Page last updated: 2024-08-26

nicotine and varenicline

nicotine has been researched along with varenicline in 364 studies

Research

Studies (364)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's81 (22.25)29.6817
2010's234 (64.29)24.3611
2020's49 (13.46)2.80

Authors

AuthorsStudies
Arnold, EP; Bashore, CG; Bianco, KE; Brooks, PR; Coe, JW; Davis, TI; Fox, CB; Lebel, LA; Mansbach, RS; O'Neill, BT; Rollema, H; Sands, SB; Schulz, DW; Tingley, FD; Vetelino, MG; Wirtz, MC1
Brieaddy, LE; Burgess, JP; Damaj, MI; Ivy Carroll, F; Lee, JR; Ma, W; Martin, BR; Navarro, HA; Yokota, Y1
Carroll, FI; Damaj, MI; Deng, L; Ma, W; Martin, BR; Navarro, HA1
Coe, JW; DeNinno, SL; Ellerbrock, B; Gorczyca, R; Horner, W; Hurst, RS; Johnson, DE; Kozak, R; Lowe, JA; MacDougall, MC; Majchrzak, MJ; Mather, RJ; McDowell, LL; Mente, S; Osgood, SM; Rollema, H; Sadlier, J; Shaffer, CL; Shrikhande, A; Tingley, FD; Tritto, T; Ward, KM; Zhang, L1
Binda, M; Bolchi, C; Fumagalli, L; Gotti, C; Pallavicini, M; Pistillo, F; Pucci, L; Valoti, E; Vistoli, G1
Brunner, D; Caldarone, B; Eaton, JB; Fedolak, A; Hanania, T; Kozikowski, AP; Lukas, RJ; Tückmantel, W; Yu, LF1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Bertrand, D; Bertrand, S; Bréthous, L; Garcia-Delgado, N; Reymond, JL; Schwartz, J1
Benson, LR; Bhatti, BS; Breining, SR; Byrd, GD; Fedorov, NB; Hepler, CD; Hooker, DN; Kiser, MN; Lucero, LM; Lukas, RJ; Melvin, M; Mitchener, JP; Reynolds, LA; Sidach, SS; Whiteaker, P; Yohannes, D; Zhang, J1
Brunner, D; Eaton, JB; Fedolak, A; Hanania, T; Kozikowski, AP; Lukas, RJ; Yu, LF; Zhang, HK1
Al-Muhtasib, N; Brown, ML; Kellar, KJ; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Richardson, J; Sahibzada, N; Sexton, HG; Tran, T; Xiao, Y; Xie, T; Yenugonda, VM1
Al-Muhtasib, N; Brown, ML; Dakshanamurthy, S; Johnson, JE; Kellar, KJ; Kong, HS; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Sahibzada, N; Slade, S; Tomita, Y; Tran, T; Wells, C; Xiao, Y; Xie, T; Yenugonda, VM1
Bartkowiak, JM; Carroll, FI; Castro, AH; Damaj, MI; Luetje, CW; Mascarella, SW; Navarro, HA; Ondachi, PW1
Brunner, D; Caldarone, BJ; Eaton, JB; Kozikowski, AP; Lukas, RJ; Onajole, OK; Thiede, L1
Carroll, FI; Castro, AH; Damaj, MI; Luetje, CW; Mascarella, SW; Navarro, HA; Ondachi, PW; Ye, Z1
Camarelles Guillem, F1
Corelli, RL; Hudmon, KS1
Burstein, AH; Clark, DJ; Faessel, HM; Gibbs, MA; Rohrbacher, K; Stolar, M1
Mogg, A; Peacey, E; Pullar, IA; Smith, JW; Szekeres, P; Tafi, E; Tricklebank, M1
Dimoulas, P; Mills, EJ; Wilson, K; Wu, P1
Chambers, LK; Coe, JW; Glowa, J; Hurst, RS; Lebel, LA; Lu, Y; Mansbach, RS; Mather, RJ; Rollema, H; Rovetti, CC; Sands, SB; Schaeffer, E; Schulz, DW; Tingley, FD; Williams, KE1
Siu, EC; Tyndale, RF1
Cahill, K; Lancaster, T; Stead, LF5
Frishman, WH1
Oberpichler-Schwenk, H1
Crane, R1
Garwood, CL; Potts, LA1
Freedman, R1
Croghan, E1
Lerman, C; Patterson, F; Schnoll, RA1
Doggrell, SA1
Hoogendoorn, M; Rutten-van Mölken, MP; Welsing, P1
George, TP; Le Foll, B1
Milbrandt, A; Ratcliffe, M; Smith, R; Spirling, LI; Stapleton, JA; Sutherland, G; Watson, L1
Cohen, AF; Dubois, EA; van Bronswijk, H; Zitman, FG1
Andrews, JO; Bennett, SM; Heath, JH1
Cahill, K; Lancaster, T; Stead, L2
Baker, CL; Bushmakin, AG; Cappelleri, JC; West, R1
Cooley, ME; Murphy, M; Sarna, L; Sipples, RL1
Aubin, HJ; Billing, CB; Bobak, A; Britton, JR; Gong, J; Oncken, C; Reeves, KR; Williams, KE1
Benowitz, NL2
Stapleton, JA1
Wonnacott, S1
Crawford, JT; Goldenberg, RL; Tolosa, JE1
Brees, DJ; Cai, JH; Elwell, MR; Finkelstein, MB; Jakowski, AB; Sands, SB; Shen, AC; Tingley, FD1
Baker, C; Boler, A; Howard, P; Knight, C1
Bölcskei, PL; Walden, K1
Tønnesen, P2
Bélisle, P; Eisenberg, MJ; Filion, KB; Gervais, A; Joseph, L; Mottillo, S; O'Loughlin, J; Paradis, G; Pilote, L; Rinfret, S; Yavin, D1
Rose, JE2
Bhowmik, A; Hillman, T; Rajakulasingam, K1
Ferguson, SG; Shiffman, S1
Reus, VI; Smith, BJ1
Filip, M; McCreary, AC; Przegaliński, E; Stefański, R; Zaniewska, M1
Carroll, FI; Corrigall, WA; LeSage, MG; Ross, JT; Shelley, D1
Bader, P; McDonald, P; Selby, P1
Hering, T2
Schunack, W1
Brace, V; Danielian, P; Rore, C; Williams, D1
Ebbert, JO; Hays, JT2
Bardo, MT; Crooks, PA; Dwoskin, LP; Joyce, BM; Neugebauer, NM; Pivavarchyk, M; Zhang, Z; Zheng, G1
Peiffer, G1
Ericson, M; Löf, E; Söderpalm, B; Stomberg, R1
McEwen, A; West, R1
Aveyard, P; Hajek, P; Inglis, J; Parsons, AC; Shraim, M1
Einarson, A; Riordan, S1
Florek, E; Piekoszewski, W1
Arora, G; Jain, M; Talwar, A1
Cornwell, J; Davis, JM; Gupta, S; Lajtha, A; Lindenmayer, JP; Noth, K; Sershen, H; Smith, RC1
Ebbert, JO1
Burke, MV; Ebbert, JO; Hays, JT; Hurt, RD1
Ferguson, SG; Gritz, ER; Henningfield, JE; Shiffman, S1
Ashby, CR; Callahan, PM; Gardner, EL; Li, X; Spiller, K; Tehim, A; Xi, ZX1
Cryan, JF; Flynn, RA; Glynn, DA; Kennedy, MP; Kent, P1
Laniado-Laborín, R2
George, TP; Lising-Enriquez, K1
Bau, CH; Bizarro, L; Dobler, CJ; Kortmann, GL1
Heimlich, L; Steinberg, ML; Williams, JM1
Aubin, HJ; Benhaddi, H; Bolin, K; de Nigris, E; Marbaix, S; Mork, AC; Wilson, K1
Deissenrieder, F; Groneberg, D; Kusma, B; Mache, S; Quarcoo, D; Welte, T1
Keiding, H1
Herman, AI; Mooney, M; Sofuoglu, M; Waters, AJ1
Maritz, GS1
Annemans, L; Bartsch, P; Marbaix, S; Nackaerts, K; Prignot, J1
Kranzler, HR; Oncken, CA1
Tonstad, S1
Davies, C; Gunnell, D; Irvine, D; Martin, RM; Wise, L1
Dufour, E; Gardier, AM; Maskos, U; Pons, S; Reperant, C; Rollema, H1
Batra, A; Friederich, HM1
Mead, AN; O'Connor, EC; Parker, D; Rollema, H1
Corelli, RL; Hudmon, KS; Prokhorov, AV1
Keating, GM; Lyseng-Williamson, KA1
Noda, K; Saku, K; Tsukahara, H1
Biala, G; Budzynska, B; Staniak, N1
Barr, JD; Bevins, RA; Murray, JE; Reichel, CM1
Costa, E; Davis, JM; Guidotti, A; Lajtha, A; Maloku, E; Sershen, H; Smith, RC; Zhubi, A1
Ainamo, A; Binnie, VI; Carr, AB; Fundak, A; Koeber, A; Koerber, A; Needleman, IG; Ohrn, K; Rosseel, J1
Beck, HN; Biazzo, LL; Campbell, SL; Froshaug, DB; Harwell, TS; Haugland, C; Helgerson, SD1
Frey, JM; Jepson, C; Lerman, C; Patterson, F; Phillips, JM; Rudnick, ND; Siegel, SJ; Strasser, AA; Turetsky, BI1
Blendy, JA; Castellano, LM; Turner, JR2
Biala, G; Staniak, N1
Hizue, M; Ishibashi, T; Nomura, S1
Bhat, A; Crain, D1
Chengappa, KN; Fonte, CA; Jain, A; Lerman, C; Mercincavage, M; Perkins, KA; Stitzer, ML1
Ioannides-Demos, LL; McNeil, JJ; Piccenna, L1
Lund, KE; McNeill, A; Scheffels, J1
Herman, AI; Sofuoglu, M1
Ruff, P1
Zeller, A1
von Garnier, C1
Ayesta Ayesta, FJ; Minué Lorenzo, C; Olano Espinosa, E1
Carroll, FI; Damaj, MI; George, O; Koob, GF; Lloyd, A1
Bover, MT; Foulds, J; Richardson, DL; Schmelzer, AC; Steinberg, MB; Williams, JM1
Gnegy, ME; Jutkiewicz, EM; Kim, MN; Zhang, M1
Johnson, TS1
Cesario, A; Galetta, D; Granone, P; Greenberg, DS; Margaritora, S; Russo, P; Rutella, S; Spaggiari, L; Veronesi, G1
Balmford, J; Borland, R; Cummings, KM; Hammond, D1
Cunningham, CS; McMahon, LR2
Weinsier, ST1
Al Rubaiy, SA; Bloom, SA; Guendisch, D; Papke, RL; Trocmé-Thibierge, C1
Ebbert, J; Erwin, PJ; Montori, VM; Stead, LF1
De Vries, TJ; De Vries, W; Pattij, T; Riga, D; Schetters, D; Schoffelmeer, AN; Stegeman, M; van Mourik, Y; Wouda, JA1
Grief, SN1
Dong, E; Guidotti, A; Kadriu, B; Maloku, E; Pibiri, F; Satta, R; Zhubi, A1
Díaz Cerezo, S; Martí Sánchez, B; Navarro Artieda, R; Sanz De Burgoa, V; Sicras Mainar, A1
Bartlett, SE; Bito-Onon, JJ; Chatterjee, S; Holgate, J; Simms, JA1
Coleman, T; Huang, Y; Langley, TE; Lewis, S; McNeill, A; Szatkowski, L1
Gur, RC; Lerman, C; Loughead, J; O'Donnell, GP; Ray, R; Ruparel, K; Senecal, N; Siegel, S; Wileyto, EP1
Simon, JA1
Aubin, HJ; Karila, L; Reynaud, M1
Bircher, R; Chen, W; DiFranza, JR; Heffernan, M; Huang, W; King, J; Rane, P; Shields, J1
Agboola, S; Coleman, T; Leonardi-Bee, J; McNeill, A; Taylor, M1
Coleman, T; Lewis, S; McNeill, A; Szatkowski, L1
Foulds, J; Gandhi, KK; Steinberg, MB; Steinberg, ML; Ulpe, R; Williams, JM1
Belcon, AL1
Marti, J1
Brooks, EA; Jutkiewicz, EM; Kynaston, AD; Rice, KC; Woods, JH1
Czoty, PW; Gould, RW; Nader, MA; Nader, SH1
Kadokura, Y; Kano, M; Kushihashi, Y; Saito, H; Shino, M; Suzaki, H; Suzuki, M; Takiguchi, S; Yamada, Y1
Barnes, C; Chakraborty-Chatterjee, M; Gamaleddin, I; Goldberg, SR; Khaled, M; Le Foll, B; Lev-Ran, S; Pushparaj, A; Yan, Y1
Baker, TB; Fiore, MC1
Caggiula, AR; Donny, EC; Levin, ME; Palmatier, MI; Sved, AF; Weaver, MT1
Ansermot, N; Choong, E; Cornuz, J; Dobrinas, M; Eap, CB; Noetzli, M1
Furberg, CD; Glenmullen, J; Maltsberger, JT; Moore, TJ; Singh, S1
Grady, SR; Marks, MJ; O'Neill, HC; Ortiz, NC1
Ammerman, S; Bailey, SR; Crew, EE; Killen, JD; Riske, EC; Robinson, TN1
Schuurmans, MM; Zellweger, JP1
Azar, MR; Cohen, A; Fox, BS; George, O; Goeders, NE; Koob, GF1
Cunningham, CS; Javors, MA; McMahon, LR1
Etter, JF; Schneider, NG1
Bordia, T; Chin, M; Hrachova, M; McIntosh, JM; Quik, M1
Gallagher, T; Haseler, CA; Rucktooa, P; Sixma, TK; Smit, AB; van Elk, R1
Papke, RL; Stokes, C1
Browning, KK; Diaz, P; Ferketich, AK; Koletar, SL; Lu, B; Reynolds, NR; Wewers, ME1
Ashare, RL; Blair, IA; Leone, F; Mesaros, AC; Strasser, AA; Tang, KZ1
Akk, G; Esch, C; Herder, P; Laughlin, JR; Li, P; Stitzel, JA; Tammimäki, A1
Blendy, JA; Cousins, V; Hussmann, GP; Kellar, KJ; Levin, ED; Lomazzo, E; Perry, DC; Rezvani, AH; Turner, JR; Venkatesh, R; Wolfe, BB; Xiao, Y; Yasuda, RP1
Garg, PK; Garg, S; Gould, RW; Nader, MA1
Holloway, AC; Nicholson, CJ; Raha, S; Woynillowicz, AK1
Mikkelsen, K; Tønnesen, P1
Anthony, JC; Behm, FM; Eaton, WW; Fisher, C; Ialongo, N; Musci, R; Rose, JE; Storr, CL; Uhl, GR; Walther, D1
Almgren, MM; Clark, KJ; Stroman, RT; Wynn, WP1
Biała, G; Budzyńska, B; Kruk-Słomka, M1
Baker, TB; Benowitz, NL; Bergen, AW; Conti, DV; Edlund, CK; Hall, S; Javitz, HS; Krasnow, R; Kwok, PY; Lee, W; Lerman, C; Liu, J; Michel, M; Nishita, D; Swan, GE; Tyndale, RF1
Dixon-McDougall, T; Nowak, C; Pereira, S; Qian, C; Sellings, L; Tyndale, RF; van der Kooy, D; Zhao, B1
Damborsky, JC; DuBois, DW; Fincher, AS; Frye, GD; Winzer-Serhan, UH1
Milnerowicz, H; Sliwińska-Mossoń, M; Zieleń, I1
Porwal, M; Tsoi, DT; Webster, AC1
Carroll, AJ; Hong, LE; Ross, TJ; Salmeron, BJ; Stein, EA; Sutherland, MT1
Brown, VL; Cinciripini, PM; Engelmann, JM; Karam-Hage, M; Lam, C; Minnix, JA; Robinson, JD; Versace, F; Wetter, DW1
Blendy, JA; Carlson, GC; Gould, TJ; Poole, RL; Turner, JR; Wilkinson, DS1
Berg, A; Foulds, J; Franzon, M; Galaznik, A; Hughes, JR; Russ, C; Yu, CR; Zou, KH1
Antilla, JC; Bickford, PC; Engberg, ME; Hudson, CE; Kang, CW; Lambert, CS; Philpot, RM; Rowell, PP; Wecker, L; Zesiewicz, TA1
Fagerström, KO; Jiménez-Ruiz, CA1
Brasic, JR; Chamroonrat, W; Dannals, RF; Gao, Y; Gean, EG; Horti, AG; Kim, J; Kuwabara, H; Mathur, A; McCaul, ME; Valentine, H; Wand, G; Willis, W; Wong, DF1
Brown, J; Kotz, D; West, R2
Hajek, P; Hartmann-Boyce, J; Jarvis, M; Lancaster, T; Stead, LF; West, R1
Alexander, JC; Bruijnzeel, AW; Igari, M; Ji, Y; Papke, RL; Qi, X1
Kaakkola, S; Tuominen, R1
Dow, WH; Rungruanghiranya, S; White, JS1
Checa-Andrés, MD; Esparza-Martín, N; García-Cantón, C; Guerra-Rodríguez, R; Ramírez-Puga, A; Suria-González, S1
Goutier, W; Kloeze, MB; McCreary, AC1
Carroll, FI; Fivel, PA; Kohut, SJ; Mello, NK1
Eapen, S; Mills, EJ; Prochaska, JJ; Thorlund, K; Wu, P1
Bertrand, D; Hurst, RS; Lee, TC; Rollema, H; Russ, C1
Blendy, JA; DeDominicis, KE; Forcelli, PA; Hussmann, GP; Kellar, KJ; Klehm, J; Lindstrom, J; Richardson, JR; Sahibzada, N; Turner, JR; Wolfe, BB; Xiao, Y; Yasuda, RP1
Gupta, T; Jain, R; Majumder, P1
Cieślewicz, A; Jabłecka, A; Korzeniowska, K1
Daughton, DM; Rennard, SI1
Buyukuysal, S; Coskun, AS; Goktalay, G; Goktalay, T; Kayir, H; Uslu, G; Uzbay, T; Yorgancioglu, A1
Ebbert, JO; Elrashidi, MY1
Argue, DP; Cousin, MA; Ebbert, JO; Ekker, SC; Klee, EW; Urban, MD; Wiinamaki, AR1
Møller, AM; Thomsen, T; Villebro, N1
Andrea, D; Braida, D; Cannazza, G; Clementi, F; Fasoli, F; Gotti, C; Manfredi, I; Papke, RL; Ponzoni, L; Pucci, L; Sala, M; Stokes, C1
Arteaga, C; Brosky, G; Oh, P; Ranger, S; Raymond, V; Selby, P1
Abdool-Gaffar, MS; Bateman, ED; Bruning, A; Emanuel, S; Esterhuizen, TM; Irusen, EM; Koegelenberg, CF; Noor, F; O'Brien, JA; Smith, C; van Zyl-Smit, RN1
Kuryatov, A; Ley, CK; Lindstrom, JM; Wang, J1
Faessel, HM; Gastonguay, MR; Lee, TC; Niaura, R; Ravva, P1
Caggiula, AR; Donny, EC; Levin, ME; Palmatier, MI; Schassburger, RL; Sved, AF; Weaver, MT1
Fisher, DC; Fletcher, PJ; Guy, EG; Higgins, GA1
Baena, A; Masuet-Aumatell, C; Morchon, S; Ramon, JM1
Steurer, J1
Abe, S; Imaizumi, S; Kawachi, E; Matsuo, Y; Miura, S; Noda, K; Saku, K; Shimizu, T; Suematsu, Y; Takata, K; Tsukahara, H; Uehara, Y; Yahiro, E; Zhang, B1
Hogarth, L; Panlilio, LV; Shoaib, M1
Ciccocioppo, R; Cippitelli, A; Gaiolini, KA; Gorman, M; Khroyan, TV; Mercatelli, D; Pascual, C; Ramirez, A; Schoch, J; Toll, L; Wu, J; Xie, XS; Yasuda, D; Zaveri, NT1
Davies, NM; Munafò, MR; Ware, JJ1
Benowitz, NL; Cinciripini, P; George, TP; Hawk, LW; Heitjan, DF; Lerman, C; Schnoll, RA; Swan, GE; Tyndale, RF; Wileyto, EP1
Hall, BJ; Levin, ED; Rose, JE; Slade, S; Wells, C1
Bergman, J; Desai, RI1
Fedota, JR; Hong, LE; Ross, TJ; Salmeron, BJ; Stein, EA; Sutherland, MT1
Baker, NL; Carpenter, MJ; Gray, KM; Hartwell, KJ; McClure, EA; Ramakrishnan, V; Saladin, ME1
Borland, R; Brady, K; Carpenter, MJ; Cummings, KM; Fong, GT; Hartwell, K; Hyland, A; Kasza, KA; McKee, SA; Smith, PH1
Chang, Q; Hanania, T; Maillet, EL; Mash, DC1
Chenoweth, MJ; Cinciripini, PM; George, TP; Hawk, LW; Lerman, C; Novalen, M; Schnoll, RA; Tyndale, RF1
Butt, CM; Grady, SR; Marks, MJ; McIntosh, JM; O'Neill, HC; Ortiz, NC; Short, CA; Simmons, EE; Wynalda-Camozzi, KM1
Tashkin, DP1
He, Y; Sun, S; Wu, L; Zeng, J1
Benowitz, NL; Prochaska, JJ1
Bevins, RA; Dwoskin, LP; Pittenger, ST; Zeplin, LC1
Coen, K; Funk, D; Lê, AD; Lo, S1
Ciccocioppo, R; Cippitelli, A; Scuppa, G; Toll, L; Ubaldi, M1
Ebbert, JO; Elrashidi, MY; Stead, LF1
Clemens, KJ; Holmes, NM; Lay, BP1
Abdullah, R; Banks, ML; Bettinger, JC; Carroll, FI; Damaj, IM; Dawson, A; Jackson, A; Miles, MF; Muldoon, PP; O'Brien, M; Slater, CA; Soll, LG; Tapper, AR1
Abe, TO; Gaya, PV; Pereira, AC; Pinheiro, GG; Santos, PC; Scholz, J; Silva, AP1
Seguí Díaz, M1
Baker, TB; Bolt, DM; Fiore, MC; Fraser, DL; Piper, ME; Smith, SS; Stein, JH1
Wise, J1
Banks, ML; Blough, BE; Smith, DA1
Clemens, KJ; Holmes, NM; Macnamara, CL; Westbrook, RF1
Prochaska, JJ1
Carroll, ME; Smethells, JR; Swalve, N1
Cahill, K; Fanshawe, TR; Lancaster, T; Lindson-Hawley, N; Thomas, KH1
Abe, TO; Amorim, C; Buzo, CG; Gaya, PV; Lopes, NH; Pereira, AC; Pierri, H; Santos, PC; Scholz, J1
Della Santa, P1
Blazekovic, S; Brubaker, TR; Hitsman, B; Hole, A; Kalhan, R; Langer, C; Leone, F; Patel, J; Price, S; Schnoll, R; Veluz-Wilkins, A; Wileyto, EP1
Ban, N; Hamajima, N; Hasegawa, Y; Murohara, T; Oguri, T; Okada, Y; Sato, M; Shimadu, S1
Besheer, J; Cannady, R; Randall, PA1
Buhidma, Y; Jackson, A; Shoaib, M; Silk, S1
Kotz, D; van der Meer, RM; van Eerd, EA; van Schayck, OC1
Emme, E; Mazure, CM; McKee, SA; Smith, PH; Weinberger, AH; Zhang, J1
Carroll, FI; Cunningham, CS; Javors, MA; McMahon, LR; Moerke, MJ1
Albillos, A; Blázquez, J; de Castro-Guerín, C; González-Enguita, C; Hone, AJ; Michael McIntosh, J; Passas, J; Rueda-Ruzafa, L1
Gass, JC; Germeroth, LJ; Hawk, LW; Moore, FE; Motschman, CA; Munoz, DA; Rhodes, JD; Schlienz, NJ; Tiffany, ST; Wray, JM1
Muheim, L1
de Moura, FB; McMahon, LR2
Izumi, T; Ohmura, Y; Sasamori, H; Tsutsui-Kimura, I; Yoshida, T; Yoshioka, M1
Clyde, M; Els, C; Pipe, A; Reid, R; Tulloch, H1
Chappell, K; Ferguson, SG; Jacobson, GA; Lu, W; Patel, R; Schüz, N; Walters, JAE1
Aronson, SE; Lesage, E; Ross, TJ; Salmeron, BJ; Stein, EA; Sutherland, MT1
Batsikadze, G; Grundey, J; Hasan, A; Kuo, MF; Nitsche, MA; Paulus, W1
Colby, SM; MacKillop, J; Martin, RA; Murphy, CM; Rohsenow, DJ; Tidey, JW1
Baraona, LK; Daniels, JL; Lovelace, D; McDaniel, L1
Acuña Izcaray, A; Alfageme Michavila, I; Buljubasich, D; Casas, A; Chatkin, JM; de Granda Orive, JI; Guerreros Benavides, A; Jiménez Ruiz, CA; Noé, V; Núñez-Sánchez, I; Paez Espinel, N; Palomar Lever, A; Riesco Miranda, JA; Sánchez-Angarita, E; Sansores, RH; Zabert, G1
Govind, AP; Green, WN; Stolz, JR; Swanson, GT; Vallejo, YF; Yan, JZ1
Benowitz, NL; Cinciripini, P; George, TP; Hawk, LW; Lerman, C; Morales, M; Nollen, NL; Peng, AR; Schnoll, R; Tyndale, RF; Wileyto, EP1
Davies, NM; Jones, T; Martin, RM; Munafò, MR; Taylor, AE; Taylor, GMJ; Thomas, KH; Windmeijer, F1
Cornuz, J; Csajka, C; Dobrinas, M; Eap, CB; Gholamrezaee, M; Glatard, A; Lubomirov, R1
Abney, L; Beaulieu, DB; Duncan, MS; Freiberg, MS; Gatskie, V; Greevy, RA; King, S; Kundu, S; Scoville, E; Tindle, HA; Tyndale, RF; Wells, QS1
Bagdas, D; Hamouda, AK; Imad Damaj, M; Jackson, A1
Ginsburg, BC; Lamb, RJ; Levy, SA1
Bardo, MT; Baxter, TA; Bell, RL; Crooks, P; Dwoskin, LP; Maggio, SE; Newman, AH; Nixon, K; Prendergast, MA; Saunders, MA; Slack, RD; Zheng, G1
Barrett, ST; Bevins, RA; Geary, TN; Steiner, AN1
Abdul-Kader, J; Airagnes, G; D'almeida, S; Le Faou, AL; Limosin, F1
Bambs S, C; Cerda L, J; Corvalán B, MP; Pavié G, J; Véjar M, L; Zagolin B, M1
Harika-Germaneau, G; Jaafari, N; Peiffer, G; Perriot, J; Underner, M1
Clark, A; Clyde, M; Els, C; Fu, A; Pipe, A; Reid, R; Tulloch, H1
Alkhlaif, Y; Bagdas, D; Carroll, FI; Damaj, MI; Ditre, JW; Jackson, A1
Clemens, KJ; Davis, A; Holmes, NM; Pan, J; Panayi, MC1
Fukumoto, K; Kusaba, M; Mizoguchi, H; Wang, T; Yamada, K1
Cinciripini, P; George, TP; Hawk, LW; Lerman, C; Peng, AR; Schnoll, R; Tyndale, RF1
Aksöyler, DY; Aksu, AE; Bitik, O; Çalış, M; Kösemehmetoğlu, K; Üstün, GG; Uzun, H1
Aveyard, P; Coleman, T; Hajek, P; Lewis, S; Lindson, N; Munafo, M1
Adams, R; Ahmed, K; Alekna, R; Anderson, EC; Anderson, R; Ataya-Williams, A; Attwood, A; Aveyard, P; Banting, M; Bisal, N; Coleman, T; Coyle, D; Coyle, K; Dickinson, A; Easey, K; Fluharty, M; Freuler, T; Hajek, P; Healy, M; Homsey, C; Hurse, M; Khan, S; Khouja, J; Lacey, L; Lewis, S; Li, J; Lindson, N; Lycett, D; McEwen, A; McRobbie, HJ; Munafò, M; Myers-Smith, K; Orton, S; Perdue, J; Phillips, A; Pokhrel, S; Przulj, D; Rai, G; Randall, C; Tearne, S; Wood, C1
McMahon, LR; Moerke, MJ1
Bedi, G; Comer, SD; Cooper, ZD; Foltin, RW; Haney, M; Herrmann, ES; Ramesh, D; Reed, SC1
Bardo, MT; Bell, RL; Crooks, PA; Dwoskin, LP; Maggio, SE; Nixon, K; Prendergast, MA; Saunders, MA; Zheng, G1
Absalom, NL; Ahring, PK; Balle, T; Chebib, M; Indurthi, DC; Lewis, TM; Liao, VW; Qudah, T1
Charntikov, S; Kazan, T1
McMahon, LR1
Leischow, SJ1
Carroll, AJ; Hitsman, B; Hole, A; Jao, NC; Kalhan, R; Langer, C; Leone, F; Lubitz, SF; Miele, A; Patel, J; Paul Wileyto, E; Schnoll, R; Veluz-Wilkins, A1
Bao, H; Bera, K; Bishara, I; Borden, PM; Chapman, ER; Cohen, B; Dougherty, DA; Jeon, J; Kim, C; Lester, HA; Looger, LL; Marvin, JS; Mulcahy, MJ; Muthusamy, AK; Nichols, AL; O'Riordan, SL; Shivange, AV1
Hajek, P; Hartmann-Boyce, J; Jarvis, M; Livingstone-Banks, J; Norris, E; West, R1
Hauser, SR; Knight, CP; McBride, WJ; Pratt, LA; Rodd, ZA; Waeiss, RA1
de Abreu, GR; de Souza Spinosa, H; Faria Waziry, PA; Flório, JC; Fukushima, AR; Lebrun, I; Moreira, N; Petrocelli, BM; Reis-Silva, TM; Ricci, EL; Sandini, TM; Zaccarelli-Magalhães, J1
Barrett, ST; Bevins, RA; Thompson, BM1
Brath, H; Fasching, P; Kaser, S; Tatschl, C1
Baker, TB; Cook, JW; Piper, ME; Schlam, TR; Smith, SS1
Dannals, RF; Kuwabara, H; McCaul, ME; Wand, GS; Wong, D; Xu, X1
Brousse, G; de Chazeron, I; Harika-Germaneau, G; Jaafari, N; Peiffer, G; Perriot, J; Schmitt, A; Underner, M1
Alayoubi, H; Alkhlaif, Y; AlOmari, D; Bagdas, D; Carper, M; Damaj, MI; Diester, CM; Poklis, JL; Riley, J1
Cornuz, J; Jacot Sadowski, I; Rat, C; Selby, K1
Le Foll, B; Trigo, JM1
Davies, NM; Itani, T; Jones, T; Martin, RM; Munafò, MR; Rai, D; Taylor, AE; Taylor, GMJ; Thomas, KH; Windmeijer, F1
Eberg, M; Filion, KB; Platt, RW; Reynier, P1
Barkat, SS; Eloma, AS; Tellier, SM1
Flannery, JS; Laird, AR; Poudel, R; Riedel, MC; Ross, TJ; Salmeron, BJ; Stein, EA; Sutherland, MT1
Inada, K; Kanaoka, Y; Kataoka, Y; Koga, M; Nakao, Y; Okamoto, M; Takayama, S; Yamauchi, A1
Davis, CM; Holtyn, AF; Weerts, EM1
Davies, NM; Itani, T; Jones, T; Martin, RM; Munafò, MR; Rai, D; Taylor, AE; Taylor, GMJ; Thomas, KH1
Havard, A; Kennedy, D; Lee, ML; Tran, DT; Welsh, A1
Lesage, E; Ross, TJ; Salmeron, BJ; Stein, EA; Sutherland, MT1
Charntikov, S; Cova, N; Kazan, T; Madore, VM; Robison, CL1
Abney, LR; Adams, DW; Beaulieu, DB; Freiberg, MS; Gatskie, V; Gurwara, S; Horst, SN; King, S; Peyton, SC; Pointer, SO; Schwartz, DA; Scoville, EA; Tindle, HA; Wells, QS1
Bardo, MT; Chandler, CM; Maggio, SE; Nixon, K; Peng, H1
Amos, CI; Baker, TB; Bierut, LJ; Bray, M; Carney, RM; Chen, J; Chen, LS; Culverhouse, RC; Jorenby, DE; Miller, JP; Saccone, NL; Smock, N; Stoneking, F1
Firth, J; Kisely, S; Siskind, DJ; Wong, TT; Wu, BT1
Ashare, RL; Bauer, AM; Flitter, A; Gross, R; Hitsman, B; Hosie Quinn, M; Leone, FT; Lubitz, SF; Schnoll, R1
Barrett, ST; Charntikov, S; Hart, E; Hertia, D1
Barrett, ST; Bevins, RA; Huynh, YW; Kwan, DA; Murray, JE; Thompson, BM1
Ding, ZM; Gao, Y; Sentir, AM; Tan, X1
Antoniu, SA; Buculei, I; Crisan Dabija, R; Mihaltan, F; Trofor, AC1
Higgins, GA; Sellers, EM1
Achenbach, C; Ashare, R; Bauer, AM; Fox, EN; Gollan, J; Gross, R; Hatzell, J; Hitsman, B; Josephson, S; Leone, F; Purnell, J; Quinn, MH; Randle, T; Rogers, T; Schnoll, R; Stevens, N; Wileyto, EP1
Albillos, A; Blázquez, J; de Los Ríos, C; González-Enguita, C; Hone, AJ; Jiménez-Pompa, A; Medina-Polo, J; Michael McIntosh, J; Rueda-Ruzafa, L; Sanz-Lázaro, S1
de Chazeron, I; Jaafari, N; Peiffer, G; Perriot, J; Ruppert, AM; Underner, M1
Choi, SKY; Einarsdottir, K; Havard, A; Jorm, LR; Kemp-Casey, A; Preen, DB; Randall, D; Tran, DT1
Chenoweth, MJ; Hawk, LW; Novalen, M; Tyndale, RF; Zhao, B1
Evers-Casey, S; Leone, FT1
Beloate, LN; Doolittle, J; Froeliger, B; Garcia-Keller, C; Kalivas, PW; Meyerink, ME; Nall, RW; Penaloza, T1
Chakraborti, Y; Coffman, DL; Piper, ME1
George, TP; Johnstone, S; Rabin, RA; Sorkhou, M1
Abramson, MJ; Bonevski, B; George, J; Gobarani, RK; Ilomäki, J; Wood, S1
Humair, JP; Papachristou, C1
Apolone, G; Boeri, M; Boffi, R; Gallus, S; Ladisa, V; Ledda, RE; Marchianò, A; Milanese, G; Munarini, E; Pastorino, U; Rolli, L; Sabia, F; Sozzi, G; Suatoni, P; Trussardo, S; Valsecchi, C1
Bendiks, S; Blokhina, E; Bryant, K; Cheng, DM; Freiberg, MS; Gnatienko, N; Hahn, J; Krupitsky, E; Lioznov, D; Patts, G; Samet, JH; So-Armah, K; Stein, MD; Tindle, HA; Yaroslavtseva, T1
Bhuiyan, M; Chen, CT; Freifelder, R; Govind, AP; Green, WN; Holderman, N; Kao, CM; Kucharski, A; Mitchell, S; Mukherjee, J; Zammit, M; Zhang, HJ; Zhuang, X1
Baliunas, D; Comans, T; Gartner, C; Hollingworth, SA; Pole, JD; Sullivan, C1
Barrett, ST; Bevins, RA; Dwoskin, LP; Huynh, YW; Thompson, BM; Tracy, ME1
Chenoweth, MJ; Knight, J; Lerman, C; Tyndale, RF1
Chow, CK; Falster, MO; Filion, KB; Havard, A; Hsu, B; Jorm, L; Pearson, SA; Robijn, AL; Woodward, M1
Buzzi, B; Damaj, MI; Koseli, E; Moncayo, L; Shoaib, M1
Burkard, T; Christ-Crain, M; Coynel, D; Erlanger, TE; Hemkens, LG; Jeanloz, N; Lengsfeld, S; Meienberg, A; Speich, B; Vogt, DR; Winzeler, B; Zanchi, D1
Canseco, JA; D'Antonio, ND; Heard, JC; Karamian, BA; Kepler, CK; Lambrechts, MJ; Levy, HA; Markova, DZ; Vaccaro, AR; Yalla, GR1
Fanshawe, TR; Hajizadeh, A; Hartman, L; Lindson, N; Livingstone-Banks, J; Theodoulou, A; Thomas, KH1
Ashburner, JM; Klemenc Ketiš, Z; Oreskovic, S; Oreskovic, T; Percac-Lima, S; Rifel, J; Tiljak, H1
Ahluwalia, JS; Cox, LS; Ellerbeck, EF; Greiner, KA; Leavens, ELS; Mayo, MS; Nollen, NL; Salzman, G; Shanks, D; Woodward, J1
Budzyńska, B; Chałas, R; Maciąg, M; Rahnama-Hezavah, M; Stachurski, P; Świątkowska, A; Świątkowski, W; Tylżanowski, P1
Dennis, BB; Devereaux, PJ; Fairbairn, N; Lu, C; Mbuagbaw, L; Ofori, S; Olasupo, OO1
Davis, JM; Masclans, L; Rose, JE1
Agrawal, S; Aveyard, P; Fanshawe, TR; Freeman, SC; Hajizadeh, A; Hartmann-Boyce, J; Lindson, N; Livingstone-Banks, J; Ordóñez-Mena, JM; Sutton, AJ; Theodoulou, A; Zhu, S1
Barnes, J; Bullen, C; Calder, A; Laking, G; Parag, V; Walker, N1
Ahluwalia, JS; Brown, A; Cruvinel, E; Funk, O; Lambart, L; Leavens, E; Mayo, MS; Nollen, NL; Sanderson Cox, L1

