nifedipine and oxadiazoles

nifedipine has been researched along with oxadiazoles in 66 studies

Research

Studies (66)

TimeframeStudies, this research(%)All Research%
pre-199038 (57.58)18.7374
1990's15 (22.73)18.2507
2000's10 (15.15)29.6817
2010's3 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hammond, C; Henderson, G; Mason, WT; Morton, AJ1
Bolger, GT; Campbell, N; Crowley, M; McKay, DW; O'Neill, SK; Triggle, CR1
Gu, XH; Nayler, WG1
Fitzpatrick, LA; Jones, JI1
Hosey, MM; McMahon, KK; Ptasienski, J1
Benavides, J; Bertrand, P; Burgevin, MC; Doble, A; Ferris, O; Gueremy, C; Le Fur, G; Menager, J; Uzan, A; Vaucher, N1
Glossmann, H; Goll, A; Moosburger, K; Striessnig, J1
Cognard, C; Fosset, M; Galizzi, JP; Lazdunski, M; Romey, G1
Carpenter, CL; Greenberg, DA; Messing, RO1
Cauvin, C; Hwang, O; van Breemen, C; Yamamoto, M1
Holck, M; Osterrieder, W1
Abram, A; Baginski, T; Banning, J; Rao, V1
DeRoth, L; Godfraind, T; Wibo, M1
Lamb, GD; Walsh, T1
Massieu, L; Tapia, R1
Akbarali, H; Gilbert, R; Hall, J; Moody-Corbett, F1
Matlib, MA1
Magill, SB; Parmar, SS; Stone, JS1
Ferry, DR; Glossmann, H; Goll, A; Linn, T1
Godfraind, T; Morel, N1
Al-Mahmood, HA; el-Khatim, MS; Gumaa, KA; Thulesius, O1
Handley, DA; Melden, MK; Saunders, RN; Van Valen, RG1
Allen, J; Jackson, NC; Pool, PE; Taylor, SH1
Hof, RP1
del Pozo, E; Sieber, C1
Navarro, J; Tauber, AI; Williamson, KC1
Barrès, C; Cerutti, C; Morin, B; Sassard, J1
Navarro, J1
Jie, K; Timmermans, PB; van Brummelen, P; van Zwieten, PA; Vermey, P1
Oswald, RE; Weiland, GA1
Church, J; Davies, SN; Lodge, D1
Sokolov, AM1
Dougherty, C; Rutsch, W; Schartl, M; Schmutzler, H1
Bichko, MV; Korabel'shchikova, NI; Rishko, NV2
Lee, HR; Roeske, WR; Yamamura, HI1
Karobath, M; Supavilai, P1
Müller-Schweinitzer, E; Neumann, P1
Cortés, R; Karobath, M; Palacios, JM; Supavilai, P1
Ferry, DR; Glossmann, H; Goll, A1
Fuchs, M; Hilger, HH; Hombach, V; Jansen, W; Osterspey, A; Tauchert, M1
Kolsky, H; Moisson, P; Witchitz, S1
Hill, RG; Longmore, J; Razzaque, Z1
Dakshinamurti, K; Lal, KJ1
Ehrenstein, G; Fitzpatrick, LA; Pocotte, SL1
Hattori, K; Maruyama, K; Nagatomo, T; Qu, YL; Sugiyama, K; Takamizawa, C; Watanabe, K1
Masuda, Y; Tanaka, S; Yamashita, T1
Fitzpatrick, LA; Maercklein, PB; Ritchie, CK1
McMurtry, IF; Morris, KG; Oka, M1
Calvino, R; Di Stilo, A; Fruttero, R; Gasco, A; Gasco, AM; Sorba, G1
Brauns, T; Glossmann, H; Haugland, RP; Kimball, SD; Prinz, H; Striessnig, J1
Cocks, TM; Satchell, DG; Selemidis, S1
Cena, C; Di Stilo, A; Ermondi, G; Gasco, A; Gasco, AM; Visentin, S1
Cocks, TM; Selemidis, S1
Lovren, F; Triggle, C1
Kan, E; Kelly, JE; Lokuta, AJ; Nishio, M; Sagawa, K; Sagawa, T; Tsai, J; Wasserstrom, JA1
Fernández, E; Jiménez, M; Tanović, A1
Paterson, WG; Zhang, Y2
Anderson, U; Keef, KD; O'Driscoll, K; Sanders, KM; Ward, SM1
Delogu, MR; Desole, MS; Esposito, G; Miele, E; Miele, M; Migheli, R; Mura, MP; Rocchitta, G; Serra, PA; Taras, MG1
Ambrosio, SR; da Costa, FB; de Oliveira, AM; Tirapelli, CR1
Favaloro, JL; Kemp-Harper, BK1
Centurión, D; Cobos-Puc, LE; González-Hernández, A; Maassenvandenbrink, A; Muñoz-Islas, E; Ramírez-Rosas, MB; Sánchez-López, A; Villalón, CM1
Piñeros, MA; Tester, M1
Blood, AB; Liu, T; Longo, LD; Power, GG; Schroeder, HJ; Terry, MH; Wilson, SM; Zhang, M1

