nicardipine and papaverine

nicardipine has been researched along with papaverine in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19905 (17.24)18.7374
1990's12 (41.38)18.2507
2000's5 (17.24)29.6817
2010's7 (24.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Kaku, Y; Kazekawa, K; Tsukahara, T; Yonekawa, Y1
Aoki, K; Kishimoto, T; Naruchi, T; Okamiya, Y; Takeshita, T; Tanabe, H1
Karasawa, A; Kubo, K; Nakamizo, N; Oka, T; Shuto, K1
Bongrani, S; Razzetti, R; Schiantarelli, P2
Endoh, M; Taira, N; Yanagisawa, T1
Arimitsu, T; Mori, K; Oda, Y; Okumura, T1
Ogihara, M1
Hayakawa, T; Ioku, M; Kataoka, K; Kuroda, R; Niiyama, K; Taneda, M; Uejima, T; Yamada, K1
Han, H; Macdonald, RL; Zhang, J1
Advenier, C; Candenas, ML; Martin, JD; Moreau, J; Naline, E; Norte, M; Palette, C; Pays, M1
Asano, T; Itoh, S; Kaizu, H; Matsui, T1
Arnaboldi, R; Benzi, G; Ghigini, B; Gorini, A; Villa, R1
Hashimoto, N; Kazekawa, K; Kobayashi, A; Tsukahara, T; Yoshimura, S1
Melon, E; Rimaniol, JM1
Cromeens, DM; Evans, GR; Gherardini, G; Gürlek, A; Joly, GA; Kilbourn, RG; Langstein, H; Lundeberg, T; Sukumaran, AV; Wang, B; Williams, J1
Blin, D; Chavanon, O; Cracowski, JL; Durand, M; Hacini, R; Noirclerc, M; Stanke, F1
Az-Ma, T; Saeki, N; Yuge, O1
Hoh, BL; Ogilvy, CS1
Abdennour, L; Boch, AL; Bonneville, F; Lejean, L; Puybasset, L1
Aggour, M; Moret, J; Pierot, L1
Koolen, PG; Lee, BT; Lin, SJ; Ricci, JA; Shah, J; Tobias, AM1

Reviews

4 review(s) available for nicardipine and papaverine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
[Pharmacological treatment of vasospasm in subarachnoid hemorrhage].
    Annales francaises d'anesthesie et de reanimation, 1996, Volume: 15, Issue:3

    Topics: Antioxidants; Humans; Ischemic Attack, Transient; Lipid Peroxides; Male; Nicardipine; Nimodipine; Papaverine; Plasminogen Activators; Pregnatrienes; Subarachnoid Hemorrhage; Tissue Plasminogen Activator; Vasodilator Agents

1996
Endovascular treatment of cerebral vasospasm: transluminal balloon angioplasty, intra-arterial papaverine, and intra-arterial nicardipine.
    Neurosurgery clinics of North America, 2005, Volume: 16, Issue:3

    Topics: Angioplasty, Balloon; Humans; Injections, Intra-Arterial; Nicardipine; Papaverine; Vasodilator Agents; Vasospasm, Intracranial

2005
Vasospasm after aneurysmal subarachnoid hemorrhage: recent advances in endovascular management.
    Current opinion in critical care, 2010, Volume: 16, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Angioplasty, Balloon; Critical Care; Endovascular Procedures; Humans; Intensive Care Units; Milrinone; Nicardipine; Papaverine; Risk Factors; Subarachnoid Hemorrhage; Vasodilator Agents; Vasospasm, Intracranial; Verapamil

2010

Trials

1 trial(s) available for nicardipine and papaverine

ArticleYear
Effect of topical vasodilators on gastroepiploic artery graft.
    The Annals of thoracic surgery, 1999, Volume: 67, Issue:5

    Topics: Administration, Topical; Aged; Arteries; Coronary Artery Bypass; Double-Blind Method; Female; Hemodynamics; Humans; Intraoperative Period; Male; Middle Aged; Molsidomine; Nicardipine; Nitroglycerin; Papaverine; Regional Blood Flow; Stomach; Vasodilator Agents

1999

Other Studies

24 other study(ies) available for nicardipine and papaverine

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Superselective intra-arterial infusion of papaverine for the treatment of cerebral vasospasm after subarachnoid hemorrhage.
    Journal of neurosurgery, 1992, Volume: 77, Issue:6

