nitrendipine and diazoxide

nitrendipine has been researched along with diazoxide in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.88)18.7374
1990's4 (23.53)18.2507
2000's7 (41.18)29.6817
2010's5 (29.41)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Topliss, JG; Yoshida, F1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Fujitani, S; Yada, T1
Kojima, I; Mine, T; Sekine, N; Shibata, H; Totsuka, Y; Yasuda, H1
Fujimoto, S; Ishida, H; Kajikawa, M; Kato, S; Mizuno, N; Mukai, E; Nishimura, M; Seino, Y; Tsuura, Y; Usami, M1
Cockburn, BN; Polonsky, KS; Pugh, W; Zhou, YP1
Miwa, I; Okinaka, M; Tanigawa, K; Taniguchi, S1
Budzko, D; Miki, T; Niki, I; Niwa, T; Senda, T; Yu, W1

Other Studies

17 other study(ies) available for nitrendipine and diazoxide

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
A novel D-phenylalanine-derivative hypoglycemic agent A-4166 increases cytosolic free Ca2+ in rat pancreatic beta-cells by stimulating Ca2+ influx.
    Endocrinology, 1994, Volume: 134, Issue:3

    Topics: Animals; Calcium; Cyclohexanes; Cytosol; Diazoxide; Dose-Response Relationship, Drug; Glucose; Hypoglycemic Agents; Islets of Langerhans; Nateglinide; Nitrendipine; Phenylalanine; Potassium Channels; Rats; Rats, Wistar; Sulfonylurea Compounds

1994
Activin A increases intracellular free calcium concentrations in rat pancreatic islets.
    FEBS letters, 1993, Aug-23, Volume: 329, Issue:1-2

    Topics: Activins; Animals; Calcium; Carbachol; Cyclic AMP; Diazoxide; Inhibins; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Nitrendipine; Rats; Rats, Wistar; Verapamil

1993
Necessity of endogenous GTP derived from glucose-6-phosphate for insulin secretion augmented by glucose under protein kinase A activation.
    Biochemical and biophysical research communications, 1998, Feb-04, Volume: 243, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Cyclic AMP-Dependent Protein Kinases; Diazoxide; Enzyme Activation; Glucose; Glucose-6-Phosphate; Glyceraldehyde 3-Phosphate; Glycolysis; Guanosine Triphosphate; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nitrendipine; Potassium Channels; Rats; Rats, Wistar; Signal Transduction

1998
Basal insulin hypersecretion in insulin-resistant Zucker diabetic and Zucker fatty rats: role of enhanced fuel metabolism.
    Metabolism: clinical and experimental, 1999, Volume: 48, Issue:7

    Topics: Animals; Blood Glucose; Calcium Channel Blockers; Diabetes Mellitus; Diazoxide; Enzyme Inhibitors; Glycolysis; Insulin; Insulin Resistance; Insulin Secretion; Islets of Langerhans; Male; Nitrendipine; Obesity; Proinsulin; Protein Kinase Inhibitors; Rats; Rats, Zucker

1999
Difference in mechanism between glyceraldehyde- and glucose-induced insulin secretion from isolated rat pancreatic islets.
    Journal of biochemistry, 2000, Volume: 127, Issue:2

    Topics: Adenosine Triphosphate; Animals; Calcium Channel Blockers; Carbachol; Cholinergic Agonists; Diazoxide; Female; Glucose; Glyceraldehyde; In Vitro Techniques; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Lactic Acid; Nitrendipine; Pyruvic Acid; Rats; Rats, Wistar; Triose-Phosphate Isomerase

2000
Ca2+ influx does not trigger glucose-induced traffic of the insulin granules and alteration of their distribution.
    Experimental biology and medicine (Maywood, N.J.), 2003, Volume: 228, Issue:10

    Topics: Calcium; Calcium Signaling; Cell Line; Cytoplasm; Diazoxide; Dose-Response Relationship, Drug; Down-Regulation; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Myosin Light Chains; Nifedipine; Nitrendipine; Phosphorylation; Tetradecanoylphorbol Acetate; Time Factors

2003