Trials

5 trial(s) available for nifedipine and oxadiazoles

ArticleYear
Efficacy of a new calcium antagonist PN 200-110 (isradipine) in angina pectoris.
    The American journal of cardiology, 1987, Jan-30, Volume: 59, Issue:3

    Topics: Angina Pectoris; Calcium Channel Blockers; Clinical Trials as Topic; Double-Blind Method; Exercise Test; Female; Humans; Isosorbide Dinitrate; Isradipine; Male; Nifedipine; Oxadiazoles; Placebos

1987
Influence of calcium entry blockade on alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in the forearm of hypertensive patients.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:2

    Topics: Adult; Azepines; Calcium Channel Blockers; Female; Forearm; Hemodynamics; Humans; Hypertension; Isradipine; Male; Methoxamine; Middle Aged; Nifedipine; Oxadiazoles; Receptors, Adrenergic, alpha; Regional Blood Flow; Vascular Resistance; Vasoconstriction

1987
Hemodynamic effects of molsidomine, isosorbide dinitrate, and nifedipine at rest and during exercise.
    American heart journal, 1985, Volume: 109, Issue:3 Pt 2

    Topics: Adult; Blood Pressure; Coronary Disease; Heart Rate; Hemodynamics; Humans; Isosorbide Dinitrate; Middle Aged; Molsidomine; Nifedipine; Oxadiazoles; Physical Exertion; Stroke Volume; Sydnones; Time Factors; Vasodilator Agents

1985
[Rheological properties of blood in patients with stenocardia during treatment with obsidan, corvatone and corinfar].
    Vrachebnoe delo, 1985, Issue:4

    Topics: Adult; Angina Pectoris; Blood Viscosity; Clinical Trials as Topic; Humans; Male; Middle Aged; Molsidomine; Nifedipine; Oxadiazoles; Propranolol; Sydnones; Vasodilator Agents

1985
Long-term treatment of patients with coronary heart disease using isosorbide dinitrate, nifedipine and molsidomine.
    Zeitschrift fur Kardiologie, 1983, Volume: 72 Suppl 3

    Topics: Adult; Blood Pressure; Coronary Disease; Drug Administration Schedule; Drug Tolerance; Hemodynamics; Humans; Isosorbide Dinitrate; Middle Aged; Molsidomine; Nifedipine; Oxadiazoles; Physical Exertion; Sydnones; Vasodilator Agents

1983

Other Studies

61 other study(ies) available for nifedipine and oxadiazoles

ArticleYear
Characterisation of the L- and N-type calcium channels in differentiated SH-SY5Y neuroblastoma cells: calcium imaging and single channel recording.
    Brain research. Molecular brain research, 1992, Volume: 13, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cadmium; Cadmium Chloride; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Differentiation; Cell Line; Cell Membrane; Chlorides; Evoked Potentials; Fura-2; Humans; Kinetics; Microscopy, Fluorescence; Neuroblastoma; Nicotinic Acids; Nifedipine; omega-Conotoxins; Oxadiazoles; Peptides, Cyclic; Potassium; Tretinoin

1992
Comparative behavioral, neurochemical and pharmacological activities of dihydropyridine calcium channel activating drugs.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcium Channel Agonists; Catecholamines; Chromatography, High Pressure Liquid; Dihydropyridines; Guinea Pigs; Injections, Intraperitoneal; Male; Mice; Motor Activity; Muscle Contraction; Muscle, Smooth; Nicotinic Acids; Nifedipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1990
(-)[3H]amlodipine binding to rat cardiac membranes.
    Journal of cardiovascular pharmacology, 1991, Volume: 17, Issue:4