    Topics: Adult; Aged; Aged, 80 and over; Aneurysm, Ruptured; Angioplasty, Balloon; Female; Humans; Infusions, Intra-Arterial; Intracranial Aneurysm; Ischemic Attack, Transient; Male; Middle Aged; Nicardipine; Papaverine; Radiography; Rupture, Spontaneous; Subarachnoid Hemorrhage; Urokinase-Type Plasminogen Activator

1992
Effect of TC-81, a new dihydropyridine derivative, on K(+)-induced contraction in rat aorta.
    European journal of pharmacology, 1991, Nov-19, Volume: 205, Issue:1

    Topics: Animals; Aorta; Calcium; Calcium Radioisotopes; Dihydropyridines; Diltiazem; In Vitro Techniques; Isometric Contraction; Male; Nicardipine; Nifedipine; Papaverine; Potassium; Rats; Rats, Inbred Strains; Vasoconstriction; Vasodilator Agents

1991
Vasodilating effects of the new calcium antagonist benidipine hydrochloride in anesthetized dogs and cats.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Blood Flow Velocity; Blood Pressure; Calcium Channel Blockers; Cats; Cerebral Cortex; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Injections, Intra-Arterial; Injections, Intravenous; Male; Nicardipine; Nifedipine; Papaverine; Vasodilation; Vasodilator Agents

1988
Regional vasodilating and cardiac effects of nicardipine in anaesthetized open chest dog.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 273, Issue:2

    Topics: Animals; Blood Pressure; Coronary Circulation; Dogs; Femoral Artery; Heart; Heart Rate; Nicardipine; Nifedipine; Papaverine; Regional Blood Flow; Vascular Resistance; Vasodilator Agents; Verapamil

1985
Dissociation of cyclic AMP and contractile responses to isoprenaline: effects of a dihydropyridine derivative, nicardipine (YC-93), on canine ventricular muscle.
    European journal of pharmacology, 1980, Oct-17, Volume: 67, Issue:2-3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Calcium; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; Gallopamil; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Nicardipine; Nifedipine; Papaverine; Pyridines; Theophylline; Vasodilator Agents

1980
In vitro effects of nicardipine on vascular and cardiac muscle preparations.
    Pharmacological research communications, 1984, Volume: 16, Issue:8

    Topics: Animals; Aorta, Thoracic; Blood Vessels; Coronary Vessels; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Nicardipine; Nifedipine; Papaverine; Rabbits; Vascular Resistance; Vasodilation; Verapamil

1984
[Sustained-release pellet of vasodilators--basic experiment].
    No shinkei geka. Neurological surgery, 1984, Volume: 12, Issue:11

    Topics: Delayed-Action Preparations; Diltiazem; Humans; Intracranial Aneurysm; Ischemic Attack, Transient; Nicardipine; Nifedipine; Papaverine; Rupture, Spontaneous; Silicone Elastomers; Subarachnoid Hemorrhage; Temperature

1984
Nifedipine and nicardipine potentiate glucagon-stimulated glycogenolysis in primary cultures of rat hepatocytes.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:9

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Caffeine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Glucagon; Glycogen; Liver; Male; Nicardipine; Nifedipine; Papaverine; Rats; Rats, Wistar

1993
Treatment of severe localized cerebral vasospasm following recurrent hemorrhage from middle cerebral artery aneurysm--case report.
    Neurologia medico-chirurgica, 1993, Volume: 33, Issue:12

    Topics: Brain; Cerebral Angiography; Cerebral Arteries; Female; Humans; Intracranial Aneurysm; Ischemic Attack, Transient; Middle Aged; Nicardipine; Papaverine; Subarachnoid Hemorrhage; Tomography, X-Ray Computed

1993
Angioplasty reduces pharmacologically mediated vasoconstriction in rabbit carotid arteries with and without vasospasm.
    Stroke, 1995, Volume: 26, Issue:6

    Topics: Acetylcholine; Analysis of Variance; Angioplasty; Animals; Carotid Arteries; In Vitro Techniques; Ischemic Attack, Transient; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Papaverine; Potassium; Rabbits; Serotonin; Time Factors; Vasoconstriction

1995
Effects of okadaic acid on the human isolated bronchus.
    European journal of pharmacology, 1994, May-02, Volume: 256, Issue:3

