nicotine has been researched along with sazetidine-a in 19 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 19 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bajjuri, KM; Brunner, D; Caldarone, B; Eaton, JB; Fedolak, A; Ghavami, A; Kozikowski, AP; Lowe, DA; Lukas, RJ; Paterson, NE; Tückmantel, W; Wang, D; Yu, LF; Yuen, PW; Zhang, H | 1 |
Al-Muhtasib, N; Brown, ML; Kellar, KJ; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Richardson, J; Sahibzada, N; Sexton, HG; Tran, T; Xiao, Y; Xie, T; Yenugonda, VM | 1 |
Al-Muhtasib, N; Brown, ML; Dakshanamurthy, S; Johnson, JE; Kellar, KJ; Kong, HS; Levin, ED; Liu, Y; Paige, M; Rezvani, AH; Sahibzada, N; Slade, S; Tomita, Y; Tran, T; Wells, C; Xiao, Y; Xie, T; Yenugonda, VM | 1 |
Brunner, D; Caldarone, BJ; Eaton, JB; Kozikowski, AP; Lukas, RJ; Onajole, OK; Thiede, L | 1 |
Binda, M; Bolchi, C; Budriesi, R; Fasoli, F; Fucile, S; Fumagalli, L; Gotti, C; Mucchietto, V; Pallavicini, M; Ruggeri, P; Sciaccaluga, M; Valoti, E | 1 |
Brown, ML; Cauley, M; Hampton, D; Kellar, KJ; Levin, ED; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Rose, JE; Slade, S; Wells, C; Xiao, Y | 1 |
Blendy, JA; Castellano, LM; Turner, JR | 1 |
Brown, ML; Kellar, KJ; Levin, ED; Li, TK; Lumeng, L; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Rose, JE; Slade, S; Wells, C; Xiao, Y | 1 |
Brown, ML; Johnson, JE; Kellar, KJ; Levin, ED; McDowell, BE; Paige, MA; Petro, A; Rezvani, AH; Sexton, H; Slade, S; Wells, C; Xiao, Y | 1 |
DeCuir, D; Gordon, CJ; Kellar, KJ; Levin, ED; Rezvani, AH; Sexton, HG; Timofeeva, O; Xiao, Y | 1 |
Blendy, JA; Cousins, V; Hussmann, GP; Kellar, KJ; Levin, ED; Lomazzo, E; Perry, DC; Rezvani, AH; Turner, JR; Venkatesh, R; Wolfe, BB; Xiao, Y; Yasuda, RP | 1 |
Blendy, JA; Carlson, GC; Gould, TJ; Poole, RL; Turner, JR; Wilkinson, DS | 1 |
Blendy, JA; DeDominicis, KE; Forcelli, PA; Hussmann, GP; Kellar, KJ; Klehm, J; Lindstrom, J; Richardson, JR; Sahibzada, N; Turner, JR; Wolfe, BB; Xiao, Y; Yasuda, RP | 1 |
Abdullah, R; Banks, ML; Bettinger, JC; Carroll, FI; Damaj, IM; Dawson, A; Jackson, A; Miles, MF; Muldoon, PP; O'Brien, M; Slater, CA; Soll, LG; Tapper, AR | 1 |
Dezfuli, G; Dretchen, KL; Gillis, RA; Kellar, KJ; Sahibzada, N; Tizabi, Y | 1 |
Bevins, RA; Charntikov, S; Dwoskin, LP; Falco, AM; Fink, K | 1 |
Lee, AM; Maertens, JJ; Mason, MM; O'Rourke, KY; Touchette, JC | 1 |
Levin, ED; Rezvani, AH; Slade, S; Wells, C | 1 |
Kellar, KJ; Levin, ED; Rezvani, AH; Slade, S; Wells, C; Xiao, Y | 1 |
19 other study(ies) available for nicotine and sazetidine-a
Article | Year |
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Chemistry and behavioral studies identify chiral cyclopropanes as selective α4β2-nicotinic acetylcholine receptor partial agonists exhibiting an antidepressant profile.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Cell Line; Crystallography, X-Ray; Drug Partial Agonism; Female; Humans; Ligands; Mice; Mice, Inbred BALB C; Molecular Conformation; Nicotinic Agonists; Radioligand Assay; Rats; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship | 2012 |
Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selective α4β2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats.
Topics: Alcohol Drinking; Animals; Ethanol; Ferrets; Ligands; Magnetic Resonance Spectroscopy; Pyridines; Rats; Receptors, Nicotinic; Spectrometry, Mass, Electrospray Ionization | 2013 |
Design, synthesis and discovery of picomolar selective α4β2 nicotinic acetylcholine receptor ligands.
Topics: Azetidines; Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Discovery; Humans; Ligands; Models, Molecular; Molecular Structure; Pyridines; Receptors, Nicotinic; Software; Structure-Activity Relationship | 2013 |
Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selective α4β2-nAChR Ligands.
Topics: | 2014 |
Chemistry and Pharmacology of a Series of Unichiral Analogues of 2-(2-Pyrrolidinyl)-1,4-benzodioxane, Prolinol Phenyl Ether, and Prolinol 3-Pyridyl Ether Designed as α4β2-Nicotinic Acetylcholine Receptor Agonists.
