niacinamide and ex 527

niacinamide has been researched along with ex 527 in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (7.14)29.6817
2010's12 (85.71)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
He, W; Jung, M; Maurer, B; Rumpf, T; Scharfe, M; Schmitt, ML; Sippl, W; Stolfa, DA; Verdin, E1
Ai, T; Chen, L; Cui, H; Kamal, Z; More, SS; Wilson, DJ; Xu, Y1
Chen, X; Go, ML; Jin, HX; Sethi, G; Yang, T1
Bai, JJ; Cao, J; Farooqi, AS; Hong, JY; Kosciuk, T; Lin, H; Lu, X; Price, IR; Yang, M; Zhao, Q1
Amouzegh, P; Barker, J; Curtis, R; DiStefano, PS; Flegg, A; Hamelin, E; Hixon, J; Jones, S; Kates, M; Keavey, K; McDonagh, T; Napper, AD; Navia, MA; Pons, JF; Saunders, JO; Thomas, RJ; Yau, WT1
Caton, PW; Corder, R; Khan, NQ; Nayuni, NK; Wood, EG1
Andersson, G; Anderstam, B; He, J; He, X; Li, Y; Lindgren, U1
Camacho-Pereira, J; Chini, CC; Chini, EN; Escande, C; Giri, S; Lou, Z; Matalonga, J; Nin, V1
Avner, ED; Denu, JM; Fan, LX; Li, X; Sweeney, WE; Zhou, X1
Jarho, E; Kokkola, T; Kokkonen, P; Lahtela-Kakkonen, M; Mellini, P; Rahnasto-Rilla, M1
Haldar, M; Mallik, S; Srivastava, DK; Yu, J1
Bartolomé, A; Benito, M; García-Aguilar, A; Guillén, C; Nellist, M1
Guarente, L; Igarashi, M; Jaksch, F; Kadowaki, T; Miura, M; Williams, E; Yamauchi, T1
Alves, EGL; Araújo, FR; Bertassoli, BM; Camara, BOS; Jorge, EC; Malm, C; Ocarino, NM; Reis, AMS; Serakides, R1

Other Studies

14 other study(ies) available for niacinamide and ex 527

ArticleYear
Inhibitors of the NAD(+)-Dependent Protein Desuccinylase and Demalonylase Sirt5.
    ACS medicinal chemistry letters, 2012, Dec-13, Volume: 3, Issue:12

    Topics:

2012
Discovery of potent and selective sirtuin 2 (SIRT2) inhibitors using a fragment-based approach.
    Journal of medicinal chemistry, 2014, Oct-23, Volume: 57, Issue:20

    Topics: Animals; Dogs; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; Enzyme Inhibitors; Humans; Ligands; Madin Darby Canine Kidney Cells; MCF-7 Cells; Molecular Structure; Niacinamide; Sirtuin 2; Structure-Activity Relationship; Sulfonic Acids; Suramin

2014
Functionalized tetrahydro-1H-pyrido[4,3-b]indoles: a novel chemotype with Sirtuin 2 inhibitory activity.
    European journal of medicinal chemistry, 2015, Mar-06, Volume: 92

    Topics: Dose-Response Relationship, Drug; Humans; Indoles; Models, Molecular; Molecular Structure; Pyridines; Sirtuin 2; Structure-Activity Relationship

2015
Novel Lysine-Based Thioureas as Mechanism-Based Inhibitors of Sirtuin 2 (SIRT2) with Anticancer Activity in a Colorectal Cancer Murine Model.
    Journal of medicinal chemistry, 2019, 04-25, Volume: 62, Issue:8

    Topics: Animals; Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Cell Proliferation; Colorectal Neoplasms; Disease Models, Animal; Drug Design; Drug Screening Assays, Antitumor; Female; Humans; Lysine; Male; Mice; Mice, Transgenic; Molecular Docking Simulation; Protein Isoforms; Sirtuin 2; Structure-Activity Relationship; Thiourea

2019
Discovery of indoles as potent and selective inhibitors of the deacetylase SIRT1.
    Journal of medicinal chemistry, 2005, Dec-15, Volume: 48, Issue:25

    Topics: Animals; Biological Availability; Carbazoles; Cell Membrane Permeability; CHO Cells; Cricetinae; Cricetulus; Drug Stability; Fluorometry; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; In Vitro Techniques; Indoles; Kinetics; Mice; Mice, Inbred C57BL; Microsomes, Liver; NAD; NAD+ Nucleosidase; Niacinamide; Rats; Recombinant Proteins; Sirtuin 1; Sirtuins; Stereoisomerism; Structure-Activity Relationship

2005
Fructose induces gluconeogenesis and lipogenesis through a SIRT1-dependent mechanism.
    The Journal of endocrinology, 2011, Volume: 208, Issue:3

