niacinamide and indomethacin

niacinamide has been researched along with indomethacin in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199010 (34.48)18.7374
1990's2 (6.90)18.2507
2000's4 (13.79)29.6817
2010's10 (34.48)24.3611
2020's3 (10.34)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Dittgen, M; Kala, H; Zessin, G1
Bolton, TB; Clapp, LH1
Behrman, HR; Preston, SL1
Bendtzen, K; Borg, LA; Eizirik, DL; Sandler, S; Strandell, E; Welsh, N1
Gross, GJ; Pieper, GM1
Glaise, D; Guillouzo, A; Ratanasavanh, D; Vandenberghe, Y1
Nakamura, Y; Sakai, K; Sugimoto, T; Yamazaki, T1
Ban, M; Enomoto, I; Hashimoto, H; Ito, T; Ogawa, K; Sakai, K1
Aniya, Y; Higuchi, M; Miyamoto, Y; Sakanashi, M; Takeo, S1
Burke, V; Gracey, M1
Monteiro-Riviere, NA; Riviere, JE; Zhang, Z1
Caputi, AP; Costantino, G; Cuzzocrea, S; Mazzon, E; RombolĂ , L; Sautebin, L1
Decker, RW; Malejka-Giganti, D; Ritter, CL1
Kamata, K; Kobayashi, T; Matsumoto, T; Wakabayashi, K1
Buczko, W; Kramkowski, K; Mogielnicki, A; Pietrzak, L1
Chuang, LM; Guo, RT; Hu, SM; Ko, TP; Wang, AH; Wu, YH1
Abdallah, DM1
Grobelski, B; Kazmierczak, P; Przygodzki, T; Watala, C1
Hirakura, Y; Terada, K; Teramura, T; Yamashita, H; Yuda, M1
Alhalaweh, A; Antzutkin, ON; Brown, SP; Iuga, D; Maruyoshi, K; Velaga, SP1
Huang, YT; Lin, HL; Lin, SY; Zhang, GC1
Box, KJ; Comer, J; Fotaki, N; Karki, S; Price, R; Ruiz, R; Taylor, R1
Biggart, GD; Clarke, GS; Ewing, AV; Hale, CR; Kazarian, SG1
Adibkia, K; Barzegar-Jalali, M; Emami, S; Siahi-Shadbad, M1
Chavan, T; Kunda, NK; Tawfeek, HM1
Cai, Y; Deng, X; Jing, P; Li, Y; Xu, G; Xu, L; Zhou, Q1
Gao, Y; Heng, W; Hu, E; Qian, S; Shen, P; Wei, Y; Zhang, C; Zhang, J1

Other Studies

29 other study(ies) available for niacinamide and indomethacin

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
[Drug liberation from imbedded forms with a polyacrylate base].
    Die Pharmazie, 1977, Volume: 32, Issue:12

    Topics: Acrylates; Chemistry, Pharmaceutical; Citrates; Creatinine; Delayed-Action Preparations; Diffusion; Indomethacin; Medazepam; Niacinamide; Phenacetin; Phenobarbital

1977
Endothelial-dependent relaxant actions of carbachol and substance P in arterial smooth muscle.
    British journal of pharmacology, 1986, Volume: 87, Issue:4

    Topics: Animals; Calcimycin; Carbachol; Endothelium; Female; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Membrane Potentials; Mesenteric Arteries; Monoamine Oxidase Inhibitors; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Potassium; Rabbits; Substance P

1986
Luteolytic actions of peroxide in rat ovarian cells.
    Endocrinology, 1989, Volume: 124, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Benzamides; Corpus Luteum; Cyclic AMP; Dinoprost; DNA Repair; Female; Hydrogen Peroxide; In Vitro Techniques; Indomethacin; Kinetics; Luteinizing Hormone; Niacinamide; Ovary; Progesterone; Rats; Sexual Maturation

1989
Studies on the mechanisms causing inhibition of insulin secretion in rat pancreatic islets exposed to human interleukin-1 beta indicate a perturbation in the mitochondrial function.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Acetophenones; Animals; Culture Techniques; Cyclosporins; Cytoplasmic Granules; DNA; Glucose; Indomethacin; Insulin; Insulin Secretion; Interleukin-1; Islets of Langerhans; Male; Masoprocol; Methylurea Compounds; Microscopy, Electron; Mitochondria; Niacinamide; Phenanthrolines; Rats; Rats, Inbred Strains; Recombinant Proteins

1989
Effect of cyclooxygenase blockade on the beneficial actions of nicorandil in the stunned myocardium of dogs.
    Pharmacology, 1989, Volume: 38, Issue:6

    Topics: Animals; Blood Pressure; Cardiomyopathies; Coronary Circulation; Cyclooxygenase Inhibitors; Dinoprostone; Dogs; Female; Heart Rate; Hemodynamics; In Vitro Techniques; Indomethacin; Male; Myocardial Reperfusion Injury; Niacinamide; Nicorandil; Prostaglandins; Thromboxane A2; Time Factors; Vasodilator Agents

