; Ultraviolet Rays

1989
Cortical dihydropyridine binding sites are unaltered in human alcoholic brain.
    Annals of neurology, 1989, Volume: 26, Issue:3

    Topics: Alcoholism; Cerebral Cortex; Dihydropyridines; Humans; Isradipine; Male; Middle Aged; Nitrendipine; Oxadiazoles

1989
Improved radioreceptor assay for the determination of plasma levels of dihydropyridine calcium channel blockers in humans.
    Therapeutic drug monitoring, 1989, Volume: 11, Issue:5

    Topics: Animals; Calcium Channel Blockers; Dihydropyridines; Isradipine; Male; Mass Spectrometry; Nicardipine; Nitrendipine; Pyridines; Radioligand Assay; Rats; Rats, Inbred Strains

1989
Molecular approach to the calcium channel.
    Advances in myocardiology, 1985, Volume: 5

    Topics: Animals; Benzothiazoles; Binding Sites; Brain; Calcium; Cattle; Chemical Phenomena; Chemistry; Diltiazem; Guinea Pigs; In Vitro Techniques; Ion Channels; Isradipine; Muscles; Myocardium; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Oxadiazoles; Thiazoles; Verapamil

1985
Depolarization of chick myotubes triggers the appearance of (+)-[3H]PN 200-110-binding sites.
    Molecular pharmacology, 1987, Volume: 32, Issue:6

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Chick Embryo; Isradipine; Muscles; Nitrendipine; Oxadiazoles; Receptors, Nicotinic

1987
Effect of divalent cation chelation on dihydropyridine binding in isolated cardiac sarcolemma vesicles.
    Biochimica et biophysica acta, 1988, Aug-18, Volume: 943, Issue:2

    Topics: Animals; Calcimycin; Calcium; Cations, Divalent; Dihydropyridines; Dogs; Edetic Acid; Hydrogen-Ion Concentration; Isradipine; Magnesium; Myocardium; Nitrendipine; Ouabain; Oxadiazoles; Phosphates; Sarcolemma

1988
Dihydropyridine [methyl-3H]PN 200-110 binding and myogenesis in intact muscle cells in vitro.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Aminoquinolines; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Chick Embryo; Isradipine; Kinetics; Muscles; Nifedipine; Nitrendipine; Oxadiazoles; Receptors, Nicotinic

1986
The mechanism of binding of dihydropyridine calcium channel blockers to rat brain membranes.
    The Journal of biological chemistry, 1985, Jul-15, Volume: 260, Issue:14

    Topics: Animals; Brain; Calcium Channel Blockers; Isomerism; Isradipine; Kinetics; Mathematics; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Time Factors

1985
High affinity specific [3H](+)PN 200-110 binding to dihydropyridine receptors associated with calcium channels in rat cerebral cortex and heart.
    Life sciences, 1984, Aug-13, Volume: 35, Issue:7

    Topics: Animals; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Ion Channels; Isradipine; Kinetics; Male; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic

1984
Differential labelling of putative skeletal muscle calcium channels by [3H]-nifedipine, [3H]-nitrendipine, [3H]-nimodipine and [3H]-PN 200 110.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 323, Issue:3

    Topics: Animals; Calcium Channel Blockers; Guinea Pigs; In Vitro Techniques; Ion Channels; Isradipine; Kinetics; Muscles; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Oxadiazoles

1983
PCA 50941, a novel Ca2+ channel agonist.
    European journal of pharmacology, 1993, Oct-12, Volume: 243, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Calcium Channel Agonists; Cardiovascular System; Dihydropyridines; Heart Atria; In Vitro Techniques; Isradipine; Mesenteric Arteries; Muscles; Nitrendipine; Rabbits; Rats; Rats, Sprague-Dawley; Swine; Thiazoles; Vasoconstriction

1993
The differential effects of felodipine and nitrendipine on cerebral dihydropyridine binding ex vivo and the ethanol withdrawal syndrome in mice.
    British journal of pharmacology, 1994, Volume: 112, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bicuculline; Binding Sites; Brain; Ethanol; Felodipine; Isradipine; Male; Mice; Nitrendipine; Substance Withdrawal Syndrome

1994
Functional properties of cardiac L-type calcium channels transiently expressed in HEK293 cells. Roles of alpha 1 and beta subunits.
    The Journal of general physiology, 1995, Volume: 105, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Barium; Calcium; Calcium Channels; Calcium Channels, L-Type; Cells, Cultured; Electrophysiology; Humans; Isradipine; Kinetics; Muscle Proteins; Myocardium; Nitrendipine; Time Factors; Transfection

1995
The voltage dependence of depolarization-induced calcium release in isolated skeletal muscle triads.
    The Journal of membrane biology, 1995, Volume: 144, Issue:3

