nicardipine has been researched along with bay-k-8644 in 67 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (23.88) | 18.7374 |
1990's | 38 (56.72) | 18.2507 |
2000's | 10 (14.93) | 29.6817 |
2010's | 3 (4.48) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H | 1 |
Baraldi, PG; Geppetti, P; Materazzi, S; Preti, D | 1 |
Hirano, Y; January, CT; Moscucci, A | 1 |
Advenier, C; Candenas, ML; Naline, E; Sarria, B | 1 |
Bergamaschi, S; Govoni, S; Grimaldi, M; Meucci, O; Schettini, G; Scorziello, A; Yasumoto, T | 1 |
Inagami, T; Ishido, M; Miyazaki, H; Murakami, K; Ohnishi, J; Shibata, T | 1 |
Alabadí, JA; Alborch, E; Miranda, FJ; Salom, JB; Torregrosa, G | 1 |
Serebryakov, V; Takeda, K | 1 |
Brisac, AM; Dubray, C; Huguet, F; Roche, A | 1 |
Advenier, C; Lagente, V; Naline, E; Puybasset, L; Sarria, B | 1 |
Calixto, JB; Rae, GA | 2 |
Florio, T; Grimaldi, M; Landolfi, E; Meucci, O; Schettini, G; Scorziello, A; Ventra, C | 1 |
Blondfield, DP; Ozaki, H; Publicover, NG; Sanders, KM; Stevens, RJ | 1 |
Clark, RB; Giles, WR; Gotoh, Y; Imaizumi, Y; Shibata, EF; Watanabe, M | 1 |
Alabadí, JA; Alborch, E; Alvarez, C; Miranda, FJ; Salom, JB; Torregrosa, G | 1 |
Baeyens, JM; Barrios, M | 1 |
Kurokawa, K; Naruse, M; Ogata, E; Uchida, S | 1 |
Baldy-Moulinier, M; Diochot, S; Nargeot, J; Richard, S; Valmier, J | 1 |
Matsuo, K; Uchida, S | 1 |
Advenier, C; Naline, E; Renier, A | 1 |
Collu, R; Lafond, J | 1 |
Matsuo, K; Uchida, MK | 1 |
Ohshika, H; Takemura, H | 1 |
Brisac, AM; Champeroux, P; Gerard, P; Huguet, F; Laurent, S; Lucet, B; Montastruc, JL; Narcisse, G; Schmitt, H | 1 |
Fukuda, Y; Hirata, Y; Kobayashi, Y; Kojima, T; Masaki, T; Yanagisawa, M; Yoshimi, H | 1 |
Akahane, K; Chiba, S; Furukawa, Y; Ogiwara, Y | 1 |
Duncan, GP; Patmore, L; Spedding, M | 1 |
D'Orleans-Juste, P; de Nucci, G; Finet, M; Vane, JR | 1 |
D'Orleans-Juste, P; De Nucci, G; Vane, JR | 1 |
Briand, V; Laurent, S; Schmitt, H | 1 |
Bloom, SR; Dollery, CT; Polak, JM; Power, RF; Turner, NC | 1 |
Goto, K; Ishikawa, T; Kasuya, Y; Kimura, S; Masaki, T; Yanagisawa, M | 1 |
Chang, CC; Chiou, LC; Hong, SJ; Huang, CY; Hwang, LL | 1 |
Groth, H; Locher, R; Neyses, L; Stimpel, M; Vetter, W | 1 |
Goldstein, M; Masuyama, Y; Nishio, I; Tsuda, K; Tsuda, S | 1 |
Akera, T; Jiang, J; Temma, K | 1 |
Brooker, G; Carlson, RO; Masco, D; Spiegel, S | 1 |
Hosoi, K; Kamioka, H; Kawata, T; Miki, Y; Sumitani, K; Tagami, K; Terai, K | 1 |
