nilutamide and dihydrotestosterone

nilutamide has been researched along with dihydrotestosterone in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19904 (21.05)18.7374
1990's6 (31.58)18.2507
2000's5 (26.32)29.6817
2010's3 (15.79)24.3611
2020's1 (5.26)2.80

Authors

AuthorsStudies
Annoot, D; Clément-Lacroix, P; Deprez, P; Duval, E; Fleury, D; Guédin, D; Hebbe, S; Lefrançois, JM; Lemoullec, JM; Michoux, L; Minet, D; Mollat, P; Nique, F; Peixoto, C; Prangé, T; Robin-Jagerschmidt, C; Thauvin, M; Triballeau, N1
Bian, J; Chen, R; Li, M; Li, Z; Tang, J; Tian, Y; Xie, Y; Xu, X; Zhang, Y; Zhang, Z1
Brand, T; Slob, AK1
Bruchovsky, N; Fletcher, T; Foekens, JA; Goldenberg, SL; Lawson, D; Rennie, PS1
Belanger, A; Cusan, L; Dupont, A; Emond, JP; Fazekas, AT; Husson, JM; Laberge, JG; Labrie, F; Lefebvre, FA; Monfette, G; Raynaud, JP1
Brown, TR; Migeon, CJ; Rothwell, SW; Sultan, C1
Kopu, H1
Bentel, JM; Birrell, SN; Hickey, TE; Horsfall, DJ; Ricciardelli, C; Tilley, WD; Weger, MA1
Govindan, MV; Koutsilieris, M; Pagé, N; Warriar, N2
Barritault, D; Caruelle, D; Caruelle, JP; Courty, J; Delbe, J; Laaroubi, K; Vacherot, F1
Balk, SP; Bubley, GJ; Fenton, MA; Fertig, AM; Kolvenbag, G; Shuster, TD; Taplin, ME1
Baltogiannis, D; Charalabopoulos, K; Giannakopoulos, X; Sofikitis, N1
Bian, Q; Chen, JF; Song, L; Sun, H; Wang, XR; Xu, LC1
Chang, CY; Chang, SY; Hsuuw, YD; Huang, CK; Huang, FJ; Huang, KE; Kang, HY; Shyr, CR1
Chen, JF; Cui, LB; Hong, X; Song, L; Sun, H; Wang, XR; Xu, LC; Xu, XL1
Dong, Z; Lu, S; Wang, A1
Hu, JX; Li, J; Li, YF; Pan, C; Wang, HM; Xu, LC; Zhang, JP1
Dong, Y; Guy, RK; Keiser, J; Lin, MF; Min, J; Muniyan, S; Vargas, M; Vennerstrom, JL; Wang, C; Wang, X; Zhao, Q1

Reviews

2 review(s) available for nilutamide and dihydrotestosterone

ArticleYear
Overview of the development of selective androgen receptor modulators (SARMs) as pharmacological treatment for osteoporosis (1998-2021).
    European journal of medicinal chemistry, 2022, Feb-15, Volume: 230

    Topics: Androgen Antagonists; Androgens; Humans; Osteoporosis; Receptors, Androgen; Structure-Activity Relationship

2022
Monotherapy in advanced prostate cancer: an overview.
    Experimental oncology, 2004, Volume: 26, Issue:3

    Topics: Adenocarcinoma; Androgen Antagonists; Anilides; Antineoplastic Agents, Hormonal; Combined Modality Therapy; Cyproterone Acetate; Dihydrotestosterone; Estrogens; Flutamide; Gonadotropin-Releasing Hormone; Humans; Imidazolidines; Male; Nitriles; Orchiectomy; Palliative Care; Progesterone Congeners; Prostatic Neoplasms; Randomized Controlled Trials as Topic; Testosterone; Tosyl Compounds

2004

Other Studies

17 other study(ies) available for nilutamide and dihydrotestosterone

ArticleYear
Discovery of diarylhydantoins as new selective androgen receptor modulators.
    Journal of medicinal chemistry, 2012, Oct-11, Volume: 55, Issue:19

    Topics: Anabolic Agents; Androgen Receptor Antagonists; Androgens; Animals; Binding, Competitive; Bone and Bones; Crystallography, X-Ray; Drug Partial Agonism; HeLa Cells; Humans; Hydantoins; Male; Models, Molecular; Muscle, Skeletal; Orchiectomy; Prostate; Rats; Receptors, Androgen; Stereoisomerism; Structure-Activity Relationship; Transcriptional Activation

