niacinamide and suramin

niacinamide has been researched along with suramin in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's5 (83.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berger, SL; Brent, M; Dang, W; Howitz, K; Jackson, B; Marmorstein, R; Sanders, BD; Schreiber, SL; Taylor, AM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Canonico, PL; Coppo, C; Galli, U; Genazzani, AA; Mesenzani, O; Sorba, G; Tron, GC1
He, W; Jung, M; Maurer, B; Rumpf, T; Scharfe, M; Schmitt, ML; Sippl, W; Stolfa, DA; Verdin, E1
He, B; Huang, W; Li, Y; Xie, T; You, L1
Ai, T; Chen, L; Cui, H; Kamal, Z; More, SS; Wilson, DJ; Xu, Y1

Other Studies

6 other study(ies) available for niacinamide and suramin

ArticleYear
Identification and characterization of novel sirtuin inhibitor scaffolds.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Drug Evaluation, Preclinical; Enzyme Inhibitors; Fibroblast Growth Factor 6; Fungal Proteins; Humans; Inhibitory Concentration 50; Kinetics; Sirtuins; Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2.
    European journal of medicinal chemistry, 2012, Volume: 55

    Topics: Cell Line, Tumor; Cell Proliferation; Drug Evaluation, Preclinical; Histone Deacetylase Inhibitors; Humans; Niacinamide; Sirtuin 1; Sirtuin 2; Sirtuin 3; Substrate Specificity

2012
Inhibitors of the NAD(+)-Dependent Protein Desuccinylase and Demalonylase Sirt5.
    ACS medicinal chemistry letters, 2012, Dec-13, Volume: 3, Issue:12

    Topics:

2012
A FRET-based assay for screening SIRT5 specific modulators.
    Bioorganic & medicinal chemistry letters, 2015, Apr-15, Volume: 25, Issue:8

    Topics: Amino Acid Sequence; Coumarins; Enzyme Assays; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Kinetics; Molecular Sequence Data; p-Dimethylaminoazobenzene; Peptides; Sirtuins; Substrate Specificity

2015
Discovery of potent and selective sirtuin 2 (SIRT2) inhibitors using a fragment-based approach.
    Journal of medicinal chemistry, 2014, Oct-23, Volume: 57, Issue:20

    Topics: Animals; Dogs; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; Enzyme Inhibitors; Humans; Ligands; Madin Darby Canine Kidney Cells; MCF-7 Cells; Molecular Structure; Niacinamide; Sirtuin 2; Structure-Activity Relationship; Sulfonic Acids; Suramin

2014