Reviews

99 review(s) available for nicotine and varenicline

ArticleYear
Pharmacologic interventions for smoking cessation.
    Critical care nursing clinics of North America, 2006, Volume: 18, Issue:1

    Topics: Administration, Cutaneous; Administration, Inhalation; Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Chewing Gum; Clonidine; Critical Care; Drug Therapy, Combination; Evidence-Based Medicine; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Nurse's Role; Patient Education as Topic; Patient Selection; Phytotherapy; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking Cessation; Smoking Prevention; United States; United States Food and Drug Administration; Varenicline

2006
Effectiveness of smoking cessation therapies: a systematic review and meta-analysis.
    BMC public health, 2006, Dec-11, Volume: 6

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Quinoxalines; Smoking Cessation; Treatment Outcome; Varenicline

2006
Non-nicotinic therapies for smoking cessation.
    Annual review of pharmacology and toxicology, 2007, Volume: 47

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Drugs, Investigational; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2007
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2007, Jan-24, Issue:1

    Topics: Alkaloids; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking Cessation; Varenicline

2007
Smoking cessation pharmacotherapy--nicotine and non-nicotine preparations.
    Preventive cardiology, 2007,Spring, Volume: 10, Issue:2 Suppl 1

    Topics: Administration, Cutaneous; Administration, Inhalation; Benzazepines; Bupropion; Chewing Gum; Clonidine; Coronary Artery Disease; Humans; Monoamine Oxidase Inhibitors; Nicotine; Nortriptyline; Piperidines; Pyrazoles; Quinoxalines; Receptors, Nicotinic; Rimonabant; Selective Serotonin Reuptake Inhibitors; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Disorder; Tobacco, Smokeless; Varenicline

2007
The most addictive drug, the most deadly substance: smoking cessation tactics for the busy clinician.
    Primary care, 2007, Volume: 34, Issue:1

    Topics: Age Factors; Benzazepines; Bupropion; Complementary Therapies; Dopamine Uptake Inhibitors; Dosage Forms; Humans; Nicotine; Nicotinic Agonists; Physician's Role; Primary Health Care; Quinoxalines; Referral and Consultation; Smoking Cessation; Tobacco Use Disorder; Varenicline

2007
Varenicline: the newest agent for smoking cessation.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2007, Jul-01, Volume: 64, Issue:13

    Topics: Animals; Benzazepines; Clinical Trials, Phase III as Topic; Drug Interactions; Humans; Nicotine; Quinoxalines; Receptors, Cholinergic; Smoking Cessation; Varenicline

2007
Optimizing on smoke free legislation making the most of the opportunity.
    British journal of community nursing, 2007, Volume: 12, Issue:8

    Topics: Benzazepines; Bupropion; Decision Trees; Dopamine Uptake Inhibitors; Drug Therapy, Combination; Health Services Needs and Demand; Humans; Nicotine; Nicotinic Agonists; Nurse's Role; Patient Care Planning; Patient Education as Topic; Practice Guidelines as Topic; Public Facilities; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Social Support; United Kingdom; Varenicline

2007
Treating tobacco dependence in women.
    Journal of women's health (2002), 2007, Volume: 16, Issue:8

    Topics: Benzazepines; Bupropion; Counseling; Dopamine Uptake Inhibitors; Female; Humans; Lung Neoplasms; Nicotine; Nicotinic Agonists; Quinoxalines; Risk Reduction Behavior; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; United States; Varenicline; Women's Health

2007
Which is the best primary medication for long-term smoking cessation--nicotine replacement therapy, bupropion or varenicline?
    Expert opinion on pharmacotherapy, 2007, Volume: 8, Issue:17

    Topics: Benzazepines; Bupropion; Combined Modality Therapy; Counseling; Dopamine Uptake Inhibitors; Drug Administration Routes; Drug Partial Agonism; Drug Therapy, Combination; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Time Factors; Treatment Outcome; Varenicline

2007
Treatment of tobacco dependence: integrating recent progress into practice.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 2007, Nov-20, Volume: 177, Issue:11

    Topics: Behavior Therapy; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Health Behavior; Health Policy; Humans; Nicotine; Nicotinic Agonists; Practice Guidelines as Topic; Quinoxalines; Tobacco Use Cessation; Tobacco Use Disorder; Varenicline

2007
Breaking the ties of nicotine dependence.
    The Nurse practitioner, 2007, Volume: 32, Issue:11

    Topics: Algorithms; Benzazepines; Bupropion; Decision Trees; Dopamine Uptake Inhibitors; Drug Costs; Evidence-Based Medicine; Global Health; Humans; Nicotine; Nicotinic Agonists; Nurse Practitioners; Nurse's Role; Nursing Assessment; Patient Acceptance of Health Care; Patient Care Planning; Patient Education as Topic; Practice Guidelines as Topic; Prevalence; Primary Health Care; Quinoxalines; Risk Factors; Smoking Cessation; Tobacco Use Disorder; Varenicline

2007
An update on therapeutics for tobacco dependence.
    Expert opinion on pharmacotherapy, 2008, Volume: 9, Issue:1

    Topics: Alkaloids; Anti-Anxiety Agents; Azocines; Benzazepines; Bupropion; Clinical Trials as Topic; Databases, Bibliographic; Humans; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Quinolizines; Quinoxalines; Review Literature as Topic; Rimonabant; Smoking; Smoking Cessation; Varenicline

2008
Effect of varenicline and bupropion SR on craving, nicotine withdrawal symptoms, and rewarding effects of smoking during a quit attempt.
    Psychopharmacology, 2008, Volume: 197, Issue:3

    Topics: Adolescent; Adult; Affect; Aged; Benzazepines; Bupropion; Clinical Trials, Phase III as Topic; Delayed-Action Preparations; Dopamine Uptake Inhibitors; Double-Blind Method; Follow-Up Studies; Humans; Middle Aged; Motivation; Multicenter Studies as Topic; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Disorder; Varenicline

2008
Smoking cessation and lung cancer: oncology nurses can make a difference.
    Seminars in oncology nursing, 2008, Volume: 24, Issue:1

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Information Services; Lung Neoplasms; Nicotine; Oncology Nursing; Quinoxalines; Smoking; Smoking Cessation; Varenicline

2008
Clinical pharmacology of nicotine: implications for understanding, preventing, and treating tobacco addiction.
    Clinical pharmacology and therapeutics, 2008, Volume: 83, Issue:4

    Topics: Antidepressive Agents; Aryl Hydrocarbon Hydroxylases; Asian; Benzazepines; Black or African American; Bupropion; Cotinine; Cues; Cytochrome P-450 CYP2A6; Drug Tolerance; Genetic Predisposition to Disease; Harm Reduction; Humans; Menthol; Mixed Function Oxygenases; Neuronal Plasticity; Nicotine; Nicotinic Agonists; Quinoxalines; Receptors, Nicotinic; Reinforcement, Psychology; Smoking; Smoking Cessation; Tobacco Use Disorder; United States; Varenicline; White People