    Topics: Acetyl-CoA Carboxylase; Animals; Carbazoles; Cholesterol; Fructose; Gluconeogenesis; Hepatocytes; Heterocyclic Compounds, 4 or More Rings; Hydroxymethylglutaryl-CoA-Reductases, NADP-dependent; Lipogenesis; Male; NAD; Niacinamide; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phosphoenolpyruvate Carboxykinase (ATP); Rats; Rats, Sprague-Dawley; RNA-Binding Proteins; Rotenone; Sirtuin 1; Sterol Regulatory Element Binding Protein 1; Transcription Factors

2011
Nicotinamide phosphoribosyltransferase (Nampt) affects the lineage fate determination of mesenchymal stem cells: a possible cause for reduced osteogenesis and increased adipogenesis in older individuals.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2011, Volume: 26, Issue:11

    Topics: Adipocytes; Adipogenesis; Aging; Animals; Bone Marrow Cells; Carbazoles; Cell Line; Cell Lineage; Culture Media; Cytokines; Humans; Intracellular Space; Male; Mesenchymal Stem Cells; Mice; Mice, Inbred C57BL; NAD; Niacinamide; Nicotinamide Phosphoribosyltransferase; Osteogenesis; Sirtuin 1; Stromal Cells

2011
Role of deleted in breast cancer 1 (DBC1) protein in SIRT1 deacetylase activation induced by protein kinase A and AMP-activated protein kinase.
    The Journal of biological chemistry, 2012, Jul-06, Volume: 287, Issue:28

    Topics: Acrylamides; Adaptor Proteins, Signal Transducing; Amino Acid Sequence; AMP-Activated Protein Kinases; Animals; Blotting, Western; Carbazoles; Cell Line, Tumor; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; HEK293 Cells; Hep G2 Cells; Humans; Mice; Mice, Knockout; Models, Biological; Mutation; NAD; Niacinamide; Phosphorylation; Piperidines; Resveratrol; RNA Interference; Signal Transduction; Sirtuin 1; Stilbenes

2012
Sirtuin 1 inhibition delays cyst formation in autosomal-dominant polycystic kidney disease.
    The Journal of clinical investigation, 2013, Volume: 123, Issue:7

    Topics: Acetylation; Animals; Apoptosis; Carbazoles; Cell Proliferation; Cells, Cultured; Drug Evaluation, Preclinical; Epithelial Cells; Female; Gene Expression Regulation, Enzymologic; Kidney; Male; Mice; Mice, Knockout; Niacinamide; Phosphorylation; Polycystic Kidney, Autosomal Dominant; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-myc; Retinoblastoma Protein; Sirtuin 1; Tumor Necrosis Factor-alpha; Tumor Suppressor Protein p53

2013
Studying SIRT6 regulation using H3K56 based substrate and small molecules.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2014, Oct-15, Volume: 63

    Topics: Acetylation; Carbazoles; Histones; Humans; Molecular Structure; Niacinamide; Peptides; Quercetin; Recombinant Proteins; Sirtuins; Structure-Activity Relationship

2014
Role of the Substrate Specificity-Defining Residues of Human SIRT5 in Modulating the Structural Stability and Inhibitory Features of the Enzyme.
    PloS one, 2016, Volume: 11, Issue:3

    Topics: Amino Acids; Biocatalysis; Calorimetry; Carbazoles; Catalytic Domain; Circular Dichroism; Enzyme Stability; Humans; Kinetics; Models, Molecular; Mutant Proteins; Mutation; Niacinamide; Protein Denaturation; Protein Structure, Secondary; Sirtuin 1; Sirtuins; Structure-Activity Relationship; Substrate Specificity; Temperature

2016
TSC2 N-terminal lysine acetylation status affects to its stability modulating mTORC1 signaling and autophagy.
    Biochimica et biophysica acta, 2016, Volume: 1863, Issue:11

    Topics: Acetylation; Animals; Autophagy; Carbazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; HEK293 Cells; Histone Deacetylase Inhibitors; Humans; Lysine; Mechanistic Target of Rapamycin Complex 1; Mice; Multiprotein Complexes; Niacinamide; Protein Domains; Protein Processing, Post-Translational; Protein Stability; Resveratrol; RNA Interference; Signal Transduction; Sirtuin 1; Stilbenes; Time Factors; TOR Serine-Threonine Kinases; Transfection; Tuberous Sclerosis Complex 2 Protein; Tumor Suppressor Proteins

2016
NAD
    Aging cell, 2019, Volume: 18, Issue:3

    Topics: Adult Stem Cells; Aging; Animals; Carbazoles; Cell Proliferation; Cells, Cultured; Dextran Sulfate; Intestinal Mucosa; Male; Mice; Mice, Inbred C57BL; NAD; Niacinamide; Pyridinium Compounds; Rejuvenation; Sirolimus

2019
Differentiation of canine adipose mesenchymal stem cells into insulin-producing cells: comparison of different culture medium compositions.
    Domestic animal endocrinology, 2021, Volume: 74

    Topics: Adipogenesis; Animals; Carbazoles; Cell Differentiation; Chondrogenesis; Culture Media; Dogs; Immunophenotyping; Insulin; Mercaptoethanol; Mesenchymal Stem Cells; Niacinamide; Osteogenesis

2021