    Topics: Adenosine Triphosphate; Animals; Benzothiazoles; Calcium; Carbocyanines; Fluorescent Dyes; In Vitro Techniques; Isradipine; Kinetics; Membrane Potentials; Muscle, Skeletal; Nitrendipine; Potassium; Rabbits; Ryanodine; Signal Transduction; Spectrometry, Fluorescence; Tritium

1995
Specific bindings of [3H](+)PN200-110 and [125I]omega-conotoxin to crude membranes from differentiated NG108-15 cells.
    Neurochemical research, 1993, Volume: 18, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Bucladesine; Cell Differentiation; Cell Membrane; Diltiazem; Glioma; Hybrid Cells; Isradipine; Mollusk Venoms; Neuroblastoma; Nitrendipine; omega-Conotoxin GVIA; Potassium Chloride; Rats; Tumor Cells, Cultured; Verapamil

1993
Dihydropyridine ligand binding decreases earlier in adolescent than in infant swine after global cerebral ischemia.
    Stroke, 1994, Volume: 25, Issue:10

    Topics: Aging; Animals; Blood Pressure; Brain Ischemia; Calcium Channels; Caudate Nucleus; Cerebral Cortex; Dihydropyridines; Hippocampus; Isradipine; Ligands; Membrane Proteins; Nitrendipine; Protein Binding; Swine; Synaptosomes; Time Factors

1994
Synthesis and antiinflammatory activity of 2,6-bis(1,1-dimethylethyl)phenol derivatives.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:10

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Binding Sites; Calcium; Carrageenan; Edema; Female; Isradipine; Male; Nitrendipine; Phenols; Rats; Rats, Sprague-Dawley; Synaptosomes

1993
Effects of calcium- and ETA-receptor antagonists on endothelin-induced vasoconstriction and levels of endothelin in the human internal mammary artery.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:1

    Topics: Calcium Channel Blockers; Cells, Cultured; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Endothelium, Vascular; Humans; In Vitro Techniques; Isradipine; Mammary Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nisoldipine; Nitrendipine; Peptides, Cyclic; Radioimmunoassay; Vasoconstriction

1994
Increased activation of L-type voltage-dependent calcium channels is associated with glycine enhancement of N-methyl-D-aspartate-stimulated dopamine release in global cerebral ischemia/reperfusion.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: Animals; Brain Ischemia; Calcium Channels; Dogs; Dopamine; Female; Glycine; Isradipine; N-Methylaspartate; Nitrendipine; Reperfusion Injury; Time Factors; Tritium

1994
Age-related changes in Ca2+ channel antagonist receptors in rabbit lower urinary tract.
    European journal of pharmacology, 1993, Mar-02, Volume: 232, Issue:2-3

    Topics: Aging; Animals; Animals, Newborn; Body Weight; Calcium Channel Agonists; Calcium Channels; Female; In Vitro Techniques; Isradipine; Male; Muscle, Smooth; Nitrendipine; Organ Size; Rabbits; Urethra; Urinary Bladder; Urinary Tract

1993
Enantiomer separation of dihydropyridine calcium antagonists with cyclodextrins as chiral selectors: structural correlation.
    Journal of chromatography. B, Biomedical applications, 1996, May-31, Volume: 681, Issue:1

    Topics: Amlodipine; Buffers; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Cyclodextrins; Dihydropyridines; Electrolytes; Electrophoresis, Capillary; Isradipine; Microspheres; Molecular Conformation; Nimodipine; Nisoldipine; Nitrendipine; Sodium Dodecyl Sulfate; Solvents; Stereoisomerism; Surface-Active Agents

1996
L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other.
    Biochemistry, 1997, Mar-25, Volume: 36, Issue:12

    Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Fluorescent Dyes; Isomerism; Isradipine; Kinetics; Nicotinic Acids; Nifedipine; Nitrendipine; Oxadiazoles; Rabbits

1997
CaV2.2 and CaV2.3 (N- and R-type) Ca2+ channels in depolarization-evoked entry of Ca2+ into mouse sperm.
    The Journal of biological chemistry, 2000, Jul-14, Volume: 275, Issue:28

    Topics: Animals; Cadmium; Calcium; Calcium Channel Blockers; Calcium Channels, N-Type; Calcium Channels, R-Type; Calcium Signaling; Ion Channel Gating; Isradipine; Kinetics; Male; Membrane Potentials; Mibefradil; Mice; Neurotoxins; Nickel; Nitrendipine; omega-Conotoxin GVIA; omega-Conotoxins; Scorpion Venoms; Spermatozoa

2000
Effect of calcium channel blockers on paraoxonase-1 (PON1) activity and oxidative stress.
    Pharmacological reports : PR, 2014, Volume: 66, Issue:1

    Topics: Amlodipine; Aryldialkylphosphatase; Calcium Channel Blockers; Humans; Isradipine; Nifedipine; Nitrendipine; Oxidative Stress

2014