2008
Smoking cessation in pregnancy: why, how, and what next...
    Clinical obstetrics and gynecology, 2008, Volume: 51, Issue:2

    Topics: Behavior Therapy; Benzazepines; Bupropion; Counseling; Female; Humans; Nicotine; Pregnancy; Pregnancy Outcome; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Varenicline

2008
[The ABC of smoking cessation].
    Medizinische Monatsschrift fur Pharmazeuten, 2008, Volume: 31, Issue:5

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Cognitive Behavioral Therapy; Humans; Hypnosis; Motivation; Nicotiana; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Varenicline

2008
Which drug to be used in smoking cessation?
    Polskie Archiwum Medycyny Wewnetrznej, 2008, Volume: 118, Issue:6

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Quinoxalines; Smoking Cessation; Treatment Outcome; Varenicline

2008
Pharmacotherapies for smoking cessation: a meta-analysis of randomized controlled trials.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 2008, Jul-15, Volume: 179, Issue:2

    Topics: Administration, Cutaneous; Administration, Inhalation; Administration, Oral; Benzazepines; Bupropion; Chewing Gum; Female; Follow-Up Studies; Humans; Male; Multivariate Analysis; Nicotine; Nicotinic Agonists; Patient Compliance; Probability; Quebec; Quinoxalines; Risk Assessment; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Treatment Outcome; Varenicline

2008
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2008, Jul-16, Issue:3

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Varenicline

2008
The relevance and treatment of cue-induced cravings in tobacco dependence.
    Journal of substance abuse treatment, 2009, Volume: 36, Issue:3

    Topics: Adaptation, Psychological; Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Cognitive Behavioral Therapy; Cues; Extinction, Psychological; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2009
Drugs for tobacco dependence.
    Treatment guidelines from the Medical Letter, 2008, Volume: 6, Issue:73

    Topics: Adrenergic alpha-Agonists; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2008
Multimodal techniques for smoking cessation: a review of their efficacy and utilisation and clinical practice guidelines.
    International journal of clinical practice, 2008, Volume: 62, Issue:11

    Topics: Benzazepines; Combined Modality Therapy; Complementary Therapies; Drug Therapy, Combination; Humans; Nicotine; Nicotinic Agonists; Practice Guidelines as Topic; Psychotherapy; Quinoxalines; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Treatment Outcome; Varenicline

2008
Pharmacology of nicotine: addiction, smoking-induced disease, and therapeutics.
    Annual review of pharmacology and toxicology, 2009, Volume: 49

    Topics: Animals; Behavior, Addictive; Benzazepines; Bupropion; Ganglionic Stimulants; Humans; Nicotine; Nicotinic Agonists; Nonprescription Drugs; Quinoxalines; Smoking; Tobacco Use Disorder; Varenicline

2009
[Modern medical support for smoking cessation].
    Der Internist, 2009, Volume: 50, Issue:1

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Practice Patterns, Physicians'; Quinoxalines; Smoking Cessation; Smoking Prevention; Varenicline

2009
[Not smoking, essential for healthy lungs].
    Pharmazie in unserer Zeit, 2008, Volume: 37, Issue:6

    Topics: Administration, Cutaneous; Benzazepines; Bupropion; Chewing Gum; Health; Humans; Lung; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Tablets; Varenicline

2008
Smoking cessation in pregnancy.
    Expert opinion on drug safety, 2008, Volume: 7, Issue:6

    Topics: Animals; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Female; Humans; Nicotine; Nicotinic Agonists; Pregnancy; Pregnancy Complications; Quinoxalines; Smoking Cessation; Varenicline

2008
Varenicline for tobacco dependence.
    The New England journal of medicine, 2008, Nov-06, Volume: 359, Issue:19

    Topics: Benzazepines; Brain; Coronary Artery Disease; Humans; Male; Middle Aged; Motivation; Nicotine; Nicotinic Agonists; Practice Guidelines as Topic; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Disorder; Varenicline

2008
New findings on nicotine addiction and treatment.
    Nebraska Symposium on Motivation. Nebraska Symposium on Motivation, 2009, Volume: 55

    Topics: Animals; Benzazepines; Bupropion; Humans; Mecamylamine; Motivation; Nicotine; Nicotinic Antagonists; Quinoxalines; Reward; Smoking Cessation; Tobacco Use Disorder; Vaccines; Varenicline

2009
Interventions for preventing weight gain after smoking cessation.
    The Cochrane database of systematic reviews, 2009, Jan-21, Issue:1

    Topics: Antidepressive Agents; Benzazepines; Exercise; Female; Humans; Male; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking Cessation; Varenicline; Weight Gain

2009
Smoking in pregnancy and lactation: a review of risks and cessation strategies.
    European journal of clinical pharmacology, 2009, Volume: 65, Issue:4

    Topics: Adult; Alkaloids; Antidepressive Agents; Azocines; Benzazepines; Breast Feeding; Bromocriptine; Cognitive Behavioral Therapy; Female; Humans; Lactation; Nicotine; Nicotinic Agonists; Pregnancy; Pregnancy Complications; Quinolizines; Quinoxalines; Risk Assessment; Risk Factors; Smoking; Smoking Cessation; Vaccines; Varenicline; Young Adult

2009
[Pharmacotherapy of smoking cessation with application of nicotine and nicotine free drugs].
    Przeglad lekarski, 2008, Volume: 65, Issue:10

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Quinoxalines; Receptors, Nicotinic; Smoking; Smoking Cessation; Tobacco Use Disorder; Varenicline

2008
A preliminary benefit-risk assessment of varenicline in smoking cessation.
    Drug safety, 2009, Volume: 32, Issue:2

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Product Surveillance, Postmarketing; Quinoxalines; Recurrence; Risk Assessment; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2009
Emerging drugs for the treatment of tobacco dependence.
    Expert opinion on emerging drugs, 2009, Volume: 14, Issue:1

    Topics: Animals; Benzazepines; Clinical Trials as Topic; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Disorder; Varenicline

2009
Tobacco dependence and withdrawal: science base, challenges and opportunities for pharmacotherapy.
    Pharmacology & therapeutics, 2009, Volume: 123, Issue:1

    Topics: Animals; Benzazepines; Bupropion; Clinical Trials as Topic; Humans; Nicotine; Quinoxalines; Receptors, Nicotinic; Substance Withdrawal Syndrome; Tobacco Use Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2009
Update on smoking cessation therapies.
    Advances in therapy, 2009, Volume: 26, Issue:4

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Cost of Illness; Drug Approval; Global Health; Humans; Morbidity; Nicotine; Nicotinic Agonists; Quinoxalines; Safety; Smoking; Smoking Cessation; Smoking Prevention; Treatment Outcome; United States; Varenicline

2009
Smoking and chronic obstructive pulmonary disease (COPD). Parallel epidemics of the 21 century.
    International journal of environmental research and public health, 2009, Volume: 6, Issue:1

    Topics: Benzazepines; Bupropion; Combined Modality Therapy; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Smoking; Smoking Cessation; Varenicline

2009
Pharmacogenetics of smoking cessation therapy.
    American journal of medical genetics. Part B, Neuropsychiatric genetics : the official publication of the International Society of Psychiatric Genetics, 2010, Jan-05, Volume: 153B, Issue:1

    Topics: Benzazepines; Bupropion; Clonidine; Genome-Wide Association Study; Humans; Nicotine; Nortriptyline; Pharmacogenetics; Quinoxalines; Smoking Cessation; Varenicline

2010
Tobacco use among individuals with intellectual or developmental disabilities: a brief review.
    Intellectual and developmental disabilities, 2009, Volume: 47, Issue:3

    Topics: Adult; Benzazepines; Bupropion; Counseling; Cross-Sectional Studies; Disabled Persons; Health Policy; Humans; Nicotine; Persons with Mental Disabilities; Quinoxalines; Smoking; Smoking Cessation; Tobacco Smoke Pollution; Tobacco Use Disorder; United States; Varenicline

2009
Are nicotine replacement therapy, varenicline or bupropion options for pregnant mothers to quit smoking? Effects on the respiratory system of the offspring.
    Therapeutic advances in respiratory disease, 2009, Volume: 3, Issue:4

    Topics: Animals; Antioxidants; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Female; Humans; Maternal-Fetal Exchange; Nicotine; Nicotinic Agonists; Pregnancy; Pregnancy Complications; Quinoxalines; Respiratory System; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Varenicline

2009
What do we know about the role of pharmacotherapy for smoking cessation before or during pregnancy?
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2009, Volume: 11, Issue:11

    Topics: Animals; Benzazepines; Bupropion; Drug Therapy; Drug-Related Side Effects and Adverse Reactions; Female; Humans; Nicotine; Pregnancy; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Varenicline

2009
Current approaches to pharmacotherapy for smoking cessation.
    Therapeutic advances in respiratory disease, 2010, Volume: 4, Issue:1

    Topics: Adolescent; Adult; Animals; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Female; Humans; Male; Nicotine; Nicotinic Agonists; Pregnancy; Quinoxalines; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; United States; Varenicline

2010
Varenicline: a pharmacoeconomic review of its use as an aid to smoking cessation.
    PharmacoEconomics, 2010, Volume: 28, Issue:3

    Topics: Benzazepines; Bupropion; Clinical Trials as Topic; Cost-Benefit Analysis; Delayed-Action Preparations; Health Care Costs; Humans; Models, Statistical; Nicotine; Nicotinic Agonists; Prevalence; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2010
Smoking cessation intervention: an evidence-based approach.
    Postgraduate medicine, 2010, Volume: 122, Issue:2

    Topics: Antidepressive Agents, Second-Generation; Behavior Therapy; Benzazepines; Bupropion; Directive Counseling; Drug Therapy, Combination; Evidence-Based Medicine; Global Health; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Varenicline

2010
Improving the effectiveness of tobacco use cessation (TUC).
    International dental journal, 2010, Volume: 60, Issue:1

    Topics: Antidepressive Agents, Second-Generation; Behavior Therapy; Benzazepines; Bupropion; Chewing Gum; Counseling; Dental Offices; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Referral and Consultation; Smoking; Tobacco Use Cessation; Varenicline

2010
[Pharmacological profile and clinical findings on varenicline tartrate (Champix tablets)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2010, Volume: 135, Issue:5

    Topics: Animals; Benzazepines; Clinical Trials, Phase III as Topic; Corpus Striatum; Dopamine; Humans; Nicotine; Nicotinic Agonists; Nucleus Accumbens; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Disorder; Varenicline

2010
Smoking cessation-recent advances.
    Cardiovascular drugs and therapy, 2010, Volume: 24, Issue:4

    Topics: Australia; Benzazepines; Bupropion; Cardiovascular Diseases; Dopamine Uptake Inhibitors; Drug Therapy, Combination; Humans; Immunotherapy, Active; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Transdermal Patch; Treatment Outcome; United Kingdom; United States; Varenicline

2010
Comparison of available treatments for tobacco addiction.
    Current psychiatry reports, 2010, Volume: 12, Issue:5

    Topics: Behavior Therapy; Benzazepines; Bupropion; Humans; Nicotine; Nortriptyline; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2010
[Preventive relapse treatment for tobacco cessation - is it worthwhile?].
    Therapeutische Umschau. Revue therapeutique, 2010, Volume: 67, Issue:8

    Topics: Antidepressive Agents; Behavior Therapy; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Secondary Prevention; Smoking Cessation; Treatment Outcome; Varenicline

2010
[Pharmacotherapies for nicotine dependence: review of scientific evidence. Spanish Society of Smoking Specialists: recommendations about election and individualization].
    Medicina clinica, 2011, Jan-29, Volume: 136, Issue:2

    Topics: Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Tobacco Use Disorder; Varenicline

2011
A brief review of pharmacotherapeutic treatment options in smoking cessation: bupropion versus varenicline.
    Journal of the American Academy of Nurse Practitioners, 2010, Volume: 22, Issue:10

    Topics: Antidepressive Agents, Second-Generation; Behavior Therapy; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Risk Factors; Smoking Cessation; Smoking Prevention; Substance-Related Disorders; Varenicline

2010
Impact of genetic variability in nicotinic acetylcholine receptors on nicotine addiction and smoking cessation treatment.
    Current medicinal chemistry, 2011, Volume: 18, Issue:1

    Topics: Benzazepines; Bupropion; Genetic Variation; Humans; Nicotine; Protein Subunits; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Disorder; Varenicline

2011
Adverse effects and tolerability of medications for the treatment of tobacco use and dependence.
    Drugs, 2010, Dec-24, Volume: 70, Issue:18

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2010
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2010, Dec-08, Issue:12

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2010
Interventions for smokeless tobacco use cessation.
    The Cochrane database of systematic reviews, 2011, Feb-16, Issue:2

    Topics: Benzazepines; Bupropion; Chewing Gum; Counseling; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Tobacco Use Cessation; Tobacco, Smokeless; Varenicline

2011
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2011, Feb-16, Issue:2

    Topics: Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2011
Nicotine dependence: health consequences, smoking cessation therapies, and pharmacotherapy.
    Primary care, 2011, Volume: 38, Issue:1

    Topics: Administration, Cutaneous; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Heart Diseases; Humans; Neoplasms; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Substance-Related Disorders; Varenicline

2011
Pharmacotherapy for smoking cessation: present and future.
    Current pharmaceutical design, 2011, Volume: 17, Issue:14

    Topics: Adolescent; Animals; Benzazepines; Bupropion; Delayed-Action Preparations; Female; Humans; Nicotine; Nicotinic Agonists; Pregnancy; Quinoxalines; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Varenicline

2011
Varenicline for tobacco dependence: panacea or plight?
    Expert opinion on pharmacotherapy, 2011, Volume: 12, Issue:11

    Topics: Animals; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Cessation; Tobacco Use Disorder; Tobacco, Smokeless; Varenicline

2011
Clinical practice. Treating smokers in the health care setting.
    The New England journal of medicine, 2011, Sep-29, Volume: 365, Issue:13

    Topics: Benzazepines; Bupropion; Cholinergic Agents; Counseling; Dopamine Uptake Inhibitors; Evidence-Based Medicine; Female; Humans; Middle Aged; Motivation; Nicotine; Patient Compliance; Physician-Patient Relations; Practice Guidelines as Topic; Quinoxalines; Smoking; Smoking Cessation; United States; Varenicline

2011
Efficacy and tolerability of pharmacotherapies to aid smoking cessation in adolescents.
    Paediatric drugs, 2012, Apr-01, Volume: 14, Issue:2

    Topics: Adolescent; Benzazepines; Bupropion; Clinical Trials as Topic; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Patient Compliance; Prescription Drugs; Quinoxalines; Randomized Controlled Trials as Topic; Safety; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2012
[Smoking cessation in medical practice--new possibilities?].
    Revue medicale suisse, 2012, Jan-25, Volume: 8, Issue:325

    Topics: Benzazepines; Bupropion; Complementary Therapies; Drugs, Investigational; General Practitioners; Humans; Nicotine; Nicotinic Agonists; Professional Practice; Quinoxalines; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2012
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2012, Apr-18, Issue:4

    Topics: Alkaloids; Azepines; Azocines; Benzazepines; Bupropion; Counseling; Heterocyclic Compounds, 4 or More Rings; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2012
The pharmacist "toolbox" for smoking cessation: a review of methods, medicines, and novel means to help patients along the path of smoking reduction to smoking cessation.
    Journal of pharmacy practice, 2012, Volume: 25, Issue:6

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Education, Pharmacy, Continuing; Humans; Nicotine; Nicotinic Agonists; Patient Acceptance of Health Care; Pharmacists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Cessation Devices; Varenicline

2012
[Drugs used to treat nicotine addiction].
    Przeglad lekarski, 2012, Volume: 69, Issue:10

    Topics: Adult; Age Distribution; Alkaloids; Azocines; Benzazepines; Bupropion; Causality; Comorbidity; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Poland; Quinolizines; Quinoxalines; Sex Distribution; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Varenicline; Young Adult

2012
Interventions for smoking cessation and reduction in individuals with schizophrenia.
    The Cochrane database of systematic reviews, 2013, Feb-28, Issue:2

    Topics: Adult; Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Reinforcement, Psychology; Schizophrenia; Schizophrenic Psychology; Smoking Cessation; Smoking Prevention; Tobacco Use Cessation Devices; Varenicline

2013
Smoking cessation and COPD.
    European respiratory review : an official journal of the European Respiratory Society, 2013, Mar-01, Volume: 22, Issue:127

    Topics: Benzazepines; Bupropion; Counseling; Humans; Nicotine; Nicotinic Agonists; Prevalence; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Risk Factors; Risk Reduction Behavior; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2013
Smoking cessation treatment for COPD smokers: the role of pharmacological interventions.
    Monaldi archives for chest disease = Archivio Monaldi per le malattie del torace, 2013, Volume: 79, Issue:1

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2013
Relapse prevention interventions for smoking cessation.
    The Cochrane database of systematic reviews, 2013, Aug-20, Issue:8

    Topics: Behavior Therapy; Benzazepines; Chewing Gum; Female; Humans; Male; Nicotine; Nicotinic Agonists; Pregnancy; Quinoxalines; Randomized Controlled Trials as Topic; Secondary Prevention; Smoking Cessation; Smoking Prevention; Varenicline

2013
[Nicotine and neurologic diseases--even a noxious substance may possess beneficial properties].
    Duodecim; laaketieteellinen aikakauskirja, 2013, Volume: 129, Issue:16

    Topics: Alzheimer Disease; Ataxia; Benzazepines; Cognitive Dysfunction; Epilepsy, Frontal Lobe; Humans; Mutation; Nicotine; Nicotinic Agonists; Parkinson Disease; Quinoxalines; Receptors, Nicotinic; Tobacco Use Cessation Devices; Varenicline

2013
Cardiovascular events associated with smoking cessation pharmacotherapies: a network meta-analysis.
    Circulation, 2014, Jan-07, Volume: 129, Issue:1

    Topics: Adult; Benzazepines; Bupropion; Cardiovascular Diseases; Dopamine Uptake Inhibitors; Female; Humans; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Risk Factors; Smoking; Smoking Cessation; Varenicline

2014
Pharmacological intervention of nicotine dependence.
    BioMed research international, 2013, Volume: 2013

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Quinoxalines; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2013
Smoking cessation.
    Clinics in chest medicine, 2014, Volume: 35, Issue:1

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2014
Emerging drugs for the treatment of tobacco dependence: 2014 update.
    Expert opinion on emerging drugs, 2014, Volume: 19, Issue:2

    Topics: Atomoxetine Hydrochloride; Benzazepines; Bupropion; Clinical Trials as Topic; Clonidine; Humans; Mecamylamine; Nicotine; Nortriptyline; Propylamines; Quinoxalines; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2014
Interventions for preoperative smoking cessation.
    The Cochrane database of systematic reviews, 2014, Mar-27, Issue:3

    Topics: Benzazepines; Humans; Nicotine; Nicotinic Agonists; Postoperative Complications; Preoperative Care; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2014
Smoking Cessation in Chronic Obstructive Pulmonary Disease.
    Seminars in respiratory and critical care medicine, 2015, Volume: 36, Issue:4

    Topics: Combined Modality Therapy; Counseling; Electronic Nicotine Delivery Systems; Humans; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Secondary Prevention; Smoking; Smoking Cessation; Treatment Outcome; Varenicline

2015
Effect of Smoking Reduction Therapy on Smoking Cessation for Smokers without an Intention to Quit: An Updated Systematic Review and Meta-Analysis of Randomized Controlled.
    International journal of environmental research and public health, 2015, Aug-25, Volume: 12, Issue:9

    Topics: Adult; Aged; Benzazepines; Bupropion; Female; Humans; Intention; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Varenicline

2015
The Past, Present, and Future of Nicotine Addiction Therapy.
    Annual review of medicine, 2016, Volume: 67

    Topics: Alkaloids; Azocines; Bupropion; Directive Counseling; Dopamine Uptake Inhibitors; Drug Therapy, Combination; Health Policy; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Social Media; Text Messaging; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2016
Interventions for smokeless tobacco use cessation.
    The Cochrane database of systematic reviews, 2015, Oct-26, Issue:10

    Topics: Benzazepines; Bupropion; Chewing Gum; Counseling; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Randomized Controlled Trials as Topic; Tobacco Use Cessation; Tobacco, Smokeless; Varenicline

2015
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2016, May-09, Issue:5

    Topics: Alkaloids; Azepines; Azocines; Benzazepines; Bupropion; Counseling; Heterocyclic Compounds, 4 or More Rings; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2016
Smoking cessation for people with chronic obstructive pulmonary disease.
    The Cochrane database of systematic reviews, 2016, Aug-20, Issue:8

    Topics: Adult; Behavior Therapy; Bupropion; Combined Modality Therapy; Female; Humans; Male; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Randomized Controlled Trials as Topic; Smoking Cessation; Varenicline

2016
Sex Differences in Smoking Cessation Pharmacotherapy Comparative Efficacy: A Network Meta-analysis.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2017, Mar-01, Volume: 19, Issue:3

    Topics: Adult; Female; Humans; Male; Nicotine; Nicotinic Agonists; Sex Distribution; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2017
Selection criteria limit generalizability of smoking pharmacotherapy studies differentially across clinical trials and laboratory studies: A systematic review on varenicline.
    Drug and alcohol dependence, 2016, Dec-01, Volume: 169

    Topics: Adult; Bupropion; Clinical Trials as Topic; Female; Humans; Laboratories; Middle Aged; Nicotine; Nicotinic Agonists; Patient Selection; Smoking; Smoking Cessation; Varenicline

2016
Tobacco Harms, Nicotine Pharmacology, and Pharmacologic Tobacco Cessation Interventions for Women.
    Journal of midwifery & women's health, 2017, Volume: 62, Issue:3

    Topics: Bupropion; Female; Fetus; Humans; Lactation; Nicotiana; Nicotine; Pregnancy; Pregnant Women; Smoking; Smoking Cessation; Tobacco Use Cessation; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2017
[Interventions for smoking cessation in 2018].
    Revue de pneumologie clinique, 2018, Volume: 74, Issue:3

    Topics: Bupropion; History, 21st Century; Humans; Nicotine; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2018
[Smoking cessation: Pharmacological strategies different from standard treatments].
    Revue de pneumologie clinique, 2018, Volume: 74, Issue:4