Fukata, F; Kanda, M; Kurahashi, K; Matsui, H; Nakamura, S; Shirahase, H; Wada, K | 1 |
Arimura, T; Kobayashi, K; Okada, T; Piccolino, M; Tachibana, M | 1 |
Nargeot, J; Neveu, D; Richard, S | 1 |
Brisac, AM; Dubar, M; Huguet, F; Ingrand, P; Piriou, A | 1 |
Awere, S; Moore, NA; Rees, G; Sanger, G | 1 |
Dupont, AG; Massart, DL; Schoors, DF; Vercruysse, I | 1 |
Brickley, K; Dolphin, AC; Galione, A; Hunt, SV; Sadighi Akha, AA; Willmott, NJ | 1 |
Albat, B; Nargeot, J; Quignard, JF; Richard, S; Ryckwaert, F | 1 |
Fujita, H; Kageyama, M; Nakata, K; Shirasawa, E | 1 |
Akishita, M; Eto, M; Hashimoto, M; Kim, S; Kozaki, K; Nagano, K; Ouchi, Y; Sudo, N; Toba, K; Watanabe, M; Yoo, HJ; Yoshizumi, M | 1 |
Cohen, C; Perrault, G; Sanger, DJ | 1 |
Ban, Y; Makita, T | 1 |
Akaike, N; Ishibashi, H; Rhee, JS | 1 |
Bertrand, PP; Clerc, N; Furness, JB; Kunze, WA | 1 |
Guo, J; Mitsuiye, T; Noma, A | 1 |
Cameron, JS; Coyne, MD; Gwathmey, JK; Kim, CS | 1 |
Ishikawa, T; Kimura, M; Nakayama, K; Obara, K; Sasase, T; Tanabe, Y | 1 |
Hattori, T; Maehashi, H | 1 |
Cathala, L; Chesnoy-Marchais, D | 1 |
Druet, P; Fournié, GJ; Gallard, A; Gomes, B; Guéry, JC; Leclerc, C; Mariamé, B; Moreau, M; Narbonnet, S; Paulet, P; Pelletier, L; Saoudi, A; Savignac, M | 1 |
Boddy, G; Daniel, EE | 1 |
Hontela, A; Lacroix, A | 1 |
Gordon, TP; Jackson, MW; Wan, EC | 1 |
Cho, WJ; Daniel, EE; Elyazbi, A; Eteraf, T; Sommer, B | 1 |
Asano, S; Bender, SB; Borbouse, L; Bratz, IN; Dick, GM; Dincer, UD; Neeb, ZP; Payne, GA; Sturek, M; Tune, JD | 1 |
Gordon, TP; Jackson, MW | 1 |
An Haack, K; Bennett, MJ; Li, H; Narayan, SB; Tan, L; Warnock, A | 1 |
Jacobson, KA; Jiang, JL; Melman, N; Olah, ME; Stiles, GL; van Rhee, AM | 1 |
1 review(s) available for nicardipine and bay-k-8644
Article | Year |
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Transient receptor potential ankyrin 1 (TRPA1) channel as emerging target for novel analgesics and anti-inflammatory agents.
Topics: Analgesics; Animals; Anti-Inflammatory Agents; Asthma; Humans; Ion Channel Gating; Neurons; Pain; Peripheral Nervous System Diseases; Pulmonary Disease, Chronic Obstructive; Transient Receptor Potential Channels | 2010 |
66 other study(ies) available for nicardipine and bay-k-8644
Article | Year |
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Small molecule regulators of autophagy identified by an image-based high-throughput screen.
Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers | 2007 |
Direct measurement of L-type Ca2+ window current in heart cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium; Calcium Channels; Dogs; Isoproterenol; Membrane Potentials; Models, Biological; Nicardipine; Nifedipine; Purkinje Fibers | 1992 |
Effect of epithelium removal and of enkephalin inhibition on the bronchoconstrictor response to three endothelins of the human isolated bronchus.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bronchi; Dose-Response Relationship, Drug; Endothelins; Epithelium; Glycopeptides; Humans; Muscle Contraction; Neprilysin; Nicardipine | 1992 |
Maitotoxin-induced intracellular calcium rise in PC12 cells: involvement of dihydropyridine-sensitive and omega-conotoxin-sensitive calcium channels and phosphoinositide breakdown.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cytosol; Dihydropyridines; Dose-Response Relationship, Drug; GTP-Binding Proteins; Marine Toxins; Nicardipine; omega-Conotoxins; Oxocins; PC12 Cells; Peptides, Cyclic; Pertussis Toxin; Phosphatidylinositols; Rats; Sodium; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1992 |
The rat angiotensin II AT1A receptor couples with three different signal transduction pathways.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Binding, Competitive; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Kinetics; Neomycin; Nicardipine; Rats; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Transfection; Type C Phospholipases | 1992 |
Comparison of the contractile effects of endothelin-1 and sarafotoxin S6b in goat isolated cerebral arteries.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cerebral Arteries; Dose-Response Relationship, Drug; Endothelins; Endothelium, Vascular; Female; Goats; Indomethacin; Nicardipine; Vasoconstriction; Vasoconstrictor Agents; Viper Venoms | 1992 |
Voltage-dependent calcium current and the effects of adrenergic modulation in rat aortic smooth muscle cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Barium; Cadmium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Cesium; Epinephrine; Male; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Nickel; Norepinephrine; Phenylephrine; Rats; Rats, Inbred WKY | 1992 |
Absence of a direct coupling of a G protein to dihydropyridine binding sites in rat heart.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Calcium Channels; Dihydropyridines; GTP-Binding Proteins; Heart; Male; Myocardium; Nicardipine; Nifedipine; Rats; Rats, Wistar | 1992 |
Contractile activity of three endothelins (ET-1, ET-2 and ET-3) on the human isolated bronchus.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amino Acid Sequence; Bronchi; Calcium Channel Blockers; Endothelins; Female; Humans; In Vitro Techniques; Indomethacin; Male; Middle Aged; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Nicardipine; Peptides | 1990 |
Effects of endothelins on nerve-mediated contractions of the mouse vas deferens.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Calcium Channels; Electric Stimulation; Endothelins; Male; Mice; Muscle Contraction; Nicardipine; Norepinephrine; Potassium Chloride; Sympathetic Nervous System; Vas Deferens | 1990 |
Dihydropyridine modulation of voltage-activated calcium channels in PC12 cells: effect of pertussis toxin pretreatment.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Gland Neoplasms; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Electrophysiology; Nicardipine; Pertussis Toxin; Pheochromocytoma; Potassium; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1991 |
Simultaneous measurement of membrane potential, cytosolic Ca2+, and tension in intact smooth muscles.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Cytosol; Dogs; Egtazic Acid; Electrophysiology; Female; In Vitro Techniques; Ionomycin; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Nicardipine; Stomach | 1991 |
Inhibition of transient outward K+ current by DHP Ca2+ antagonists and agonists in rabbit cardiac myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Dihydropyridines; Dose-Response Relationship, Drug; Electrophysiology; Heart; In Vitro Techniques; Myocardium; Nicardipine; Potassium; Rabbits | 1991 |
Effects of endothelins, Bay K 8644 and other oxytocics in non-pregnant and late pregnant rat isolated uterus.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dinoprost; Endothelins; Female; In Vitro Techniques; Nicardipine; Oxytocics; Pregnancy; Pregnancy, Animal; Rats; Rats, Inbred Strains; Serotonin; Uterine Contraction; Uterus | 1991 |
Effects of endothelin-1 on the cerebrovascular bed of the goat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Radioisotopes; Cerebrovascular Circulation; Endothelins; Female; Goats; In Vitro Techniques; Isometric Contraction; Muscle, Smooth, Vascular; Nicardipine; Potassium | 1991 |
Differential effects of L-type calcium channel blockers and stimulants on naloxone-precipitated withdrawal in mice acutely dependent on morphine.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Female; Mice; Morphine Dependence; Naloxone; Nicardipine; Postural Balance; Substance Withdrawal Syndrome; Verapamil | 1991 |
Endothelin 1 increases cell calcium in mouse collecting tubule cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine Vasopressin; Calcium; Dose-Response Relationship, Drug; Endothelins; In Vitro Techniques; Kidney Tubules, Collecting; Male; Mice; Nicardipine; Osmolar Concentration | 1991 |
Inhibition of T-type calcium currents by dihydropyridines in mouse embryonic dorsal root ganglion neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dihydropyridines; Electric Conductivity; Electric Stimulation; Electrophysiology; Ganglia, Spinal; Mice; Neurons; Nicardipine | 1991 |
[Synergism of the calcium reversal phenomenon of potassium depolarizing in the rat uterine muscle by Bay k-8644, a calcium agonist].