    Topics: Amlodipine; Animals; Female; Gallopamil; Hydrogen-Ion Concentration; In Vitro Techniques; Isradipine; Kinetics; Membranes; Myocardium; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains; Stereoisomerism; Temperature

1991
Binding of [125I]iodipine to parathyroid cell membranes: evidence of a dihydropyridine-sensitive calcium channel.
    Endocrinology, 1990, Volume: 126, Issue:4

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Dihydropyridines; Iodine Radioisotopes; Iodobenzenes; Kinetics; Ligands; Nicotinic Acids; Nifedipine; Oxadiazoles; Parathyroid Glands; Stereoisomerism

1990
High and low affinity states of the dihydropyridine and phenylalkylamine receptors on the cardiac calcium channel and their interconversion by divalent cations.
    Biochemical and biophysical research communications, 1985, Jun-28, Volume: 129, Issue:3

    Topics: Animals; Calcium; Cations, Divalent; Chickens; Dihydropyridines; Heart; Ion Channels; Isradipine; Magnesium; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Pyridines; Receptors, Drug; Verapamil

1985
Dihydropyridine and peripheral type benzodiazepine binding sites: subcellular distribution and molecular size determination.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Fractionation; Dogs; Ion Channels; Isoquinolines; Isradipine; Male; Molecular Weight; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Nicotinic; Sarcolemma; Sarcoplasmic Reticulum; Verapamil

1985
Purified calcium channels have three allosterically coupled drug receptors.
    FEBS letters, 1986, Mar-03, Volume: 197, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Allosteric Regulation; Amines; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Diltiazem; Guinea Pigs; Ion Channels; Isradipine; Muscles; Nifedipine; Oxadiazoles; Pyridines; Receptors, Drug; Verapamil

1986
Dihydropyridine-sensitive Ca2+ channels in mammalian skeletal muscle cells in culture: electrophysiological properties and interactions with Ca2+ channel activator (Bay K8644) and inhibitor (PN 200-110).
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Cells, Cultured; Electric Conductivity; Ion Channels; Isradipine; Membrane Potentials; Muscles; Nifedipine; Oxadiazoles; Rats

1986
Depolarization-dependent binding of the calcium channel antagonist, (+)-[3H]PN200-110, to intact cultured PC12 cells.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Cells, Cultured; Isradipine; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Onium Compounds; Organophosphorus Compounds; Oxadiazoles; Potassium; Pyridines; Tritium

1986
Effects of dihydropyridines on tension and calcium-45 influx in isolated mesenteric resistance vessels from spontaneously hypertensive and normotensive rats.
    The American journal of cardiology, 1987, Jan-30, Volume: 59, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Radioisotopes; Female; Ion Channels; Isradipine; Mesenteric Arteries; Nifedipine; Nisoldipine; Norepinephrine; Oxadiazoles; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Vascular Resistance

1987
Inhibition of myocardial Ca2+ channels by three dihydropyridines with different structural features: potential-dependent blockade by Ro 18-3981.
    British journal of pharmacology, 1987, Volume: 91, Issue:1

    Topics: Animals; Calcium Channel Blockers; Dihydropyridines; Female; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Isradipine; Male; Membrane Potentials; Myocardial Contraction; Myocardium; Nifedipine; Oxadiazoles; Potassium; Pyridines

1987
Effect of daunorubicin on dihydropyridine-sensitive binding sites in cardiac sarcolemma.
    Biochemical pharmacology, 1987, Dec-15, Volume: 36, Issue:24

    Topics: Animals; Calcium; Cricetinae; Daunorubicin; Dihydropyridines; Female; In Vitro Techniques; Ion Channels; Isradipine; Male; Myocardial Contraction; Myocardium; Nifedipine; Oxadiazoles; Sarcolemma

1987
Pharmacologic relevance of dihydropyridine binding sites in membranes from rat aorta: kinetic and equilibrium studies.
    Circulation research, 1988, Volume: 62, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Binding, Competitive; Calcium; Calcium Channels; Ion Channels; Isradipine; Kinetics; Muscle, Smooth, Vascular; Nifedipine; Nisoldipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Stereoisomerism