1989
Influence of medium composition and culture conditions on glutathione S-transferase activity in adult rat hepatocytes during culture.
    In vitro cellular & developmental biology : journal of the Tissue Culture Association, 1988, Volume: 24, Issue:4

    Topics: Animals; Cell Survival; Cells, Cultured; Culture Media; Cysteine; Cytochrome P-450 Enzyme System; Dimethyl Sulfoxide; Glutathione Transferase; Indomethacin; Liver; Niacinamide; Rats; Selenium

1988
Protective effects of the antianginal agent nicorandil on arachidonate-induced sudden death in rats: comparison with several antianginal agents and cyclooxygenase inhibitors.
    Japanese journal of pharmacology, 1985, Volume: 37, Issue:1

    Topics: Angina Pectoris; Animals; Arachidonic Acid; Arachidonic Acids; Aspirin; Cyclooxygenase Inhibitors; Death, Sudden; Diltiazem; Indomethacin; Male; Mice; Niacinamide; Nicorandil; Nitroglycerin; Rats; Rats, Inbred Strains; Vasodilator Agents

1985
SG-75 induction of increased coronary outflow and PGE1 from ischemic areas in dogs with experimental myocardial infarction.
    Japanese heart journal, 1982, Volume: 23, Issue:4

    Topics: Alprostadil; Animals; Coronary Circulation; Dinoprostone; Dogs; Indomethacin; Lactates; Myocardial Infarction; Myocardium; Niacinamide; Nicorandil; Prostaglandins E; Vasodilator Agents

1982
Effects of 2-nicotinamidoethyl nitrate (SG-75, nicorandil) on indomethacin-induced contractions of isolated dog coronary arteries.
    Japanese heart journal, 1983, Volume: 24, Issue:2

    Topics: Animals; Coronary Vessels; Depression, Chemical; Dogs; Epoprostenol; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Tranylcypromine

1983
Studies with enterotoxigenic microorganisms: effects of candidate antidiarrhoeals in experimental animals in vivo.
    Journal of pediatric gastroenterology and nutrition, 1984, Volume: 3, Issue:4

    Topics: Aluminum Hydroxide; Animals; Antidiarrheals; Aspirin; Bacterial Infections; Charcoal; Chlorpromazine; Cholestyramine Resin; Diarrhea; Drug Combinations; Enterotoxins; Indomethacin; Loperamide; Male; Niacinamide; Rats; Rats, Inbred Strains; Water-Electrolyte Balance

1984
Evaluation of protective effects of sodium thiosulfate, cysteine, niacinamide and indomethacin on sulfur mustard-treated isolated perfused porcine skin.
    Chemico-biological interactions, 1995, Jun-14, Volume: 96, Issue:3

    Topics: Animals; Cysteine; Dinoprostone; Female; Indomethacin; Mustard Gas; Niacinamide; Skin; Skin Diseases; Swine; Thiosulfates

1995
Regulation of prostaglandin production by inhibition of poly (ADP-ribose) synthase in carrageenan-induced pleurisy.
    Life sciences, 1999, Volume: 65, Issue:12

    Topics: Animals; Anti-Inflammatory Agents; Benzamides; Carrageenan; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indomethacin; Niacinamide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Pleurisy; Poly(ADP-ribose) Polymerase Inhibitors; Prostaglandins; Rats

1999
Reductions of nitro and 9-Oxo groups of environmental nitrofluorenes by the rat mammary gland in vitro.
    Chemical research in toxicology, 2000, Volume: 13, Issue:8

    Topics: Air Pollutants; Allopurinol; Animals; Breast; Cytosol; Dicumarol; Female; Fluorenes; Hypoxanthine; Indomethacin; Microsomes; Niacinamide; Oxidation-Reduction; Oxygen; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Rutin; Vitamin K; Xanthine

2000
Alterations in vascular endothelial function in the aorta and mesenteric artery in type II diabetic rats.
    Canadian journal of physiology and pharmacology, 2004, Volume: 82, Issue:3

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Biological Factors; Chlorides; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Hyperglycemia; Indomethacin; Insulin; Isotonic Solutions; Male; Mesenteric Artery, Superior; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nitric Oxide; Nitroarginine; Nitroprusside; Norepinephrine; Phenylephrine; Potassium; Rats; Rats, Wistar; Sodium

2004
N-methylnicotinamide inhibits arterial thrombosis in hypertensive rats.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2007, Volume: 58, Issue:3

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Blood Flow Velocity; Blood Pressure; Carotid Arteries; Collagen; Dose-Response Relationship, Drug; Epoprostenol; Fibrinolysis; Heart Rate; Hypertension, Renal; Indomethacin; Injections, Intravenous; Male; NG-Nitroarginine Methyl Ester; Niacinamide; Nitric Oxide Synthase; Platelet Aggregation; Platelet Aggregation Inhibitors; Rats; Rats, Wistar; Thrombosis

