nipecotic acid and baclofen

nipecotic acid has been researched along with baclofen in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19907 (21.88)18.7374
1990's15 (46.88)18.2507
2000's9 (28.13)29.6817
2010's1 (3.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chambon, JP; Desarmenien, M; Feltz, P; Humblet, C; Mann, A; Schlichter, R; Wermuth, CG1
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Dutia, MB; Johnston, AR; McQueen, DS1
Barolet, AW; Morris, ME1
Andrioli, GC; Bonanno, G; Raiteri, M; Ruelle, A1
Dun, NJ; Wang, MY1
Sved, AF; Sved, JC2
Bernardi, G; Calabresi, P; De Murtas, M; Mercuri, NB1
Dutar, P; Lamour, Y; Rascol, O1
Arakawa, T; Okada, Y1
Catelli, JM; Sved, AF1
Classen, K; Göthert, M; Schlicker, E1
Cherubini, E; North, RA1
el Manira, A; Grillner, S; Matsushima, T; Tegnér, J1
Gayet, J; Ginefri-Gayet, M1
Draguhn, A; Heinemann, U; Meierkord, H; Pfeiffer, M1
Hashimoto, T; Kuriyama, K1
Kelley, AE; Stratford, TR1
Abraini, JH; Bouquet, C; Cagniard, B; Kriem, B; Rostain, JC1
Cherubini, E; Martina, M; Sciancalepore, M; Strata, F1
Hemmings, HC; Murugaiah, KD1
Durgam, VR; Mifflin, SW; Vitela, M1
Ferreira, M; Gillis, RA; Hernandez, YM; Sahibzada, N; Wasserman, AM1
Bungo, T; Furuse, M; Izumi, T; Kawamura, K; Takagi, T; Ueda, H1
Frosini, M; Sgaragli, G; Valoti, M1
Isogai, O; Ito, S; Masubuchi, Y; Saito, S; Tsukamoto, K; Uchiyama, T; Yajima, Y1
Cremers, TI; Rea, K; Westerink, BH1
Galik, J; Hefferan, MP; Kakinohana, M; Kakinohana, O; Marsala, J; Marsala, M; Nakamura, S; Tomori, Z; Yaksh, TL1
Marino, V; Nassery, K; Parker, DA1
Arisawa, M; Hayakawa, W; Ide, S; Ito, Y; Katayama, T; Kawamura, S; Kobayashi, T; Masuda, E; Minami, M; Nakada, K; Shuto, S; Suemasa, A; Yamada, S; Yoshikawa, M1

Other Studies

32 other study(ies) available for nipecotic acid and baclofen

ArticleYear
Synthesis and activity of 5-(aminomethylene)-1,3-cyclohexanediones: enolic analogues of gamma-aminobutyric acid.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:10

    Topics: Action Potentials; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Cyclohexanes; Cyclohexanones; Molecular Conformation; Rats; Receptors, GABA-A; Structure-Activity Relationship

1985
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Tonic activity of rat medial vestibular nucleus neurones in vitro and its inhibition by GABA.
    Experimental brain research, 1992, Volume: 88, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Cobalt; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Neurons; Nipecotic Acids; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Vestibular Nuclei

1992
Changes in extracellular K+ evoked by GABA, THIP and baclofen in the guinea-pig hippocampal slice.
    Experimental brain research, 1991, Volume: 84, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electrodes; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Isoxazoles; Nipecotic Acids; Potassium; Proline; Receptors, GABA-A; Temperature

1991
Cholinergic nerve terminals of human cerebral cortex possess a GABA transporter whose activation induces release of acetylcholine.
    Brain research, 1991, Jan-25, Volume: 539, Issue:2

    Topics: Acetylcholine; Anticonvulsants; Baclofen; Bicuculline; Biotransformation; Carrier Proteins; Cerebral Cortex; Choline; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Male; Membrane Proteins; Membrane Transport Proteins; Middle Aged; Muscimol; Nerve Endings; Nerve Tissue Proteins; Nipecotic Acids; Organic Anion Transporters; Parasympathetic Nervous System; Proline; Synaptosomes

1991
Phaclofen-insensitive presynaptic inhibitory action of (+/-)-baclofen in neonatal rat motoneurones in vitro.
    British journal of pharmacology, 1990, Volume: 99, Issue:2

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Evoked Potentials; Glutamates; In Vitro Techniques; Membrane Potentials; Motor Neurons; Nipecotic Acids; Potassium Channels; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior; Synapses

1990
Endogenous GABA acts on GABAB receptors in nucleus tractus solitarius to increase blood pressure.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vigabatrin