1988
Calcium currents, charge movement and dihydropyridine binding in fast- and slow-twitch muscles of rat and rabbit.
    The Journal of physiology, 1987, Volume: 393

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; In Vitro Techniques; Ion Channels; Isradipine; Muscles; Nifedipine; Oxadiazoles; Rabbits; Rats; Time Factors

1987
Relationship of dihydropyridine binding sites with calcium-dependent neurotransmitter release in synaptosomes.
    Journal of neurochemistry, 1988, Volume: 51, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; gamma-Aminobutyric Acid; Ion Channels; Isradipine; Lanthanum; Male; Mice; Neurotransmitter Agents; Nifedipine; Nitrendipine; Oxadiazoles; Potassium; Receptors, Nicotinic; Ruthenium Red; Synaptosomes

1988
Calcium current in embryonic Xenopus muscle cells in culture.
    Canadian journal of physiology and pharmacology, 1989, Volume: 67, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Cells, Cultured; Embryo, Nonmammalian; Isradipine; Muscles; Nifedipine; Oxadiazoles; Xenopus

1989
Relaxation of potassium chloride-induced contractions by amlodipine and its interaction with the 1,4-dihydropyridine-binding site in pig coronary artery.
    The American journal of cardiology, 1989, Nov-07, Volume: 64, Issue:17

    Topics: Amlodipine; Animals; Binding Sites; Calcium Channel Blockers; Coronary Vessels; Dihydropyridines; Isradipine; Nifedipine; Oxadiazoles; Potassium Chloride; Sarcolemma; Stereoisomerism; Swine; Vasoconstriction; Vasodilation

1989
High affinity binding of the calcium channel blocker, (+)-[methyl-3H]PN200-110(3HPN) in rat brain.
    Physiology & behavior, 1989, Volume: 46, Issue:1

    Topics: Animals; Brain; Calcium Channel Blockers; Calcium Channels; Isradipine; Male; Nifedipine; Oxadiazoles; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Synaptosomes

1989
Molecular approach to the calcium channel.
    Advances in myocardiology, 1985, Volume: 5

    Topics: Animals; Benzothiazoles; Binding Sites; Brain; Calcium; Cattle; Chemical Phenomena; Chemistry; Diltiazem; Guinea Pigs; In Vitro Techniques; Ion Channels; Isradipine; Muscles; Myocardium; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Oxadiazoles; Thiazoles; Verapamil

1985
Selective modulation by membrane potential of the interaction of some calcium entry blockers with calcium channels in rat mesenteric artery.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Flunarizine; In Vitro Techniques; Isradipine; Membrane Potentials; Membranes; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1988
The effect of calcium-blockers nicardipine, darodipine, PN-200-110 and nifedipine on insulin release from isolated rat pancreatic islets.
    Acta physiologica Scandinavica, 1986, Volume: 126, Issue:2

    Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Isradipine; Male; Nicardipine; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1986
Suppression of rat carotid lesion development by the calcium channel blocker PN 200-110.
    The American journal of pathology, 1986, Volume: 124, Issue:1

    Topics: Angioplasty, Balloon; Animals; Arteriosclerosis; Blood Platelets; Blood Pressure; Carotid Arteries; Hypotension; Isradipine; Male; Muscle, Smooth, Vascular; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1986
Comparison of cardiodepressant and vasodilator effects of PN 200-110 (isradipine), nifedipine and diltiazem in anesthetized rabbits.
    The American journal of cardiology, 1987, Jan-30, Volume: 59, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Blood Pressure; Calcium Channel Blockers; Coronary Circulation; Diltiazem; Dose-Response Relationship, Drug; Heart; Isradipine; Myocardial Contraction; Nifedipine; Oxadiazoles; Rabbits; Vasodilation

1987
Failure of a new calcium-antagonist PN 200-110 and nifedipine to affect exercise stimulated GH-secretion in healthy volunteers.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1987, Volume: 19, Issue:6

    Topics: Adult; Calcium Channel Blockers; Growth Hormone; Humans; Isradipine; Male; Nifedipine; Oxadiazoles; Physical Exertion

