Page last updated: 2024-08-26

nicotine and sazetidine-a

nicotine has been researched along with sazetidine-a in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's19 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bajjuri, KM; Brunner, D; Caldarone, B; Eaton, JB; Fedolak, A; Ghavami, A; Kozikowski, AP; Lowe, DA; Lukas, RJ; Paterson, NE; Tückmantel, W; Wang, D; Yu, LF; Yuen, PW; Zhang, H1
Al-Muhtasib, N; Brown, ML; Kellar, KJ; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Richardson, J; Sahibzada, N; Sexton, HG; Tran, T; Xiao, Y; Xie, T; Yenugonda, VM1
Al-Muhtasib, N; Brown, ML; Dakshanamurthy, S; Johnson, JE; Kellar, KJ; Kong, HS; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Sahibzada, N; Slade, S; Tomita, Y; Tran, T; Wells, C; Xiao, Y; Xie, T; Yenugonda, VM1
Brunner, D; Caldarone, BJ; Eaton, JB; Kozikowski, AP; Lukas, RJ; Onajole, OK; Thiede, L1
Binda, M; Bolchi, C; Budriesi, R; Fasoli, F; Fucile, S; Fumagalli, L; Gotti, C; Mucchietto, V; Pallavicini, M; Ruggeri, P; Sciaccaluga, M; Valoti, E1
Brown, ML; Cauley, M; Hampton, D; Kellar, KJ; Levin, ED; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Rose, JE; Slade, S; Wells, C; Xiao, Y1
Blendy, JA; Castellano, LM; Turner, JR1
Brown, ML; Kellar, KJ; Levin, ED; Li, TK; Lumeng, L; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Rose, JE; Slade, S; Wells, C; Xiao, Y1
Brown, ML; Johnson, JE; Kellar, KJ; Levin, ED; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Sexton, H; Slade, S; Wells, C; Xiao, Y1
DeCuir, D; Gordon, CJ; Kellar, KJ; Levin, ED; Rezvani, AH; Sexton, HG; Timofeeva, O; Xiao, Y1
Blendy, JA; Cousins, V; Hussmann, GP; Kellar, KJ; Levin, ED; Lomazzo, E; Perry, DC; Rezvani, AH; Turner, JR; Venkatesh, R; Wolfe, BB; Xiao, Y; Yasuda, RP1
Blendy, JA; Carlson, GC; Gould, TJ; Poole, RL; Turner, JR; Wilkinson, DS1
Blendy, JA; DeDominicis, KE; Forcelli, PA; Hussmann, GP; Kellar, KJ; Klehm, J; Lindstrom, J; Richardson, JR; Sahibzada, N; Turner, JR; Wolfe, BB; Xiao, Y; Yasuda, RP1
Abdullah, R; Banks, ML; Bettinger, JC; Carroll, FI; Damaj, IM; Dawson, A; Jackson, A; Miles, MF; Muldoon, PP; O'Brien, M; Slater, CA; Soll, LG; Tapper, AR1
Dezfuli, G; Dretchen, KL; Gillis, RA; Kellar, KJ; Sahibzada, N; Tizabi, Y1
Bevins, RA; Charntikov, S; Dwoskin, LP; Falco, AM; Fink, K1
Lee, AM; Maertens, JJ; Mason, MM; O'Rourke, KY; Touchette, JC1
Levin, ED; Rezvani, AH; Slade, S; Wells, C1
Kellar, KJ; Levin, ED; Rezvani, AH; Slade, S; Wells, C; Xiao, Y1

Other Studies

19 other study(ies) available for nicotine and sazetidine-a

ArticleYear
Chemistry and behavioral studies identify chiral cyclopropanes as selective α4β2-nicotinic acetylcholine receptor partial agonists exhibiting an antidepressant profile.
    Journal of medicinal chemistry, 2012, Jan-26, Volume: 55, Issue:2

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Cell Line; Crystallography, X-Ray; Drug Partial Agonism; Female; Humans; Ligands; Mice; Mice, Inbred BALB C; Molecular Conformation; Nicotinic Agonists; Radioligand Assay; Rats; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2012
Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective α4β2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats.
    Journal of medicinal chemistry, 2013, Apr-11, Volume: 56, Issue:7

    Topics: Alcohol Drinking; Animals; Ethanol; Ferrets; Ligands; Magnetic Resonance Spectroscopy; Pyridines; Rats; Receptors, Nicotinic; Spectrometry, Mass, Electrospray Ionization

2013
Design, synthesis and discovery of picomolar selective α4β2 nicotinic acetylcholine receptor ligands.
    Journal of medicinal chemistry, 2013, Nov-14, Volume: 56, Issue:21

    Topics: Azetidines; Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Discovery; Humans; Ligands; Models, Molecular; Molecular Structure; Pyridines; Receptors, Nicotinic; Software; Structure-Activity Relationship

2013
Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selective α4β2-nAChR Ligands.
    ACS medicinal chemistry letters, 2014, Nov-13, Volume: 5, Issue:11

    Topics:

2014
Chemistry and Pharmacology of a Series of Unichiral Analogues of 2-(2-Pyrrolidinyl)-1,4-benzodioxane, Prolinol Phenyl Ether, and Prolinol 3-Pyridyl Ether Designed as α4β2-Nicotinic Acetylcholine Receptor Agonists.
    Journal of medicinal chemistry, 2015, Aug-27, Volume: 58, Issue:16