    Topics: Bupropion; Humans; Nicotine; Smoking; Smoking Cessation; Smoking Cessation Agents; Standard of Care; Tobacco Use Cessation Devices; Varenicline

2018
Green tobacco sickness: mecamylamine, varenicline, and nicotine vaccine as clinical research tools and potential therapeutics.
    Expert review of clinical pharmacology, 2019, Volume: 12, Issue:3

    Topics: Agricultural Workers' Diseases; Humans; Mecamylamine; Nicotiana; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Plant Leaves; Vaccines; Varenicline

2019
Relapse prevention interventions for smoking cessation.
    The Cochrane database of systematic reviews, 2019, 02-13, Volume: 2

    Topics: Behavior Therapy; Bupropion; Chewing Gum; Female; Humans; Male; Nicotine; Nicotinic Agonists; Pregnancy; Randomized Controlled Trials as Topic; Secondary Prevention; Smoking Cessation; Smoking Cessation Agents; Smoking Prevention; Varenicline

2019
[Smoking, alcohol and diabetes (Update 2019)].
    Wiener klinische Wochenschrift, 2019, Volume: 131, Issue:Suppl 1

    Topics: Alcohol Drinking; Benzazepines; Bupropion; Diabetes Mellitus; Humans; Nicotine; Practice Guidelines as Topic; Quinoxalines; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2019
[Stopping and reducing smoking in patients with schizophrenia].
    L'Encephale, 2019, Volume: 45, Issue:4

    Topics: Bupropion; Cognitive Behavioral Therapy; Electronic Nicotine Delivery Systems; Humans; Nicotine; Reinforcement, Psychology; Schizophrenia; Smoking Cessation; Tobacco Smoking; Tobacco Use Cessation Devices; Varenicline

2019
[Smoking cessation: How can we involve patients better in treatment choice?]
    Revue des maladies respiratoires, 2019, Volume: 36, Issue:5

    Topics: Bupropion; Choice Behavior; Counseling; Decision Making, Shared; Humans; Nicotine; Patient Participation; Patient Selection; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2019
Pharmacological interventions for smoking cessation among people with schizophrenia spectrum disorders: a systematic review, meta-analysis, and network meta-analysis.
    The lancet. Psychiatry, 2020, Volume: 7, Issue:9

    Topics: Antidepressive Agents, Second-Generation; Bupropion; Humans; Network Meta-Analysis; Nicotine; Nicotinic Agonists; Randomized Controlled Trials as Topic; Schizophrenia; Schizophrenic Psychology; Smoking Cessation; Varenicline

2020
Pharmacological strategies for smoking cessation in patients with chronic obstructive pulmonary disease: a pragmatic review.
    Expert opinion on pharmacotherapy, 2021, Volume: 22, Issue:7

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Pulmonary Disease, Chronic Obstructive; Quinoxalines; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2021
[Combinations of pharmacological treatments in smoking cessation. A systematic review].
    Revue des maladies respiratoires, 2021, Volume: 38, Issue:7

    Topics: Bupropion; Humans; Nicotine; Smoking; Smoking Cessation; Varenicline

2021
Tobacco Use Disorder.
    The Medical clinics of North America, 2022, Volume: 106, Issue:1

    Topics: Behavior, Addictive; Bupropion; Combined Modality Therapy; Counseling; Drug Therapy; Electronic Nicotine Delivery Systems; Humans; Morbidity; Neurobiology; Nicotine; Nicotinic Agonists; Phenotype; Prevalence; Smoking Cessation; Smoking Cessation Agents; Tobacco Use Cessation Devices; Tobacco Use Disorder; United States; Varenicline

2022
Nicotine receptor partial agonists for smoking cessation.
    The Cochrane database of systematic reviews, 2023, 05-05, Volume: 5

    Topics: Alkaloids; Bupropion; Electronic Nicotine Delivery Systems; Humans; Nicotine; Nicotinic Agonists; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2023
Cytisine for smoking cessation: A systematic review and meta-analysis.
    Drug and alcohol dependence, 2023, 10-01, Volume: 251

    Topics: Adult; Alkaloids; Azocines; Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Varenicline

2023
Pharmacological and electronic cigarette interventions for smoking cessation in adults: component network meta-analyses.
    The Cochrane database of systematic reviews, 2023, 09-12, Volume: 9

    Topics: Adult; Bupropion; Electronic Nicotine Delivery Systems; Female; Humans; Network Meta-Analysis; Nicotine; Nortriptyline; Pregnancy; Smoking Cessation; Varenicline

2023

Trials

52 trial(s) available for nicotine and varenicline

ArticleYear
Multiple-dose pharmacokinetics of the selective nicotinic receptor partial agonist, varenicline, in healthy smokers.
    Journal of clinical pharmacology, 2006, Volume: 46, Issue:12

    Topics: Administration, Oral; Adolescent; Adult; Area Under Curve; Benzazepines; Cotinine; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Half-Life; Headache; Humans; Hypotension, Orthostatic; Male; Metabolic Clearance Rate; Middle Aged; Nausea; Nicotine; Patient Dropouts; Quinoxalines; Receptors, Nicotinic; Smoking; Smoking Cessation; Smoking Prevention; Tablets; Varenicline; Vomiting

2006
Varenicline versus transdermal nicotine patch for smoking cessation: results from a randomised open-label trial.
    Thorax, 2008, Volume: 63, Issue:8

    Topics: Administration, Cutaneous; Adolescent; Adult; Aged; Benzazepines; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Patient Compliance; Quinoxalines; Reinforcement, Psychology; Smoking Cessation; Smoking Prevention; Substance Withdrawal Syndrome; Treatment Outcome; Varenicline

2008
Cognitive and antismoking effects of varenicline in patients with schizophrenia or schizoaffective disorder.
    Schizophrenia research, 2009, Volume: 110, Issue:1-3

    Topics: Adult; Analysis of Variance; Antipsychotic Agents; Benzazepines; Carbon Dioxide; Cognition; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Neuropsychological Tests; Nicotine; Prospective Studies; Psychiatric Status Rating Scales; Psychotic Disorders; Quinoxalines; Schizophrenia; Schizophrenic Psychology; Smoking; Time Factors; Varenicline

2009
Varenicline attenuates some of the subjective and physiological effects of intravenous nicotine in humans.
    Psychopharmacology, 2009, Volume: 207, Issue:1

    Topics: Adult; Affect; Benzazepines; Blood Pressure; Cognition Disorders; Cotinine; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Female; Heart Rate; Humans; Injections, Intravenous; Male; Middle Aged; Neuropsychological Tests; Nicotine; Nicotinic Agonists; Quinoxalines; Severity of Illness Index; Smoking Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2009
A randomized controlled open comparative trial of varenicline vs nicotine patch in adult smokers: efficacy, safety and withdrawal symptoms (the VN-SEESAW study).
    Circulation journal : official journal of the Japanese Circulation Society, 2010, Volume: 74, Issue:4

    Topics: Administration, Cutaneous; Adult; Benzazepines; Emotions; Endpoint Determination; Female; Humans; Incidence; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Risk Factors; Smoking; Smoking Cessation; Stress, Psychological; Substance Withdrawal Syndrome; Treatment Outcome; Varenicline

2010
Mouse model predicts effects of smoking and varenicline on event-related potentials in humans.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2010, Volume: 12, Issue:6

    Topics: Adult; Animals; Benzazepines; Cross-Over Studies; Evoked Potentials; Female; Humans; Male; Mice; Mice, Inbred C57BL; Nicotine; Placebo Effect; Quinoxalines; Smoking; Varenicline; Young Adult

2010
Cross-validation of a new procedure for early screening of smoking cessation medications in humans.
    Clinical pharmacology and therapeutics, 2010, Volume: 88, Issue:1

    Topics: Administration, Cutaneous; Adult; Benzazepines; Cross-Over Studies; Data Interpretation, Statistical; Double-Blind Method; Drug Evaluation, Preclinical; Female; Humans; Male; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Reproducibility of Results; Research Design; Smoking; Smoking Cessation; Surveys and Questionnaires; Varenicline

2010
Brain activity and emotional processing in smokers treated with varenicline.
    Addiction biology, 2013, Volume: 18, Issue:4

    Topics: Adolescent; Adult; Affect; Aged; Amygdala; Analysis of Variance; Benzazepines; Brain; Cross-Over Studies; Double-Blind Method; Emotions; Facial Expression; Female; Functional Neuroimaging; Humans; Linear Models; Magnetic Resonance Imaging; Male; Middle Aged; Nicotine; Nicotinic Agonists; Oxygen; Photic Stimulation; Placebos; Quinoxalines; Reaction Time; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Treatment Outcome; Varenicline; Young Adult

2013
Safety of varenicline among smokers enrolled in the lung HIV study.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2013, Volume: 15, Issue:1

    Topics: Adult; Benzazepines; Female; HIV Infections; Humans; Male; Middle Aged; Nicotine; Prospective Studies; Quinoxalines; Smoking Cessation; Treatment Outcome; Varenicline

2013
Effects of 21 days of varenicline versus placebo on smoking behaviors and urges among non-treatment seeking smokers.
    Journal of psychopharmacology (Oxford, England), 2012, Volume: 26, Issue:10

    Topics: Adult; alpha7 Nicotinic Acetylcholine Receptor; Behavior, Addictive; Benzazepines; Biomarkers; Cotinine; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Middle Aged; Nausea; Nicotine; Nicotinic Agonists; Patient Acceptance of Health Care; Pennsylvania; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Time Factors; Varenicline; Young Adult

2012
Varenicline to stop long-term nicotine replacement use: a double-blind, randomized, placebo-controlled trial.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2013, Volume: 15, Issue:2

    Topics: Benzazepines; Body Weight; Double-Blind Method; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Antagonists; Placebos; Quinoxalines; Smoking Cessation; Substance Withdrawal Syndrome; Surveys and Questionnaires; Varenicline

2013
Smoking quit success genotype score predicts quit success and distinct patterns of developmental involvement with common addictive substances.
    Molecular psychiatry, 2014, Volume: 19, Issue:1

    Topics: Adolescent; Benzazepines; Bupropion; Case-Control Studies; Cohort Studies; Dose-Response Relationship, Drug; Female; Genotype; Humans; Male; Nicotine; Outcome Assessment, Health Care; Polymorphism, Single Nucleotide; Quinoxalines; Reproducibility of Results; Risk Factors; Smoking Cessation; Substance-Related Disorders; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline; Young Adult

2014
Nicotinic acetylcholine receptor variation and response to smoking cessation therapies.
    Pharmacogenetics and genomics, 2013, Volume: 23, Issue:2

    Topics: Adult; Antidepressive Agents, Second-Generation; Behavior Therapy; Benzazepines; Bupropion; Female; Genotype; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Polymorphism, Single Nucleotide; Quinoxalines; Receptors, Nicotinic; Recurrence; Smoking; Smoking Cessation; Varenicline

2013
Down-regulation of amygdala and insula functional circuits by varenicline and nicotine in abstinent cigarette smokers.
    Biological psychiatry, 2013, Oct-01, Volume: 74, Issue:7

    Topics: Adolescent; Adult; Amygdala; Benzazepines; Brain Mapping; Cerebral Cortex; Double-Blind Method; Down-Regulation; Female; Humans; Magnetic Resonance Imaging; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Rest; Smoking Cessation; Varenicline; Young Adult

2013
Effects of varenicline and bupropion sustained-release use plus intensive smoking cessation counseling on prolonged abstinence from smoking and on depression, negative affect, and other symptoms of nicotine withdrawal.
    JAMA psychiatry, 2013, Volume: 70, Issue:5

    Topics: Adolescent; Adult; Affect; Aged; Benzazepines; Bupropion; Combined Modality Therapy; Counseling; Delayed-Action Preparations; Depression; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Treatment Outcome; Varenicline; Young Adult

2013
Effect of varenicline on individual nicotine withdrawal symptoms: a combined analysis of eight randomized, placebo-controlled trials.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2013, Volume: 15, Issue:11

    Topics: Adult; Aged; Benzazepines; Double-Blind Method; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Sleep Wake Disorders; Smoking Cessation; Smoking Prevention; Substance Withdrawal Syndrome; Varenicline

2013
Commitment contracts and team incentives: a randomized controlled trial for smoking cessation in Thailand.
    American journal of preventive medicine, 2013, Volume: 45, Issue:5

    Topics: Adult; Aged; Benzazepines; Contracts; Cost-Benefit Analysis; Counseling; Female; Humans; Male; Middle Aged; Motivation; Nicotine; Quinoxalines; Rural Population; Smoking Cessation; Thailand; Time Factors; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2013
A pragmatic, randomized, controlled study evaluating the impact of access to smoking cessation pharmacotherapy coverage on the proportion of successful quitters in a Canadian population of smokers motivated to quit (ACCESSATION).
    BMC public health, 2014, May-07, Volume: 14

    Topics: Benzazepines; Bupropion; Canada; Female; Health Services Accessibility; Humans; Insurance, Health; Male; Middle Aged; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2014
Efficacy of varenicline combined with nicotine replacement therapy vs varenicline alone for smoking cessation: a randomized clinical trial.
    JAMA, 2014, Volume: 312, Issue:2

    Topics: Adult; Benzazepines; Breath Tests; Carbon Monoxide; Cholinergic Agents; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Quinoxalines; Smoking Cessation; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2014
Pharmacokinetic-pharmacodynamic modeling of the effect of varenicline on nicotine craving in adult smokers.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2015, Volume: 17, Issue:1

    Topics: Adolescent; Adult; Benzazepines; Craving; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Surveys and Questionnaires; Varenicline

2015
Combining varenicline and nicotine patches: a randomized controlled trial study in smoking cessation.
    BMC medicine, 2014, Oct-08, Volume: 12

    Topics: Administration, Cutaneous; Adolescent; Adult; Benzazepines; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Cessation Devices; Tobacco Use Disorder; Treatment Outcome; Varenicline

2014
[Smoking cessation: varenicline/nicotine patch combination more effective than varenicline alone].
    Praxis, 2014, Oct-15, Volume: 103, Issue:21

    Topics: Administration, Cutaneous; Adolescent; Adult; Aged; Benzazepines; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Quinoxalines; Smoking Cessation; Treatment Outcome; Varenicline; Young Adult

2014
Impact of cigarette smoking cessation on high-density lipoprotein functionality.
    Circulation journal : official journal of the Japanese Circulation Society, 2014, Volume: 78, Issue:12

    Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Administration, Cutaneous; Adult; Apolipoprotein A-I; Benzazepines; Cardiovascular Diseases; Cholesterol; Cholesterol, HDL; Cholinergic Agonists; Female; Humans; Inflammation; Lipid Peroxidation; Lipids; Lipoproteins, HDL; Macrophages; Male; Malondialdehyde; Middle Aged; Nicotine; Oxidation-Reduction; Quinoxalines; Receptors, Nicotinic; Risk Factors; Smoking; Smoking Cessation; Varenicline

2014
Use of the nicotine metabolite ratio as a genetically informed biomarker of response to nicotine patch or varenicline for smoking cessation: a randomised, double-blind placebo-controlled trial.
    The Lancet. Respiratory medicine, 2015, Volume: 3, Issue:2

    Topics: Adult; Biomarkers; Cotinine; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Smoking Cessation; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2015
Increasing progesterone levels are associated with smoking abstinence among free-cycling women smokers who receive brief pharmacotherapy.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2015, Volume: 17, Issue:4

    Topics: Adolescent; Adult; Benzazepines; Estradiol; Female; Humans; Menstrual Cycle; Middle Aged; Nicotine; Nicotinic Agonists; Progesterone; Quinoxalines; Smoking Cessation; Transdermal Patch; Treatment Outcome; Varenicline; Women's Health

2015
The Nicotine Metabolite Ratio is Associated With Early Smoking Abstinence Even After Controlling for Factors That Influence the Nicotine Metabolite Ratio.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2016, Volume: 18, Issue:4

    Topics: Adult; Female; Humans; Male; Middle Aged; Nicotine; Prospective Studies; Smoking; Smoking Cessation; Time Factors; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2016
Effects of Nicotine Patch vs Varenicline vs Combination Nicotine Replacement Therapy on Smoking Cessation at 26 Weeks: A Randomized Clinical Trial.
    JAMA, 2016, Jan-26, Volume: 315, Issue:4

    Topics: Adult; Carbon Monoxide; Counseling; Female; Humans; Intention to Treat Analysis; Male; Medication Adherence; Middle Aged; Nicotine; Nicotinic Agonists; Outcome Assessment, Health Care; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Time Factors; Tobacco Use Cessation Devices; Varenicline

2016
    Praxis, 2016, Volume: 105, Issue:24

    Topics: Adolescent; Adult; Aged; Anxiety Disorders; Bupropion; Cohort Studies; Comorbidity; Double-Blind Method; Female; Humans; Male; Middle Aged; Mood Disorders; Nicotine; Smoking Cessation; Varenicline; Young Adult

2016
Factor structure of the Smoking Cessation Self-Efficacy Questionnaire among smokers with and without a psychiatric diagnosis.
    Psychology of addictive behaviors : journal of the Society of Psychologists in Addictive Behaviors, 2017, Volume: 31, Issue:2

    Topics: Adult; Factor Analysis, Statistical; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Outcome Assessment, Health Care; Self Efficacy; Smoking Cessation; Surveys and Questionnaires; Tobacco Use Cessation Devices; Varenicline

2017
Neural Signatures of Cognitive Flexibility and Reward Sensitivity Following Nicotinic Receptor Stimulation in Dependent Smokers: A Randomized Trial.
    JAMA psychiatry, 2017, 06-01, Volume: 74, Issue:6

    Topics: Adult; Cerebral Cortex; Cross-Over Studies; Double-Blind Method; Executive Function; Female; Humans; Impulsive Behavior; Limbic System; Male; Motivation; Nicotine; Receptors, Nicotinic; Reversal Learning; Reward; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2017
Effects of varenicline versus transdermal nicotine replacement therapy on cigarette demand on quit day in individuals with substance use disorders.
    Psychopharmacology, 2017, Volume: 234, Issue:16

    Topics: Administration, Cutaneous; Adult; Craving; Double-Blind Method; Female; Humans; Male; Middle Aged; Nicotine; Reinforcement, Psychology; Smoking; Smoking Cessation; Smoking Prevention; Substance-Related Disorders; Treatment Outcome; Varenicline

2017
Nicotine Metabolism-informed Care for Smoking Cessation: A Pilot Precision RCT.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2018, 11-15, Volume: 20, Issue:12

    Topics: Adult; Female; Follow-Up Studies; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Pilot Projects; Precision Medicine; Smoking Cessation; Smoking Cessation Agents; Tobacco Smoking; Tobacco Use Cessation Devices; Varenicline

2018
Nicotine metabolite ratio and smoking outcomes using nicotine replacement therapy and varenicline among smokers with and without psychiatric illness.
    Journal of psychopharmacology (Oxford, England), 2018, Volume: 32, Issue:9

    Topics: Female; Humans; Male; Mental Disorders; Middle Aged; Nicotine; Smoking; Smoking Cessation; Smoking Cessation Agents; Time Factors; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2018
Predicting smoking abstinence with biological and self-report measures of adherence to varenicline: Impact on pharmacogenetic trial outcomes.
    Drug and alcohol dependence, 2018, 09-01, Volume: 190

    Topics: Adult; Female; Humans; Male; Medication Adherence; Middle Aged; Nicotine; Nicotinic Agonists; Pharmacogenetics; Predictive Value of Tests; Self Report; Smoking; Smoking Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2018
Mediators of the effect of nicotine pre-treatment on quitting smoking.
    Addiction (Abingdon, England), 2018, Volume: 113, Issue:12

    Topics: Adult; Behavior Therapy; Bupropion; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Premedication; Smoking; Smoking Cessation; Smoking Cessation Agents; Tobacco Use Cessation Devices; Varenicline

2018
Nicotine preloading for smoking cessation: the Preloading RCT.
    Health technology assessment (Winchester, England), 2018, Volume: 22, Issue:41

    Topics: Adult; Aged; Cost-Benefit Analysis; Female; Humans; Male; Middle Aged; Nicotine; Smoking Cessation; Smoking Cessation Agents; State Medicine; United Kingdom; Varenicline

2018
A randomized controlled trial of 24 weeks of varenicline for tobacco use among cancer patients: Efficacy, safety, and adherence.
    Psycho-oncology, 2019, Volume: 28, Issue:3

    Topics: Adult; Benzazepines; Counseling; Female; Humans; Male; Medication Adherence; Middle Aged; Neoplasms; Nicotine; Smoking; Smoking Cessation; Smoking Cessation Agents; Substance Withdrawal Syndrome; Treatment Outcome; Varenicline

2019
Anxiety Sensitivity and Distress Tolerance in Smokers: Relations With Tobacco Dependence, Withdrawal, and Quitting Success†.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2020, 01-27, Volume: 22, Issue:1

    Topics: Adolescent; Adult; Anxiety Disorders; Child; Ecological Momentary Assessment; Female; Humans; Male; Middle Aged; Motivation; Nicotine; Nicotinic Agonists; Smokers; Smoking Cessation; Stress, Psychological; Substance Withdrawal Syndrome; Surveys and Questionnaires; Tobacco Use Disorder; Varenicline; Young Adult

2020
The Relationship of Varenicline Agonism of α4β2 Nicotinic Acetylcholine Receptors and Nicotine-Induced Dopamine Release in Nicotine-Dependent Humans.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2020, 05-26, Volume: 22, Issue:6

    Topics: Adolescent; Adult; Brain; Dopamine; Double-Blind Method; Female; Humans; Male; Maryland; Middle Aged; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline; Young Adult

2020
Genetic Variant in CHRNA5 and Response to Varenicline and Combination Nicotine Replacement in a Randomized Placebo-Controlled Trial.
    Clinical pharmacology and therapeutics, 2020, Volume: 108, Issue:6

    Topics: Administration, Cutaneous; Administration, Oral; Adult; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Missouri; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Pharmacogenetics; Pharmacogenomic Variants; Prospective Studies; Race Factors; Receptors, Nicotinic; Smokers; Smoking Cessation; Smoking Cessation Agents; Time Factors; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2020
Medication adherence and rate of nicotine metabolism are associated with response to treatment with varenicline among smokers with HIV.
    Addictive behaviors, 2021, Volume: 112

    Topics: Adolescent; Benzazepines; HIV Infections; Humans; Medication Adherence; Nicotine; Nicotinic Agonists; Quinoxalines; Smokers; Varenicline