1987
Nisoldepine inhibits formyl-methionyl-leucyl-phenylalanine (fMet-Leu-Phe) receptor-coupled calcium transport in human neutrophils.
    Journal of leukocyte biology, 1987, Volume: 42, Issue:3

    Topics: Adult; Biological Transport; Calcium; Calcium Channel Blockers; Humans; In Vitro Techniques; Isradipine; Neutrophils; Nifedipine; Nisoldipine; Oxadiazoles; Receptors, Formyl Peptide; Receptors, Immunologic

1987
Cardiovascular effects of two new calcium antagonists, PY 108-068 and PN 200-110, in conscious spontaneously hypertensive rats.
    British journal of pharmacology, 1988, Volume: 93, Issue:1

    Topics: Animals; Blood Pressure; Calcium Channel Blockers; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Isradipine; Male; Nifedipine; Nitroglycerin; Oxadiazoles; Phenylephrine; Pressoreceptors; Rats; Rats, Inbred SHR; Reflex

1988
Dihydropyridine [methyl-3H]PN 200-110 binding and myogenesis in intact muscle cells in vitro.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Aminoquinolines; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Chick Embryo; Isradipine; Kinetics; Muscles; Nifedipine; Nitrendipine; Oxadiazoles; Receptors, Nicotinic

1986
The mechanism of binding of dihydropyridine calcium channel blockers to rat brain membranes.
    The Journal of biological chemistry, 1985, Jul-15, Volume: 260, Issue:14

    Topics: Animals; Brain; Calcium Channel Blockers; Isomerism; Isradipine; Kinetics; Mathematics; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Time Factors

1985
Non-pharmacological effects of the use of microelectrophoresis and pressure ejection of drugs in combination.
    Journal of neuroscience methods, 1987, Volume: 20, Issue:3

    Topics: Amino Acids; Animals; Aspartic Acid; Electrophoresis; Ibotenic Acid; Kainic Acid; Microelectrodes; N-Methylaspartate; Neurons; Nifedipine; Oxadiazoles; Quisqualic Acid; Rats; Spinal Cord

1987
[Effect of molsidomin and nifedipine on tolerance of physical exertion among rheumatic fever patients in the initial stage of heart failure].
    Vrachebnoe delo, 1986, Issue:1

    Topics: Adult; Female; Heart Failure; Heart Valve Diseases; Humans; Male; Middle Aged; Molsidomine; Nifedipine; Oxadiazoles; Rheumatic Heart Disease; Sydnones; Vasodilator Agents

1986
[Effectiveness of treating stenocardia patients with obzidan, corvaton and corinfar based on the indices of spirometric bicycle ergometry and of central hemodynamics].
    Vrachebnoe delo, 1985, Issue:8

    Topics: Adult; Angina Pectoris; Drug Evaluation; Exercise Test; Hemodynamics; Humans; Male; Middle Aged; Molsidomine; Nifedipine; Oxadiazoles; Propranolol; Spirometry; Sydnones; Vasodilator Agents

1985
High affinity specific [3H](+)PN 200-110 binding to dihydropyridine receptors associated with calcium channels in rat cerebral cortex and heart.
    Life sciences, 1984, Aug-13, Volume: 35, Issue:7

    Topics: Animals; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Ion Channels; Isradipine; Kinetics; Male; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic

1984
The interaction of [3H]PY 108-068 and of [3H]PN 200-110 with calcium channel binding sites in rat brain.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Brain; In Vitro Techniques; Ion Channels; Isradipine; Kinetics; Male; Membranes; Molecular Conformation; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1984
In vitro effects of calcium antagonists PN 200-110, nifedipine, and nimodipine on human and canine cerebral arteries.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1983, Volume: 3, Issue:3

    Topics: Animals; Basilar Artery; Blood Physiological Phenomena; Calcium Channel Blockers; Cerebral Arteries; Dogs; Humans; In Vitro Techniques; Isradipine; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nicotinic Acids; Nifedipine; Nimodipine; Oxadiazoles; Serotonin; Vasoconstriction

1983
Calcium antagonist binding sites in the rat brain: quantitative autoradiographic mapping using the 1,4-dihydropyridines [3H]PN 200-110 and [3H]PY 108-068.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Autoradiography; Binding Sites; Brain; Calcium Channel Blockers; Isradipine; Male; Nifedipine; Oxadiazoles; Rats; Rats, Inbred Strains