    Topics: Animals; Brain Chemistry; Cell Line; Dioxanes; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Conformation; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Phenyl Ethers; Pyridines; Pyrrolidines; Rats; Receptors, Nicotinic; Structure-Activity Relationship

2015
Sazetidine-A, a selective alpha4beta2 nicotinic receptor desensitizing agent and partial agonist, reduces nicotine self-administration in rats.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:3

    Topics: Animals; Azetidines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Partial Agonism; Food; Male; Motivation; Motor Activity; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration

2010
Nicotinic partial agonists varenicline and sazetidine-A have differential effects on affective behavior.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 334, Issue:2

    Topics: Animals; Anxiety; Azetidines; Behavior, Animal; Benzazepines; Chimera; Depression; Drug Partial Agonism; Male; Mice; Mood Disorders; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Varenicline

2010
Effects of sazetidine-A, a selective alpha4beta2 nicotinic acetylcholine receptor desensitizing agent on alcohol and nicotine self-administration in selectively bred alcohol-preferring (P) rats.
    Psychopharmacology, 2010, Volume: 211, Issue:2

    Topics: Animals; Azetidines; Dose-Response Relationship, Drug; Drug Administration Schedule; Ethanol; Male; Naltrexone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Pyridines; Rats; Receptors, Nicotinic; Reward; Saccharin; Self Administration

2010
Assessing the effects of chronic sazetidine-A delivery on nicotine self-administration in both male and female rats.
    Psychopharmacology, 2012, Volume: 222, Issue:2

    Topics: Animals; Azetidines; Dose-Response Relationship, Drug; Female; Male; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Sex Factors; Smoking Cessation

2012
Effects of sazetidine-A, a selective α4β2* nicotinic receptor desensitizing agent, on body temperature regulation in mice and rats.
    European journal of pharmacology, 2012, May-05, Volume: 682, Issue:1-3

    Topics: Aconitine; Animals; Azetidines; Body Temperature Regulation; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Nicotine; Nicotinic Antagonists; Pyridines; Rats; Receptors, Nicotinic

2012
Chronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 343, Issue:2

    Topics: Animals; Azetidines; Behavior, Animal; Benzazepines; Binding Sites; Brain Chemistry; Cerebral Cortex; Dose-Response Relationship, Drug; Female; Male; Membranes; Neurons; Nicotine; Nicotinic Agonists; Pregnancy; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Up-Regulation; Varenicline

2012
Divergent functional effects of sazetidine-a and varenicline during nicotine withdrawal.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:10

    Topics: Animals; Anxiety; Azetidines; Benzazepines; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Partial Agonism; Evoked Potentials; Hippocampus; Male; Mice; Microinjections; Motor Activity; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Up-Regulation; Varenicline

2013
Chronic sazetidine-A maintains anxiolytic effects and slower weight gain following chronic nicotine without maintaining increased density of nicotinic receptors in rodent brain.
    Journal of neurochemistry, 2014, Volume: 129, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azetidines; Benzazepines; Brain Chemistry; Drug Evaluation, Preclinical; Feeding Behavior; Gene Expression Regulation; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Substance Withdrawal Syndrome; Tobacco Use Cessation; Tobacco Use Disorder; Up-Regulation; Varenicline; Weight Gain

2014
Nicotine Enhances the Hypnotic and Hypothermic Effects of Alcohol in the Mouse.
    Alcoholism, clinical and experimental research, 2016, Volume: 40, Issue:1

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Azetidines; Body Temperature; Central Nervous System Depressants; Drug Interactions; Ethanol; Hypnotics and Sedatives; Hypothermia; Ketamine; Mecamylamine; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Pyridines; Receptors, Nicotinic; Reflex, Righting; Varenicline

2016
Evidence for the role of β2* nAChR desensitization in regulating body weight in obese mice.
    Neuropharmacology, 2016, Volume: 110, Issue:Pt A

    Topics: Animals; Azetidines; Body Weight; Eating; Infusion Pumps; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Mice, Transgenic; Nicotine; Pyridines; Receptors, Nicotinic

2016
The effect of sazetidine-A and other nicotinic ligands on nicotine controlled goal-tracking in female and male rats.
    Neuropharmacology, 2017, Volume: 113, Issue:Pt A

    Topics: Animals; Azetidines; Discrimination Learning; Female; Goals; Ligands; Male; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Sex Factors

2017
The nicotinic receptor drug sazetidine-A reduces alcohol consumption in mice without affecting concurrent nicotine consumption.
    Neuropharmacology, 2018, 05-01, Volume: 133

    Topics: Alcohol Drinking; Animals; Azetidines; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Female; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Pyridines; Self Administration; Substance Withdrawal Syndrome; Time Factors; Tobacco Use Disorder

2018
Mutually augmenting interactions of dextromethorphan and sazetidine-A for reducing nicotine self-administration in rats.
    Pharmacology, biochemistry, and behavior, 2018, Volume: 166

    Topics: Animals; Azetidines; Behavior, Addictive; Dextromethorphan; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Excitatory Amino Acid Antagonists; Female; Locomotion; Nicotine; Pyridines; Rats; Rats, Sprague-Dawley; Self Administration; Smoking Cessation Agents

2018
Oral sazetidine-A, a selective α4β2* nicotinic receptor desensitizing agent, reduces nicotine self-administration in rats.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 179

    Topics: Administration, Oral; Animals; Azetidines; Female; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic

2019