nipecotic acid has been researched along with baclofen in 32 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (21.88) | 18.7374 |
1990's | 15 (46.88) | 18.2507 |
2000's | 9 (28.13) | 29.6817 |
2010's | 1 (3.13) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chambon, JP; Desarmenien, M; Feltz, P; Humblet, C; Mann, A; Schlichter, R; Wermuth, CG | 1 |
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Dutia, MB; Johnston, AR; McQueen, DS | 1 |
Barolet, AW; Morris, ME | 1 |
Andrioli, GC; Bonanno, G; Raiteri, M; Ruelle, A | 1 |
Dun, NJ; Wang, MY | 1 |
Sved, AF; Sved, JC | 2 |
Bernardi, G; Calabresi, P; De Murtas, M; Mercuri, NB | 1 |
Dutar, P; Lamour, Y; Rascol, O | 1 |
Arakawa, T; Okada, Y | 1 |
Catelli, JM; Sved, AF | 1 |
Classen, K; Göthert, M; Schlicker, E | 1 |
Cherubini, E; North, RA | 1 |
el Manira, A; Grillner, S; Matsushima, T; Tegnér, J | 1 |
Gayet, J; Ginefri-Gayet, M | 1 |
Draguhn, A; Heinemann, U; Meierkord, H; Pfeiffer, M | 1 |
Hashimoto, T; Kuriyama, K | 1 |
Kelley, AE; Stratford, TR | 1 |
Abraini, JH; Bouquet, C; Cagniard, B; Kriem, B; Rostain, JC | 1 |
Cherubini, E; Martina, M; Sciancalepore, M; Strata, F | 1 |
Hemmings, HC; Murugaiah, KD | 1 |
Durgam, VR; Mifflin, SW; Vitela, M | 1 |
Ferreira, M; Gillis, RA; Hernandez, YM; Sahibzada, N; Wasserman, AM | 1 |
Bungo, T; Furuse, M; Izumi, T; Kawamura, K; Takagi, T; Ueda, H | 1 |
Frosini, M; Sgaragli, G; Valoti, M | 1 |
Isogai, O; Ito, S; Masubuchi, Y; Saito, S; Tsukamoto, K; Uchiyama, T; Yajima, Y | 1 |
Cremers, TI; Rea, K; Westerink, BH | 1 |
Galik, J; Hefferan, MP; Kakinohana, M; Kakinohana, O; Marsala, J; Marsala, M; Nakamura, S; Tomori, Z; Yaksh, TL | 1 |
Marino, V; Nassery, K; Parker, DA | 1 |
Arisawa, M; Hayakawa, W; Ide, S; Ito, Y; Katayama, T; Kawamura, S; Kobayashi, T; Masuda, E; Minami, M; Nakada, K; Shuto, S; Suemasa, A; Yamada, S; Yoshikawa, M | 1 |
32 other study(ies) available for nipecotic acid and baclofen
Article | Year |
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Synthesis and activity of 5-(aminomethylene)-1,3-cyclohexanediones: enolic analogues of gamma-aminobutyric acid.
Topics: Action Potentials; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Cyclohexanes; Cyclohexanones; Molecular Conformation; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1985 |
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles | 2005 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Tonic activity of rat medial vestibular nucleus neurones in vitro and its inhibition by GABA.
Topics: Action Potentials; Animals; Baclofen; Cobalt; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Neurons; Nipecotic Acids; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Vestibular Nuclei | 1992 |
Changes in extracellular K+ evoked by GABA, THIP and baclofen in the guinea-pig hippocampal slice.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electrodes; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Isoxazoles; Nipecotic Acids; Potassium; Proline; Receptors, GABA-A; Temperature | 1991 |
Cholinergic nerve terminals of human cerebral cortex possess a GABA transporter whose activation induces release of acetylcholine.
Topics: Acetylcholine; Anticonvulsants; Baclofen; Bicuculline; Biotransformation; Carrier Proteins; Cerebral Cortex; Choline; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Male; Membrane Proteins; Membrane Transport Proteins; Middle Aged; Muscimol; Nerve Endings; Nerve Tissue Proteins; Nipecotic Acids; Organic Anion Transporters; Parasympathetic Nervous System; Proline; Synaptosomes | 1991 |
Phaclofen-insensitive presynaptic inhibitory action of (+/-)-baclofen in neonatal rat motoneurones in vitro.
Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Evoked Potentials; Glutamates; In Vitro Techniques; Membrane Potentials; Motor Neurons; Nipecotic Acids; Potassium Channels; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior; Synapses | 1990 |
Endogenous GABA acts on GABAB receptors in nucleus tractus solitarius to increase blood pressure.
Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vigabatrin | 1990 |
Endogenous GABA mediates presynaptic inhibition of spontaneous and evoked excitatory synaptic potentials in the rat neostriatum.
Topics: Animals; Baclofen; Corpus Striatum; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Synapses; Tetrodotoxin | 1990 |
Cardiovascular responses elicited by gamma-aminobutyric acid in the nucleus tractus solitarius: evidence for action at the GABAB receptor.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; gamma-Aminobutyric Acid; Hemodynamics; Injections; Male; Medulla Oblongata; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasopressins | 1989 |
Rhythmical bursting activity and GABAergic mechanisms in the medial septum of normal and pertussis toxin-pretreated rats.
Topics: Action Potentials; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Neurons; Nipecotic Acids; Pertussis Toxin; Proline; Rats; Rats, Inbred Strains; Septum Pellucidum; Virulence Factors, Bordetella | 1989 |
Excitatory and inhibitory action of GABA on synaptic transmission in slices of guinea pig superior colliculus.
Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Muscimol; Nipecotic Acids; Perfusion; Proline; Receptors, GABA-A; Superior Colliculi; Synaptic Membranes; Synaptic Transmission | 1988 |
Enhanced pressor response to GABA in the nucleus tractus solitarii of the spontaneously hypertensive rat.
Topics: Animals; Baclofen; Blood Pressure; Brain Stem; gamma-Aminobutyric Acid; Heart Rate; Hypertension; Male; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred SHR; Rats, Inbred Strains | 1988 |
GABAB receptor-mediated inhibition of serotonin release in the rat brain.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Brain Chemistry; Cerebral Cortex; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Nipecotic Acids; Phentolamine; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin | 1984 |
Actions of gamma-aminobutyric acid on neurones of guinea-pig myenteric plexus.
Topics: Acetylcholine; Alanine; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glycine; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscimol; Myenteric Plexus; Neural Conduction; Neuromuscular Depolarizing Agents; Neurons; Nipecotic Acids; Picrotoxin; Proline; Tetrodotoxin | 1984 |
The spinal GABA system modulates burst frequency and intersegmental coordination in the lamprey: differential effects of GABAA and GABAB receptors.
Topics: Animals; Baclofen; Bicuculline; Culture Techniques; Diazepam; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Lampreys; Locomotion; Motor Neurons; Muscimol; Muscles; N-Methylaspartate; Nerve Net; Neurons; Nipecotic Acids; Proline; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission | 1993 |
Hypothermia induced by infusion of methionine sulfoximine into the dorsal raphe nucleus of the rat: involvement of 5-HT1A and GABAB receptors.
Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Bicuculline; Body Temperature Regulation; Hypothermia; Infusions, Parenteral; Ketanserin; Male; Methionine Sulfoximine; Nipecotic Acids; Pindolol; Proline; Raphe Nuclei; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Vigabatrin | 1993 |
Effects of gamma-aminobutyric acid (GABA) agonists and GABA uptake inhibitors on pharmacosensitive and pharmacoresistant epileptiform activity in vitro.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Entorhinal Cortex; Epilepsy; Female; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Muscimol; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Proline; Rats; Rats, Wistar; Tiagabine | 1996 |
GABAA receptor-mediated K(+)-evoked GABA release from globus pallidus--analysis using microdialysis.
Topics: Animals; Baclofen; Dinucleoside Phosphates; GABA Agonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Muscimol; Nipecotic Acids; Potassium Chloride; Proline; Rats; Rats, Wistar; Receptors, GABA-A | 1997 |
GABA in the nucleus accumbens shell participates in the central regulation of feeding behavior.
Topics: Animals; Baclofen; Eating; Enzyme Inhibitors; Feeding Behavior; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Nucleus Accumbens; Proline; Rats; Rats, Sprague-Dawley; Vigabatrin | 1997 |
Modulation by GABA transmission in the substantia nigra compacta and reticulata of locomotor activity in rats exposed to high pressure.