2012
On the organization of partner preference behavior in female Wistar rats.
    Physiology & behavior, 1991, Volume: 49, Issue:3

    Topics: Androgen Antagonists; Animals; Copulation; Dihydrotestosterone; Dose-Response Relationship, Drug; Estradiol; Female; Flutamide; Imidazoles; Imidazolidines; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Sex Differentiation; Sexual Behavior, Animal; Sexual Maturation; Social Environment; Testosterone

1991
Relative effectiveness of alternative androgen withdrawal therapies in initiating regression of rat prostate.
    The Journal of urology, 1988, Volume: 139, Issue:6

    Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Gonadotropin-Releasing Hormone; Imidazoles; Imidazolidines; Leuprolide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen

1988
New hormonal treatment in cancer of the prostate: combined administration of an LHRH agonist and an antiandrogen.
    Journal of steroid biochemistry, 1983, Volume: 19, Issue:1C

    Topics: Androgen Antagonists; Animals; Buserelin; Castration; Dihydrotestosterone; Drug Therapy, Combination; Gonadotropin-Releasing Hormone; Hormones; Humans; Imidazoles; Imidazolidines; Male; Prostate; Prostatic Neoplasms; Rats; Seminal Vesicles; Testosterone

1983
Inhibition of androgen binding in human foreskin fibroblasts by antiandrogens.
    Steroids, 1981, Volume: 37, Issue:6

    Topics: Androgen Antagonists; Androgens; Binding, Competitive; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Estrenes; Fibroblasts; Humans; Imidazoles; Imidazolidines; Infant, Newborn; Male; Metribolone; Penis; Receptors, Androgen; Receptors, Steroid; Subcellular Fractions; Testosterone

1981
5 alpha-Dihydrotestosterone-induced uteroglobin synthesis in rabbit uterus is not inhibited by antiandrogen administration but is prevented by estradiol.
    Biochimica et biophysica acta, 1981, Jul-27, Volume: 654, Issue:2

    Topics: Androgen Antagonists; Animals; Dihydrotestosterone; Estradiol; Female; Glycoproteins; Imidazoles; Imidazolidines; In Vitro Techniques; Rabbits; Receptors, Progesterone; RNA, Messenger; Uteroglobin; Uterus

1981
Androgens induce divergent proliferative responses in human breast cancer cell lines.
    The Journal of steroid biochemistry and molecular biology, 1995, Volume: 52, Issue:5

    Topics: Androgen Receptor Antagonists; Androgens; Breast Neoplasms; Cell Division; Dihydrotestosterone; Flutamide; Humans; Imidazoles; Imidazolidines; Nandrolone; Oligonucleotides, Antisense; Receptors, Androgen; Tumor Cells, Cultured

1995
Antiandrogens inhibit human androgen receptor-dependent gene transcription activation in the human prostate cancer cells LNCaP.
    The Prostate, 1994, Volume: 24, Issue:4

    Topics: Amino Acid Sequence; Androgen Antagonists; Binding, Competitive; Blotting, Western; Chloramphenicol O-Acetyltransferase; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Gene Expression Regulation, Viral; Humans; Imidazoles; Imidazolidines; Male; Mammary Tumor Virus, Mouse; Molecular Sequence Data; Promoter Regions, Genetic; Prostatic Neoplasms; Receptors, Androgen; Transcription, Genetic; Transfection; Tumor Cells, Cultured

1994
Interaction of antiandrogen-androgen receptor complexes with DNA and transcription activation.
    The Journal of steroid biochemistry and molecular biology, 1993, Volume: 46, Issue:6

    Topics: Androgen Antagonists; Animals; Binding, Competitive; Blotting, Western; Cell Line; Chloramphenicol O-Acetyltransferase; Chlorocebus aethiops; Cyproterone Acetate; Dihydrotestosterone; DNA; Flutamide; Gene Expression Regulation; Humans; Imidazoles; Imidazolidines; Kidney; Kinetics; Mammary Tumor Virus, Mouse; Metribolone; Receptors, Androgen; Recombinant Proteins; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection

1993
Upregulation of heparin-affin regulatory peptide by androgen.
    In vitro cellular & developmental biology. Animal, 1995, Volume: 31, Issue:9

    Topics: Androgen Antagonists; Animals; Carrier Proteins; Cell Line; Cytokines; Dihydrotestosterone; Gene Expression Regulation; Growth Substances; Humans; Imidazoles; Imidazolidines; RNA, Messenger; Up-Regulation

1995
Functional characterization of mutant androgen receptors from androgen-independent prostate cancer.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 1997, Volume: 3, Issue:8

    Topics: Amino Acid Substitution; Androgen Antagonists; Androgens; Androstenedione; Animals; beta-Galactosidase; Cell Line; Dihydrotestosterone; Estradiol; Flutamide; Genes, Reporter; Imidazoles; Imidazolidines; Luciferases; Male; Point Mutation; Progesterone; Prostatic Neoplasms; Receptors, Androgen; Recombinant Fusion Proteins; Transfection

1997
Androgen receptor activities of p,p'-DDE, fenvalerate and phoxim detected by androgen receptor reporter gene assay.
    Toxicology letters, 2006, Jan-05, Volume: 160, Issue:2

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Animals; Biological Assay; Cell Line; Cercopithecus; Dexamethasone; Dichlorodiphenyl Dichloroethylene; Dihydrotestosterone; Genes, Reporter; Humans; Imidazolidines; Insecticides; Mammary Tumor Virus, Mouse; Mice; Nitriles; Organothiophosphorus Compounds; Plasmids; Pyrethrins; Receptors, Androgen; Transfection

2006
Androgenic and antiandrogenic effects and expression of androgen receptor in mouse embryonic stem cells.
    Fertility and sterility, 2006, Volume: 85 Suppl 1

    Topics: Androgen Antagonists; Androgens; Animals; Blastocyst; Cell Differentiation; Cell Proliferation; Cells, Cultured; Dihydrotestosterone; Gene Expression Regulation, Developmental; Imidazolidines; Mice; Mice, Inbred ICR; Receptors, Adrenergic; Stem Cells; Testosterone

2006
Antiandrogenic activity of pyrethroid pesticides and their metabolite in reporter gene assay.
    Chemosphere, 2007, Volume: 66, Issue:3

    Topics: Androgen Antagonists; Animals; Cell Line; Cell Proliferation; Cell Survival; Dexamethasone; Dihydrotestosterone; Flutamide; Humans; Imidazolidines; Luciferases; Molecular Structure; Nitriles; Permethrin; Pesticides; Pyrethrins; Receptors, Androgen; Recombinant Fusion Proteins; Response Elements; Transfection

2007
A novel synthetic compound that interrupts androgen receptor signaling in human prostate cancer cells.
    Molecular cancer therapeutics, 2007, Volume: 6, Issue:7

    Topics: Androgen Receptor Antagonists; Androgens; Anilides; Antineoplastic Agents; Cell Proliferation; Dihydrotestosterone; Drug Resistance, Neoplasm; Drug Synergism; Flutamide; Gene Expression Regulation, Neoplastic; HeLa Cells; Humans; Imidazolidines; Male; Nitriles; Prostate-Specific Antigen; Prostatic Neoplasms; Receptors, Androgen; Signal Transduction; Tosyl Compounds; Transcription, Genetic

2007
Anti-androgen effects of cypermethrin on the amino- and carboxyl-terminal interaction of the androgen receptor.
    Toxicology, 2012, Feb-26, Volume: 292, Issue:2-3

    Topics: Androgen Antagonists; Androgen Receptor Antagonists; Cell Line; Dihydrotestosterone; Humans; Imidazolidines; Insecticides; Plasmids; Pyrethrins; Receptors, Androgen; Recombinant Proteins; Two-Hybrid System Techniques

2012
Antischistosomal versus antiandrogenic properties of aryl hydantoin Ro 13-3978.
    The American journal of tropical medicine and hygiene, 2014, Volume: 90, Issue:6

    Topics: Androgen Receptor Antagonists; Animals; Cell Line, Tumor; Cell Proliferation; Dihydrotestosterone; Disease Models, Animal; Humans; Hydantoins; Imidazolidines; Male; Mice; Schistosoma mansoni; Schistosomiasis mansoni; Schistosomicides

2014