niacinamide and sirtinol

niacinamide has been researched along with sirtinol in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (30.77)29.6817
2010's18 (69.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Järvinen, T; Kyrylenko, S; Leppänen, J; Niskanen, P; Nyrönen, TH; Poso, A; Salminen, A; Tervo, AJ1
Goekjian, P; Jochum, A; Jung, M; Kunick, C; Marshall, B; Meier, R; Saunders, L; Sippl, W; Trapp, J; Verdin, E1
Hruby, H; Jung, M; Meier, R; Neugebauer, RC; Sippl, W; Uchiechowska, U; Valkov, V; Verdin, E1
Berger, SL; Brent, M; Dang, W; Howitz, K; Jackson, B; Marmorstein, R; Sanders, BD; Schreiber, SL; Taylor, AM1
Zheng, W1
He, W; Jung, M; Maurer, B; Rumpf, T; Scharfe, M; Schmitt, ML; Sippl, W; Stolfa, DA; Verdin, E1
He, B; Huang, W; Li, Y; Xie, T; You, L1
He, B; Huang, W; Li, Y; Liu, J; You, L; Zhu, H1
Chauhan, S; Kumar, A1
Forgione, M; Hailu, GS; Mai, A; Robaa, D; Rotili, D; Sippl, W1
Alcendor, RR; Imai, S; Kirshenbaum, LA; Sadoshima, J; Vatner, SF1
Ahmad, N; Jung-Hynes, B; Nihal, M; Zhong, W1
He, QY; Li, DD; Li, Y; Xu, R; Zhang, XM1
Fujioka, H; Fujita, N; Hayashi, S; Ishida, K; Kubo, S; Kuroda, R; Kurosaka, M; Matsumoto, T; Matsushita, T; Sasaki, K; Takayama, K; Tei, K1
Davidson, NE; Gu, Y; Li, H; Yao, Y; Zhou, Q1
Black, JC; Boss, O; Dyson, NJ; Elson, SL; Hart, AC; Hirsch, ML; Israelian, K; Ji, JY; Jiang, K; Kadyk, LC; Li, X; Mostoslavsky, R; Mulligan, P; Näär, AM; Najafi-Shoushtari, H; Puigserver, P; Purushotham, A; Ribich, S; Rodgers, JT; Shioda, T; Smith, JJ; Thakur, JK; Walker, AK; Watts, JL; Westphal, CH; Whetstine, JR; Yang, F1
Ancrenaz, V; Camins, A; Folch, J; Junyent, F; Pallàs, M; Pizarro, JG; Sureda, F; Verdaguer, E1
Kang, YG; Kim, EC; Kim, SJ; Lee, SI; Lee, YM; Park, KH1
Cheong, SA; Hyun, SH; Jeon, Y; Kwak, SS; Yoon, JD1
Ji, M; Li, Y; Lin, Q; Lin, R; Ren, F; Wang, W; Zhang, J1
Bai, L; Ji, M; Lin, R; Lu, Y; Qiao, H; Ren, F; Wang, W; Yang, L; Zhang, J1
Gao, SJ; He, M; Li, Q; Ye, F; Zhou, F1
Hu, J; Jing, H; Lin, H1
Chang, YZ; Chen, MY; Hu, ML; Song, TY; Yang, NC1
Ding, X; Hu, J; Ma, R; Xu, Y; Zhang, L1
Li, YJ; Wang, YH; Zheng, GX1

Reviews

4 review(s) available for niacinamide and sirtinol

ArticleYear
Sirtuins as emerging anti-parasitic targets.
    European journal of medicinal chemistry, 2013, Volume: 59

    Topics: Animals; Antiparasitic Agents; Drug Delivery Systems; Enzyme Activation; Enzyme Inhibitors; Humans; Molecular Structure; Parasites; Sirtuins

2013
How much successful are the medicinal chemists in modulation of SIRT1: A critical review.
    European journal of medicinal chemistry, 2016, Aug-25, Volume: 119

    Topics: Animals; Chemistry, Pharmaceutical; Drug Discovery; Enzyme Activation; Histone Deacetylase Inhibitors; Humans; Sirtuin 1

2016
Lysine Deacetylase Inhibitors in Parasites: Past, Present, and Future Perspectives.
    Journal of medicinal chemistry, 2017, 06-22, Volume: 60, Issue:12