1990
Endogenous GABA mediates presynaptic inhibition of spontaneous and evoked excitatory synaptic potentials in the rat neostriatum.
    Neuroscience letters, 1990, Oct-02, Volume: 118, Issue:1

    Topics: Animals; Baclofen; Corpus Striatum; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Synapses; Tetrodotoxin

1990
Cardiovascular responses elicited by gamma-aminobutyric acid in the nucleus tractus solitarius: evidence for action at the GABAB receptor.
    Neuropharmacology, 1989, Volume: 28, Issue:5

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; gamma-Aminobutyric Acid; Hemodynamics; Injections; Male; Medulla Oblongata; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasopressins

1989
Rhythmical bursting activity and GABAergic mechanisms in the medial septum of normal and pertussis toxin-pretreated rats.
    Experimental brain research, 1989, Volume: 77, Issue:2

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Neurons; Nipecotic Acids; Pertussis Toxin; Proline; Rats; Rats, Inbred Strains; Septum Pellucidum; Virulence Factors, Bordetella

1989
Excitatory and inhibitory action of GABA on synaptic transmission in slices of guinea pig superior colliculus.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Muscimol; Nipecotic Acids; Perfusion; Proline; Receptors, GABA-A; Superior Colliculi; Synaptic Membranes; Synaptic Transmission

1988
Enhanced pressor response to GABA in the nucleus tractus solitarii of the spontaneously hypertensive rat.
    European journal of pharmacology, 1988, Jul-07, Volume: 151, Issue:2

    Topics: Animals; Baclofen; Blood Pressure; Brain Stem; gamma-Aminobutyric Acid; Heart Rate; Hypertension; Male; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred SHR; Rats, Inbred Strains

1988
GABAB receptor-mediated inhibition of serotonin release in the rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 326, Issue:2

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Brain Chemistry; Cerebral Cortex; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Nipecotic Acids; Phentolamine; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin

1984
Actions of gamma-aminobutyric acid on neurones of guinea-pig myenteric plexus.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Acetylcholine; Alanine; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glycine; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscimol; Myenteric Plexus; Neural Conduction; Neuromuscular Depolarizing Agents; Neurons; Nipecotic Acids; Picrotoxin; Proline; Tetrodotoxin

1984
The spinal GABA system modulates burst frequency and intersegmental coordination in the lamprey: differential effects of GABAA and GABAB receptors.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Culture Techniques; Diazepam; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Lampreys; Locomotion; Motor Neurons; Muscimol; Muscles; N-Methylaspartate; Nerve Net; Neurons; Nipecotic Acids; Proline; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission

1993
Hypothermia induced by infusion of methionine sulfoximine into the dorsal raphe nucleus of the rat: involvement of 5-HT1A and GABAB receptors.
    European journal of pharmacology, 1993, Apr-28, Volume: 235, Issue:2-3

    Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Bicuculline; Body Temperature Regulation; Hypothermia; Infusions, Parenteral; Ketanserin; Male; Methionine Sulfoximine; Nipecotic Acids; Pindolol; Proline; Raphe Nuclei; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Vigabatrin

1993
Effects of gamma-aminobutyric acid (GABA) agonists and GABA uptake inhibitors on pharmacosensitive and pharmacoresistant epileptiform activity in vitro.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Entorhinal Cortex; Epilepsy; Female; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Muscimol; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Proline; Rats; Rats, Wistar; Tiagabine

1996
GABAA receptor-mediated K(+)-evoked GABA release from globus pallidus--analysis using microdialysis.
    Neurochemistry international, 1997, Volume: 30, Issue:3

    Topics: Animals; Baclofen; Dinucleoside Phosphates; GABA Agonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Muscimol; Nipecotic Acids; Potassium Chloride; Proline; Rats; Rats, Wistar; Receptors, GABA-A

1997
GABA in the nucleus accumbens shell participates in the central regulation of feeding behavior.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jun-01, Volume: 17, Issue:11

    Topics: Animals; Baclofen; Eating; Enzyme Inhibitors; Feeding Behavior; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Nucleus Accumbens; Proline; Rats; Rats, Sprague-Dawley; Vigabatrin

1997
Modulation by GABA transmission in the substantia nigra compacta and reticulata of locomotor activity in rats exposed to high pressure.
    Neuroreport, 1998, May-11, Volume: 9, Issue:7

    Topics: Animals; Baclofen; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Helium; High Pressure Neurological Syndrome; Male; Motor Activity; Muscimol; Myoclonus; Nipecotic Acids; Proline; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra; Synaptic Transmission; Time Factors; Vigabatrin

1998
GABA excites immature CA3 pyramidal cells through bicuculline-sensitive and -insensitive chloride-dependent receptors.
    Perspectives on developmental neurobiology, 1998, Volume: 5, Issue:2-3

