nicardipine and nilvadipine

nicardipine has been researched along with nilvadipine in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19905 (23.81)18.7374
1990's11 (52.38)18.2507
2000's3 (14.29)29.6817
2010's2 (9.52)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aisaka, K; Cho, H; Hamaguchi, M; Hayashimatsu, M; Hidaka, T; Mizuno, A; Ohnaka, Y; Shima, K; Takeuchi, Y; Ueda, M1
Coassolo, P; Lavé, T; Schneider, G1
Topliss, JG; Yoshida, F1
Horinouchi, M; Komada, F; Nishiguchi, K; Ohmoto, N; Ohnishi, N; Okumura, K; Sakaeda, T; Takara, K; Tanigawara, Y; Yokoyama, T1
Sun, H1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Fujiwara, T; Kohsaka, M; Mori, J; Satoh, H; Sogabe, K; Takakura, S; Tokuma, Y; Totsuka, Z1
Furuichi, Y; Kohsaka, M; Mori, J; Satoh, H; Takakura, S1
Handa, J; Mori, J; Satoh, H; Shiino, A; Susumu, T; Takakura, S1
Handa, J; Inubushi, T; Kido, C; Matsuda, M; Morikawa, S; Shiino, A; Susumu, T1
Furui, H; Furumichi, T; Saito, H; Yamada, Y; Yamauchi, K; Yokota, M1
Furuta, T1
Koibuchi, Y; Miura, S; Ohtsuka, M; Ono, T; Sakai, S; Shibayama, F1
Kuwaki, T; Nishimura, T; Ono, T; Satoh, H; Shibayama, F; Yamashita, T1
Ishii, A; Nakamizo, N; Nishida, K; Oka, T1
Sanada, H1
Kikuchi, K; Sugawara, H; Tobise, K1
Akaike, N; Ishibashi, H; Rhee, JS1
Hayasaka, S; Hiraki, S; Zhang, XY1
Matsuda, Y; Tsukuda, E1
Dezawa, M; Ishikawa, F; Ishikawa, H; Mamiya, K; Metoki, T; Nakazawa, M; Ohguro, H; Ohguro, I; Takano, Y; Yamazaki, H1

Other Studies

21 other study(ies) available for nicardipine and nilvadipine

ArticleYear
Dihydropyrimidines: novel calcium antagonists with potent and long-lasting vasodilative and antihypertensive activity.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:10

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Dogs; Female; Heart Rate; Indicators and Reagents; Male; Molecular Structure; Pyrimidines; Rats; Rats, Inbred SHR; Receptors, Nicotinic; Structure-Activity Relationship; Vasodilator Agents

1989
Combining in vitro and in vivo pharmacokinetic data for prediction of hepatic drug clearance in humans by artificial neural networks and multivariate statistical techniques.
    Journal of medicinal chemistry, 1999, Dec-16, Volume: 42, Issue:25

    Topics: Animals; Biological Availability; Dogs; Humans; Least-Squares Analysis; Liver; Multivariate Analysis; Neural Networks, Computer; Pharmacokinetics; Rats

1999
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Effects of 12 Ca2+ antagonists on multidrug resistance, MDR1-mediated transport and MDR1 mRNA expression.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2002, Volume: 16, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cell Line; Digoxin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Gene Expression; Humans; Nifedipine; Paclitaxel; RNA, Messenger; Swine; Tritium; Tumor Cells, Cultured; Verapamil; Vinblastine

2002
Capture hydrolysis signals in the microsomal stability assay: molecular mechanisms of the alkyl ester drug and prodrug metabolism.
    Bioorganic & medicinal chemistry letters, 2012, Jan-15, Volume: 22, Issue:2

    Topics: Carboxylic Acids; Cytochrome P-450 Enzyme System; Esters; Humans; Hydrolysis; Microsomes; Models, Molecular; Molecular Structure; Prodrugs; Quantum Theory; Signal Transduction

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Nilvadipine as a neuroprotective calcium entry blocker in a rat model of global cerebral ischemia. A comparative study with nicardipine hydrochloride.
    Neuroscience letters, 1992, Jul-20, Volume: 141, Issue:2

    Topics: Animals; Brain; Brain Ischemia; Calcium Channel Blockers; Decerebrate State; Fatty Acids, Nonesterified; Male; Nicardipine; Nifedipine; Rats; Rats, Sprague-Dawley

1992
Effects of nilvadipine on neuronal function in the ischemic cat brain.
    Surgical neurology, 1992, Volume: 37, Issue:4

    Topics: Animals; Brain; Brain Ischemia; Calcium Channel Blockers; Cats; Cerebrovascular Circulation; Evoked Potentials, Somatosensory; Female; Male; Neurons; Nicardipine; Nifedipine

1992
Nilvadipine, a new calcium channel blocker, reduces ischemic brain injury in rats.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:4

    Topics: Animals; Brain Ischemia; Calcium Channel Blockers; Cerebral Infarction; Nicardipine; Nifedipine; Rats; Rats, Inbred SHR

1991
[Ca++ antagonist and acute brain ischemia: effects of nilvadipine and nicardipine on middle cerebral artery occlusion in rats].
    Nihon geka hokan. Archiv fur japanische Chirurgie, 1991, Jan-01, Volume: 60, Issue:1