1984
Differential labelling of putative skeletal muscle calcium channels by [3H]-nifedipine, [3H]-nitrendipine, [3H]-nimodipine and [3H]-PN 200 110.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 323, Issue:3

    Topics: Animals; Calcium Channel Blockers; Guinea Pigs; In Vitro Techniques; Ion Channels; Isradipine; Kinetics; Muscles; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Oxadiazoles

1983
[Molsidomine in exertion angina].
    Annales de cardiologie et d'angeiologie, 1983, Volume: 32, Issue:8

    Topics: Angina Pectoris; Exercise Test; Hemodynamics; Humans; Isosorbide Dinitrate; Molsidomine; Nifedipine; Oxadiazoles; Sydnones

1983
Differences in the effects of ketanserin and GR127935 on 5-HT-receptor mediated responses in rabbit saphenous vein and guinea-pig jugular vein.
    European journal of pharmacology, 1995, Sep-05, Volume: 283, Issue:1-3

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Jugular Veins; Ketanserin; Male; Myenteric Plexus; Nifedipine; Oxadiazoles; Piperazines; Rabbits; Saphenous Vein; Serotonin; Serotonin Antagonists; Sumatriptan

1995
Calcium channels in vitamin B6 deficiency-induced hypertension.
    Journal of hypertension, 1993, Volume: 11, Issue:12

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Pressure; Calcium Channel Blockers; Calcium Channels; Diltiazem; Hypertension; Male; Nicotinic Acids; Nifedipine; Oxadiazoles; Rats; Rats, Sprague-Dawley; Verapamil; Vitamin B 6 Deficiency

1993
Role of calcium channels in parathyroid hormone secretion.
    Bone, 1995, Volume: 16, Issue:4 Suppl

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cattle; Cyclic AMP; Electrophoresis, Polyacrylamide Gel; Ionomycin; Isotope Labeling; Nicotinic Acids; Nifedipine; Oxadiazoles; Parathyroid Glands; Parathyroid Hormone; Pertussis Toxin; Phosphorylation; Potassium; Radioimmunoassay; Stereoisomerism; Verapamil; Virulence Factors, Bordetella

1995
Residual inhibition in density of [3H]isradipine binding sites in rat brain membrane pretreated with amlodipine.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1995, Volume: 16, Issue:4

    Topics: Amlodipine; Animals; Binding Sites; Brain; Calcium Channel Blockers; Dihydropyridines; Isradipine; Male; Nifedipine; Oxadiazoles; Radioligand Assay; Rats; Rats, Wistar

1995
Potassium channel openers relax A23187-induced nifedipine-resistant contraction of rat aorta.
    Journal of cardiovascular pharmacology, 1994, Volume: 24, Issue:6

    Topics: Animals; Aorta; Benzopyrans; Calcimycin; Cromakalim; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Nifedipine; Oxadiazoles; Piperidines; Pyrroles; Rats; Rats, Wistar; Vasoconstriction; Vasodilator Agents

1994
Direct effect of calcium channel antagonists on osteoclast function: alterations in bone resorption and intracellular calcium concentrations.
    Endocrinology, 1994, Volume: 135, Issue:3

    Topics: Animals; Bone Resorption; Calcium; Calcium Channel Blockers; Cells, Cultured; Intracellular Membranes; Isomerism; Isradipine; Nicotinic Acids; Nifedipine; Osmolar Concentration; Osteoclasts; Oxadiazoles; Rats; Whales

1994
NIP-121 is more effective than nifedipine in acutely reversing chronic pulmonary hypertension.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 75, Issue:3

    Topics: Altitude; Animals; Chronic Disease; Glyburide; Hemodynamics; Hypertension, Pulmonary; Hypoxia; Male; Nifedipine; Oxadiazoles; Piperidines; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasodilation

1993
Pharmacochemistry of the furoxan ring: recent developments.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:2

    Topics: Animals; Blood Platelets; Calcium Channel Blockers; Cyclic GMP; Guinea Pigs; Heart Rate; Humans; In Vitro Techniques; Myocardial Contraction; Nifedipine; Oxadiazoles; Platelet Aggregation Inhibitors; Prazosin; Vasodilator Agents