2021
Rationale and design of a randomized factorial clinical trial of pharmacogenetic and adherence optimization strategies to promote tobacco cessation among persons with HIV.
    Contemporary clinical trials, 2021, Volume: 110

    Topics: HIV Infections; Humans; Nicotine; Nicotinic Agonists; Pharmacogenetics; Tobacco Use Cessation; Varenicline

2021
Time-Varying Mediation of Pharmacological Smoking Cessation Treatments on Smoking Lapse via Craving, Cessation Fatigue, and Negative Mood.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2022, 10-17, Volume: 24, Issue:10

    Topics: Craving; Fatigue; Humans; Nicotine; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Smoking; Varenicline

2022
Cytisine Therapy Improved Smoking Cessation in the Randomized Screening and Multiple Intervention on Lung Epidemics Lung Cancer Screening Trial.
    Journal of thoracic oncology : official publication of the International Association for the Study of Lung Cancer, 2022, Volume: 17, Issue:11

    Topics: Alkaloids; Azocines; Early Detection of Cancer; Humans; Lung; Lung Neoplasms; Nicotine; Quinolizines; Smoking Cessation; Varenicline

2022
Effectiveness of Varenicline and Cytisine for Alcohol Use Reduction Among People With HIV and Substance Use: A Randomized Clinical Trial.
    JAMA network open, 2022, 08-01, Volume: 5, Issue:8

    Topics: Adult; Alcoholism; Alkaloids; Azocines; Benzazepines; Female; HIV Infections; Humans; Male; Nicotine; Nicotinic Agonists; Quinolizines; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2022
Influence of CYP2A6 Genetic Variation, Nicotine Dependence Severity, and Treatment on Smoking Cessation Success.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2023, 05-22, Volume: 25, Issue:6

    Topics: Adult; Cytochrome P-450 CYP2A6; Female; Genetic Variation; Humans; Male; Nicotine; Smoking Cessation; Tobacco Use Disorder; Varenicline

2023
Glucagon-like peptide-1 analogues: a new way to quit smoking? (SKIP)-a structured summary of a study protocol for a randomized controlled study.
    Trials, 2023, Apr-20, Volume: 24, Issue:1

    Topics: Double-Blind Method; Glucagon-Like Peptide 1; Humans; Nicotine; Randomized Controlled Trials as Topic; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline; Weight Gain

2023
Cytisine Versus Varenicline for Smoking Cessation in a Primary Care Setting: A Randomized Non-inferiority Trial.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2023, 08-19, Volume: 25, Issue:9

    Topics: Alkaloids; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Primary Health Care; Quinolizines; Smoking Cessation; Treatment Outcome; Varenicline

2023
Multiple Pharmacotherapy Adaptations for Smoking Cessation Based on Treatment Response in Black Adults Who Smoke: A Randomized Clinical Trial.
    JAMA network open, 2023, 06-01, Volume: 6, Issue:6

    Topics: Adult; Bupropion; Ethnicity; Female; Humans; Male; Middle Aged; Minority Groups; Nicotine; Smoking; Smoking Cessation; Varenicline

2023
Adaptive Smoking Cessation Using Precessation Varenicline or Nicotine Patch: A Randomized Clinical Trial.
    JAMA network open, 2023, 09-05, Volume: 6, Issue:9

    Topics: Bupropion; COVID-19; Female; Humans; Male; Middle Aged; Nicotine; Pandemics; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2023
Effectiveness of nicotine salt vapes, cytisine, and a combination of these products, for smoking cessation in New Zealand: protocol for a three-arm, pragmatic, community-based randomised controlled trial.
    BMC public health, 2023, 09-11, Volume: 23, Issue:1

    Topics: Electronic Nicotine Delivery Systems; Humans; New Zealand; Nicotine; Quality of Life; Randomized Controlled Trials as Topic; Smoking Cessation; Sodium Chloride, Dietary; Tobacco Use Cessation Devices; Vaping; Varenicline

2023
The impact of blunt use on smoking abstinence among Black adults: Secondary analysis from randomized controlled smoking cessation clinical trial.
    Addictive behaviors, 2024, Volume: 148

    Topics: Adult; Aged; Aged, 80 and over; Black or African American; Female; Humans; Male; Middle Aged; Nicotine; Smoking; Smoking Cessation; Varenicline; Young Adult

2024

Other Studies

213 other study(ies) available for nicotine and varenicline

ArticleYear
3,5-Bicyclic aryl piperidines: a novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation.
    Bioorganic & medicinal chemistry letters, 2005, Nov-15, Volume: 15, Issue:22

    Topics: Animals; Cyclization; Molecular Structure; Piperidines; Rats; Receptors, Nicotinic; Smoking Cessation; Structure-Activity Relationship

2005
Synthesis, nicotinic acetylcholine receptor binding, and pharmacological properties of 3'-(substituted phenyl)deschloroepibatidine analogs.
    Bioorganic & medicinal chemistry, 2008, Jan-15, Volume: 16, Issue:2

    Topics: Analgesics; Animals; Body Temperature; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Disease Models, Animal; Dose-Response Relationship, Drug; Mice; Molecular Structure; Nicotinic Antagonists; Pain; Protein Binding; Pyridines; Radioligand Assay; Receptors, Nicotinic; Structure-Activity Relationship

2008
Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 3'-(substituted phenyl)epibatidine analogues. Nicotinic partial agonists.
    Journal of natural products, 2010, Mar-26, Volume: 73, Issue:3

    Topics: Analgesics; Animals; Bridged Bicyclo Compounds, Heterocyclic; Male; Mice; Molecular Structure; Nicotinic Agonists; Pyridines; Rats; Receptors, Nicotinic

2010
A novel series of [3.2.1] azabicyclic biaryl ethers as alpha3beta4 and alpha6/4beta4 nicotinic receptor agonists.
    Bioorganic & medicinal chemistry letters, 2010, Aug-15, Volume: 20, Issue:16

    Topics: Azabicyclo Compounds; Nicotinic Agonists; Receptors, Nicotinic; Structure-Activity Relationship; Sulfonamides

2010
Unichiral 2-(2'-pyrrolidinyl)-1,4-benzodioxanes: the 2R,2'S diastereomer of the N-methyl-7-hydroxy analogue is a potent α4β2- and α6β2-nicotinic acetylcholine receptor partial agonist.
    Journal of medicinal chemistry, 2011, Nov-10, Volume: 54, Issue:21

    Topics: Animals; Binding Sites; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine; Drug Partial Agonism; HEK293 Cells; Humans; In Vitro Techniques; Male; Models, Molecular; Nicotinic Agonists; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2011
Identification of novel α4β2-nicotinic acetylcholine receptor (nAChR) agonists based on an isoxazole ether scaffold that demonstrate antidepressant-like activity.
    Journal of medicinal chemistry, 2012, Jan-26, Volume: 55, Issue:2

    Topics: Animals; Antidepressive Agents; Blood Proteins; Cytochrome P-450 Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; HEK293 Cells; Humans; Isoxazoles; Male; Mice; Mice, Inbred BALB C; Microsomes, Liver; Nicotinic Agonists; Protein Binding; Radioligand Assay; Rats; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Synthesis and nicotinic receptor activity of chemical space analogues of N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chlorobenzamide (PNU-282,987) and 1,4-diazabicyclo[3.2.2]nonane-4-carboxylic acid 4-bromophenyl ester (SSR180711).
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Allosteric Regulation; Animals; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Databases, Factual; Female; Humans; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Patch-Clamp Techniques; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship; Xenopus

2012
Structure-activity studies of 7-heteroaryl-3-azabicyclo[3.3.1]non-6-enes: a novel class of highly potent nicotinic receptor ligands.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cells, Cultured; Electrophysiology; Humans; Kidney; Ligands; Molecular Structure; Neuroblastoma; Nicotine; Protein Subunits; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2012
Discovery of highly potent and selective α4β2-nicotinic acetylcholine receptor (nAChR) partial agonists containing an isoxazolylpyridine ether scaffold that demonstrate antidepressant-like activity. Part II.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Animals; Antidepressive Agents; Humans; Isoxazoles; Male; Mice; Mice, Inbred BALB C; Motor Activity; Neuroblastoma; Nicotinic Agonists; Protein Binding; Radioligand Assay; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship; Swimming

2012
Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective α4β2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats.
    Journal of medicinal chemistry, 2013, Apr-11, Volume: 56, Issue:7

    Topics: Alcohol Drinking; Animals; Ethanol; Ferrets; Ligands; Magnetic Resonance Spectroscopy; Pyridines; Rats; Receptors, Nicotinic; Spectrometry, Mass, Electrospray Ionization

2013
Design, synthesis and discovery of picomolar selective α4β2 nicotinic acetylcholine receptor ligands.
    Journal of medicinal chemistry, 2013, Nov-14, Volume: 56, Issue:21

    Topics: Azetidines; Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Discovery; Humans; Ligands; Models, Molecular; Molecular Structure; Pyridines; Receptors, Nicotinic; Software; Structure-Activity Relationship

2013
Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted pyridinyl)-7-deschloroepibatidine analogues.
    Journal of medicinal chemistry, 2014, Feb-13, Volume: 57, Issue:3

    Topics: Analgesics; Animals; Body Temperature; Bridged Bicyclo Compounds, Heterocyclic; Contraindications; Female; Male; Mice; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Pain; Patch-Clamp Techniques; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Structure-Activity Relationship; Xenopus

2014
Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selective α4β2-nAChR Ligands.
    ACS medicinal chemistry letters, 2014, Nov-13, Volume: 5, Issue:11

    Topics:

2014
Synthesis, nicotinic acetylcholine receptor binding, in vitro and in vivo pharmacology properties of 3'-(substituted pyridinyl)-deschloroepibatidine analogs.
    Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Humans; Mice; Molecular Structure; Nicotiana; Pyridines; Rats; Receptors, Nicotinic; Structure-Activity Relationship

2015
[Medication for ending tobacco dependency. Current state].
    Atencion primaria, 2005, Jun-30, Volume: 36, Issue:2

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Cannabinoid Receptor Antagonists; Humans; Nicotine; Piperidines; Pyrazoles; Quinoxalines; Receptors, Nicotinic; Rimonabant; Smoking Cessation; Time Factors; Tobacco Use Disorder; Varenicline

2005
Ligands selective for alpha4beta2 but not alpha3beta4 or alpha7 nicotinic receptors generalise to the nicotine discriminative stimulus in the rat.
    Psychopharmacology, 2007, Volume: 190, Issue:2

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Appetitive Behavior; Azetidines; Benzazepines; Corpus Striatum; Cystine; Discrimination Learning; Dose-Response Relationship, Drug; Male; Motivation; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Tobacco Use Disorder; Varenicline

2007
Pharmacological profile of the alpha4beta2 nicotinic acetylcholine receptor partial agonist varenicline, an effective smoking cessation aid.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Animals; Behavior, Animal; Benzazepines; Brain; Cell Line, Transformed; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; In Vitro Techniques; Male; Membrane Potentials; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Protein Binding; Quinoxalines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Self Administration; Smoking Cessation; Transfection; Varenicline

2007
[The path from cigarettes--with support it works better].
    Medizinische Monatsschrift fur Pharmazeuten, 2007, Volume: 30, Issue:3

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Varenicline

2007
Exacerbation of schizophrenia by varenicline.
    The American journal of psychiatry, 2007, Volume: 164, Issue:8

    Topics: Acute Disease; Benzazepines; Cognition Disorders; Comorbidity; Female; Humans; Middle Aged; Nicotine; Quinoxalines; Recurrence; Schizophrenia; Schizophrenic Psychology; Self Medication; Smoking; Smoking Cessation; Varenicline

2007
Cost-effectiveness of varenicline compared with bupropion, NRT, and nortriptyline for smoking cessation in the Netherlands.
    Current medical research and opinion, 2008, Volume: 24, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Benzazepines; Bupropion; Cost-Benefit Analysis; Female; Health Care Costs; Humans; Male; Middle Aged; Models, Theoretical; Netherlands; Nicotine; Nortriptyline; Quality of Life; Quinoxalines; Smoking; Smoking Cessation; Varenicline

2008
Varenicline in the routine treatment of tobacco dependence: a pre-post comparison with nicotine replacement therapy and an evaluation in those with mental illness.
    Addiction (Abingdon, England), 2008, Volume: 103, Issue:1

    Topics: Adult; Benzazepines; Cohort Studies; Drug Combinations; Female; Follow-Up Studies; Humans; London; Male; Mental Disorders; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Disorder; Treatment Outcome; Varenicline

2008
[New drugs; varenicline].
    Nederlands tijdschrift voor geneeskunde, 2007, Nov-10, Volume: 151, Issue:45

    Topics: Benzazepines; Humans; Nausea; Nicotine; Nicotinic Agonists; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline

2007
The truth about smoking cessation.
    The Johns Hopkins medical letter health after 50, 2007, Volume: 19, Issue:8

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Counseling; Humans; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Varenicline

2007
Breaking away from a narrow prescribing protocol for medicinal nicotine.
    Addiction (Abingdon, England), 2008, Volume: 103, Issue:4

    Topics: Administration, Cutaneous; Adult; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Patient Acceptance of Health Care; Quinoxalines; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2008
Stat bite: Medicaid coverage of tobacco-dependence treatments.
    Journal of the National Cancer Institute, 2008, Apr-02, Volume: 100, Issue:7

    Topics: Administration, Cutaneous; Administration, Intranasal; Administration, Oral; Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Counseling; Dopamine Uptake Inhibitors; Female; Humans; Insurance Coverage; Male; Medicaid; Nicotine; Nicotinic Agonists; Pregnancy; Pregnancy Complications; Quinoxalines; Tobacco Use Disorder; United States; Varenicline

2008
Smoking cessation 2008.
    IDrugs : the investigational drugs journal, 2008, Volume: 11, Issue:4

    Topics: Benzazepines; Cannabinoid Receptor Antagonists; Drug Prescriptions; Humans; Marketing of Health Services; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking; Smoking Cessation; Smoking Prevention; Vaccines; Varenicline

2008
Pharmacological effects of nicotine on norepinephrine metabolism in rat brown adipose tissue: relevance to nicotinic therapies for smoking cessation.
    Toxicologic pathology, 2008, Volume: 36, Issue:4

    Topics: Adipose Tissue, Brown; Animals; Benzazepines; Dose-Response Relationship, Drug; Female; Lipoma; Male; Mediastinal Neoplasms; Nicotine; Nicotinic Agonists; Norepinephrine; Quinoxalines; Rats; Rats, Sprague-Dawley; Sex Factors; Smoking Cessation; Varenicline

2008
Cost-utility analysis of varenicline versus existing smoking cessation strategies using the BENESCO Simulation model: application to a population of US adult smokers.
    PharmacoEconomics, 2008, Volume: 26, Issue:6

    Topics: Adolescent; Adult; Benzazepines; Bupropion; Costs and Cost Analysis; Drug Costs; Female; Humans; Male; Markov Chains; Middle Aged; Models, Statistical; Nicotine; Quinoxalines; Smoking; Smoking Cessation; United States; Varenicline

2008
Pre-cessation varenicline treatment vs post-cessation NRT: an uneven playing field.
    Thorax, 2008, Volume: 63, Issue:8

    Topics: Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Smoking Prevention; Varenicline

2008
Clinically significant outcomes in smoking cessation.
    Thorax, 2008, Volume: 63, Issue:8

    Topics: Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Smoking Prevention; Treatment Outcome; Varenicline

2008
Effect of varenicline on the acute and repeated locomotor responses to nicotine in rats.
    Synapse (New York, N.Y.), 2008, Volume: 62, Issue:12

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Benzazepines; Drug Administration Schedule; Male; Motor Activity; Nicotine; Quinoxalines; Rats; Rats, Wistar; Receptors, Nicotinic; Varenicline

2008
Effects of the nicotinic receptor partial agonists varenicline and cytisine on the discriminative stimulus effects of nicotine in rats.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 91, Issue:3

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Conditioning, Operant; Data Interpretation, Statistical; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Rats, Long-Evans; Receptors, Nicotinic; Varenicline

2009
An algorithm for tailoring pharmacotherapy for smoking cessation: results from a Delphi panel of international experts.
    Tobacco control, 2009, Volume: 18, Issue:1

    Topics: Algorithms; Behavior Therapy; Benzazepines; Bupropion; Combined Modality Therapy; Consensus; Decision Support Techniques; Delphi Technique; Humans; Nicotine; Nicotinic Agonists; Practice Patterns, Physicians'; Quinoxalines; Smoking Cessation; Varenicline

2009
Targeting reward-relevant nicotinic receptors in the discovery of novel pharmacotherapeutic agents to treat tobacco dependence.
    Nebraska Symposium on Motivation. Nebraska Symposium on Motivation, 2009, Volume: 55

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Benzazepines; Brain; Bupropion; Dopamine; Dose-Response Relationship, Drug; Drugs, Investigational; Male; Neurons; Nicotine; Nicotinic Antagonists; Picolines; Quaternary Ammonium Compounds; Quinoxalines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, Nicotinic; Reward; Smoking Cessation; Structure-Activity Relationship; Tobacco Use Disorder; Varenicline; Ventral Tegmental Area

2009
[Drug treatment for smoking and marijuana abuse].
    Revue des maladies respiratoires, 2008, Volume: 25, Issue:10

    Topics: Antidepressive Agents, Second-Generation; Benzazepines; Humans; Marijuana Abuse; Nicotine; Nicotinic Agonists; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline

2008
The smoking cessation medication varenicline attenuates alcohol and nicotine interactions in the rat mesolimbic dopamine system.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 329, Issue:1

    Topics: Animals; Benzazepines; Central Nervous System Depressants; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Limbic System; Male; Microdialysis; Nicotine; Nucleus Accumbens; Quinoxalines; Rats; Rats, Wistar; Smoking Cessation; Varenicline

2009
Do implementation issues influence the effectiveness of medications? The case of nicotine replacement therapy and bupropion in UK Stop Smoking Services.
    BMC public health, 2009, Jan-21, Volume: 9

    Topics: Administration, Cutaneous; Adult; Benzazepines; Bupropion; Cohort Studies; Community Health Services; Female; Follow-Up Studies; Humans; Logistic Models; Male; Middle Aged; Multivariate Analysis; Nicotine; Nicotinic Agonists; Patient Participation; Probability; Program Evaluation; Quinoxalines; Randomized Controlled Trials as Topic; Risk Factors; Smoking; Smoking Cessation; Smoking Prevention; Treatment Outcome; United Kingdom; Varenicline; Young Adult

2009
A reader responds to "Seven pharmacotherapies do promote smoking abstinence at 6 and 12 months".
    Medscape journal of medicine, 2008, Volume: 10, Issue:12

    Topics: Administration, Cutaneous; Administration, Inhalation; Administration, Oral; Benzazepines; Bupropion; Chewing Gum; Female; Follow-Up Studies; Humans; Male; Multivariate Analysis; Nicotine; Nicotinic Agonists; Patient Compliance; Probability; Quebec; Quinoxalines; Risk Assessment; Smoking; Smoking Cessation; Smoking Prevention; Tobacco Use Disorder; Treatment Outcome; Varenicline

2008
Combination treatment with varenicline and nicotine replacement therapy.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2009, Volume: 11, Issue:5

    Topics: Adult; Aged; Benzazepines; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Outcome Assessment, Health Care; Quinoxalines; Smoking Cessation; Varenicline

2009
Varenicline attenuates nicotine-enhanced brain-stimulation reward by activation of alpha4beta2 nicotinic receptors in rats.
    Neuropharmacology, 2009, Volume: 57, Issue:1

    Topics: Animals; Benzazepines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Male; Medial Forebrain Bundle; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Rats; Rats, Long-Evans; Receptors, Nicotinic; Reward; Varenicline

2009
Treatment of comorbid tobacco use in people with serious mental illness.
    Journal of psychiatry & neuroscience : JPN, 2009, Volume: 34, Issue:3

    Topics: Adult; Benzazepines; Bupropion; Comorbidity; Counseling; Dopamine Uptake Inhibitors; Female; Follow-Up Studies; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Schizophrenia, Paranoid; Smoking; Smoking Cessation; Varenicline

2009
Cost-effectiveness of varenicline compared with nicotine patches for smoking cessation--results from four European countries.
    European journal of public health, 2009, Volume: 19, Issue:6

    Topics: Adolescent; Adult; Aged; Benzazepines; Cost-Benefit Analysis; Europe; Female; Heart Diseases; Humans; Incidence; Lung Neoplasms; Male; Markov Chains; Middle Aged; Models, Statistical; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Quality-Adjusted Life Years; Quinoxalines; Smoking; Smoking Cessation; Stroke; Varenicline; Young Adult

2009
[Current and future medical drugs for smoking cessation].
    Laryngo- rhino- otologie, 2009, Volume: 88, Issue:6

    Topics: Adrenergic alpha-Agonists; Antidepressive Agents; Behavior Therapy; Benzazepines; Bupropion; Cannabinoid Receptor Antagonists; Clinical Trials as Topic; Clonidine; Combined Modality Therapy; Counseling; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking Cessation; Tobacco Use Disorder; Vaccines; Varenicline

2009
Cost-effectiveness of varenicline for smoking cessation.
    Expert review of pharmacoeconomics & outcomes research, 2009, Volume: 9, Issue:3

    Topics: Benzazepines; Bupropion; Clinical Trials as Topic; Cost Savings; Cost-Benefit Analysis; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Varenicline

2009
Cost effectiveness of varenicline in Belgium, compared with bupropion, nicotine replacement therapy, brief counselling and unaided smoking cessation: a BENESCO Markov cost-effectiveness analysis.
    Clinical drug investigation, 2009, Volume: 29, Issue:10

    Topics: Adolescent; Adult; Age Factors; Aged; Antidepressive Agents, Second-Generation; Belgium; Benzazepines; Bupropion; Computer Simulation; Cost-Benefit Analysis; Counseling; Female; Humans; Male; Markov Chains; Middle Aged; Models, Statistical; Nicotine; Nicotinic Agonists; Quinoxalines; Recurrence; Smoking; Smoking Cessation; Treatment Outcome; Varenicline; Young Adult

2009
Smoking cessation: how to advise the patient.
    Heart (British Cardiac Society), 2009, Volume: 95, Issue:19

    Topics: Ambulatory Care; Behavior Therapy; Benzazepines; Bupropion; Counseling; Dopamine Uptake Inhibitors; Humans; Motivation; Nicotine; Nicotinic Agonists; Patient Education as Topic; Physician-Patient Relations; Quinoxalines; Secondary Prevention; Smoking Cessation; Smoking Prevention; Varenicline