Topics: Animals; Brain Chemistry; Cell Line; Dioxanes; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Conformation; Nicotine; Nicotinic Agonists; Patch-Clamp Techniques; Phenyl Ethers; Pyridines; Pyrrolidines; Rats; Receptors, Nicotinic; Structure-Activity Relationship | 2015 |
Sazetidine-A, a selective alpha4beta2 nicotinic receptor desensitizing agent and partial agonist, reduces nicotine self-administration in rats.
Topics: Animals; Azetidines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Partial Agonism; Food; Male; Motivation; Motor Activity; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration | 2010 |
Nicotinic partial agonists varenicline and sazetidine-A have differential effects on affective behavior.
Topics: Animals; Anxiety; Azetidines; Behavior, Animal; Benzazepines; Chimera; Depression; Drug Partial Agonism; Male; Mice; Mood Disorders; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Varenicline | 2010 |
Effects of sazetidine-A, a selective alpha4beta2 nicotinic acetylcholine receptor desensitizing agent on alcohol and nicotine self-administration in selectively bred alcohol-preferring (P) rats.
Topics: Animals; Azetidines; Dose-Response Relationship, Drug; Drug Administration Schedule; Ethanol; Male; Naltrexone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Pyridines; Rats; Receptors, Nicotinic; Reward; Saccharin; Self Administration | 2010 |
Assessing the effects of chronic sazetidine-A delivery on nicotine self-administration in both male and female rats.
Topics: Animals; Azetidines; Dose-Response Relationship, Drug; Female; Male; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Sex Factors; Smoking Cessation | 2012 |
Effects of sazetidine-A, a selective α4β2* nicotinic receptor desensitizing agent, on body temperature regulation in mice and rats.
Topics: Aconitine; Animals; Azetidines; Body Temperature Regulation; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Nicotine; Nicotinic Antagonists; Pyridines; Rats; Receptors, Nicotinic | 2012 |
Chronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain.
Topics: Animals; Azetidines; Behavior, Animal; Benzazepines; Binding Sites; Brain Chemistry; Cerebral Cortex; Dose-Response Relationship, Drug; Female; Male; Membranes; Neurons; Nicotine; Nicotinic Agonists; Pregnancy; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Self Administration; Up-Regulation; Varenicline | 2012 |
Divergent functional effects of sazetidine-a and varenicline during nicotine withdrawal.
Topics: Animals; Anxiety; Azetidines; Benzazepines; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Partial Agonism; Evoked Potentials; Hippocampus; Male; Mice; Microinjections; Motor Activity; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Receptors, Nicotinic; Smoking Cessation; Substance Withdrawal Syndrome; Up-Regulation; Varenicline | 2013 |
Chronic sazetidine-A maintains anxiolytic effects and slower weight gain following chronic nicotine without maintaining increased density of nicotinic receptors in rodent brain.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Azetidines; Benzazepines; Brain Chemistry; Drug Evaluation, Preclinical; Feeding Behavior; Gene Expression Regulation; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Substance Withdrawal Syndrome; Tobacco Use Cessation; Tobacco Use Disorder; Up-Regulation; Varenicline; Weight Gain | 2014 |
Nicotine Enhances the Hypnotic and Hypothermic Effects of Alcohol in the Mouse.
Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Azetidines; Body Temperature; Central Nervous System Depressants; Drug Interactions; Ethanol; Hypnotics and Sedatives; Hypothermia; Ketamine; Mecamylamine; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Pyridines; Receptors, Nicotinic; Reflex, Righting; Varenicline | 2016 |
Evidence for the role of β2* nAChR desensitization in regulating body weight in obese mice.
Topics: Animals; Azetidines; Body Weight; Eating; Infusion Pumps; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Mice, Transgenic; Nicotine; Pyridines; Receptors, Nicotinic | 2016 |
The effect of sazetidine-A and other nicotinic ligands on nicotine controlled goal-tracking in female and male rats.
Topics: Animals; Azetidines; Discrimination Learning; Female; Goals; Ligands; Male; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Sex Factors | 2017 |
The nicotinic receptor drug sazetidine-A reduces alcohol consumption in mice without affecting concurrent nicotine consumption.
Topics: Alcohol Drinking; Animals; Azetidines; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Female; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Pyridines; Self Administration; Substance Withdrawal Syndrome; Time Factors; Tobacco Use Disorder | 2018 |
Mutually augmenting interactions of dextromethorphan and sazetidine-A for reducing nicotine self-administration in rats.
Topics: Animals; Azetidines; Behavior, Addictive; Dextromethorphan; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Excitatory Amino Acid Antagonists; Female; Locomotion; Nicotine; Pyridines; Rats; Rats, Sprague-Dawley; Self Administration; Smoking Cessation Agents | 2018 |
Oral sazetidine-A, a selective α4β2* nicotinic receptor desensitizing agent, reduces nicotine self-administration in rats.
Topics: Administration, Oral; Animals; Azetidines; Female; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic | 2019 |