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dose-Response Relationship, Drug; Drug Synergism; Female; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nicardipine; Nifedipine; Oxytocin; Potassium; Rats; Uterus | 1985 |
Effects of Bay K 8644 on contraction of the human isolated bronchus and guinea-pig isolated trachea.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Bronchi; Calcium; Calcium Channel Blockers; Guinea Pigs; Histamine; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nicardipine; Nifedipine; Potassium Chloride; Trachea; Verapamil | 1986 |
Role of calcium and sodium ions in the inhibitory control of baseline and stimulated prolactin release.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Dopamine; Female; Nicardipine; Nifedipine; Phorbol Esters; Prolactin; Rats; Rats, Inbred Strains; Sodium; Thyrotropin-Releasing Hormone | 1986 |
Opposite effects of Bay k 8644 and nicardipine on the inhibitory effect of Ca2+ on rat myometrium.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Female; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myometrium; Nicardipine; Ovariectomy; Rats; Rats, Inbred Strains | 1987 |
Effects of Ca2+ agonist and antagonists on cytosolic free Ca2+ concentration: studies on Ca2+ channels in rat parotid cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Diltiazem; In Vitro Techniques; Ion Channels; Kinetics; Male; Methoxamine; Nicardipine; Parotid Gland; Potassium; Rats; Rats, Inbred Strains; Verapamil | 1987 |
Central interactions between dihydropyridines and cholinergic systems in the control of blood pressure in rat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Atropine Derivatives; Blood Pressure; Cerebral Ventricles; Dihydropyridines; Hemicholinium 3; Hexamethonium; Hexamethonium Compounds; Hippocampus; In Vitro Techniques; Male; Nicardipine; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Reference Values; Species Specificity | 1987 |
Endothelin is a potent secretagogue for atrial natriuretic peptide in cultured rat atrial myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Natriuretic Factor; Cells, Cultured; Drug Synergism; Endothelins; Heart Atria; Myocardium; Nicardipine; Peptides; Rats; Swine; Tetradecanoylphorbol Acetate | 1988 |
Different antagonism of the positive chronotropic and inotropic responses of the isolated, blood-perfused dog atrium to Bay k 8644 by nicardipine and verapamil.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Function; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Myocardial Contraction; Nicardipine; Propranolol; Verapamil | 1988 |
The effects of calcium antagonists on calcium overload contractures in embryonic chick myocytes induced by ouabain and veratrine.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Chick Embryo; Electrophysiology; Flunarizine; Myocardial Contraction; Myocardium; Nicardipine; Ouabain; Tetrodotoxin; Veratrine | 1989 |
Pharmacology of endothelin-1 in isolated vessels: effect of nicardipine, methylene blue, hemoglobin, and gossypol.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Calcium Channels; Endothelins; Gossypol; Hemoglobins; In Vitro Techniques; Indomethacin; Male; Methylene Blue; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Peptides; Rabbits; Rats; Rats, Inbred Strains; Veins | 1989 |
Endothelin-1 contracts isolated vessels independently of dihydropyridine-sensitive Ca2+ channel activation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channels; Captopril; Dihydropyridines; Dogs; Endothelins; In Vitro Techniques; Male; Methylene Blue; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Peptides; Rabbits | 1989 |
Interaction between isoproterenol and dihydropyridines in heart cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cells, Cultured; Chick Embryo; Dihydropyridines; Heart; Isoproterenol; Myocardial Contraction; Myocardium; Nicardipine; Nifedipine; Time Factors | 1989 |
Endothelin-induced contractions of tracheal smooth muscle and identification of specific endothelin binding sites in the trachea of the rat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Autoradiography; Calcium Channels; Endothelins; In Vitro Techniques; Male; Methacholine Compounds; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Nicardipine; Peptides; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Endothelin; Trachea | 1989 |
Mechanism of contraction to endothelin in isolated porcine coronary artery.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channels; Coronary Vessels; Dinoprost; Endothelins; Endothelium, Vascular; Histamine; In Vitro Techniques; Kinetics; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Peptides; Potassium Chloride; Receptors, Nicotinic; Swine; Vasoconstriction | 1989 |