    Topics: Animals; Antiparasitic Agents; Drug Repositioning; Helminth Proteins; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Leishmania; Plasmodium; Protozoan Proteins; Schistosoma; Toxoplasma; Trypanosoma

2017
Sirtuin inhibitors as anticancer agents.
    Future medicinal chemistry, 2014, Volume: 6, Issue:8

    Topics: Animals; Antineoplastic Agents; Benzamides; Enzyme Inhibitors; Humans; Naphthols; Neoplasms; Niacinamide; Protein Binding; Reactive Oxygen Species; Sirtuins

2014

Other Studies

22 other study(ies) available for niacinamide and sirtinol

ArticleYear
An in silico approach to discovering novel inhibitors of human sirtuin type 2.
    Journal of medicinal chemistry, 2004, Dec-02, Volume: 47, Issue:25

    Topics: Anthraquinones; Benzene Derivatives; Binding Sites; Crystallography, X-Ray; Databases, Factual; Models, Molecular; Molecular Structure; Phenols; Pyridines; Sirtuin 2; Sirtuins; Triazoles

2004
Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition.
    Journal of medicinal chemistry, 2006, Dec-14, Volume: 49, Issue:25

    Topics: Acetylation; Adenosine; Binding Sites; Cell Line, Tumor; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Models, Molecular; Molecular Mimicry; Protein Kinase Inhibitors; Sirtuins; Structure-Activity Relationship; Tubulin

2006
Structure-activity studies on splitomicin derivatives as sirtuin inhibitors and computational prediction of binding mode.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Acetylation; Antineoplastic Agents; Catalytic Domain; Cell Line, Tumor; Databases, Factual; Drug Screening Assays, Antitumor; Humans; Hydrogen Bonding; Models, Molecular; Naphthalenes; Protein Binding; Pyrones; Recombinant Proteins; Sirtuin 2; Sirtuins; Stereoisomerism; Structure-Activity Relationship; Thermodynamics; Tubulin

2008
Identification and characterization of novel sirtuin inhibitor scaffolds.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Drug Evaluation, Preclinical; Enzyme Inhibitors; Fibroblast Growth Factor 6; Fungal Proteins; Humans; Inhibitory Concentration 50; Kinetics; Sirtuins; Structure-Activity Relationship

2009
Inhibitors of the NAD(+)-Dependent Protein Desuccinylase and Demalonylase Sirt5.
    ACS medicinal chemistry letters, 2012, Dec-13, Volume: 3, Issue:12

    Topics:

2012
A FRET-based assay for screening SIRT5 specific modulators.
    Bioorganic & medicinal chemistry letters, 2015, Apr-15, Volume: 25, Issue:8

    Topics: Amino Acid Sequence; Coumarins; Enzyme Assays; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Kinetics; Molecular Sequence Data; p-Dimethylaminoazobenzene; Peptides; Sirtuins; Substrate Specificity

2015
A FRET-based assay for screening SIRT6 modulators.
    European journal of medicinal chemistry, 2015, Volume: 96

    Topics: Coumarins; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Humans; Molecular Structure; Sirtuins; Structure-Activity Relationship

2015
Silent information regulator 2alpha, a longevity factor and class III histone deacetylase, is an essential endogenous apoptosis inhibitor in cardiac myocytes.
    Circulation research, 2004, Nov-12, Volume: 95, Issue:10

    Topics: Acetylation; Alkaloids; Animals; Apoptosis; Atrial Natriuretic Factor; Benzamides; Benzophenanthridines; Cell Nucleus; Cell Size; Cell Survival; Cells, Cultured; Culture Media, Serum-Free; Cysteine Proteinase Inhibitors; Dogs; Gene Silencing; Genes, Dominant; Genes, p53; Heart Failure; Heart Ventricles; Hydroxamic Acids; Hypertrophy; Hypertrophy, Left Ventricular; Longevity; Mice; Myocytes, Cardiac; Naphthols; Niacinamide; Phenanthridines; Protein Processing, Post-Translational; Rats; Rats, Wistar; Recombinant Fusion Proteins; Sirtuin 1; Sirtuins; Transcription, Genetic; Tumor Suppressor Protein p53

2004
Role of sirtuin histone deacetylase SIRT1 in prostate cancer. A target for prostate cancer management via its inhibition?
    The Journal of biological chemistry, 2009, Feb-06, Volume: 284, Issue:6