1993
L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other.
    Biochemistry, 1997, Mar-25, Volume: 36, Issue:12

    Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Fluorescent Dyes; Isomerism; Isradipine; Kinetics; Nicotinic Acids; Nifedipine; Nitrendipine; Oxadiazoles; Rabbits

1997
Evidence that NO acts as a redundant NANC inhibitory neurotransmitter in the guinea-pig isolated taenia coli.
    British journal of pharmacology, 1997, Volume: 121, Issue:3

    Topics: Adenosine Triphosphate; Animals; Apamin; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Intestines; Male; Neurotransmitter Agents; Nifedipine; Nitric Oxide; Nitroarginine; Nitroprusside; Oxadiazoles; Oxyhemoglobins; Quinoxalines

1997
New 1,4-dihydropyridines conjugated to furoxanyl moieties, endowed with both nitric oxide-like and calcium channel antagonist vasodilator activities.
    Journal of medicinal chemistry, 1998, Dec-31, Volume: 41, Issue:27

    Topics: Animals; Aorta, Thoracic; Binding, Competitive; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Male; Methylene Blue; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitric Oxide Donors; Oxadiazoles; Quinoxalines; Radioligand Assay; Rats; Rats, Wistar; Structure-Activity Relationship; Vasodilator Agents

1998
Nitrergic relaxation of the mouse gastric fundus is mediated by cyclic GMP-dependent and ryanodine-sensitive mechanisms.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine Triphosphate; Animals; Caffeine; Calcium Channel Blockers; Cyclic GMP; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Gastric Fundus; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Muscle Relaxation; Muscle, Smooth; Nifedipine; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Nitroprusside; Oxadiazoles; Quinoxalines; Ryanodine

2000
Nitric oxide and sodium nitroprusside-induced relaxation of the human umbilical artery.
    British journal of pharmacology, 2000, Volume: 131, Issue:3

    Topics: Calcium Channels; Cyclic GMP; Enzyme Inhibitors; Guanylate Cyclase; Humans; In Vitro Techniques; Nifedipine; Nitric Oxide; Nitroprusside; Oxadiazoles; Oxygen; Potassium; Potassium Channel Blockers; Potassium Channels; Quinoxalines; Receptors, Atrial Natriuretic Factor; Umbilical Arteries; Vasodilation; Vasodilator Agents

2000
Activation of purified cardiac ryanodine receptors by dihydropyridine agonists.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; Dogs; Membrane Potentials; Myocardium; Nicotinic Acids; Nifedipine; Oxadiazoles; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Stereoisomerism

2001
Actions of NO donors and endogenous nitrergic transmitter on the longitudinal muscle of rat ileum in vitro: mechanisms involved.
    Life sciences, 2001, Jul-27, Volume: 69, Issue:10

    Topics: Animals; Apamin; Atropine; Calcium Channels; Charybdotoxin; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ileum; Molsidomine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Nitric Oxide; Nitroprusside; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Tetrodotoxin

2001
Nitric oxide contracts longitudinal smooth muscle of opossum oesophagus via excitation-contraction coupling.
    The Journal of physiology, 2001, Oct-01, Volume: 536, Issue:Pt 1

    Topics: Anesthetics, Local; Animals; Calcium Channel Blockers; Cyclic GMP; Enzyme Inhibitors; Esophagus; Female; In Vitro Techniques; Isometric Contraction; Male; Microelectrodes; Muscle, Smooth; Nifedipine; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Opossums; Oxadiazoles; Quinoxalines; Signal Transduction; Tetrodotoxin; Triazenes

2001
Electrical activity induced by nitric oxide in canine colonic circular muscle.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Colon; Dogs; Electric Conductivity; Enteric Nervous System; Enzyme Inhibitors; Female; Gastrointestinal Motility; In Vitro Techniques; Indoles; Male; Membrane Potentials; Mitochondria; Muscle, Smooth; Nickel; Nifedipine; Nitric Oxide; Nitric Oxide Donors; Nitroarginine; Nitroprusside; Oxadiazoles; Potassium; Quinoxalines; Uncoupling Agents

2002
Role of sarcoplasmic reticulum in control of membrane potential and nitrergic response in opossum lower esophageal sphincter.
    British journal of pharmacology, 2003, Volume: 140, Issue:6