Nicardipine inhibits axon conduction but causes dual changes of acetylcholine release in the mouse motor nerve.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Action Potentials; Animals; Axonal Transport; Axons; Chick Embryo; Diaphragm; Diltiazem; Female; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Motor Neurons; Muscle Contraction; Nicardipine; Nifedipine; Sodium Channels; Succinylcholine; Verapamil | 1989 |
Human red blood cells--an ideal model system for the action of calcium agonists and antagonists.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Erythrocytes; Humans; Ion Channels; Nicardipine; Nifedipine; Nitrendipine; Pyridines; Stimulation, Chemical; Verapamil | 1984 |
Effects of bradykinin on [3H]-norepinephrine release in rat hypothalamus.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bradykinin; Central Nervous System; Drug Interactions; Hypothalamus; Male; Nicardipine; Norepinephrine; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Synaptic Transmission; Tritium | 1993 |
Dual effects of nicardipine: evidence from intracellular Ca2+ transients and twitch contractions observed in single myocytes obtained from rat heart.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Cells, Cultured; Electric Stimulation; Female; Heart Ventricles; Male; Myocardial Contraction; Nicardipine; Rats | 1994 |
Endogenous ganglioside GM1 modulates L-type calcium channel activity in N18 neuroblastoma cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Line; Cholera Toxin; Dihydropyridines; Egtazic Acid; Fura-2; G(M1) Ganglioside; G(M3) Ganglioside; Manganese; Mice; Microscopy, Fluorescence; Neuroblastoma; Nicardipine; Nickel; Potassium; Tumor Cells, Cultured | 1994 |
Extracellular calcium causes the release of calcium from intracellular stores in chick osteocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Chick Embryo; Cytosol; Gallic Acid; Nicardipine; Nifedipine; Osteocytes | 1995 |
Effects of the novel water-soluble calcium antagonist (+/-)-3-(4-allyl-1-piperazinyl)-2,2-dimethylpropyl methyl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylate dihydrochloride on the responses of isolated canine arteries.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Dihydropyridines; Dogs; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nicardipine; Nifedipine; Norepinephrine; Potassium Chloride; Vasoconstrictor Agents; Vasodilator Agents | 1995 |
Dihydropyridine-sensitive calcium current mediates neurotransmitter release from bipolar cells of the goldfish retina.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Fura-2; Goldfish; In Vitro Techniques; Kinetics; Neurons; Nicardipine; Nifedipine; omega-Conotoxins; Peptides; Retina | 1993 |
Two high-voltage-activated, dihydropyridine-sensitive Ca2+ channel currents with distinct electrophysiological and pharmacological properties in cultured rat aortic myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Barium; Calcium Channels; Cell Membrane Permeability; Cells, Cultured; Dihydropyridines; Electric Conductivity; Electrophysiology; Male; Muscle, Smooth, Vascular; Nicardipine; Rats; Rats, Wistar | 1993 |
Endothelin modulates dihydropyridine receptor decreased binding in hippocampal slices from normotensive and spontaneously hypertensive rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Endothelins; Hippocampus; Hypertension; In Vitro Techniques; Isradipine; Male; Membranes; Muscle Proteins; Nicardipine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Wistar | 1993 |
Effect of L-type calcium channel modulators on stimulant-induced hyperactivity.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amphetamine; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Central Nervous System Stimulants; Cocaine; Drug Interactions; Male; Motor Activity; Nicardipine; Rats | 1993 |
Influences of the calcium antagonists nicardipine and nifedipine, and the calcium agonist BAY-K-8644, on the pharmacokinetics of propranolol in rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Administration, Oral; Animals; Biological Availability; Calcium Channel Agonists; Calcium Channel Blockers; Drug Interactions; Injections, Intravenous; Male; Nicardipine; Nifedipine; Propranolol; Rats; Rats, Wistar | 1993 |
Anti-Ig-induced calcium influx in rat B lymphocytes mediated by cGMP through a dihydropyridine-sensitive channel.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antibodies; B-Lymphocytes; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cell Membrane; Cell Separation; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Egtazic Acid; Elapid Venoms; Immunoglobulin D; Immunoglobulin M; Kinetics; Lymph Nodes; Nicardipine; Rats | 1996 |