2007
Structural basis for catalytic and inhibitory mechanisms of human prostaglandin reductase PTGR2.
    Structure (London, England : 1993), 2008, Nov-12, Volume: 16, Issue:11

    Topics: 15-Oxoprostaglandin 13-Reductase; Alcohol Dehydrogenase; Amino Acid Sequence; Animals; Catalysis; Dinoprostone; Guinea Pigs; Humans; Indomethacin; Kinetics; Mice; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Niacinamide; Protein Binding; Sequence Alignment; Sequence Homology, Amino Acid

2008
Nicotinamide alleviates indomethacin-induced gastric ulcers: a novel antiulcer agent.
    European journal of pharmacology, 2010, Feb-10, Volume: 627, Issue:1-3

    Topics: Animals; Anti-Ulcer Agents; Antioxidants; Capillary Permeability; Gastric Mucosa; Indomethacin; Male; Niacinamide; Rats; Rats, Wistar; Stomach Ulcer; Sucralfate

2010
N-Methyl-2-pyridone-5-carboxamide is 1-methylnicotinamide metabolite of low cyclooxygenase-dependent vasodilating activity.
    Journal of physiology and biochemistry, 2012, Volume: 68, Issue:3

    Topics: Animals; Bradykinin; Human Umbilical Vein Endothelial Cells; Humans; Indomethacin; Male; Niacinamide; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Sprague-Dawley; Transfection; Vasodilation

2012
Detection of cocrystal formation based on binary phase diagrams using thermal analysis.
    Pharmaceutical research, 2013, Volume: 30, Issue:1

    Topics: Caffeine; Calorimetry, Differential Scanning; Camphor; Carbamazepine; Crystallization; Heating; Indomethacin; Niacinamide; Pharmaceutical Preparations; Phase Transition; Piroxicam; Powder Diffraction; Salicylic Acid; Theophylline; X-Ray Diffraction

2013
Identifying the intermolecular hydrogen-bonding supramolecular synthons in an indomethacin-nicotinamide cocrystal by solid-state NMR.
    Chemical communications (Cambridge, England), 2012, Nov-14, Volume: 48, Issue:88

    Topics: Crystallization; Hydrogen Bonding; Indomethacin; Magnetic Resonance Spectroscopy; Niacinamide

2012
An investigation of indomethacin-nicotinamide cocrystal formation induced by thermal stress in the solid or liquid state.
    Journal of pharmaceutical sciences, 2014, Volume: 103, Issue:8

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Calorimetry, Differential Scanning; Crystallization; Indomethacin; Niacinamide; Spectroscopy, Fourier Transform Infrared; Temperature; Vitamin B Complex

2014
Small-Scale Assays for Studying Dissolution of Pharmaceutical Cocrystals for Oral Administration.
    AAPS PharmSciTech, 2016, Volume: 17, Issue:2

    Topics: Administration, Oral; Biological Assay; Carbamazepine; Chemical Precipitation; Crystallization; Indomethacin; Niacinamide; Pharmaceutical Preparations; Saccharin; Solubility; Tablets

2016
Comparison of pharmaceutical formulations: ATR-FTIR spectroscopic imaging to study drug-carrier interactions.
    International journal of pharmaceutics, 2015, Nov-10, Volume: 495, Issue:1

    Topics: Chemistry, Pharmaceutical; Drug Carriers; Drug Liberation; Indomethacin; Mannitol; Niacinamide; Spectroscopy, Fourier Transform Infrared; Urea

2015
Feasibility of electrospray deposition for rapid screening of the cocrystal formation and single step, continuous production of pharmaceutical nanococrystals.
    Drug development and industrial pharmacy, 2018, Volume: 44, Issue:6

    Topics: Crystallization; Indomethacin; Niacinamide; Saccharin; Solvents; X-Ray Diffraction

2018
Effect of Spray Drying on Amorphization of Indomethacin Nicotinamide Cocrystals; Optimization, Characterization, and Stability Study.
    AAPS PharmSciTech, 2020, Jun-30, Volume: 21, Issue:5

    Topics: Calorimetry, Differential Scanning; Desiccation; Drug Compounding; Drug Stability; Indomethacin; Molecular Structure; Niacinamide; Powders; Solubility; X-Ray Diffraction

2020
Terahertz spectroscopic characterizations and DFT calculations of indomethacin cocrystals with nicotinamide and saccharin.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2021, Mar-15, Volume: 249

    Topics: Density Functional Theory; Indomethacin; Niacinamide; Saccharin; Solubility; Terahertz Spectroscopy

2021
Switch between Cocrystal and Coamorphous Forms Depending on Thermal Modulation of Hot-Melt Extrusion.
    Molecular pharmaceutics, 2023, 07-03, Volume: 20, Issue:7

    Topics: Drug Compounding; Hot Temperature; Indomethacin; Niacinamide; Solubility; Solvents

2023