    Topics: Acetylcholine; Bronchi; Cadmium; Cadmium Compounds; Caffeine; Dose-Response Relationship, Drug; Ethers, Cyclic; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Nicardipine; Okadaic Acid; Papaverine; Phosphatidylinositols; Potassium Chloride; Sulfates; Vasoconstrictor Agents

1994
The role of active smooth-muscle contraction in the occurrence of chronic vasospasm in the canine two-hemorrhage model.
    Journal of neurosurgery, 1994, Volume: 80, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Basilar Artery; Dogs; Female; Ischemic Attack, Transient; Isoquinolines; Male; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Papaverine; Piperazines; Protein Kinase C; Radiography; Subarachnoid Hemorrhage; Vasodilation

1994
Effect of intermittent mild hypoxia and drug treatment on synaptosomal nonmitochondrial ATPase activities.
    Journal of neuroscience research, 1993, Apr-15, Volume: 34, Issue:6

    Topics: Adenosine Triphosphatases; Animals; Cerebral Cortex; Energy Metabolism; Hypoxia; In Vitro Techniques; Lipid Metabolism; Male; Morpholines; Nicardipine; Oxygen Consumption; Papaverine; Phosphatidylcholines; Rats; Rats, Wistar; Synaptic Membranes; Synaptosomes; Thiophenes

1993
Intra-arterial infusion of papaverine combined with intravenous administration of high-dose nicardipine for cerebral vasospasm.
    Acta neurochirurgica, 1995, Volume: 135, Issue:3-4

    Topics: Adult; Aged; Aneurysm, Ruptured; Calcium Channel Blockers; Cerebral Angiography; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Infusions, Intra-Arterial; Infusions, Intravenous; Intracranial Aneurysm; Ischemic Attack, Transient; Male; Middle Aged; Nicardipine; Papaverine; Subarachnoid Hemorrhage; Ultrasonography, Doppler, Transcranial; Vasodilator Agents

1995
Drug-induced vasodilation in an in vitro and in vivo study: the effects of nicardipine, papaverine, and lidocaine on the rabbit carotid artery.
    Plastic and reconstructive surgery, 1997, Volume: 100, Issue:6

    Topics: Administration, Topical; Anastomosis, Surgical; Animals; Blood Pressure; Carotid Arteries; Dose-Response Relationship, Drug; Follow-Up Studies; Ischemia; Isotonic Solutions; Lidocaine; Microcirculation; Microsurgery; Monitoring, Physiologic; Nicardipine; Norepinephrine; Papaverine; Rabbits; Regional Blood Flow; Single-Blind Method; Surgical Flaps; Ultrasonography, Doppler; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

1997
Differential action of spasmolytic vasodilators on platelet aggregation and endothelial cell-dependent anti-aggregation.
    Acta anaesthesiologica Scandinavica, 2000, Volume: 44, Issue:4

    Topics: Alprostadil; Animals; Aorta; Cells, Cultured; Diltiazem; Dose-Response Relationship, Drug; Endothelium, Vascular; Nicardipine; Nitroglycerin; Nitroprusside; Papaverine; Pentobarbital; Platelet Aggregation; Platelet Aggregation Inhibitors; Swine; Sympatholytics; Vasodilator Agents

2000
[Endovascular treatment of vasospasm following subarachnoid aneurysmal haemorrhage].
    Annales francaises d'anesthesie et de reanimation, 2007, Volume: 26, Issue:11

    Topics: Calcium Channel Blockers; Humans; Intracranial Aneurysm; Nicardipine; Nimodipine; Nitroprusside; Papaverine; Phosphodiesterase Inhibitors; Subarachnoid Hemorrhage; Vasospasm, Intracranial

2007
Comparing the Outcomes of Different Agents to Treat Vasospasm at Microsurgical Anastomosis during the Papaverine Shortage.
    Plastic and reconstructive surgery, 2016, Volume: 138, Issue:3

    Topics: Administration, Topical; Aged; Anastomosis, Surgical; Drug Substitution; Female; Free Tissue Flaps; Graft Survival; Humans; Intraoperative Complications; Lidocaine; Microsurgery; Middle Aged; Nicardipine; Outcome Assessment, Health Care; Papaverine; Parasympatholytics; Retrospective Studies; Vasoconstriction

2016