    Topics: Acute Disease; Animals; Calcium Channel Blockers; Cerebral Infarction; Constriction; Ischemic Attack, Transient; Magnetic Resonance Imaging; Male; Nicardipine; Nifedipine; Rats; Rats, Inbred Strains

1991
Protective effects of calcium channel blockers on hydrogen peroxide induced increases in endothelial permeability.
    Cardiovascular research, 1990, Volume: 24, Issue:12

    Topics: Albumins; Calcium Channel Blockers; Capillary Permeability; Cell Membrane Permeability; Cells, Cultured; Diltiazem; Electric Conductivity; Endothelium, Vascular; Humans; Hydrogen Peroxide; Nicardipine; Nifedipine; Verapamil

1990
Prolonged inhibitory effects of nilvadipine (FR34235) following washout in isolated rabbit aorta and mesenteric artery.
    Journal of cardiovascular pharmacology, 1988, Volume: 11, Issue:2

    Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Diltiazem; Female; In Vitro Techniques; Male; Mesenteric Arteries; Nicardipine; Nifedipine; Norepinephrine; Potassium Chloride; Rabbits; Vasodilator Agents

1988
Suppression of atherogenesis in cholesterol-fed rabbits treated with nilvadipine, a new vasoselective calcium entry blocker.
    Atherosclerosis, 1989, Volume: 79, Issue:2-3

    Topics: Animals; Aorta, Thoracic; Arteriosclerosis; Blood Pressure; Calcium; Calcium Channel Blockers; Cholesterol; Liver; Male; Myocardium; Nicardipine; Nifedipine; Rabbits

1989
Nilvadipine attenuates ischemic degradation of gerbil brain cytoskeletal proteins.
    Stroke, 1989, Volume: 20, Issue:1

    Topics: Animals; Brain; Brain Ischemia; Calmodulin-Binding Proteins; Clathrin; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Gerbillinae; Male; Microtubule-Associated Proteins; Nicardipine; Nifedipine; Nimodipine

1989
Slow dissociation of the new slow-onset and long-acting calcium antagonist benidipine hydrochloride from 3H-nitrendipine binding sites.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Male; Nicardipine; Nifedipine; Nisoldipine; Nitrendipine; Rats; Rats, Inbred Strains

1988
[Effects of calcium antagonists on prostaglandin E2 production in cultured human amnion cells].
    Nihon Sanka Fujinka Gakkai zasshi, 1994, Volume: 46, Issue:2

    Topics: Amnion; Calcium Channel Blockers; Cells, Cultured; Depression, Chemical; Diltiazem; Dinoprostone; Dose-Response Relationship, Drug; Egtazic Acid; Female; Humans; Interleukin-1; Nicardipine; Nifedipine; Phospholipases A; Phospholipases A2; Pregnancy; Verapamil

1994
Antioxidant effects of calcium antagonists on rat myocardial membrane lipid peroxidation.
    Hypertension research : official journal of the Japanese Society of Hypertension, 1996, Volume: 19, Issue:4

    Topics: Adenosine Diphosphate; Animals; Antioxidants; Calcium Channel Blockers; Cell Membrane; Dihydropyridines; Diltiazem; Felodipine; Fumarates; Heart; Iron; Lipid Peroxidation; Male; Myocardium; Nicardipine; Nifedipine; Nisoldipine; Nitrendipine; Oxidation-Reduction; Rats; Rats, Sprague-Dawley; Verapamil

1996
Effect of nilvadipine on high-voltage activated Ca2+ channels in rat CNS neurons.
    Neuroreport, 1997, Mar-03, Volume: 8, Issue:4

    Topics: Animals; Brain; Cadmium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; In Vitro Techniques; Kinetics; Membrane Potentials; Nerve Tissue Proteins; Neurons; Nicardipine; Nifedipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Rats; Rats, Wistar; Spider Venoms

1997
Nilvadipine inhibits acute rise of aqueous flare and intraocular pressure induced by prostaglandin E2 in pigmented rabbits.
    Ophthalmic research, 1998, Volume: 30, Issue:3

    Topics: Animals; Anterior Eye Segment; Aqueous Humor; Calcium Channel Blockers; Dinoprostone; Dose-Response Relationship, Drug; Eye Proteins; Injections, Intravenous; Intraocular Pressure; Male; Nicardipine; Nifedipine; Ophthalmic Solutions; Rabbits; Tonometry, Ocular

1998
Effect of benidipine on depolarizing stimulation-induced increase of intracellular calcium concentration in cultured mouse hippocampal neurons.
    Japanese journal of pharmacology, 1999, Volume: 81, Issue:4

    Topics: Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Dihydropyridines; Electric Stimulation; Hippocampus; Mice; Neurons; Nicardipine; Nifedipine

1999
Study of drug effects of calcium channel blockers on retinal degeneration of rd mouse.
    Biochemical and biophysical research communications, 2004, Jan-23, Volume: 313, Issue:4

    Topics: Animals; Calcium Channel Blockers; Caspases; Diltiazem; Electroretinography; Fibroblast Growth Factor 2; Gene Expression; Membrane Proteins; Mice; Mice, Mutant Strains; Microscopy, Electron; Nerve Tissue Proteins; Nicardipine; Nifedipine; Photoreceptor Cells, Vertebrate; Retinal Degeneration; Retinitis Pigmentosa; Synaptogyrins

2004