A novel tetrodotoxin-sensitive Na+ current in cultured human coronary myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adult; Calcium Channel Agonists; Calcium Channel Blockers; Cnidarian Venoms; Coronary Vessels; Dose-Response Relationship, Drug; Humans; Ion Channel Gating; Lidocaine; Male; Middle Aged; Muscle, Smooth, Vascular; Neurotoxins; Nicardipine; Patch-Clamp Techniques; Sodium Channels; Tetrodotoxin; Veratridine | 1997 |
Involvement of both L- and N-type voltage-dependent Ca2+ channels in KCl- and veratridine-evoked transmitter release from non-adrenergic, non-cholinergic nerves in the rabbit iris sphincter muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesics; Animals; Atropine; Calcium Channel Blockers; Calcium Channels; Capsaicin; Iris; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nicardipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Peptides; Potassium Chloride; Rabbits; Receptors, Tachykinin; Sodium Channels; Spider Venoms; Substance P; Synaptic Transmission; Veratridine | 1997 |
Augmented Ca2+ influx is involved in the mechanism of enhanced proliferation of cultured vascular smooth muscle cells from spontaneously diabetic Goto-Kakizaki rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Aorta, Thoracic; Blood Glucose; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cell Count; Cell Division; Cells, Cultured; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Insulin; Male; Muscle, Smooth, Vascular; Nicardipine; Rats; Rats, Wistar; Vasoconstrictor Agents; Verapamil | 1997 |
Effects of dihydropyridine Ca2+ channel blockers on the discriminative stimulus and the motor impairing effects of (+/-)-Bay K 8644.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Discrimination, Psychological; Male; Mice; Motor Activity; Nicardipine; Nifedipine; Nimodipine | 1997 |
A calcium agonist, Bay k 8644, suppresses the embryotoxic effects induced by dihydropyridines calcium channel blockers in cultured rat embryos.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Culture Techniques; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Female; Male; Nicardipine; Nifedipine; Nitrendipine; Rats; Rats, Sprague-Dawley | 1998 |
Calcium channels in the GABAergic presynaptic nerve terminals projecting to meynert neurons of the rat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cholinergic Fibers; Electrophysiology; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Nicardipine; omega-Conotoxin GVIA; omega-Conotoxins; Organ Culture Techniques; Peptides; Presynaptic Terminals; Rats; Rats, Wistar; Ryanodine; Substantia Innominata; Tetrodotoxin; Thapsigargin | 1999 |
Contractile activity in intestinal muscle evokes action potential discharge in guinea-pig myenteric neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Axons; Calcium Channel Agonists; Denervation; Gadolinium; Gastrointestinal Motility; Guinea Pigs; Ileum; Immunohistochemistry; Muscle, Smooth; Myenteric Plexus; Neurons; Nicardipine; Paralysis; Physical Stimulation; Stereoisomerism | 1999 |
Nicardipine-sensitive Na+-mediated single channel currents in guinea-pig sinoatrial node pacemaker cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Guinea Pigs; In Vitro Techniques; Ion Channels; Kinetics; Membrane Potentials; Nicardipine; Patch-Clamp Techniques; Sinoatrial Node; Sodium | 1999 |
Effects of temperature and calcium availability on ventricular myocardium from rainbow trout.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Adrenergic beta-Agonists; Animals; Body Temperature; Cadmium; Caffeine; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Central Nervous System Stimulants; Cold Temperature; Heart Ventricles; Isometric Contraction; Isoproterenol; Myocardial Contraction; Myocardium; Nicardipine; Oncorhynchus mykiss; Oxygen Consumption; Patch-Clamp Techniques; Ryanodine; Sarcolemma; Ventricular Function | 2000 |
Specific inhibition of stretch-induced increase in L-type calcium channel currents by herbimycin A in canine basilar arterial myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Basilar Artery; Benzoquinones; Calcium Channel Agonists; Calcium Channels, L-Type; Cell Size; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Genistein; Hypotonic Solutions; Isoflavones; Isotonic Solutions; Lactams, Macrocyclic; Male; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Osmolar Concentration; Patch-Clamp Techniques; Phenols; Physical Stimulation; Protein-Tyrosine Kinases; Quinones; Rifabutin; Vanadates | 2000 |
Facilitation of calcium influx by propylene glycol through the voltage-dependent calcium channels in PC12 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium Chloride; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Electric Stimulation; Nicardipine; omega-Conotoxins; PC12 Cells; Propylene Glycol; Rats | 1999 |
