niacinamide and pyrazole

niacinamide has been researched along with pyrazole in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kasuya, Y; Kawanishi, T; Ohno, Y; Omori, Y; Takahashi, A; Takanaka, A1
Decker, RW; Malejka-Giganti, D; Ritter, CL1
Getlik, M; Grütter, C; Pawar, V; Rabiller, M; Rauh, D; Simard, JR; Wulfert, S1
Hah, JM; Kim, H; Kim, M; Kim, MH; Sim, T; Yoo, KH; Yu, H1

Other Studies

4 other study(ies) available for niacinamide and pyrazole

ArticleYear
Nature of N-nitrosodimethylamine demethylase in hepatic microsomes of rats.
    Archives of toxicology, 1984, Volume: 56, Issue:1

    Topics: Aminoacetonitrile; Aminopyrine N-Demethylase; Aniline Compounds; Animals; Benzoflavones; Cytochrome P-450 CYP2E1; Cytochrome P-450 Enzyme System; Imidazoles; In Vitro Techniques; Kinetics; Male; Methylcholanthrene; Metyrapone; Microsomes, Liver; Monoamine Oxidase; Niacinamide; Oxidoreductases, N-Demethylating; Phenobarbital; Proadifen; Pyrazoles; Rats; Rats, Inbred Strains; Tranylcypromine

1984
Reductions of nitro and 9-Oxo groups of environmental nitrofluorenes by the rat mammary gland in vitro.
    Chemical research in toxicology, 2000, Volume: 13, Issue:8

    Topics: Air Pollutants; Allopurinol; Animals; Breast; Cytosol; Dicumarol; Female; Fluorenes; Hypoxanthine; Indomethacin; Microsomes; Niacinamide; Oxidation-Reduction; Oxygen; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Rutin; Vitamin K; Xanthine

2000
Development of a fluorescent-tagged kinase assay system for the detection and characterization of allosteric kinase inhibitors.
    Journal of the American Chemical Society, 2009, Sep-23, Volume: 131, Issue:37

    Topics: Adenosine Triphosphate; Allosteric Regulation; Amino Acid Sequence; Benzenesulfonates; Binding, Competitive; Catalytic Domain; Crystallography, X-Ray; Drug Evaluation, Preclinical; Enzyme Activation; Enzyme Stability; Fluorescent Dyes; Humans; Kinetics; Models, Molecular; Molecular Sequence Data; Niacinamide; p38 Mitogen-Activated Protein Kinases; Phenylurea Compounds; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Reproducibility of Results; Small Molecule Libraries; Sorafenib; Structure-Activity Relationship

2009
Structure based design and syntheses of amino-1H-pyrazole amide derivatives as selective Raf kinase inhibitors in melanoma cells.
    Bioorganic & medicinal chemistry, 2011, Mar-15, Volume: 19, Issue:6

    Topics: Amides; Antineoplastic Agents; Benzenesulfonates; Binding Sites; Cell Line, Tumor; Computer Simulation; Humans; Melanoma; Niacinamide; Phenylurea Compounds; Protein Kinase Inhibitors; Pyrazoles; Pyridines; raf Kinases; Sorafenib; Structure-Activity Relationship

2011