nevirapine has been researched along with r-82913 in 27 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 23 (85.19) | 18.2507 |
2000's | 4 (14.81) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Balani, SK; Ciccarone, TM; Condra, JH; Emini, EA; Goldman, ME; Greenlee, WJ; Kauffman, LR; MacTough, SC; Rooney, CS; Williams, TM | 1 |
Bell, FW; Cantrell, AS; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kinnick, MD; Lind, P; Morin, JM; Noréen, R | 1 |
Cantrell, AS; Engelhardt, P; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kangasmetsä, J; Kinnick, MD; Lind, P; Morin, JM; Muesing, MA; Noreén, R; Oberg, B; Pranc, P; Sahlberg, C; Ternansky, RJ; Vasileff, RT; Vrang, L; West, SJ; Zhang, H | 1 |
Andreola, ML; Aubertin, AM; Bisagni, E; Dollé, V; Kirn, A; Legraverend, M; Nguyen, CH; Tarrago-Litvak, L; Ventura, M | 1 |
Jorgensen, WL; Rizzo, RC; Tirado-Rives, J; Wang, DP | 1 |
Jorgensen, WL; Kroeger Smith, MB; Rizzo, RC; Smith, RH; Tirado-Rives, J; Udier-Blagović, M; Wang, DP; Watkins, EK | 1 |
De Corte, BL | 1 |
Larder, BA | 1 |
Deibel, MR; Dueweke, TJ; Kézdy, FJ; Tarpley, WG; Waszak, GA | 1 |
Adams, J; Hargrave, KD; Jacober, SP; Mui, PW | 1 |
Colonno, RJ; Condra, JH; Emini, EA; Gotlib, L; Graham, DJ; Sardana, VV; Schlabach, AJ; Wolfgang, JA | 1 |
Condra, JH; Emini, EA; Gotlib, L; Graham, DJ; Lineberger, DW; Long, WJ; Sardana, VV; Schlabach, AJ; Wolfgang, JA | 1 |
Bacolla, A; Griffin, JA; Hansen, GL; Rose, JM; Shih, CK; Wu, JC | 1 |
Alam, M; Bechtold, CM; Colonno, RJ; Gant, TG; Li, H; Lin, PF; Meyers, AI; Patick, AK; Skoog, MT; Trimble, J | 1 |
De Clercq, E | 1 |
Byrnes, VW; Condra, JH; Emini, EA; Sardana, VV; Schleif, WA | 1 |
Bäckbro, K; Noréen, R; Oberg, B; Unge, T; Vrang, L; Zhang, H | 1 |
Anderson, KS; Johnson, KA; Kati, WM; Spence, RA | 1 |
Evans, DB; Fan, N; Rank, KB; Sharma, SK; Tarpley, WG; Thomas, RC | 1 |
Friebe, WG; Leinert, H; Mertens, A; Nuber, B; Poll, T; Schäfer, W; von der Saal, W; Ziegler, ML; Zilch, H | 1 |
Chen, IS; Dueweke, TJ; Poppe, SM; Pushkarskaya, T; Stevenson, M; Swaney, SM; Tarpley, WG; Zhao, JQ | 1 |
Balzarini, J; Camarasa, MJ; De Clercq, E; Karlsson, A; Pérez-Pérez, MJ; Tarpley, WG | 1 |
Balzarini, J; Camarasa, MJ; De Clercq, E; Karlsson, A; Pérez-Pérez, MJ | 1 |
Esnouf, R; Hopkins, A; Jones, Y; Ren, J; Ross, C; Stammers, D; Stuart, D | 1 |
Balzarini, J; De Clercq, E; Kleim, JP; Pelemans, H; Riess, G; Roesner, M; Winkler, I | 1 |
Fujiwara, T; Hayami, M; Isaka, Y; Kawauchi, S; Miki, S; Sato, A; Suyama, A | 1 |
Ekstrand, DH; Gronowitz, JS; Källander, CF; Rytting, AS; Shao, X; Vrang, L | 1 |
3 review(s) available for nevirapine and r-82913
Article | Year |
---|---|
From 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk](1,4)benzodiazepin-2(1H)-one (TIBO) to etravirine (TMC125): fifteen years of research on non-nucleoside inhibitors of HIV-1 reverse transcriptase.
Topics: Anti-HIV Agents; Benzodiazepines; Drug Design; Drug Resistance, Viral; HIV Reverse Transcriptase; Imidazoles; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors | 2005 |
HIV resistance to reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Dideoxynucleosides; Dose-Response Relationship, Drug; Drug Resistance; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Mutation; Nevirapine; Pyridines; Reverse Transcriptase Inhibitors; Thymine | 1994 |
The genetic and functional basis of HIV-1 resistance to nonnucleoside reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Benzoxazoles; Clinical Trials as Topic; Drug Resistance, Microbial; Genetic Variation; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1994 |
24 other study(ies) available for nevirapine and r-82913
Article | Year |
---|---|
5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.