Topics: Animals; Baclofen; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Helium; High Pressure Neurological Syndrome; Male; Motor Activity; Muscimol; Myoclonus; Nipecotic Acids; Proline; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra; Synaptic Transmission; Time Factors; Vigabatrin | 1998 |
GABA excites immature CA3 pyramidal cells through bicuculline-sensitive and -insensitive chloride-dependent receptors.
Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Chloride Channels; Culture Techniques; Evoked Potentials; gamma-Aminobutyric Acid; Kynurenic Acid; Nipecotic Acids; Patch-Clamp Techniques; Picrotoxin; Proline; Pyramidal Cells; Rats; Receptors, GABA-A; Receptors, GABA-B; Zinc | 1998 |
Effects of intravenous general anesthetics on [3H]GABA release from rat cortical synaptosomes.
Topics: Aminobutyrates; Anesthesia, General; Anesthetics, Intravenous; Animals; Baclofen; Bicuculline; Calcium; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Nerve Endings; Nipecotic Acids; Picrotoxin; Potassium Chloride; Proline; Propofol; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Synaptic Transmission; Synaptosomes; Tritium | 1998 |
Enhanced gamma-aminobutyric acid-B receptor agonist responses and mRNA within the nucleus of the solitary tract in hypertension.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Agonists; GABA Antagonists; Hypertension, Renovascular; Male; Muscimol; Nephrectomy; Nipecotic Acids; Phosphinic Acids; Proline; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Solitary Nucleus; Transcription, Genetic | 1999 |
GABA-mediated neurotransmission in the ventrolateral NTS plays a role in respiratory regulation in the rat.
Topics: Animals; Apnea; Baclofen; Bicuculline; Cardiovascular System; Fluorescent Antibody Technique; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Kynurenic Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA; Respiration; Synaptic Transmission; Ventral Thalamic Nuclei | 2002 |
Intracerebroventricular injection of muscimol, baclofen or nipecotic acid stimulates food intake in layer-type, but not meat-type, chicks.
Topics: Animals; Animals, Newborn; Baclofen; Behavior, Animal; Chickens; Dose-Response Relationship, Drug; Eating; GABA Agonists; Injections, Intraventricular; Male; Muscimol; Nipecotic Acids; Species Specificity | 2003 |
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex | 2004 |
Effect of a high-salt diet on gamma-aminobutyric acid-mediated responses in the nucleus tractus solitarius of Sprague-Dawley rats.
Topics: Animals; Baclofen; Baroreflex; Bicuculline; Blood Pressure; Cardiovascular Physiological Phenomena; Dose-Response Relationship, Drug; Food, Formulated; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Heart Rate; Male; Muscimol; Neural Inhibition; Nipecotic Acids; Nitroprusside; Organophosphorus Compounds; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Sodium Chloride, Dietary; Solitary Nucleus | 2004 |
HPLC conditions are critical for the detection of GABA by microdialysis.
Topics: Anesthetics, Local; Animals; Baclofen; Benzylamines; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Nipecotic Acids; Phosphinic Acids; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Time Factors | 2005 |
Development of GABA-sensitive spasticity and rigidity in rats after transient spinal cord ischemia: a qualitative and quantitative electrophysiological and histopathological study.
Topics: Acetyltransferases; Analysis of Variance; Animals; Baclofen; Dose-Response Relationship, Radiation; Drug Delivery Systems; Electric Stimulation; Electromyography; Evoked Potentials, Motor; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression; H-Reflex; Immunohistochemistry; Male; Muscle Rigidity; Muscle Spasticity; Muscle, Skeletal; Neurologic Examination; Nipecotic Acids; Rats; Rats, Sprague-Dawley; Rhizotomy; Spinal Cord Ischemia; Vesicular Glutamate Transport Protein 1; Vesicular Glutamate Transport Protein 2 | 2006 |
Uptake and release of [(3)H]GABA in human dental pulp.
Topics: Adult; Autoreceptors; Baclofen; Dental Pulp; Electric Stimulation; Female; GABA Agents; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Male; Morpholines; Nipecotic Acids; Oximes; Radiopharmaceuticals; Receptors, GABA; Time Factors; Tritium | 2007 |
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.
Topics: Animals; Anticonvulsants; Brain; Cyclopropanes; GABA Modulators; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ligands; Mice; Protein Binding; Rats; Seizures; Stereoisomerism; Structure-Activity Relationship | 2013 |