nitrendipine and gallopamil

nitrendipine has been researched along with gallopamil in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-199021 (70.00)18.7374
1990's6 (20.00)18.2507
2000's0 (0.00)29.6817
2010's3 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dietel, M; Höllt, V; Kouba, M; Vogt, G1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Janis, RA; Triggle, DJ1
Campillo, NE; Guerra, A; Páez, JA1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Brouillette, WJ; Brown, GB; Zha, C1
Hadley, RW; Lederer, WJ1
Blanck, TJ; Drenger, B; Hoehner, P; Quigg, M; Runge, SR1
Fricke, U; Klaus, W; Kojda, G; Werner, G1
Garcia, ML; Han, GQ; Himmel, D; Kaczorowski, GJ; King, VF; Lam, YK; Pan, JX; Reuben, JP1
Fischbach, W; Mössner, J; Schwarz, J1
Prives, J; Rapuano, M; Ross, AF1
Best, PM; Fill, MD1
Isenberg, G; Klöckner, U; Trieschmann, U1
Garcia, ML; Kaczorowski, GJ; King, VF; Morgan, G; Scott, AL; Siegl, PK1
Nielsen, PJ; Nyborg, NC1
Bolger, GT; Ruzycky, A; Triggle, DJ; Yousif, FB1
Lim, SL; May, PB; Sutter, MC1
Bengtsson, B; Khan, AR; Weiber, R1
Freedman, SB; Miller, DM; Miller, RJ; Tindall, DR1
Freedman, SB; Miller, RJ1
Lee, KS; Tsien, RW1
Pelto, DJ; Rapoport, SI; Suarez-Isla, BA; Thompson, JM1
Gopalakrishnan, V; Triggle, CR1
Moscona-Amir, E; Sokolovsky, M1
Garthoff, B; Kazda, S; Knorr, A1
Ehlert, FJ; Itoga, E; Roeske, WR; Yamamura, HI1
Pert, CB; Quirion, R1
Alabaster, VA; Cheeseman, HE; Cooper, K; deSouza, RN; Keir, RF; Parry, MJ1
Caldirola, P; Timmerman, H; Zhang, MQ1

Reviews

1 review(s) available for nitrendipine and gallopamil

ArticleYear
New developments in Ca2+ channel antagonists.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:6

    Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Calmodulin; Electrophysiology; Heart; Humans; Ion Channels; Muscle Relaxation; Muscle, Smooth; Potassium; Sodium; Structure-Activity Relationship; Substrate Specificity

1983

Other Studies

29 other study(ies) available for nitrendipine and gallopamil

ArticleYear
Stereoisomers of calcium antagonists which differ markedly in their potencies as calcium blockers are equally effective in modulating drug transport by P-glycoprotein.
    Biochemical pharmacology, 1992, Jun-23, Volume: 43, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Biological Transport; Calcium Channel Blockers; Cell Line; Dihydropyridines; Drug Resistance; Haplorhini; Immunoblotting; Membrane Glycoproteins; Mice; RNA, Messenger; Stereoisomerism; Verapamil; Vinblastine

1992
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
Properties of L-type calcium channel gating current in isolated guinea pig ventricular myocytes.
    The Journal of general physiology, 1991, Volume: 98, Issue:2

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cell Separation; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Heart Ventricles; Ion Channel Gating; Myocardium; Nitrendipine

1991
Halothane inhibits binding of calcium channel blockers to cardiac sarcolemma.
    Advances in experimental medicine and biology, 1991, Volume: 301

    Topics: Animals; Binding Sites; Calcium Channel Blockers; Cattle; Depression, Chemical; Dogs; Gallopamil; Halothane; Heart; In Vitro Techniques; Myocardium; Nitrendipine; Sarcolemma

1991
Hydrophobic properties of novel dihydronaphthyridine calcium antagonists and biological activity in porcine isolated cardiac and vascular smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:3

    Topics: Animals; Calcium Channel Blockers; Chemical Phenomena; Chemistry, Physical; Coronary Vessels; Depression, Chemical; Female; Gallopamil; Heart; Kinetics; Muscle, Smooth, Vascular; Myocardial Contraction; Naphthyridines; Nisoldipine; Nitrendipine; Potassium; Swine; Vasodilator Agents