Topics: Animals; Antiviral Agents; Base Sequence; Biological Availability; HIV; HIV Reverse Transcriptase; HIV-1; Indoles; Macaca mulatta; Molecular Sequence Data; Molecular Structure; Reverse Transcriptase Inhibitors; Sulfoxides | 1993 |
Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of PETT analogs.
Topics: Animals; Antiviral Agents; Cell Line; HIV-1; Humans; Isothiocyanates; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles; Thiourea | 1995 |
Phenethylthiazolylthiourea (PETT) compounds as a new class of HIV-1 reverse transcriptase inhibitors. 2. Synthesis and further structure-activity relationship studies of PETT analogs.
Topics: Animals; Anti-HIV Agents; Cells, Cultured; HIV Reverse Transcriptase; Intercalating Agents; Structure-Activity Relationship; Thiazoles; Thiourea | 1996 |
Synthesis and antiviral activity of 4-benzyl pyridinone derivatives as potent and selective non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors.
Topics: Anti-HIV Agents; Cell Line; Cells, Cultured; Drug Resistance, Microbial; HIV-1; Humans; Pyridones; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship; Virion; Virus Replication | 2000 |
Antiviral drug design: computational analyses of the effects of the L100I mutation for HIV-RT on the binding of NNRTIs.
Topics: Drug Design; HIV Reverse Transcriptase; Models, Molecular; Mutation; Reverse Transcriptase Inhibitors | 2001 |
Prediction of activity for nonnucleoside inhibitors with HIV-1 reverse transcriptase based on Monte Carlo simulations.
Topics: Alkynes; Anilides; Benzoxazines; Computer Simulation; Cyclopropanes; HIV Reverse Transcriptase; Hydrogen Bonding; Models, Molecular; Monte Carlo Method; Nevirapine; Oxazines; Protein Binding; Quinoxalines; Regression Analysis; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Uracil | 2002 |
3'-Azido-3'-deoxythymidine resistance suppressed by a mutation conferring human immunodeficiency virus type 1 resistance to nonnucleoside reverse transcriptase inhibitors.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Cloning, Molecular; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Pyridines; Reverse Transcriptase Inhibitors; Zidovudine | 1992 |
The binding of a novel bisheteroarylpiperazine mediates inhibition of human immunodeficiency virus type 1 reverse transcriptase.
Topics: Benzodiazepines; Binding, Competitive; Dideoxynucleosides; Foscarnet; HIV-1; Imidazoles; Indoles; Nevirapine; Phosphonoacetic Acid; Piperazines; Pyridines; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1992 |
Crystal structure of nevirapine, a non-nucleoside inhibitor of HIV-1 reverse transcriptase, and computational alignment with a structurally diverse inhibitor.
Topics: Azepines; Benzodiazepines; Binding Sites; Crystallography; HIV-1; Imidazoles; Models, Molecular; Molecular Conformation; Nevirapine; Pyridines; Reverse Transcriptase Inhibitors; X-Ray Diffraction | 1992 |
Identification of the human immunodeficiency virus reverse transcriptase residues that contribute to the activity of diverse nonnucleoside inhibitors.
Topics: Antiviral Agents; Azepines; Benzodiazepines; Benzoxazoles; Drug Resistance, Microbial; Escherichia coli; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Nevirapine; Phenotype; Pyridines; Pyridones; Reverse Transcriptase Inhibitors | 1992 |
Functional analysis of HIV-1 reverse transcriptase amino acids involved in resistance to multiple nonnucleoside inhibitors.
Topics: Amino Acid Sequence; Antiviral Agents; Azepines; Benzodiazepines; Benzoxazoles; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Nevirapine; Pyridines; Pyridones; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship | 1992 |
Chimeric human immunodeficiency virus type 1/type 2 reverse transcriptases display reversed sensitivity to nonnucleoside analog inhibitors.
Topics: Affinity Labels; Amino Acid Sequence; Azepines; Benzodiazepines; Binding Sites; DNA Mutational Analysis; HIV-1; HIV-2; Imidazoles; Molecular Sequence Data; Nevirapine; Pyridines; Recombinant Fusion Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship; Tyrosine | 1991 |
Substituted naphthalenones as a new structural class of HIV-1 reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Cell Line; Dose-Response Relationship, Drug; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Naphthalenes; Nevirapine; Oxazoles; Pyridines; Reverse Transcriptase Inhibitors; T-Lymphocytes | 1993 |
Enzymatic properties and sensitivity to inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase with Glu-138-->Arg and Tyr-188-->His mutations.