    Topics: Animals; Anthracenes; Atropine; Azepines; Caffeine; Calcium; Chloride Channels; Enzyme Inhibitors; Esophagogastric Junction; Female; Guanethidine; In Vitro Techniques; Indoles; Male; Membrane Potentials; Muscle, Smooth; Myosin-Light-Chain Kinase; Nifedipine; Niflumic Acid; Nitric Oxide; Opossums; Oxadiazoles; Quinoxalines; Ryanodine; Sarcoplasmic Reticulum; Substance P; Tetraethylammonium

2003
Role of the nitric oxide/cyclic GMP pathway and ascorbic acid in 3-morpholinosydnonimine (SIN-1)-induced increases in dopamine secretion from PC12 cells. A microdialysis in vitro study.
    Neuroscience letters, 2003, Dec-15, Volume: 353, Issue:1

    Topics: Animals; Antioxidants; Ascorbic Acid; Calcium; Calcium Channel Blockers; Cyclic GMP; Dialysis; Dopamine; Drug Interactions; In Vitro Techniques; Molsidomine; Nifedipine; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; PC12 Cells; Potassium; Rats; Signal Transduction; Time Factors

2003
Evidence for the mechanisms underlying the effects of pimaradienoic acid isolated from the roots of Viguiera arenaria on rat aorta.
    Pharmacology, 2004, Volume: 70, Issue:1

    Topics: Animals; Aorta, Thoracic; Asteraceae; Brazil; Diterpenes; Dose-Response Relationship, Drug; Endothelium, Vascular; Ethanol; Indomethacin; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nifedipine; Oxadiazoles; Phenylephrine; Plant Extracts; Plant Roots; Quinoxalines; Rats; Rats, Wistar; Tetraethylammonium; Vasoconstriction; Vasodilation

2004
The nitroxyl anion (HNO) is a potent dilator of rat coronary vasculature.
    Cardiovascular research, 2007, Feb-01, Volume: 73, Issue:3

    Topics: Acetylcholine; Animals; Anions; Antioxidants; Calcitonin Gene-Related Peptide; Coronary Vessels; Dose-Response Relationship, Drug; Guanylate Cyclase; Heart Rate; Isoproterenol; Male; Myocardial Contraction; Nifedipine; Nitrites; Nitrogen Oxides; Oxadiazoles; Oxidation-Reduction; Peptide Fragments; Perfusion; Potassium; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium Nitrite; Vasodilation

2007
Pharmacological evidence that Ca²+ channels and, to a lesser extent, K+ channels mediate the relaxation of testosterone in the canine basilar artery.
    Steroids, 2011, Volume: 76, Issue:4

    Topics: 4-Aminopyridine; Adenine; Aminoglutethimide; Androgen Receptor Antagonists; Animals; Aromatase Inhibitors; Barium Compounds; Basilar Artery; Calcium Channel Blockers; Calcium Channels; Chlorides; Cycloheximide; Dactinomycin; Dogs; Enzyme Inhibitors; Flutamide; In Vitro Techniques; Male; Nifedipine; Nucleic Acid Synthesis Inhibitors; Oxadiazoles; Potassium Channel Blockers; Potassium Channels; Protein Synthesis Inhibitors; Quinoxalines; Testosterone; Vasodilation; Vasodilator Agents

2011
Calcium inhibits dihydropyridine-stimulated increases in opening and unitary conductance of a plant Ca²+ channel.
    The Journal of membrane biology, 2011, Volume: 240, Issue:1

    Topics: Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Dihydropyridines; Lipid Bilayers; Membrane Potentials; Membranes, Artificial; Nicotinic Acids; Nifedipine; Oxadiazoles; Plant Roots; Triticum

2011
S-nitrosothiols dilate the mesenteric artery more potently than the femoral artery by a cGMP and L-type calcium channel-dependent mechanism.
    Nitric oxide : biology and chemistry, 2016, 08-31, Volume: 58

    Topics: Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Cyclic GMP; Cysteine; Diltiazem; Female; Femoral Artery; Fetus; Indazoles; Male; Mesenteric Arteries; Nifedipine; Oxadiazoles; Quinoxalines; S-Nitrosoglutathione; S-Nitrosothiols; Sheep; Soluble Guanylyl Cyclase; Vasodilation; Vasodilator Agents

2016