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Chloride Channels; Culture Techniques; Evoked Potentials; gamma-Aminobutyric Acid; Kynurenic Acid; Nipecotic Acids; Patch-Clamp Techniques; Picrotoxin; Proline; Pyramidal Cells; Rats; Receptors, GABA-A; Receptors, GABA-B; Zinc

1998
Effects of intravenous general anesthetics on [3H]GABA release from rat cortical synaptosomes.
    Anesthesiology, 1998, Volume: 89, Issue:4

    Topics: Aminobutyrates; Anesthesia, General; Anesthetics, Intravenous; Animals; Baclofen; Bicuculline; Calcium; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Nerve Endings; Nipecotic Acids; Picrotoxin; Potassium Chloride; Proline; Propofol; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Synaptic Transmission; Synaptosomes; Tritium

1998
Enhanced gamma-aminobutyric acid-B receptor agonist responses and mRNA within the nucleus of the solitary tract in hypertension.
    Hypertension (Dallas, Tex. : 1979), 1999, Volume: 33, Issue:1 Pt 2

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Agonists; GABA Antagonists; Hypertension, Renovascular; Male; Muscimol; Nephrectomy; Nipecotic Acids; Phosphinic Acids; Proline; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Solitary Nucleus; Transcription, Genetic

1999
GABA-mediated neurotransmission in the ventrolateral NTS plays a role in respiratory regulation in the rat.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 283, Issue:6

    Topics: Animals; Apnea; Baclofen; Bicuculline; Cardiovascular System; Fluorescent Antibody Technique; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Kynurenic Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA; Respiration; Synaptic Transmission; Ventral Thalamic Nuclei

2002
Intracerebroventricular injection of muscimol, baclofen or nipecotic acid stimulates food intake in layer-type, but not meat-type, chicks.
    Brain research, 2003, Dec-12, Volume: 993, Issue:1-2

    Topics: Animals; Animals, Newborn; Baclofen; Behavior, Animal; Chickens; Dose-Response Relationship, Drug; Eating; GABA Agonists; Injections, Intraventricular; Male; Muscimol; Nipecotic Acids; Species Specificity

2003
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex

2004
Effect of a high-salt diet on gamma-aminobutyric acid-mediated responses in the nucleus tractus solitarius of Sprague-Dawley rats.
    Brain research bulletin, 2004, Sep-30, Volume: 64, Issue:3

    Topics: Animals; Baclofen; Baroreflex; Bicuculline; Blood Pressure; Cardiovascular Physiological Phenomena; Dose-Response Relationship, Drug; Food, Formulated; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Heart Rate; Male; Muscimol; Neural Inhibition; Nipecotic Acids; Nitroprusside; Organophosphorus Compounds; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Sodium Chloride, Dietary; Solitary Nucleus

2004
HPLC conditions are critical for the detection of GABA by microdialysis.
    Journal of neurochemistry, 2005, Volume: 94, Issue:3

    Topics: Anesthetics, Local; Animals; Baclofen; Benzylamines; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Nipecotic Acids; Phosphinic Acids; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Time Factors

2005
Development of GABA-sensitive spasticity and rigidity in rats after transient spinal cord ischemia: a qualitative and quantitative electrophysiological and histopathological study.
    Neuroscience, 2006, Sep-01, Volume: 141, Issue:3

    Topics: Acetyltransferases; Analysis of Variance; Animals; Baclofen; Dose-Response Relationship, Radiation; Drug Delivery Systems; Electric Stimulation; Electromyography; Evoked Potentials, Motor; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression; H-Reflex; Immunohistochemistry; Male; Muscle Rigidity; Muscle Spasticity; Muscle, Skeletal; Neurologic Examination; Nipecotic Acids; Rats; Rats, Sprague-Dawley; Rhizotomy; Spinal Cord Ischemia; Vesicular Glutamate Transport Protein 1; Vesicular Glutamate Transport Protein 2

2006
Uptake and release of [(3)H]GABA in human dental pulp.
    Archives of oral biology, 2007, Volume: 52, Issue:7

    Topics: Adult; Autoreceptors; Baclofen; Dental Pulp; Electric Stimulation; Female; GABA Agents; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Male; Morpholines; Nipecotic Acids; Oximes; Radiopharmaceuticals; Receptors, GABA; Time Factors; Tritium

2007
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.
    Bioorganic & medicinal chemistry, 2013, Sep-01, Volume: 21, Issue:17

    Topics: Animals; Anticonvulsants; Brain; Cyclopropanes; GABA Modulators; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ligands; Mice; Protein Binding; Rats; Seizures; Stereoisomerism; Structure-Activity Relationship

2013