    Topics: Adult; Aged; Benzamides; Cell Line, Tumor; Forkhead Box Protein O1; Forkhead Transcription Factors; Gene Expression Regulation, Developmental; Gene Expression Regulation, Neoplastic; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Male; Middle Aged; Naphthols; Neoplasm Proteins; Niacinamide; Prostatic Neoplasms; Sirtuin 1; Sirtuins; Vitamin B Complex

2009
[Mechanism of apoptosis induced by SIRT1 deacetylase inhibitors in human breast cancer MCF-7 drug-resistant cells].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2008, Volume: 43, Issue:10

    Topics: Apoptosis; Benzamides; Breast Neoplasms; Caspases; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Female; Humans; Naphthols; Niacinamide; Sirtuin 1

2008
SIRT1 regulation of apoptosis of human chondrocytes.
    Arthritis and rheumatism, 2009, Volume: 60, Issue:9

    Topics: Adult; Apoptosis; bcl-2-Associated X Protein; Benzamides; Case-Control Studies; Caspase 3; Caspase 9; Cells, Cultured; Chondrocytes; Enzyme Inhibitors; Humans; Male; Naphthols; Niacinamide; Nitric Oxide; Osteoarthritis, Knee; Poly(ADP-ribose) Polymerases; Proto-Oncogene Proteins c-bcl-2; Resveratrol; RNA, Small Interfering; Sirtuin 1; Sirtuins; Stilbenes

2009
Inhibition of SIRT1 deacetylase suppresses estrogen receptor signaling.
    Carcinogenesis, 2010, Volume: 31, Issue:3

    Topics: Animals; Benzamides; Breast Neoplasms; Cell Line, Tumor; Cells, Cultured; Estradiol; Estrogen Receptor alpha; Female; Fibroblasts; Humans; Mammary Glands, Animal; Mice; Mice, Knockout; Naphthols; Neoplasm Proteins; Niacinamide; Promoter Regions, Genetic; Recombinant Fusion Proteins; RNA, Messenger; RNA, Neoplasm; RNA, Small Interfering; Signal Transduction; Sirtuin 1; Specific Pathogen-Free Organisms; Transcription, Genetic

2010
Conserved role of SIRT1 orthologs in fasting-dependent inhibition of the lipid/cholesterol regulator SREBP.
    Genes & development, 2010, Jul-01, Volume: 24, Issue:13

    Topics: Acetylation; Animals; Benzamides; Caenorhabditis elegans; Cell Line; Cholesterol; Down-Regulation; Fasting; HeLa Cells; Heterocyclic Compounds, 4 or More Rings; Humans; Lipids; Mice; Naphthols; Niacinamide; Protein Stability; Sirtuin 1; Sirtuins; Sterol Regulatory Element Binding Protein 1; Sterol Regulatory Element Binding Protein 2

2010
Resveratrol inhibits proliferation and promotes apoptosis of neuroblastoma cells: role of sirtuin 1.
    Neurochemical research, 2011, Volume: 36, Issue:2

    Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Benzamides; Cell Cycle; Cell Line, Tumor; Cell Proliferation; DNA Fragmentation; Humans; Naphthols; Neuroblastoma; NF-kappa B; Niacinamide; Proto-Oncogene Proteins c-akt; Resveratrol; Sirtuin 1; Stilbenes; Tumor Suppressor Protein p53; Vitamin B Complex

2011
Mechanical stress-activated immune response genes via Sirtuin 1 expression in human periodontal ligament cells.
    Clinical and experimental immunology, 2012, Volume: 168, Issue:1

    Topics: Acetylcysteine; Benzamides; Cell Line; Chemokines; Cytokines; Defensins; Extracellular Signal-Regulated MAP Kinases; Glutathione; Humans; JNK Mitogen-Activated Protein Kinases; Naphthols; NF-kappa B; Niacinamide; p38 Mitogen-Activated Protein Kinases; Periodontal Ligament; Protein Kinase C; Proto-Oncogene Proteins c-akt; Reactive Oxygen Species; Resveratrol; RNA Interference; Signal Transduction; Sirtuin 1; Stilbenes; Stress, Mechanical; Toll-Like Receptors