1991
Interaction of tetrandrine with slowly inactivating calcium channels. Characterization of calcium channel modulation by an alkaloid of Chinese medicinal herb origin.
    The Journal of biological chemistry, 1988, Feb-15, Volume: 263, Issue:5

    Topics: Alkaloids; Animals; Benzylisoquinolines; Calcium; Diltiazem; Drugs, Chinese Herbal; Gallopamil; Ion Channels; Kinetics; Myocardium; Nitrendipine; Plants, Medicinal; Sarcolemma; Swine

1988
Influence of "calcium2+-channel blockers" on exocrine pancreatic secretion by isolated rat acini.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1988, Volume: 188, Issue:4

    Topics: Amylases; Animals; Calcium; Calcium Channel Blockers; Carbachol; Gallopamil; In Vitro Techniques; Male; Nitrendipine; Pancreas; Pancreatic Juice; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Reference Values; Second Messenger Systems; Sincalide

1988
Opposing effects of calcium entry and phorbol esters on fusion of chick muscle cells.
    Developmental biology, 1989, Volume: 134, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium Channel Blockers; Cell Fusion; Cells, Cultured; Chick Embryo; Egtazic Acid; Gallopamil; Kinetics; Muscles; Myosin Subfragments; Myosin-Light-Chain Kinase; Myosins; Nitrendipine; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Tetradecanoylphorbol Acetate

1989
Block of contracture in skinned frog skeletal muscle fibers by calcium antagonists.
    The Journal of general physiology, 1989, Volume: 93, Issue:3

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Gallopamil; In Vitro Techniques; Muscle Contraction; Nitrendipine; Rana pipiens; Receptors, Nicotinic; Temperature

1989
Pharmacological modulation of calcium and potassium channels in isolated vascular smooth muscle cells.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:1A

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Nitrendipine; Potassium Channels; Swine

1989
Interactions of DPI 201-106, a novel cardiotonic agent, with cardiac calcium channels.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:6

    Topics: Animals; Calcium; Calcium Channels; Cardiotonic Agents; Cinnarizine; Diltiazem; Gallopamil; In Vitro Techniques; Membranes; Muscle Contraction; Myocardial Contraction; Myocardium; Nitrendipine; Papillary Muscles; Piperazines; Potassium; Swine

1988
Calcium antagonist-induced relaxation of the prostaglandin-F2 alpha response of isolated calf retinal resistance arteries.
    Experimental eye research, 1989, Volume: 48, Issue:3

    Topics: Animals; Cattle; Dinoprost; Gallopamil; Muscle Relaxation; Nitrendipine; Potassium; Retinal Artery

1989
Ca2+ channel antagonist actions in bladder smooth muscle: comparative pharmacologic and [3H]nitrendipine binding studies.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:5

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Diltiazem; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Microsomes; Muscarine; Muscle Contraction; Muscle, Smooth; Nicotinic Acids; Nifedipine; Nimodipine; Nisoldipine; Nitrendipine; Potassium; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Urinary Bladder

1985
Manganese can inhibit or potentiate contractile responses in mesenteric portal vein.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:6

    Topics: Animals; Barium; Calcium; Felodipine; Gallopamil; In Vitro Techniques; Male; Manganese; Mesenteric Veins; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Spectrophotometry, Atomic; Strontium; Tissue Distribution; Verapamil

1988
Low potency of Ca antagonists in smooth muscle from different levels of the respiratory tract.
    Acta physiologica Scandinavica, 1987, Volume: 131, Issue:2

    Topics: Animals; Bronchi; Calcium Channel Blockers; Felodipine; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Respiratory Muscles; Trachea; Verapamil

1987
Interactions of maitotoxin with voltage-sensitive calcium channels in cultured neuronal cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:14

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium; Calcium; Cell Line; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Ion Channels; Marine Toxins; Neurons; Nifedipine; Nitrendipine; Oxocins; Potassium

1984
Calcium channel activation: a different type of drug action.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:17