Modulation of glycine responses by dihydropyridines and verapamil in rat spinal neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cells, Cultured; Chloride Channels; Dihydropyridines; Drug Interactions; Glycine; Neural Inhibition; Neurons; Nicardipine; Nifedipine; Nitrendipine; Rats; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Synaptic Transmission; Verapamil | 2001 |
Dihydropyridine receptors are selective markers of Th2 cells and can be targeted to prevent Th2-dependent immunopathological disorders.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Autoimmune Diseases; Biomarkers; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Differentiation; Chronic Disease; Encephalomyelitis, Autoimmune, Experimental; Graft vs Host Disease; Injections, Intraperitoneal; Interleukin-4; Male; Metals, Heavy; Mice; Mice, Inbred BALB C; Mice, Transgenic; Nicardipine; Rats; Rats, Inbred BN; Rats, Inbred Lew; Th1 Cells; Th2 Cells | 2004 |
Role of l-Ca(2+) channels in intestinal pacing in wild-type and W/W(V) mice.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Electric Stimulation; Ileum; Intestines; Jejunum; Linear Models; Male; Mice; Mice, Inbred BALB C; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Nicardipine; Proto-Oncogene Proteins c-kit | 2005 |
Role of calcium channels in cadmium-induced disruption of cortisol synthesis in rainbow trout (Oncorhynchus mykiss).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Adrenocorticotropic Hormone; Animals; Cadmium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Hydrocortisone; Nicardipine; Oncorhynchus mykiss; Pregnenolone; Water Pollutants, Chemical | 2006 |
Autoantibody-mediated bladder dysfunction in type 1 diabetes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Autoantibodies; Calcium Channels, L-Type; Diabetes Mellitus, Type 1; Male; Mice; Mice, Inbred BALB C; Nicardipine; Tetrodotoxin; Urinary Bladder; Urinary Bladder Diseases | 2007 |
The role of caveolae and caveolin 1 in calcium handling in pacing and contraction of mouse intestine.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium-Transporting ATPases; Caveolae; Caveolin 1; Chelating Agents; Egtazic Acid; Intestinal Mucosa; Intestines; Male; Mice; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Nicardipine; Sarcoplasmic Reticulum | 2009 |
Impaired function of coronary BK(Ca) channels in metabolic syndrome.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 2-Chloroadenosine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arterioles; Benzimidazoles; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Coronary Circulation; Coronary Vessels; Diet, Atherogenic; Disease Models, Animal; Dose-Response Relationship, Drug; Large-Conductance Calcium-Activated Potassium Channel alpha Subunits; Large-Conductance Calcium-Activated Potassium Channel beta Subunits; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Metabolic Syndrome; Microcirculation; Muscle, Smooth, Vascular; Mycotoxins; Nicardipine; Peptides; Phenotype; Potassium Channel Blockers; Swine; Swine, Miniature; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2009 |
A novel impedance-based cellular assay for the detection of anti-calcium channel autoantibodies in type 1 diabetes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Autoantibodies; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Adhesion; Cell Line; Diabetes Mellitus, Type 1; Electric Impedance; Humans; Immunoglobulin G; Nicardipine; Rats | 2010 |
Screening for calcium channel modulators in CLN3 siRNA knock down SH-SY5Y neuroblastoma cells reveals a significant decrease of intracellular calcium levels by selected L-type calcium channel blockers.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amlodipine; Blotting, Western; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line, Tumor; Child; Drug Evaluation, Preclinical; Flunarizine; Humans; Intracellular Space; Membrane Glycoproteins; Molecular Chaperones; Neuroblastoma; Neuronal Ceroid-Lipofuscinoses; Nicardipine; Nifedipine; Nimodipine; Potassium Chloride; RNA Interference; RNA, Small Interfering | 2011 |
Interaction of 1,4-dihydropyridine and pyridine derivatives with adenosine receptors: selectivity for A3 receptors.
Topics: Adenylyl Cyclase Inhibitors; Animals; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Cerebral Cortex; CHO Cells; Cricetinae; Dihydropyridines; Enzyme Inhibitors; Guinea Pigs; Humans; Isradipine; Molecular Structure; Purinergic P1 Receptor Antagonists; Pyridines; Rats; Receptors, Purinergic P1; Recombinant Proteins; Stereoisomerism; Structure-Activity Relationship | 1996 |