nicardipine and bupivacaine

nicardipine has been researched along with bupivacaine in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (33.33)18.2507
2000's5 (41.67)29.6817
2010's3 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bruno-Blanch, L; Gálvez, J; García-Domenech, R1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chang, G; Di, L; Huang, Y; Lin, Z; Liston, TE; Scott, DO; Troutman, MD; Umland, JP1
Artursson, P; Mateus, A; Matsson, P1
Kambam, JR; Kinney, WW; Matsuda, F; Wright, W1
Attolini, L; Bruguerolle, B; Gantenbein, M; Grignon, S; Jacob, D1
Strichartz, GR; Xiong, Z1
Kurata, Y; Matsuda, T1
Asada, A; Funao, T; Oda, Y; Tanaka, K1

Other Studies

12 other study(ies) available for nicardipine and bupivacaine

ArticleYear
Topological virtual screening: a way to find new anticonvulsant drugs from chemical diversity.
    Bioorganic & medicinal chemistry letters, 2003, Aug-18, Volume: 13, Issue:16

    Topics: Anticonvulsants; Computer Simulation; Databases, Factual; Discriminant Analysis; Drug Design; Molecular Structure; Quantitative Structure-Activity Relationship

2003
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Species independence in brain tissue binding using brain homogenates.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:7

    Topics: Animals; Brain; Dogs; Guinea Pigs; Humans; Macaca fascicularis; Mice; Rats; Species Specificity

2011
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
Nicardipine reduces the cardio-respiratory toxicity of intravenously administered bupivacaine in rats.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1990, Volume: 37, Issue:8

    Topics: Analysis of Variance; Anesthesia, Conduction; Animals; Apnea; Arrhythmias, Cardiac; Bupivacaine; Heart; Heart Rate; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intravenous; Male; Nicardipine; Pentobarbital; Rats; Rats, Inbred Strains; Respiration; Survival Rate

1990
Effects of calcium antagonists on binding of local anesthetics to plasma proteins and erythrocytes in mice.
    Pharmacology, 1996, Volume: 53, Issue:4

    Topics: Anesthetics, Local; Animals; Blood Proteins; Bupivacaine; Calcium Channel Blockers; Diltiazem; Erythrocytes; In Vitro Techniques; Lidocaine; Male; Mice; Nicardipine; Protein Binding; Verapamil

1996
Inhibition by local anesthetics of Ca2+ channels in rat anterior pituitary cells.
    European journal of pharmacology, 1998, Dec-11, Volume: 363, Issue:1

    Topics: Anesthetics, Local; Animals; Bupivacaine; Calcium Channel Blockers; Clone Cells; Dihydropyridines; Dose-Response Relationship, Drug; Lidocaine; Membrane Potentials; Nicardipine; Patch-Clamp Techniques; Pituitary Gland, Anterior; Rats

1998
Effects of nicardipine and bupivacaine on early after depolarization in rabbit sinoatrial node cells: a possible mechanism of bupivacaine-induced arrhythmias.
    General pharmacology, 1999, Volume: 33, Issue:2

    Topics: Action Potentials; Anesthetics, Local; Animals; Arrhythmia, Sinus; Bupivacaine; Calcium Channel Blockers; Models, Cardiovascular; Nicardipine; Rabbits; Sinoatrial Node

1999
Vasodilation increases the threshold for bupivacaine-induced convulsions in rats.
    Anesthesia and analgesia, 2004, Volume: 98, Issue:3

    Topics: Adrenergic alpha-Antagonists; Anesthetics, Local; Animals; Blood Gas Analysis; Blood Pressure; Brain; Bupivacaine; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Heart Rate; Male; Nicardipine; Phentolamine; Rats; Rats, Sprague-Dawley; Seizures; Vasodilation; Vasodilator Agents

2004