Topics: Amino Acids; Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Binding, Competitive; Deoxyguanine Nucleotides; Dideoxynucleotides; Foscarnet; HIV Reverse Transcriptase; Humans; Imidazoles; Kinetics; Molecular Sequence Data; Mutation; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sensitivity and Specificity | 1994 |
Mechanism of inhibition of HIV-1 reverse transcriptase by nonnucleoside inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Binding Sites; Deoxyadenine Nucleotides; DNA; HIV Reverse Transcriptase; HIV-1; Imidazoles; Kinetics; Magnesium; Nevirapine; Protein Conformation; Pyridines; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1995 |
Simultaneous mutations at Tyr-181 and Tyr-188 in HIV-1 reverse transcriptase prevents inhibition of RNA-dependent DNA polymerase activity by the bisheteroarylpiperazine (BHAP) U-90152s.
Topics: Amino Acid Sequence; Antiviral Agents; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; HIV Reverse Transcriptase; HIV-1; HIV-2; Imidazoles; Indoles; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Point Mutation; Pyridines; Pyridones; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Tyrosine | 1995 |
Non-nucleoside inhibitors of HIV-1 reverse transcriptase: molecular modeling and X-ray structure investigations.
Topics: Benzodiazepines; Crystallography; Drug Design; HIV Reverse Transcriptase; Imidazoles; Kinetics; Models, Molecular; Molecular Conformation; Nevirapine; Pyridines; Reverse Transcriptase Inhibitors; Stereoisomerism; Structure-Activity Relationship | 1993 |
A mutation in reverse transcriptase of bis(heteroaryl)piperazine-resistant human immunodeficiency virus type 1 that confers increased sensitivity to other nonnucleoside inhibitors.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; Drug Resistance; HIV Reverse Transcriptase; Imidazoles; Indoles; Molecular Sequence Data; Mutation; Nevirapine; Oligodeoxyribonucleotides; Piperazines; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1993 |
Treatment of human immunodeficiency virus type 1 (HIV-1)-infected cells with combinations of HIV-1-specific inhibitors results in a different resistance pattern than does treatment with single-drug therapy.
Topics: Amino Acid Sequence; Antiviral Agents; Benzodiazepines; Cell Line; Dideoxynucleosides; Drug Interactions; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Mutagenesis; Nevirapine; Piperazines; Pyridines; Pyridones; RNA-Directed DNA Polymerase; Spiro Compounds; Thymidine; Uridine | 1993 |
Knocking-out concentrations of HIV-1-specific inhibitors completely suppress HIV-1 infection and prevent the emergence of drug-resistant virus.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Cells, Cultured; Dose-Response Relationship, Drug; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Microbial Sensitivity Tests; Molecular Sequence Data; Nevirapine; Piperazines; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sequence Analysis; Spiro Compounds; Thymidine; Thymine; Uridine; Virus Replication | 1993 |
The structure of HIV-1 reverse transcriptase complexed with 9-chloro-TIBO: lessons for inhibitor design.
Topics: Benzodiazepines; Binding Sites; Crystallography, X-Ray; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Metals; Models, Molecular; Mutation; Nevirapine; Protein Conformation; Pyridines; Reverse Transcriptase Inhibitors; Ribonuclease H; RNA-Directed DNA Polymerase; Thymine | 1995 |
Retention of marked sensitivity to (S)-4-isopropoxycarbonyl-6-methoxy-3-(methylthiomethyl)-3,4-di hydroquin oxaline-2(1H)-thione (HBY 097) by an azidothymidine (AZT)-resistant human immunodeficiency virus type 1 (HIV-1) strain subcultured in the combined
Topics: Anti-HIV Agents; Antiviral Agents; Benzodiazepines; Cell Line; Delavirdine; Drug Resistance, Microbial; Furans; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Lamivudine; Microbial Sensitivity Tests; Mutagenesis, Site-Directed; Mutation; Nevirapine; Quinoxalines; Recombinant Proteins; Reverse Transcriptase Inhibitors; Zidovudine | 1998 |
Construction of the chimeric reverse transcriptase of simian immunodeficiency virus sensitive to nonnucleoside reverse transcriptase inhibitor.
Topics: Amino Acid Sequence; Benzodiazepines; Cells, Cultured; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Kinetics; Molecular Sequence Data; Nevirapine; Reassortant Viruses; Recombinant Fusion Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Simian Immunodeficiency Virus; Transfection; Uracil | 1998 |
Colorimetric assays for evaluation of the mode of action of human immunodeficiency virus type 1 non-nucleoside reverse transcriptase inhibitors.
Topics: Amino Acid Sequence; Anti-HIV Agents; Benzodiazepines; Colorimetry; Delavirdine; Drug Evaluation; Enzyme-Linked Immunosorbent Assay; HIV Reverse Transcriptase; HIV-1; Imidazoles; Molecular Sequence Data; Nevirapine; Pyridines; Recombinant Proteins; Reverse Transcriptase Inhibitors; Templates, Genetic; Thiourea | 1998 |