2012
Expression patterns of sirtuin genes in porcine preimplantation embryos and effects of sirtuin inhibitors on in vitro embryonic development after parthenogenetic activation and in vitro fertilization.
    Theriogenology, 2012, Oct-15, Volume: 78, Issue:7

    Topics: Animals; Benzamides; Blastocyst; Embryo Culture Techniques; Embryonic Development; Fertilization in Vitro; Gene Expression Profiling; Naphthols; Niacinamide; Nuclear Transfer Techniques; Parthenogenesis; RNA, Messenger; Sirtuins; Swine

2012
PPARα agonist fenofibrate attenuates TNF-α-induced CD40 expression in 3T3-L1 adipocytes via the SIRT1-dependent signaling pathway.
    Experimental cell research, 2013, Jun-10, Volume: 319, Issue:10

    Topics: 3T3-L1 Cells; Adipocytes; AMP-Activated Protein Kinases; Animals; Benzamides; Blotting, Western; CD40 Antigens; Fenofibrate; Mice; Naphthols; NF-kappa B; Niacinamide; Oxazoles; PPAR alpha; Pyrrolidines; RNA, Messenger; Signal Transduction; Sirtuin 1; Thiocarbamates; Tumor Necrosis Factor-alpha; Tyrosine

2013
The protective effect of fenofibrate against TNF-α-induced CD40 expression through SIRT1-mediated deacetylation of NF-κB in endothelial cells.
    Inflammation, 2014, Volume: 37, Issue:1

    Topics: Acetylation; Antioxidants; Benzamides; CD40 Antigens; Cells, Cultured; Fenofibrate; Human Umbilical Vein Endothelial Cells; Humans; Hypolipidemic Agents; Inflammation; Naphthols; Niacinamide; Oxazoles; PPAR alpha; Pyrrolidines; RNA Interference; RNA, Small Interfering; Signal Transduction; Sirtuin 1; Thiocarbamates; Transcription Factor RelA; Tumor Necrosis Factor-alpha; Tyrosine; Up-Regulation

2014
Activation of Kaposi's sarcoma-associated herpesvirus (KSHV) by inhibitors of class III histone deacetylases: identification of sirtuin 1 as a regulator of the KSHV life cycle.
    Journal of virology, 2014, Volume: 88, Issue:11

    Topics: Benzamides; Blotting, Western; Cell Line, Tumor; Chromatin Immunoprecipitation; DNA Primers; Gene Expression Regulation, Viral; Gene Knockdown Techniques; Herpesvirus 8, Human; Humans; Immediate-Early Proteins; Immunoprecipitation; Luciferases; Microscopy, Confocal; Naphthols; Niacinamide; Reverse Transcriptase Polymerase Chain Reaction; RNA, Small Interfering; Sirtuin 1; Trans-Activators; Virus Activation; Virus Latency

2014
Up-regulation of nicotinamide phosphoribosyltransferase and increase of NAD+ levels by glucose restriction extend replicative lifespan of human fibroblast Hs68 cells.
    Biogerontology, 2015, Volume: 16, Issue:1

    Topics: Acrylamides; Benzamides; Cell Line; Cell Proliferation; Cell Survival; Cells, Cultured; Cellular Senescence; Cytokines; Dose-Response Relationship, Drug; Fibroblasts; Glucose; Humans; NAD; Naphthols; Niacinamide; Nicotinamide Phosphoribosyltransferase; Piperidines; Sirtuin 1; Up-Regulation

2015
Sirtuin Inhibition Adversely Affects Porcine Oocyte Meiosis.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Actins; Animals; Benzamides; Cell Polarity; Chromosomes, Mammalian; Cumulus Cells; Female; Histone Deacetylase Inhibitors; Meiosis; Naphthols; Niacinamide; Oocytes; Ovary; Polar Bodies; Primary Cell Culture; Sirtuins; Spindle Apparatus; Swine

2015
Giardia duodenalis GlSir2.2, homolog of SIRT1, is a nuclear-located and NAD(+)-dependent deacethylase.
    Experimental parasitology, 2016, Volume: 169

    Topics: Amino Acid Sequence; Benzamides; Cell Nucleus; Fluorescent Antibody Technique, Indirect; Giardia lamblia; Group III Histone Deacetylases; Humans; Inhibitory Concentration 50; Naphthalenes; Naphthols; Niacinamide; Phylogeny; Pyrones; Sequence Alignment; Sirtuins

2016