2009
Varenicline and suicidal behaviour: a cohort study based on data from the General Practice Research Database.
    BMJ (Clinical research ed.), 2009, Oct-01, Volume: 339

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Benzazepines; Bupropion; Cohort Studies; Dopamine Uptake Inhibitors; Family Practice; Female; Ganglionic Stimulants; Humans; Male; Middle Aged; Nicotine; Quinoxalines; Smoking Cessation; Suicide; Varenicline; Young Adult

2009
Effect of the alpha4beta2* nicotinic acetylcholine receptor partial agonist varenicline on dopamine release in beta2 knock-out mice with selective re-expression of the beta2 subunit in the ventral tegmental area.
    Neuropharmacology, 2010, Volume: 58, Issue:2

    Topics: Animals; Benzazepines; Dopamine; Extracellular Space; Genetic Vectors; Green Fluorescent Proteins; Lentivirus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Nicotine; Nicotinic Agonists; Nucleus Accumbens; Quinoxalines; Receptors, Nicotinic; Varenicline

2010
[Drug treatment of tobacco dependence].
    Deutsche medizinische Wochenschrift (1946), 2009, Volume: 134, Issue:47

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Humans; Meta-Analysis as Topic; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2009
The alpha4beta2 nicotinic acetylcholine-receptor partial agonist varenicline inhibits both nicotine self-administration following repeated dosing and reinstatement of nicotine seeking in rats.
    Psychopharmacology, 2010, Volume: 208, Issue:3

    Topics: Animals; Association Learning; Behavior, Animal; Benzazepines; Conditioning, Operant; Cues; Dose-Response Relationship, Drug; Exploratory Behavior; Food; Male; Models, Animal; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Receptors, Nicotinic; Recurrence; Reinforcement, Psychology; Self Administration; Tobacco Use Disorder; Varenicline

2010
Effects of varenicline and mecamylamine on the acquisition, expression, and reinstatement of nicotine-conditioned place preference by drug priming in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2010, Volume: 381, Issue:4

    Topics: Animals; Benzazepines; Conditioning, Classical; Dose-Response Relationship, Drug; Male; Mecamylamine; Morphine; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Rats; Rats, Wistar; Receptors, Nicotinic; Reward; Tobacco Use Disorder; Varenicline

2010
Extinction with varenicline and nornicotine, but not ABT-418, weakens conditioned responding evoked by the interoceptive stimulus effects of nicotine.
    Neuropharmacology, 2010, Volume: 58, Issue:8

    Topics: Animals; Benzazepines; Conditioning, Classical; Discrimination, Psychological; Extinction, Psychological; Generalization, Psychological; Isoxazoles; Ligands; Male; Nicotine; Nicotinic Agonists; Pyrrolidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Varenicline

2010
Varenicline treatment decreases DNMT1 mRNA expression in lymphocytes of schizophrenic patients who are cigarette smokers.
    Schizophrenia research, 2010, Volume: 119, Issue:1-3

    Topics: Benzazepines; Cotinine; DNA (Cytosine-5-)-Methyltransferase 1; DNA (Cytosine-5-)-Methyltransferases; Gene Expression; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; RNA, Messenger; Schizophrenia; Smoking Cessation; Varenicline

2010
Characteristics and abstinence outcomes among tobacco quitline enrollees using varenicline or nicotine replacement therapy.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2010, Volume: 12, Issue:6

    Topics: Adolescent; Adult; Benzazepines; Counseling; Female; Humans; Male; Montana; Nicotine; Nicotinic Agonists; Quinoxalines; Retrospective Studies; Smoking Cessation; Telephone; Tobacco Use Disorder; Treatment Outcome; Varenicline; Young Adult

2010
Nicotinic partial agonists varenicline and sazetidine-A have differential effects on affective behavior.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 334, Issue:2

    Topics: Animals; Anxiety; Azetidines; Behavior, Animal; Benzazepines; Chimera; Depression; Drug Partial Agonism; Male; Mice; Mood Disorders; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Varenicline

2010
Varenicline and mecamylamine attenuate locomotor sensitization and cross-sensitization induced by nicotine and morphine in mice.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 96, Issue:2

    Topics: Analgesics, Opioid; Animals; Benzazepines; Dose-Response Relationship, Drug; Drug Interactions; Male; Mecamylamine; Mice; Morphine; Motor Activity; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Varenicline

2010
Current treatment options in smoking cessation.
    Hospital practice (1995), 2010, Volume: 38, Issue:1

    Topics: Adrenergic alpha-Agonists; Antidepressive Agents; Behavior Therapy; Benzazepines; Bupropion; Clonidine; Combined Modality Therapy; Counseling; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Patient Selection; Piperidines; Practice Guidelines as Topic; Pyrazoles; Quinoxalines; Rimonabant; Self-Help Groups; Smoking Cessation; Tobacco Use Disorder; United States; Vaccines; Varenicline

2010
The use of snus for quitting smoking compared with medicinal products.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2010, Volume: 12, Issue:8

    Topics: Adult; Benzazepines; Chewing Gum; Data Collection; Humans; Male; Middle Aged; Nicotine; Quinoxalines; Regression Analysis; Smoking Cessation; Tobacco, Smokeless; Varenicline

2010
[The management of patients with nicotine dependence - the role of the general practitioners].
    Therapeutische Umschau. Revue therapeutique, 2010, Volume: 67, Issue:8

    Topics: Behavior Therapy; Benzazepines; Bupropion; Combined Modality Therapy; Disease Management; Dopamine Uptake Inhibitors; Family Practice; Humans; Motivation; Nicotine; Nicotinic Agonists; Physician-Patient Relations; Quinoxalines; Secondary Prevention; Smoking Cessation; Switzerland; Tobacco Use Disorder; Varenicline

2010
[Medical therapy for smoking cessation].
    Therapeutische Umschau. Revue therapeutique, 2010, Volume: 67, Issue:8

    Topics: Administration, Cutaneous; Administration, Inhalation; Administration, Oral; Antidepressive Agents; Benzazepines; Bupropion; Chewing Gum; Drug Therapy, Combination; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2010
Varenicline blocks nicotine intake in rats with extended access to nicotine self-administration.
    Psychopharmacology, 2011, Volume: 213, Issue:4

    Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Male; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Wistar; Receptors, Nicotinic; Reinforcement, Psychology; Self Administration; Varenicline

2011
Abstinence and psychological distress in co-morbid smokers using various pharmacotherapies.
    Drug and alcohol dependence, 2011, Mar-01, Volume: 114, Issue:1

    Topics: Adult; Aged; Benzazepines; Bupropion; Cohort Studies; Comorbidity; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nicotine; Quinoxalines; Retrospective Studies; Smoking; Smoking Cessation; Stress, Psychological; Treatment Outcome; Varenicline; Young Adult

2011
The sensitizing effect of acute nicotine on amphetamine-stimulated behavior and dopamine efflux requires activation of β2 subunit-containing nicotinic acetylcholine receptors and glutamate N-methyl-D-aspartate receptors.
    Neuropharmacology, 2011, Volume: 60, Issue:7-8

    Topics: Aconitine; Amphetamine; Animals; Behavior, Animal; Benzazepines; Central Nervous System Stimulants; Dizocilpine Maleate; Dopamine; Excitatory Amino Acid Antagonists; Female; Male; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Nicotinic; Varenicline

2011
Parallel anxiolytic-like effects and upregulation of neuronal nicotinic acetylcholine receptors following chronic nicotine and varenicline.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2011, Volume: 13, Issue:1

    Topics: Animals; Benzazepines; Cerebral Cortex; Hippocampus; Male; Mice; Nicotine; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Thalamus; Up-Regulation; Varenicline

2011
Adherence to and reasons for premature discontinuation from stop-smoking medications: data from the ITC Four-Country Survey.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2011, Volume: 13, Issue:2

    Topics: Adolescent; Adult; Aged; Australia; Benzazepines; Bupropion; Canada; Cohort Studies; Data Collection; Female; Humans; Male; Medication Adherence; Middle Aged; Nicotine; Nonprescription Drugs; Prescription Drugs; Prevalence; Quinoxalines; Smoking Cessation; Time Factors; Tobacco Use Disorder; Treatment Outcome; United Kingdom; United States; Varenicline; Young Adult

2011
The effects of nicotine, varenicline, and cytisine on schedule-controlled responding in mice: differences in α4β2 nicotinic receptor activation.
    European journal of pharmacology, 2011, Mar-01, Volume: 654, Issue:1

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Conditioning, Operant; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Reinforcement Schedule; Smoking Cessation; Time Factors; Varenicline

2011
Integrating results from smoking cessation drug research and development into clinical occupational health practice.
    AAOHN journal : official journal of the American Association of Occupational Health Nurses, 2011, Volume: 59, Issue:2

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Occupational Health Nursing; Practice Guidelines as Topic; Quinoxalines; Smoking Cessation; Tobacco Use Disorder; Varenicline

2011
Electrophysiological perspectives on the therapeutic use of nicotinic acetylcholine receptor partial agonists.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 337, Issue:2

    Topics: Acetylcholine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Azocines; Benzazepines; Bupropion; DNA, Complementary; Dopamine Uptake Inhibitors; Electrophysiological Phenomena; Humans; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Pyridinium Compounds; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline; Xenopus

2011
Varenicline attenuates cue-induced relapse to alcohol, but not nicotine seeking, while reducing inhibitory response control.
    Psychopharmacology, 2011, Volume: 216, Issue:2

    Topics: Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Cues; Dose-Response Relationship, Drug; Ethanol; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Wistar; Reaction Time; Recurrence; Reinforcement Schedule; Self Administration; Sucrose; Varenicline

2011
Selective α4β2 nicotinic acetylcholine receptor agonists target epigenetic mechanisms in cortical GABAergic neurons.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:7

    Topics: Analysis of Variance; Animals; Azetidines; Behavior, Animal; Benzazepines; Cerebral Cortex; Conditioning, Classical; Cues; DNA (Cytosine-5-)-Methyltransferase 1; DNA (Cytosine-5-)-Methyltransferases; Epigenomics; Exploratory Behavior; Fear; Freezing Reaction, Cataleptic; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Male; Mecamylamine; Methyl-CpG-Binding Protein 2; Mice; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Promoter Regions, Genetic; Quinoxalines; Receptors, Nicotinic; RNA, Messenger; Varenicline

2011
[Abstinence rates with varenicline compared to bupropion and nicotine replacement therapy for quitting smoking in primary care].
    Atencion primaria, 2011, Volume: 43, Issue:9

    Topics: Adolescent; Adult; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Female; Humans; Longitudinal Studies; Male; Middle Aged; Nicotine; Nicotinic Agonists; Primary Health Care; Quinoxalines; Retrospective Studies; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline; Young Adult

2011
Varenicline, a partial agonist at neuronal nicotinic acetylcholine receptors, reduces nicotine-induced increases in 20% ethanol operant self-administration in Sprague-Dawley rats.
    Addiction biology, 2011, Volume: 16, Issue:3

    Topics: Alcohol Drinking; Animals; Benzazepines; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Neurons; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Stimulation, Chemical; Varenicline

2011
Prescribing of smoking cessation medication in England since the introduction of varenicline.
    Addiction (Abingdon, England), 2011, Volume: 106, Issue:7

    Topics: Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Drug Prescriptions; Electronic Health Records; England; Family Practice; Humans; Models, Statistical; Nicotine; Nicotinic Agonists; Practice Guidelines as Topic; Practice Patterns, Physicians'; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; State Medicine; Time Factors; Varenicline

2011
Smoking cessation interventions: a primer for physicians: Comment on "Use of varenicline for 4 weeks before quitting smoking".
    Archives of internal medicine, 2011, Apr-25, Volume: 171, Issue:8

    Topics: Benzazepines; Bupropion; Chewing Gum; Counseling; Delayed-Action Preparations; Drug Administration Schedule; Drug Therapy, Combination; Humans; Nasal Sprays; Nebulizers and Vaporizers; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Substance Withdrawal Syndrome; Time Factors; Transdermal Patch; Treatment Outcome; Varenicline

2011
A comparison of brain and behavioral effects of varenicline and nicotine in rats.
    Behavioural brain research, 2011, Sep-30, Volume: 223, Issue:1

    Topics: Animals; Benzazepines; Brain; Brain Mapping; Drug Administration Schedule; Drug Tolerance; Injections, Intravenous; Injections, Subcutaneous; Magnetic Resonance Imaging; Male; Maze Learning; Motor Activity; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Varenicline

2011
Cost effectiveness of interventions to reduce relapse to smoking following smoking cessation.
    Addiction (Abingdon, England), 2011, Volume: 106, Issue:10

    Topics: Benzazepines; Bupropion; Cost-Benefit Analysis; Dopamine Uptake Inhibitors; England; Epidemiologic Methods; Health Care Costs; Humans; Nicotine; Nicotinic Agonists; Quinoxalines; Secondary Prevention; Smoking; Smoking Cessation; Treatment Outcome; Varenicline; Wales

2011
The impact of the introduction of smoke-free legislation on prescribing of stop-smoking medications in England.
    Addiction (Abingdon, England), 2011, Volume: 106, Issue:10

    Topics: Adolescent; Adult; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Drug Prescriptions; Electronic Health Records; England; Family Practice; Female; Humans; Male; Middle Aged; Models, Statistical; Nicotine; Nicotinic Agonists; Practice Patterns, Physicians'; Quinoxalines; Smoking; Smoking Cessation; State Medicine; Time Factors; Varenicline; Young Adult

2011
Smoking cessation pharmacotherapy: a concise overview.
    Advance for NPs & PAs, 2011, Volume: 2, Issue:4

    Topics: Adrenergic alpha-2 Receptor Agonists; Antidepressive Agents; Benzazepines; Bupropion; Clonidine; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Quinoxalines; Smoking; Smoking Cessation; Varenicline

2011
Assessing preferences for improved smoking cessation medications: a discrete choice experiment.
    The European journal of health economics : HEPAC : health economics in prevention and care, 2012, Volume: 13, Issue:5

    Topics: Adolescent; Adult; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Female; Humans; Logistic Models; Male; Middle Aged; Models, Econometric; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Substance-Related Disorders; Surveys and Questionnaires; Switzerland; Varenicline; Young Adult

2012
Patterns of nicotinic receptor antagonism: nicotine discrimination studies.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 339, Issue:1

    Topics: Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cytosine; Data Interpretation, Statistical; Dihydro-beta-Erythroidine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Mecamylamine; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Varenicline

2011
Breaking free from nicotine dependence. A combination of strategies boosts the odds of success.
    The Harvard mental health letter, 2011, Volume: 27, Issue:10

    Topics: Administration, Cutaneous; Administration, Intranasal; Adult; Antidepressive Agents, Second-Generation; Behavior Therapy; Benzazepines; Bupropion; Cognitive Behavioral Therapy; Cross-Sectional Studies; Female; Humans; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Self-Help Groups; Smoking Cessation; Tobacco Use Disorder; Varenicline

2011
Effects of varenicline on the reinforcing and discriminative stimulus effects of cocaine in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 339, Issue:2

    Topics: Animals; Benzazepines; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Discrimination Learning; Discrimination, Psychological; Dopamine Uptake Inhibitors; Macaca mulatta; Male; Mecamylamine; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Reinforcement, Psychology; Self Administration; Time Factors; Varenicline

2011
[Clinical study of smoking cessation clinic subjects].
    Nihon Jibiinkoka Gakkai kaiho, 2011, Volume: 114, Issue:8

    Topics: Adult; Aged; Aged, 80 and over; Benzazepines; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Outpatient Clinics, Hospital; Outpatients; Quinoxalines; Smoking Cessation; Varenicline

2011
Varenicline decreases nicotine self-administration and cue-induced reinstatement of nicotine-seeking behaviour in rats when a long pretreatment time is used.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:9

    Topics: Animals; Benzazepines; Conditioning, Operant; Cues; Data Interpretation, Statistical; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Feeding Behavior; Male; Motivation; Nicotine; Quinoxalines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Reinforcement Schedule; Self Administration; Tobacco Use Disorder; Varenicline

2012
[Smoking cessation--assistance for the general practitioner].
    MMW Fortschritte der Medizin, 2011, Apr-07, Volume: 153, Issue:14

    Topics: Benzazepines; Bupropion; Combined Modality Therapy; Complementary Therapies; Cost-Benefit Analysis; Drug Costs; Fee Schedules; Germany; Humans; Myocardial Infarction; National Health Programs; Nicotine; Nicotinic Agonists; Physician's Role; Polymethacrylic Acids; Polyvinyls; Psychotherapy, Group; Quinoxalines; Smoking Cessation; Social Support; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2011
Varenicline dose dependently enhances responding for nonpharmacological reinforcers and attenuates the reinforcement-enhancing effects of nicotine.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2012, Volume: 14, Issue:3

    Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Smoking Cessation; Tobacco Use Disorder; Varenicline

2012
Quantification of nicotine, cotinine, trans-3'-hydroxycotinine and varenicline in human plasma by a sensitive and specific UPLC-tandem mass-spectrometry procedure for a clinical study on smoking cessation.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2011, Nov-15, Volume: 879, Issue:30

    Topics: Benzazepines; Chromatography, High Pressure Liquid; Cotinine; Drug Stability; Humans; Linear Models; Nicotine; Quinoxalines; Reproducibility of Results; Sensitivity and Specificity; Smoking Cessation; Tandem Mass Spectrometry; Varenicline

2011
Suicidal behavior and depression in smoking cessation treatments.
    PloS one, 2011, Volume: 6, Issue:11

    Topics: Adult; Benzazepines; Bupropion; Depression; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking Cessation; Suicide; Varenicline

2011
Varenicline blocks β2*-nAChR-mediated response and activates β4*-nAChR-mediated responses in mice in vivo.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2012, Volume: 14, Issue:6

    Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Female; Genotype; Hexamethonium; Hypothermia; Inhibitory Concentration 50; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Motor Activity; Mutation; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Ondansetron; Quinoxalines; Receptors, Nicotinic; Receptors, Serotonin, 5-HT3; Varenicline

2012
Effects of the combination of metyrapone and oxazepam on intravenous nicotine self-administration in rats.
    Psychopharmacology, 2012, Volume: 223, Issue:1

    Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Drug Therapy, Combination; Enzyme Inhibitors; Hypnotics and Sedatives; Infusions, Intravenous; Male; Metyrapone; Nicotine; Oxazepam; Quinoxalines; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Smoking Cessation; Varenicline

2012
Pharmacologic characterization of a nicotine-discriminative stimulus in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 341, Issue:3

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Cocaine; Conditioning, Operant; Discrimination Learning; Dopamine Uptake Inhibitors; Drug Interactions; Female; Hypnotics and Sedatives; Macaca mulatta; Male; Mecamylamine; Midazolam; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Varenicline

2012
An internet survey of use, opinions and preferences for smoking cessation medications: nicotine, varenicline, and bupropion.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2013, Volume: 15, Issue:1

    Topics: Administration, Inhalation; Adolescent; Adult; Aged; Benzazepines; Bupropion; Data Collection; Educational Status; Female; Humans; Internet; Male; Middle Aged; Nicotine; Patient Compliance; Patient Satisfaction; Quinoxalines; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline; Young Adult

2013
Varenicline is a potent partial agonist at α6β2* nicotinic acetylcholine receptors in rat and monkey striatum.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 342, Issue:2

    Topics: Animals; Benzazepines; Corpus Striatum; Dopamine; Male; Nicotine; Protein Binding; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Saimiri; Smoking Cessation; Synaptosomes; Varenicline

2012
Structural characterization of binding mode of smoking cessation drugs to nicotinic acetylcholine receptors through study of ligand complexes with acetylcholine-binding protein.
    The Journal of biological chemistry, 2012, Jul-06, Volume: 287, Issue:28

    Topics: Acetylcholine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Aplysia; Azocines; Benzazepines; Binding Sites; Binding, Competitive; Carrier Proteins; Cell Line; HEK293 Cells; Humans; Kinetics; Ligands; Models, Molecular; Mutation; Nicotine; Nicotinic Agonists; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Varenicline

2012
Use of an α3β4 nicotinic acetylcholine receptor subunit concatamer to characterize ganglionic receptor subtypes with specific subunit composition reveals species-specific pharmacologic properties.
    Neuropharmacology, 2012, Volume: 63, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Benzazepines; Drug Partial Agonism; Evoked Potentials; Ganglia; Humans; Ligands; Mutagenesis, Site-Directed; Mutant Proteins; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Protein Subunits; Quinolizines; Quinoxalines; Rats; Receptors, Nicotinic; Recombinant Fusion Proteins; Species Specificity; Varenicline; Xenopus laevis

2012
Impact of human D398N single nucleotide polymorphism on intracellular calcium response mediated by α3β4α5 nicotinic acetylcholine receptors.
    Neuropharmacology, 2012, Volume: 63, Issue:6

    Topics: Acetylcholine; Aequorin; Algorithms; Benzazepines; Calcium; Data Interpretation, Statistical; Enzyme-Linked Immunosorbent Assay; HEK293 Cells; Humans; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Permeability; Polymorphism, Single Nucleotide; Quinoxalines; Receptors, Nicotinic; Varenicline

2012
Chronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 343, Issue:2

    Topics: Animals; Azetidines; Behavior, Animal; Benzazepines; Binding Sites; Brain Chemistry; Cerebral Cortex; Dose-Response Relationship, Drug; Female; Male; Membranes; Neurons; Nicotine; Nicotinic Agonists; Pregnancy; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Up-Regulation; Varenicline

2012
Effects of nicotinic acetylcholine receptor agonists on cognition in rhesus monkeys with a chronic cocaine self-administration history.
    Neuropharmacology, 2013, Volume: 64

    Topics: Animals; Behavior, Animal; Benzamides; Benzazepines; Bridged Bicyclo Compounds; Cocaine; Cocaine-Related Disorders; Cognition Disorders; Dopamine Uptake Inhibitors; Hippocampus; Learning; Ligands; Macaca mulatta; Male; Memory, Short-Term; Nerve Tissue Proteins; Neurons; Nicotine; Nicotinic Agonists; Nootropic Agents; Quinoxalines; Receptors, Nicotinic; Reversal Learning; Self Administration; Varenicline

2013
The effect of smoking cessation pharmacotherapies on pancreatic beta cell function.
    Toxicology and applied pharmacology, 2012, Nov-15, Volume: 265, Issue:1