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium; Calcium; Calcium Channel Blockers; Cell Line; Diltiazem; Gallopamil; Glioma; Hybrid Cells; Ion Channels; Kinetics; Mice; Neuroblastoma; Nifedipine; Nitrendipine; Pyridines; Rats

1984
Mechanism of calcium channel blockade by verapamil, D600, diltiazem and nitrendipine in single dialysed heart cells.
    Nature, 1983, Apr-28, Volume: 302, Issue:5911

    Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Cats; Diltiazem; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Verapamil

1983
Blockers of calcium permeability inhibit neurite extension and formation of neuromuscular synapses in cell culture.
    Brain research, 1984, Volume: 316, Issue:2

    Topics: Age Factors; Animals; Cadmium; Calcium Channel Blockers; Chick Embryo; Cobalt; Gallopamil; Lanthanum; Manganese; Neuromuscular Junction; Nifedipine; Nitrendipine; Retina; Verapamil

1984
Specific high affinity binding of the calcium channel antagonist, [3H]nitrendipine, to rat liver microsomes.
    Canadian journal of physiology and pharmacology, 1984, Volume: 62, Issue:9

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Gallopamil; In Vitro Techniques; Lanthanum; Male; Microsomes, Liver; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Tritium

1984
Interactions between Ca2+-antagonist binding sites in rat adenohypophysis: dependence on estrous cycle.
    Life sciences, 1984, Sep-03, Volume: 35, Issue:10

    Topics: Animals; Binding Sites; Binding, Competitive; Calcium; Estrus; Female; Gallopamil; Kinetics; Male; Nifedipine; Nitrendipine; Pituitary Gland, Anterior; Pregnancy; Rats

1984
Nitrendipine and other calcium entry blockers (calcium antagonists) in hypertension.
    Federation proceedings, 1983, Volume: 42, Issue:2

    Topics: Animals; Blood Pressure; Calcium; Calcium Channel Blockers; Dogs; Gallopamil; Heart; Hypertension; Male; Nifedipine; Nitrendipine; Organ Size; Potassium; Pyridines; Rats; Rats, Inbred Strains; Vasoconstriction

1983
The interaction of [3H]nitrendipine with receptors for calcium antagonists in the cerebral cortex and heart of rats.
    Biochemical and biophysical research communications, 1982, Feb-11, Volume: 104, Issue:3

    Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Chloride; Cerebral Cortex; Diltiazem; Gallopamil; Kinetics; Lanthanum; Male; Myocardium; Nifedipine; Nitrendipine; Pyridines; Rats; Rats, Inbred Strains; Receptors, Drug; Verapamil

1982
Certain calcium antagonists are potent displacers of [3H]phencyclidine (PCP) binding in rat brain.
    European journal of pharmacology, 1982, Sep-10, Volume: 83, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain; Calcium Channel Blockers; Gallopamil; In Vitro Techniques; Nifedipine; Nitrendipine; Olfactory Bulb; Phencyclidine; Rats; Verapamil

1982
Pharmacological profile of UK-74,505, a novel and selective PAF antagonist with potent and prolonged oral activity.
    Journal of lipid mediators and cell signalling, 1994, Volume: 10, Issue:3

    Topics: Administration, Oral; Animals; Aorta; Azepines; Blood Platelets; Brain; Calcium Channels, L-Type; Capillary Permeability; Cattle; Dihydropyridines; Diltiazem; Gallopamil; Guinea Pigs; Hypotension; Imidazoles; In Vitro Techniques; Kinetics; Male; Membranes; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle Proteins; Nitrendipine; Platelet Activating Factor; Platelet Aggregation; Platelet Aggregation Inhibitors; Potassium Chloride; Rabbits; Rats; Rats, Sprague-Dawley; Skin; Triazoles; Tritium

1994
Calcium antagonism and structure-affinity relationships of terfenadine, a histamine H1 antagonist, and some related compounds.
    The Journal of pharmacy and pharmacology, 1993, Volume: 45, Issue:1

    Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Cerebral Cortex; Gallopamil; Histamine H1 Antagonists; In Vitro Techniques; Male; Nitrendipine; Rats; Rats, Wistar; Structure-Activity Relationship; Terfenadine

1993