    Topics: Animals; Benzazepines; Bupropion; Dopamine Uptake Inhibitors; Electron Transport; Gene Expression; Glucose; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mitochondria; Nicotine; Nicotinic Agonists; Oxidative Stress; Pancreatic Function Tests; Quinoxalines; Rats; Signal Transduction; Smoking; Smoking Cessation; Varenicline

2012
Varenicline and bupropion: suicide.
    Prescrire international, 2012, Volume: 21, Issue:131

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Patient Safety; Prescription Drug Misuse; Quinoxalines; Risk Assessment; Risk Factors; Smoking Cessation; Suicide; Varenicline

2012
Involvement of cholinergic receptors in the different stages of memory measured in the modified elevated plus maze test in mice.
    Pharmacological reports : PR, 2012, Volume: 64, Issue:5

    Topics: Animals; Benzazepines; Male; Maze Learning; Mecamylamine; Memory; Mice; Motor Activity; Nicotine; Quinoxalines; Receptors, Cholinergic; Scopolamine; Varenicline

2012
Nicotine-motivated behavior in Caenorhabditis elegans requires the nicotinic acetylcholine receptor subunits acr-5 and acr-15.
    The European journal of neuroscience, 2013, Volume: 37, Issue:5

    Topics: Age Factors; Animals; Behavior, Animal; Benzazepines; Butanones; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Chemotaxis; Chlorides; Fasting; Mecamylamine; Muscles; Mutation; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Protein Subunits; Quinoxalines; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Nicotinic; Reward; Sodium; Taste; Time Factors; Varenicline

2013
Varenicline and nicotine enhance GABAergic synaptic transmission in rat CA1 hippocampal and medial septum/diagonal band neurons.
    Life sciences, 2013, Mar-14, Volume: 92, Issue:6-7

    Topics: Animals; Benzazepines; CA1 Region, Hippocampal; Female; GABAergic Neurons; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Neurons; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Sprague-Dawley; Septal Nuclei; Synaptic Transmission; Varenicline

2013
Multiple nicotine training doses in mice as a basis for differentiating the effects of smoking cessation aids.
    Psychopharmacology, 2013, Volume: 228, Issue:2

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Dihydro-beta-Erythroidine; Discrimination Learning; Dose-Response Relationship, Drug; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Midazolam; Morphine; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2013
Divergent functional effects of sazetidine-a and varenicline during nicotine withdrawal.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:10

    Topics: Animals; Anxiety; Azetidines; Benzazepines; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Partial Agonism; Evoked Potentials; Hippocampus; Male; Mice; Microinjections; Motor Activity; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Up-Regulation; Varenicline

2013
Neuronal nicotinic receptor agonists improve gait and balance in olivocerebellar ataxia.
    Neuropharmacology, 2013, Volume: 73

    Topics: Animals; Ataxia; Benzazepines; Cerebellum; Dose-Response Relationship, Drug; Gait; Male; Mecamylamine; Motor Activity; Nerve Degeneration; Neural Pathways; Niacinamide; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Olivary Nucleus; Postural Balance; Pyridines; Quinoxalines; Rats; Rotarod Performance Test; Varenicline

2013
PET imaging of high-affinity α4β2 nicotinic acetylcholine receptors in humans with 18F-AZAN, a radioligand with optimal brain kinetics.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2013, Volume: 54, Issue:8

    Topics: 2,2'-Dipyridyl; Adult; Animals; Azabicyclo Compounds; Benzazepines; Binding, Competitive; Brain; Female; Humans; Kinetics; Ligands; Male; Middle Aged; Nicotine; Nicotinic Agonists; Papio; Positron-Emission Tomography; Quinoxalines; Radiometry; Receptors, Nicotinic; Reproducibility of Results; Varenicline

2013
Effectiveness of varenicline versus nicotine replacement therapy for smoking cessation with minimal professional support: evidence from an English population study.
    Psychopharmacology, 2014, Volume: 231, Issue:1

    Topics: Adult; Aged; Benzazepines; Cross-Sectional Studies; Data Collection; Data Interpretation, Statistical; England; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Population; Prescription Drugs; Quinoxalines; Smoking; Smoking Cessation; Treatment Outcome; Varenicline

2014
Varenicline and cytisine diminish the dysphoric-like state associated with spontaneous nicotine withdrawal in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:2

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Infusion Pumps, Implantable; Male; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Varenicline

2014
Effect of allopurinol on smoking.
    Nefrologia : publicacion oficial de la Sociedad Espanola Nefrologia, 2013, Nov-13, Volume: 33, Issue:6

    Topics: Acetylcholine; Allopurinol; Benzazepines; Brain Chemistry; Bupropion; Causality; Comorbidity; Diabetic Nephropathies; Humans; Hypoxanthine; Molecular Structure; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Structure-Activity Relationship; Varenicline; Xanthine Oxidase

2013
The effect of varenicline on the development and expression of nicotine-induced behavioral sensitization and cross-sensitization in rats.
    Addiction biology, 2015, Volume: 20, Issue:2

    Topics: Animals; Benzazepines; Motor Activity; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Smoking Cessation; Varenicline

2015
Effects of chronic varenicline treatment on nicotine, cocaine, and concurrent nicotine+cocaine self-administration.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:5

    Topics: Animals; Benzazepines; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Feeding Behavior; Female; Macaca mulatta; Male; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Reinforcement, Psychology; Self Administration; Tobacco Use Disorder; Varenicline

2014
Functional interactions of varenicline and nicotine with nAChR subtypes implicated in cardiovascular control.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2014, Volume: 16, Issue:6

    Topics: Animals; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Oocytes; Protein Binding; Quinoxalines; Receptors, Nicotinic; Tobacco Use Disorder; Varenicline; Xenopus laevis

2014
Chronic sazetidine-A maintains anxiolytic effects and slower weight gain following chronic nicotine without maintaining increased density of nicotinic receptors in rodent brain.
    Journal of neurochemistry, 2014, Volume: 129, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azetidines; Benzazepines; Brain Chemistry; Drug Evaluation, Preclinical; Feeding Behavior; Gene Expression Regulation; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Substance Withdrawal Syndrome; Tobacco Use Cessation; Tobacco Use Disorder; Up-Regulation; Varenicline; Weight Gain

2014
[Safety of nicotine addiction treatment].
    Przeglad lekarski, 2013, Volume: 70, Issue:10

    Topics: Abdominal Pain; Adult; Alkaloids; Azocines; Benzazepines; Boredom; Bupropion; Female; Headache; Humans; Male; Middle Aged; Nicotine; Patient Compliance; Quinolizines; Quinoxalines; Sleep Wake Disorders; Smoking Cessation; Tobacco Use Disorder; Varenicline; Xerostomia

2013
Varenicline disrupts prepulse inhibition only in high-inhibitory rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2014, Aug-04, Volume: 53

    Topics: Acoustic Stimulation; Acoustics; Analysis of Variance; Animals; Apomorphine; Benzazepines; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Nicotine; Nicotinic Agonists; Prepulse Inhibition; Quinoxalines; Rats; Rats, Sprague-Dawley; Reflex, Startle; Varenicline

2014
Larval zebrafish model for FDA-approved drug repositioning for tobacco dependence treatment.
    PloS one, 2014, Volume: 9, Issue:3

    Topics: Animals; Benzazepines; Drug Repositioning; Models, Animal; Nicotine; Quinoxalines; Tobacco Use Disorder; United States; United States Food and Drug Administration; Varenicline; Zebrafish

2014
The cytisine derivatives, CC4 and CC26, reduce nicotine-induced conditioned place preference in zebrafish by acting on heteromeric neuronal nicotinic acetylcholine receptors.
    Psychopharmacology, 2014, Volume: 231, Issue:24

    Topics: Alkaloids; Animals; Benzazepines; Conditioning, Operant; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Quinoxalines; Receptors, Nicotinic; Varenicline; Zebrafish

2014
Efficient expression of functional (α6β2)2β3 AChRs in Xenopus oocytes from free subunits using slightly modified α6 subunits.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Cholinergic Agonists; Female; Gene Expression; Humans; Membrane Potentials; Nicotine; Nicotinic Agonists; Oocytes; Patch-Clamp Techniques; Quinolizines; Receptors, Nicotinic; Recombinant Fusion Proteins; Varenicline; Xenopus laevis

2014
Differentiating the primary reinforcing and reinforcement-enhancing effects of varenicline.
    Psychopharmacology, 2015, Volume: 232, Issue:5

    Topics: Animals; Benzazepines; Conditioning, Operant; Cues; Dose-Response Relationship, Drug; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Smoking Cessation; Varenicline

2015
Examination of the effects of varenicline, bupropion, lorcaserin, or naltrexone on responding for conditioned reinforcement in nicotine-exposed rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:8

    Topics: Animals; Benzazepines; Bupropion; Cholinergic Agents; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Male; Naltrexone; Narcotic Antagonists; Nicotine; Quinoxalines; Rats; Rats, Long-Evans; Reinforcement, Psychology; Varenicline

2014
Concurrent access to nicotine and sucrose in rats.
    Psychopharmacology, 2015, Volume: 232, Issue:8

    Topics: Animals; Behavior, Addictive; Benzazepines; Conditioning, Operant; Male; Nicotine; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration; Sucrose; Varenicline

2015
Prospective cohort study of the effectiveness of varenicline versus nicotine replacement therapy for smoking cessation in the "real world".
    BMC public health, 2014, Nov-12, Volume: 14

    Topics: Adolescent; Adult; Benzazepines; Cohort Studies; Cross-Sectional Studies; Female; Humans; Longitudinal Studies; Male; Middle Aged; Netherlands; Nicotine; Nicotinic Agonists; Patient Compliance; Prospective Studies; Quinoxalines; Smoking Cessation; Surveys and Questionnaires; Treatment Outcome; Varenicline

2014
AT-1001: a high-affinity α3β4 nAChR ligand with novel nicotine-suppressive pharmacology.
    British journal of pharmacology, 2015, Volume: 172, Issue:7

    Topics: Animals; Cell Line; Drug-Seeking Behavior; Ethanol; Humans; Ligands; Male; Motor Activity; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oligopeptides; Rats, Sprague-Dawley; Receptors, Nicotinic; Varenicline

2015
Importance of national context in the translation of personalised treatments for smoking cessation.
    The Lancet. Respiratory medicine, 2015, Volume: 3, Issue:2

    Topics: Female; Humans; Male; Nicotine; Nicotinic Agonists; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2015
Bupropion-varenicline interactions and nicotine self-administration behavior in rats.
    Pharmacology, biochemistry, and behavior, 2015, Volume: 130

    Topics: Animals; Bupropion; Dose-Response Relationship, Drug; Drug Synergism; Female; Nicotine; Rats; Self Administration; Varenicline

2015
Effects of the Nanoparticle-Based Vaccine, SEL-068, on Nicotine Discrimination in Squirrel Monkeys.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:9

    Topics: Analysis of Variance; Animals; Berberine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Immunization; Immunologic Factors; Male; Nanoparticles; Nicotine; Nicotinic Agonists; Saimiri; Time Factors; Vaccines; Varenicline

2015
Reward Anticipation Is Differentially Modulated by Varenicline and Nicotine in Smokers.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:8

    Topics: Adolescent; Adult; Brain; Case-Control Studies; Cross-Over Studies; Double-Blind Method; Female; Humans; Image Processing, Computer-Assisted; Male; Middle Aged; Motivation; Nicotine; Nicotinic Agonists; Oxygen; Reaction Time; Reward; Smoking; Varenicline; Young Adult

2015
Gender differences in medication use and cigarette smoking cessation: results from the International Tobacco Control Four Country Survey.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2015, Volume: 17, Issue:4

    Topics: Adolescent; Adult; Australia; Benzazepines; Canada; Female; Gender Identity; Humans; Longitudinal Studies; Male; Middle Aged; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Smoking; Smoking Cessation; Smoking Prevention; Substance Withdrawal Syndrome; United Kingdom; United States; Varenicline

2015
Noribogaine reduces nicotine self-administration in rats.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Ibogaine; Male; Nicotine; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Smoking Cessation; Tobacco Use Disorder; Varenicline

2015
Chronic treatment with varenicline changes expression of four nAChR binding sites in mice.
    Neuropharmacology, 2015, Volume: 99

    Topics: Animals; Autoradiography; Binding Sites; Brain; Dose-Response Relationship, Drug; Gene Expression; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Tobacco Use Cessation Devices; Varenicline

2015
The effect of switching pharmacological intervention during extinction on nicotine-evoked conditioned responding in rats.
    Psychopharmacology, 2015, Volume: 232, Issue:23

    Topics: Animals; Conditioning, Psychological; Discrimination Learning; Dose-Response Relationship, Drug; Drug Substitution; Extinction, Psychological; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Smoking Cessation; Varenicline

2015
Effects of varenicline on operant self-administration of alcohol and/or nicotine in a rat model of co-abuse.
    Behavioural brain research, 2016, Jan-01, Volume: 296

    Topics: Animals; Behavior, Addictive; Behavior, Animal; Conditioning, Operant; Disease Models, Animal; Drug Interactions; Ethanol; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Wistar; Substance-Related Disorders; Varenicline

2016
Varenicline decreases nicotine but not alcohol self-administration in genetically selected Marchigian Sardinian alcohol-preferring (msP) rats.
    Drug and alcohol dependence, 2015, Nov-01, Volume: 156

    Topics: Alcohol Drinking; Animals; Behavior, Animal; Central Nervous System Depressants; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Male; Nicotine; Nicotinic Agonists; Rats; Self Administration; Varenicline

2015
Extended nicotine self-administration increases sensitivity to nicotine, motivation to seek nicotine and the reinforcing properties of nicotine-paired cues.
    Addiction biology, 2017, Volume: 22, Issue:2

    Topics: Animals; Behavior, Animal; Cues; Drug-Seeking Behavior; Male; Motivation; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration; Tobacco Use Disorder; Varenicline

2017
Nicotine Enhances the Hypnotic and Hypothermic Effects of Alcohol in the Mouse.
    Alcoholism, clinical and experimental research, 2016, Volume: 40, Issue:1

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Azetidines; Body Temperature; Central Nervous System Depressants; Drug Interactions; Ethanol; Hypnotics and Sedatives; Hypothermia; Ketamine; Mecamylamine; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Pyridines; Receptors, Nicotinic; Reflex, Righting; Varenicline

2016
Influence of smoking cessation drugs on blood pressure and heart rate in patients with cardiovascular disease or high risk score: real life setting.
    BMC cardiovascular disorders, 2016, Jan-05, Volume: 16

    Topics: Adult; Aged; Blood Pressure; Brazil; Bupropion; Cardiovascular Diseases; Comorbidity; Coronary Artery Disease; Diabetes Mellitus; Diastole; Dopamine Uptake Inhibitors; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Nicotine; Nicotinic Agonists; Risk Factors; Smoking; Smoking Cessation; Systole; Tobacco Use Cessation Devices; Varenicline

2016
[Varenicline in nicotine replacement therapy: Does it really increase the risk of cardiovascular and neuropsychiatric events?].
    Semergen, 2016, Volume: 42, Issue:6

    Topics: Bupropion; Humans; Nicotine; Nicotinic Agonists; Smoking; Varenicline

2016
Similar quit rates are found with three smoking cessation options.
    BMJ (Clinical research ed.), 2016, Jan-26, Volume: 352

    Topics: Female; Humans; Male; Nicotine; Nicotinic Agonists; Smoking; Tobacco Use Cessation Devices; Varenicline

2016
Methamphetamine-like discriminative stimulus effects of bupropion and its two hydroxy metabolites in male rhesus monkeys.
    Behavioural pharmacology, 2016, Volume: 27, Issue:2-3 Spec I

    Topics: Animals; Antidepressive Agents, Second-Generation; Bupropion; Central Nervous System Stimulants; Conditioning, Operant; Discrimination Learning; Dopamine Antagonists; Dose-Response Relationship, Drug; Macaca mulatta; Male; Methamphetamine; Nicotine; Nicotinic Agonists; Reinforcement, Psychology; Risperidone; Time Factors; Varenicline

2016
Varenicline impairs extinction and enhances reinstatement across repeated cycles of nicotine self-administration in rats.
    Neuropharmacology, 2016, Volume: 105

    Topics: Animals; Catheters, Indwelling; Disease Models, Animal; Drug-Seeking Behavior; Extinction, Psychological; Male; Motor Activity; Nicotine; Nicotinic Agonists; Rats, Sprague-Dawley; Self Administration; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2016
Commentary on Roberts et al. (2016): Bupropion and varenicline are efficacious and well-tolerated cessation medications for smokers with serious mental illness.
    Addiction (Abingdon, England), 2016, Volume: 111, Issue:4

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Nicotinic Agonists; Smoking; Smoking Cessation; Tobacco Use Disorder; Varenicline

2016
Sex differences in attenuation of nicotine reinstatement after individual and combined treatments of progesterone and varenicline.
    Behavioural brain research, 2016, 07-15, Volume: 308

    Topics: Animals; Disease Models, Animal; Drug Combinations; Drug-Seeking Behavior; Extinction, Psychological; Female; Male; Nicotine; Nicotinic Agonists; Progesterone; Progestins; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Sex Factors; Smoking Cessation; Varenicline

2016
Effects of aging on the effectiveness of smoking cessation medication.
    Oncotarget, 2016, May-24, Volume: 7, Issue:21

    Topics: Adult; Age Factors; Aged; Brazil; Bupropion; Drug Therapy, Combination; Female; Half-Life; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Precision Medicine; Smoking Cessation; Treatment Outcome; Varenicline

2016
[Not Available].
    Revue medicale suisse, 2016, Mar-23, Volume: 12, Issue:511

    Topics: Female; Humans; Male; Nicotine; Nicotinic Agonists; Smoking; Tobacco Use Cessation Devices; Varenicline

2016
The use of varenicline to treat nicotine dependence among patients with cancer.
    Psycho-oncology, 2017, Volume: 26, Issue:10

    Topics: Adult; Benzazepines; Bupropion; Counseling; Feasibility Studies; Female; Humans; Male; Middle Aged; Neoplasms; Nicotine; Nicotinic Agonists; Smoking; Smoking Cessation; Tobacco Use Disorder; Treatment Outcome; Varenicline

2017
Factors influencing sustainable efficacy of smoking cessation treatment with varenicline beyond nine months.
    Nagoya journal of medical science, 2016, Volume: 78, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Bupropion; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Smoking; Smoking Cessation; Varenicline

2016
The nicotine + alcohol interoceptive drug state: contribution of the components and effects of varenicline in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Animals; Central Nervous System Depressants; Conditioning, Classical; Cues; Dose-Response Relationship, Drug; Ethanol; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Long-Evans; Receptors, Nicotinic; Smoking Cessation; Varenicline

2016
Varenicline, the clinically effective smoking cessation agent, restores probabilistic response reversal performance during withdrawal from nicotine.
    Addiction biology, 2017, Volume: 22, Issue:5

    Topics: Animals; Male; Nicotine; Nicotinic Agonists; Probability Learning; Psychomotor Performance; Rats; Reaction Time; Substance Withdrawal Syndrome; Tobacco Use Disorder; Varenicline

2017
Attenuated nicotine-like effects of varenicline but not other nicotinic ACh receptor agonists in monkeys receiving nicotine daily.
    British journal of pharmacology, 2016, Volume: 173, Issue:24

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Nicotine; Nicotinic Agonists; Pyridines; Receptors, Nicotinic; Structure-Activity Relationship; Varenicline

2016
Therapeutic concentrations of varenicline in the presence of nicotine increase action potential firing in human adrenal chromaffin cells.
    Journal of neurochemistry, 2017, Volume: 140, Issue:1

    Topics: Action Potentials; Adrenal Cortex; Adult; Aged; Animals; Chromaffin Cells; Dose-Response Relationship, Drug; Drug Synergism; Female; Humans; Male; Middle Aged; Nicotine; Nicotinic Agonists; Varenicline; Xenopus laevis

2017
The contribution of α4β2 and non-α4β2 nicotinic acetylcholine receptors to the discriminative stimulus effects of nicotine and varenicline in mice.
    Psychopharmacology, 2017, Volume: 234, Issue:5

    Topics: Aconitine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Azocines; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dihydro-beta-Erythroidine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Hypnotics and Sedatives; Ibogaine; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Midazolam; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Varenicline

2017
Varenicline provokes impulsive action by stimulating α4β2 nicotinic acetylcholine receptors in the infralimbic cortex in a nicotine exposure status-dependent manner.
    Pharmacology, biochemistry, and behavior, 2017, Volume: 154

    Topics: Administration, Oral; Animals; Appetite; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Drug Interactions; Hypodermoclysis; Impulsive Behavior; Limbic Lobe; Male; Microinjections; Nicotine; Nicotinic Agonists; Rats; Receptors, Nicotinic; Varenicline

2017
The effect of varenicline and nicotine patch on smoking rate and satisfaction with smoking: an examination of the mechanism of action of two pre-quit pharmacotherapies.
    Psychopharmacology, 2017, Volume: 234, Issue:13

    Topics: Humans; Nicotine; Nicotinic Agonists; Personal Satisfaction; Research Design; Smartphone; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Smoking; Tobacco Use Cessation Devices; Varenicline

2017
Compromised neuroplasticity in cigarette smokers under nicotine withdrawal is restituted by the nicotinic α
    Scientific reports, 2017, 05-03, Volume: 7, Issue:1

    Topics: Adult; Cigarette Smoking; Electric Stimulation; Evoked Potentials, Motor; Female; Humans; Male; Motor Cortex; Neuronal Plasticity; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Substance Withdrawal Syndrome; Transcranial Direct Current Stimulation; Varenicline; Young Adult

2017
Using PICO Methodology to Answer Questions About Smoking in COPD Patients.
    Archivos de bronconeumologia, 2017, Volume: 53, Issue:11

    Topics: Biomarkers; Bupropion; Clinical Trials as Topic; Cost-Benefit Analysis; Counseling; Evidence-Based Medicine; Humans; Motivation; Nicotine; Nicotinic Agonists; Pulmonary Disease, Chronic Obstructive; Randomized Controlled Trials as Topic; Smoking; Smoking Cessation; Spirometry; Surveys and Questionnaires; Varenicline

2017
Selective and regulated trapping of nicotinic receptor weak base ligands and relevance to smoking cessation.
    eLife, 2017, 07-18, Volume: 6

    Topics: HEK293 Cells; Humans; Hydrogen-Ion Concentration; Ligands; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Smoking Cessation; Up-Regulation; Varenicline

2017
Measures and predictors of varenicline adherence in the treatment of nicotine dependence.
    Addictive behaviors, 2017, Volume: 75

    Topics: Adult; Affect; Craving; Female; Humans; Logistic Models; Male; Medication Adherence; Middle Aged; Nicotine; Nicotinic Agonists; Randomized Controlled Trials as Topic; Saliva; Self Report; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Disorder; Varenicline

2017
The effectiveness of varenicline versus nicotine replacement therapy on long-term smoking cessation in primary care: a prospective cohort study of electronic medical records.
    International journal of epidemiology, 2017, 12-01, Volume: 46, Issue:6

    Topics: Adult; Electronic Health Records; England; Female; Follow-Up Studies; Humans; Logistic Models; Male; Middle Aged; Multivariate Analysis; Nicotine; Primary Health Care; Propensity Score; Prospective Studies; Smoking Cessation; Social Class; Time Factors; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2017
Association of nicotine metabolism and sex with relapse following varenicline and nicotine replacement therapy.
    Experimental and clinical psychopharmacology, 2017, Volume: 25, Issue:5

    Topics: Adult; Cotinine; Cytochrome P-450 CYP2A6; Female; Genotype; Humans; Longitudinal Studies; Male; Middle Aged; Nicotine; Recurrence; Smoking; Smoking Cessation; Tobacco Products; Varenicline

2017
Reversal of Nicotine Withdrawal Signs Through Positive Allosteric Modulation of α4β2 Nicotinic Acetylcholine Receptors in Male Mice.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2018, 06-07, Volume: 20, Issue:7

    Topics: Allosteric Regulation; Animals; Hydrocarbons, Brominated; Indole Alkaloids; Infusion Pumps, Implantable; Male; Mice; Mice, Inbred ICR; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Varenicline

2018
Nicotine as a discriminative stimulus for ethanol use.
    Drug and alcohol dependence, 2018, 01-01, Volume: 182

    Topics: Alcohol Drinking; Animals; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Ethanol; Male; Nicotine; Rats; Rats, Inbred Lew; Reaction Time; Reinforcement, Psychology; Varenicline

2018
Effects of the nicotinic agonist varenicline, nicotinic antagonist r-bPiDI, and DAT inhibitor (R)-modafinil on co-use of ethanol and nicotine in female P rats.
    Psychopharmacology, 2018, Volume: 235, Issue:5

    Topics: Alcohol Drinking; Animals; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Ethanol; Female; Modafinil; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Rats; Receptors, Nicotinic; Self Administration; Smoking Cessation; Varenicline

2018
A behavioral economic analysis of the value-enhancing effects of nicotine and varenicline and the role of nicotinic acetylcholine receptors in male and female rats.
    Behavioural pharmacology, 2018, Volume: 29, Issue:6

    Topics: Animals; Conditioning, Operant; Cues; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Economics, Behavioral; Female; Locomotion; Male; Nicotine; Nicotinic Agonists; Photic Stimulation; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Reinforcement, Psychology; Sex Characteristics; Varenicline

2018
[Clinical Practice Guidelines for Smoking Cessation].
    Revista medica de Chile, 2017, Volume: 145, Issue:11

    Topics: Bupropion; Chile; Evidence-Based Medicine; Humans; Nicotine; Smoking Cessation; Varenicline

2017
New insights on the effects of varenicline on nicotine reward, withdrawal and hyperalgesia in mice.
    Neuropharmacology, 2018, Volume: 138

    Topics: Animals; Dose-Response Relationship, Drug; Female; Hyperalgesia; Male; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Transgenic; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Reward; Smoking Cessation Agents; Substance Withdrawal Syndrome; Tobacco Use Disorder; Varenicline

2018
Rats choose high doses of nicotine in order to compensate for changes in its price and availability.
    Addiction biology, 2019, Volume: 24, Issue:5

    Topics: Animals; Behavior, Animal; Choice Behavior; Infusions, Intravenous; Nicotine; Nicotinic Agonists; Public Policy; Rats; Self Administration; Smoke-Free Policy; Smoking Cessation Agents; Tobacco Products; Varenicline

2019
Nicotine and varenicline ameliorate changes in reward-based choice strategy and altered decision-making in methamphetamine-treated rats.
    Behavioural brain research, 2019, 02-01, Volume: 359

    Topics: Animals; Central Nervous System Stimulants; Conditioning, Operant; Decision Making; Dose-Response Relationship, Drug; Male; Methamphetamine; Nicotine; Nicotinic Agonists; Rats; Rats, Wistar; Reward; Risk-Taking; Time Factors; Varenicline

2019
Varenicline increases random flap survival in rats submitted to nicotine.
    Journal of plastic surgery and hand surgery, 2018, Volume: 52, Issue:5

    Topics: Angiography; Animals; Graft Survival; Microcirculation; Microscopy; Models, Animal; Nicotine; Nicotinic Agonists; Rats, Wistar; Smoking Cessation Agents; Surgical Flaps; Varenicline

2018
Rapid nicotine tolerance and cross-tolerance to varenicline in rhesus monkeys: Drug discrimination.
    Experimental and clinical psychopharmacology, 2018, Volume: 26, Issue:6

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Tolerance; Female; Macaca mulatta; Male; Nicotine; Nicotinic Agonists; Smoking Cessation; Tobacco Use Disorder; Varenicline

2018
Varenicline and nabilone in tobacco and cannabis co-users: effects on tobacco abstinence, withdrawal and a laboratory model of cannabis relapse.
    Addiction biology, 2019, Volume: 24, Issue:4

    Topics: Adult; Cigarette Smoking; Comorbidity; Dronabinol; Female; Humans; Male; Marijuana Abuse; Nicotine; Nicotinic Agonists; Smoking Cessation; Smoking Cessation Agents; Substance Withdrawal Syndrome; Varenicline; Young Adult

2019
An improved model of ethanol and nicotine co-use in female P rats: Effects of naltrexone, varenicline, and the selective nicotinic α6β2* antagonist r-bPiDI.
    Drug and alcohol dependence, 2018, 12-01, Volume: 193

    Topics: Alcohol Deterrents; Alcohol Drinking; Animals; Disease Models, Animal; Ethanol; Female; Naltrexone; Nicotine; Nicotinic Antagonists; Picolines; Pyridinium Compounds; Rats; Self Administration; Smoking Cessation Agents; Tobacco Use Disorder; Treatment Outcome; Varenicline

2018
Differential cross-tolerance to the effects of nicotinic acetylcholine receptor drugs in C57BL/6J mice following chronic varenicline.
    Behavioural pharmacology, 2019, Volume: 30, Issue:5

    Topics: Alkaloids; Animals; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Conditioning, Operant; Drug Tolerance; Female; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Reinforcement, Psychology; Smoking Cessation; Varenicline

2019
Revisiting autosomal dominant nocturnal frontal lobe epilepsy (ADNFLE) mutations in the nicotinic acetylcholine receptor reveal an increase in efficacy regardless of stochiometry.
    Pharmacological research, 2019, Volume: 139

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Epilepsy, Frontal Lobe; Female; Mutation; Nicotine; Nicotinic Agonists; Oocytes; Quinolizines; Receptors, Nicotinic; Varenicline; Xenopus laevis

2019
Individual differences in responding to bupropion or varenicline in a preclinical model of nicotine self-administration vary according to individual demand for nicotine.
    Neuropharmacology, 2019, Volume: 148

    Topics: Animals; Bupropion; Dose-Response Relationship, Drug; Extinction, Psychological; Individuality; Male; Nicotine; Rats; Reinforcement Schedule; Self Administration; Sucrose; Varenicline

2019
Increasing Smoking Cessation in the United States: Expanding the Availability of Over-the-Counter Medications.
    JAMA, 2019, Feb-12, Volume: 321, Issue:6

    Topics: Behavior Therapy; Bupropion; Humans; Nicotine; Nonprescription Drugs; Smoking Cessation; Smoking Cessation Agents; Tobacco Use Cessation Devices; United States; Varenicline

2019
Determining the pharmacokinetics of nicotinic drugs in the endoplasmic reticulum using biosensors.
    The Journal of general physiology, 2019, 06-03, Volume: 151, Issue:6

    Topics: Animals; Biosensing Techniques; Cell Line; Cell Line, Tumor; Cell Membrane; Endoplasmic Reticulum; Female; HEK293 Cells; HeLa Cells; Hippocampus; Humans; Mammals; Mice; Neurons; Nicotine; Pregnancy; Protein Transport; Receptors, Nicotinic; Smoking; Varenicline

2019
Therapeutic challenges for concurrent ethanol and nicotine consumption: naltrexone and varenicline fail to alter simultaneous ethanol and nicotine intake by female alcohol-preferring (P) rats.
    Psychopharmacology, 2019, Volume: 236, Issue:6

    Topics: Alcohol Deterrents; Alcohol Drinking; Animals; Ethanol; Female; Injections, Subcutaneous; Naltrexone; Nicotine; Random Allocation; Rats; Self Administration; Smoking Cessation Agents; Tobacco Use Disorder; Varenicline

2019
Prolonged exposure of rats to varenicline increases anxiety and alters serotonergic system, but has no effect on memory.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 181

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Analysis of Variance; Animals; Anxiety; Behavior, Animal; Cognition; gamma-Aminobutyric Acid; Hippocampus; Male; Memory; Models, Animal; Motor Activity; Nicotine; Nicotinic Agonists; Rats; Rats, Wistar; Serotonergic Neurons; Serotonin; Smoking; Smoking Cessation; Varenicline

2019
Exploring the interoceptive stimulus effects of nicotine and varenicline.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 181

    Topics: Animals; Appetitive Behavior; Conditioning, Classical; Discrimination Learning; Discrimination, Psychological; Drug Substitution; Extinction, Psychological; Injections, Subcutaneous; Interoception; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Saline Solution; Smoking Cessation; Substance Withdrawal Syndrome; Sucrose; Varenicline

2019
Assessing nicotine dependence using an oral nicotine free-choice paradigm in mice.
    Neuropharmacology, 2019, Volume: 157

    Topics: Animals; Behavior, Addictive; Choice Behavior; Dose-Response Relationship, Drug; Drug Interactions; Female; Male; Mice; Mice, Knockout; Nicotine; Nucleus Accumbens; Quinine; Receptors, Nicotinic; Self Administration; Sex Characteristics; Substance Withdrawal Syndrome; Tobacco Use Disorder; Tyrosine 3-Monooxygenase; Varenicline

2019
Nicotine Self-Administration as Paradigm for Medication Discovery for Smoking Cessation: Recent Findings in Medications Targeting the Cholinergic System.
    Methods in molecular biology (Clifton, N.J.), 2019, Volume: 2011

    Topics: Animals; Behavior, Addictive; Cholinergic Agents; Gene Knockout Techniques; Humans; Models, Animal; Nicotine; Nicotinic Antagonists; Receptors, Nicotinic; Self Administration; Smoking Cessation; Varenicline

2019
Prescribing Prevalence, Effectiveness, and Mental Health Safety of Smoking Cessation Medicines in Patients With Mental Disorders.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2020, 01-27, Volume: 22, Issue:1

    Topics: Drug Prescriptions; Female; Humans; Male; Mental Disorders; Mental Health; Middle Aged; Nicotine; Nicotinic Agonists; Prospective Studies; Smoking Cessation; Tobacco Use Cessation Devices; Tobacco Use Disorder; Varenicline

2020
Estimation of high-dimensional propensity scores with multiple exposure levels.
    Pharmacoepidemiology and drug safety, 2020, Volume: 29 Suppl 1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Algorithms; Bupropion; Cohort Studies; Female; Humans; Male; Middle Aged; Myocardial Infarction; Nicotine; Pharmacoepidemiology; Propensity Score; Proportional Hazards Models; Retrospective Studies; Smoking Cessation; United Kingdom; Varenicline; Young Adult

2020
Varenicline for cessation from nicotine-containing electronic cigarettes.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2019, Nov-13, Volume: 76, Issue:23

    Topics: Behavior, Addictive; Humans; Male; Middle Aged; Nicotine; Severity of Illness Index; Smoking Cessation; Treatment Outcome; Vaping; Varenicline

2019
Habenular and striatal activity during performance feedback are differentially linked with state-like and trait-like aspects of tobacco use disorder.
    Science advances, 2019, Volume: 5, Issue:10

    Topics: Adolescent; Adult; Brain; Brain Mapping; Corpus Striatum; Feedback, Physiological; Female; Habenula; Humans; Magnetic Resonance Imaging; Male; Middle Aged; Nicotine; Placebo Effect; Smokers; Task Performance and Analysis; Tobacco Use Disorder; Varenicline; Young Adult

2019
Varenicline aggravates atherosclerotic plaque formation in nicotine-pretreated ApoE knockout mice due to enhanced oxLDL uptake by macrophages through downregulation of ABCA1 and ABCG1 expression.
    Journal of pharmacological sciences, 2020, Volume: 142, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter 1; ATP Binding Cassette Transporter, Subfamily G, Member 1; Down-Regulation; Gene Expression Regulation; Lipoproteins, LDL; Macrophages; Mice; Mice, Inbred C57BL; Mice, Knockout, ApoE; Nicotine; Plaque, Atherosclerotic; RAW 264.7 Cells; Smoking Cessation Agents; Varenicline

2020
Development of a novel alcohol and nicotine concurrent access (ANCA) self-administration procedure in baboons.
    Drug and alcohol dependence, 2020, 01-01, Volume: 206

    Topics: Administration, Intravenous; Administration, Oral; Animals; Drug Interactions; Ethanol; Male; Models, Animal; Nicotine; Papio; Self Administration; Varenicline

2020
Long-term effectiveness and safety of varenicline and nicotine replacement therapy in people with neurodevelopmental disorders: A prospective cohort study.
    Scientific reports, 2019, 12-20, Volume: 9, Issue:1

    Topics: Cohort Studies; Confidence Intervals; Female; Humans; Male; Neurodevelopmental Disorders; Nicotine; Propensity Score; Prospective Studies; Smoking Cessation; Varenicline

2019
Health-care providers' concern regarding smoking cessation pharmacotherapies during pregnancy: Calls to a teratology information service.
    Drug and alcohol review, 2020, Volume: 39, Issue:3

    Topics: Australia; Behavior Therapy; Bupropion; Call Centers; Female; Health Personnel; Humans; Information Services; Nicotine; Pregnancy; Smoking; Smoking Cessation; Teratology; Tobacco Use Cessation Devices; Varenicline

2020
Nicotine dependence (trait) and acute nicotinic stimulation (state) modulate attention but not inhibitory control: converging fMRI evidence from Go-Nogo and Flanker tasks.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2020, Volume: 45, Issue:5

    Topics: Adolescent; Adult; Attention; Brain; Brain Mapping; Cross-Over Studies; Double-Blind Method; Executive Function; Female; Humans; Inhibition, Psychological; Magnetic Resonance Imaging; Male; Middle Aged; Nicotine; Nicotinic Agonists; Smoking Cessation; Tobacco Use Disorder; Varenicline; Young Adult

2020
Assessment of individual differences in response to acute bupropion or varenicline treatment using a long-access nicotine self-administration model and behavioral economics in female rats.
    Behavioural brain research, 2020, 05-15, Volume: 385

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Behavior, Animal; Bupropion; Conditioning, Psychological; Economics, Behavioral; Extinction, Psychological; Female; Individuality; Nicotine; Nicotinic Agonists; Rats; Self Administration; Smoking Cessation Agents; Varenicline; Yohimbine

2020
Precision nicotine metabolism-informed care for smoking cessation in Crohn's disease: A pilot study.
    PloS one, 2020, Volume: 15, Issue:3

    Topics: Adult; Bupropion; Crohn Disease; Female; Humans; Male; Middle Aged; Nicotine; Patient Compliance; Pilot Projects; Prevalence; Randomized Controlled Trials as Topic; Severity of Illness Index; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Treatment Outcome; Varenicline

2020
Effects of ethanol, naltrexone, nicotine and varenicline in an ethanol and nicotine co-use model in Sprague-Dawley rats.
    Drug and alcohol dependence, 2020, 07-01, Volume: 212

    Topics: Alcohol Deterrents; Alcohol Drinking; Animals; Ethanol; Female; Male; Naltrexone; Nicotine; Rats; Rats, Sprague-Dawley; Self Administration; Smoking Cessation Agents; Tobacco Use Disorder; Varenicline

2020
Varenicline rescues nicotine-induced decrease in motivation for sucrose reinforcement.
    Behavioural brain research, 2021, 01-15, Volume: 397

    Topics: Animals; Behavior, Animal; Drug Interactions; Economics, Behavioral; Feeding Behavior; Male; Motivation; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Reinforcement, Psychology; Smoking Cessation Agents; Sucrose; Varenicline

2021
The importance of acquisition learning on nicotine and varenicline drug substitution in a drug-discriminated goal-tracking task.
    Pharmacology, biochemistry, and behavior, 2020, Volume: 199

    Topics: Animals; Discrimination Learning; Drug Substitution; Goals; Male; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Smoking Cessation Agents; Varenicline

2020
Self-Administration of Cotinine in Wistar Rats: Comparisons to Nicotine.
    The Journal of pharmacology and experimental therapeutics, 2021, Volume: 376, Issue:3

    Topics: Animals; Cotinine; Dose-Response Relationship, Drug; Drug Interactions; Female; Male; Mecamylamine; Nicotine; Rats; Rats, Wistar; Receptors, Nicotinic; Self Administration; Varenicline

2021
5-HT
    Progress in brain research, 2021, Volume: 259

    Topics: Humans; Molecular Targeted Therapy; Nicotine; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2021
Therapeutic concentrations of varenicline increases exocytotic release of catecholamines from human and rat adrenal chromaffin cells in the presence of nicotine.
    Neuropharmacology, 2021, 09-01, Volume: 195

    Topics: Acetylcholine; Adrenal Glands; Animals; Catecholamines; Cattle; Chromaffin Cells; Exocytosis; Humans; Nicotine; Nicotinic Agonists; Rats; Varenicline

2021
The Comparative Effectiveness of Varenicline and Nicotine Patches for Smoking Abstinence During Pregnancy: Evidence From a Population-based Cohort Study.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2021, 08-29, Volume: 23, Issue:10

    Topics: Australia; Cohort Studies; Female; Humans; Nicotine; Pregnancy; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2021
Stability of Varenicline Concentration in Saliva Over 21 Days at Three Storage Temperatures.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2022, 02-01, Volume: 24, Issue:2

    Topics: Cotinine; Humans; Nicotine; Saliva; Smoking Cessation; Temperature; Varenicline

2022
Assessing combined effects of varenicline and N-acetylcysteine on reducing nicotine seeking in rats.
    Addiction biology, 2022, Volume: 27, Issue:2

    Topics: Acetylcysteine; Animals; Nicotine; Rats; Smoking Cessation; Tobacco Use Disorder; Varenicline

2022
Dose-dependent effects of Varenicline on tobacco craving and withdrawal in tobacco smokers with and without schizophrenia.
    Drug and alcohol dependence, 2022, 05-01, Volume: 234

    Topics: Craving; Double-Blind Method; Humans; Nicotiana; Nicotine; Nicotinic Agonists; Schizophrenia; Smokers; Smoking; Substance Withdrawal Syndrome; Varenicline

2022
Characterising the use of varenicline: an analysis of the Australian dispensing claims data.
    Addiction (Abingdon, England), 2022, Volume: 117, Issue:10

    Topics: Aged; Australia; Benzazepines; Bupropion; Humans; Male; Nicotine; Nicotinic Agonists; Quinoxalines; Retrospective Studies; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2022
[Tobacco cessation treatment for people with schizophrenia].
    Revue medicale suisse, 2022, Jun-22, Volume: 18, Issue:787

    Topics: Benzazepines; Bupropion; Humans; Nicotine; Quinoxalines; Schizophrenia; Smoking Cessation; Tobacco Use Cessation; Tobacco Use Cessation Devices; Varenicline

2022
Trapping of Nicotinic Acetylcholine Receptor Ligands Assayed by
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2023, 01-04, Volume: 43, Issue:1

    Topics: Animals; Brain; Female; Ligands; Male; Mice; Nicotine; Positron-Emission Tomography; Receptors, Nicotinic; Tobacco Use Disorder; Varenicline

2023
Publicly subsidised smoking cessation medicines in times of COVID-19 in Australia: An interrupted time series analysis.
    Drug and alcohol review, 2023, Volume: 42, Issue:1

    Topics: Bupropion; COVID-19; Humans; Interrupted Time Series Analysis; Nicotine; Nicotinic Agonists; Pandemics; Pharmaceutical Preparations; Smoking; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2023
Varenicline serves as the training stimulus in the drug-discriminated goal-tracking task with rats: initial evaluation of potential neuropharmacological processes.
    Behavioural pharmacology, 2023, 02-01, Volume: 34, Issue:1

    Topics: Animals; Benzazepines; Bupropion; Goals; Motivation; Nicotine; Nicotinic Agonists; Quinoxalines; Rats; Receptors, Nicotinic; Smoking Cessation Agents; Varenicline

2023
Comparative effect of varenicline and nicotine patches on preventing repeat cardiovascular events.
    Heart (British Cardiac Society), 2023, 06-14, Volume: 109, Issue:13

    Topics: Aftercare; Cardiovascular Diseases; Cohort Studies; Female; Humans; Male; Nicotine; Nicotinic Agonists; Patient Discharge; Smoking Cessation; Tobacco Use Cessation Devices; Varenicline

2023
Role of neuronal nicotinic acetylcholine receptors in cannabinoid dependence.
    Pharmacological research, 2023, Volume: 191

    Topics: Cannabinoid Receptor Agonists; Cannabinoids; Humans; Nicotine; Nicotinic Agonists; Receptors, Nicotinic; Varenicline

2023
Varenicline mitigates the increased risk of pseudarthrosis associated with nicotine.
    The spine journal : official journal of the North American Spine Society, 2023, Volume: 23, Issue:8

    Topics: Animals; Male; Nicotine; Pseudarthrosis; Rats; Rats, Sprague-Dawley; Smoking Cessation; Varenicline

2023
Nicotine and Cytisine Embryotoxicity in the Experimental Zebrafish Model.
    International journal of molecular sciences, 2023, Jul-28, Volume: 24, Issue:15

    Topics: Alkaloids; Animals; Azocines; Benzazepines; Humans; Nicotine; Nicotinic Agonists; Quinolizines; Quinoxalines; Receptors, Nicotinic; Varenicline; Zebrafish

2023