nevirapine has been researched along with l-697661 in 23 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 21 (91.30) | 18.2507 |
2000's | 2 (8.70) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bamberger, DL; Fisher, TE; Goldman, ME; Hoffman, JM; Jones, JH; Rooney, CS; Saari, WS; Smith, AM; Thomas, CM; Wai, JS | 1 |
Fisher, TE; Goldman, ME; Hoffman, JM; Nunberg, JH; O'Brien, JA; Rooney, CS; Saari, WS; Smith, AM; Thomas, CM; Wai, JS | 1 |
Bethell, RC; Cammack, N; Green, DV; Hancock, AP; Hann, MM; Lamont, RB; Livermore, DG; Noble, SA; Orr, DC; Payne, JJ | 1 |
Ball, RG; Britcher, SF; Goldman, ME; Lumma, WC; Lyle, TA; O'Brien, JA; Sanders, WM; Tucker, TJ; Wiscount, CM; Young, SD | 1 |
Bethell, RC; Cammack, N; Charon, D; Dodic, N; Dumaitre, B; Evans, DN; Green, DV; Hopewell, PL; Humber, DC; Wyatt, PG | 1 |
Bamberger, DL; Fisher, TE; Hoffman, JM; Hudcosky, RJ; MacTough, SC; Rooney, CS; Saari, WS; Thomas, CM; Wai, JS; Williams, TM | 1 |
Balani, SK; Ciccarone, TM; Condra, JH; Emini, EA; Goldman, ME; Greenlee, WJ; Kauffman, LR; MacTough, SC; Rooney, CS; Williams, TM | 1 |
Althaus, IW; Biles, C; Busso, M; Genin, MJ; Morge, RA; Resnick, L; Reusser, F; Romero, DL; Tarpley, WG; Thomas, RC | 1 |
Kampe, W; König, B; Leinert, H; Leser, U; Mertens, A; Poll, T; Schäfer, W; Seidel, H; Zilch, H | 1 |
Bell, FW; Cantrell, AS; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kinnick, MD; Lind, P; Morin, JM; Noréen, R | 1 |
Altamura, S; Campiani, G; De Filippis, MP; Di Renzo, L; Fiorini, I; Garofalo, A; Greco, G; Nacci, V; Novellino, E | 1 |
Adams, WJ; Biles, C; Evans, DB; Friis, JM; Hosley, JD; Keiser, BJ; Kopta, LA; Morge, RA; Morris, J; Olmsted, RA; Poel, TJ; Romero, DL; Sharma, SK; Stefanski, KJ; Stehle, RG; Tarpley, WG; Thomas, RC; Voorman, RL; Wishka, DG; Yagi, Y | 1 |
Cantrell, AS; Engelhardt, P; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kangasmetsä, J; Kinnick, MD; Lind, P; Morin, JM; Muesing, MA; Noreén, R; Oberg, B; Pranc, P; Sahlberg, C; Ternansky, RJ; Vasileff, RT; Vrang, L; West, SJ; Zhang, H | 1 |
Engelhardt, P; Högberg, M; Kangasmetsä, J; Noréen, R; Sahlberg, C; Vrang, L; Zhang, H | 1 |
Biles, C; Genin, MJ; Keiser, BJ; Poppe, SM; Romero, DL; Swaney, SM; Tarpley, WG; Yagi, Y | 1 |
Dornadula, G; Grobler, JA; Hazuda, DJ; Miller, MD; Rice, MR; Simcoe, AL | 1 |
Condra, JH; Emini, EA; Gotlib, L; Graham, DJ; Lineberger, DW; Long, WJ; Sardana, VV; Schlabach, AJ; Wolfgang, JA | 1 |
Bender, R; Kirsch, R; Kleim, JP; Meichsner, C; Paessens, A; Riess, G | 1 |
Byrnes, VW; Condra, JH; Emini, EA; Sardana, VV; Schleif, WA | 1 |
Bäckbro, K; Noréen, R; Oberg, B; Unge, T; Vrang, L; Zhang, H | 1 |
Evans, DB; Fan, N; Rank, KB; Sharma, SK; Tarpley, WG; Thomas, RC | 1 |
Chen, IS; Dueweke, TJ; Poppe, SM; Pushkarskaya, T; Stevenson, M; Swaney, SM; Tarpley, WG; Zhao, JQ | 1 |
Kilby, JM; Saag, MS | 1 |
2 review(s) available for nevirapine and l-697661
Article | Year |
---|---|
The genetic and functional basis of HIV-1 resistance to nonnucleoside reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Benzoxazoles; Clinical Trials as Topic; Drug Resistance, Microbial; Genetic Variation; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1994 |
Clinical experience with non-nucleoside reverse transcriptase inhibitors: L-697,661 and nevirapine.
Topics: Benzoxazoles; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1996 |
21 other study(ies) available for nevirapine and l-697661
Article | Year |
---|---|
Synthesis and evaluation of 2-pyridinone derivatives as HIV-1-specific reverse transcriptase inhibitors. 2. Analogues of 3-aminopyridin-2(1H)-one.
Topics: Aminopyridines; Antiviral Agents; Benzoxazoles; Cells, Cultured; HIV Reverse Transcriptase; HIV-1; Pyridones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 1992 |
2-Pyridinone derivatives: a new class of nonnucleoside, HIV-1-specific reverse transcriptase inhibitors.
Topics: Antiviral Agents; HIV-1; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1991 |
Synthesis and anti-HIV-1 activity of a series of imidazo[1,5-b]pyridazines.
Topics: Antiviral Agents; Cell Division; Cell Line; Crystallization; HIV Reverse Transcriptase; HIV-1; Imidazoles; Molecular Structure; Pyridazines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Virus Replication; Zidovudine | 1993 |
Synthesis of a series of 4-(arylethynyl)-6-chloro-4-cyclopropyl-3,4-dihydroquinazolin-2(1H)-ones as novel non-nucleoside HIV-1 reverse transcriptase inhibitors.
Topics: Cells, Cultured; Crystallography, X-Ray; HIV Reverse Transcriptase; HIV-1; Humans; Quinazolines; Reverse Transcriptase Inhibitors | 1994 |
Benzophenone derivatives: a novel series of potent and selective inhibitors of human immunodeficiency virus type 1 reverse transcriptase.
Topics: Benzophenones; Cell Line; Crystallography, X-Ray; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 1995 |
Synthesis and evaluation of 2-pyridinone derivatives as specific HIV-1 reverse transcriptase inhibitors. 3. Pyridyl and phenyl analogs of 3-aminopyridin-2(1H)-one.
Topics: Aminopyridines; Animals; Antiviral Agents; Cells, Cultured; Haplorhini; HIV Reverse Transcriptase; Pyridones; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 1993 |
5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.
Topics: Animals; Antiviral Agents; Base Sequence; Biological Availability; HIV; HIV Reverse Transcriptase; HIV-1; Indoles; Macaca mulatta; Molecular Sequence Data; Molecular Structure; Reverse Transcriptase Inhibitors; Sulfoxides | 1993 |
Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogues and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)-carbonyl]-4-[3- [(1-methylethyl)amino]-pyridinyl]pi
Topics: Antiviral Agents; Delavirdine; Indoles; Piperazines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Virus Replication | 1993 |
Selective non-nucleoside HIV-1 reverse transcriptase inhibitors. New 2,3-dihydrothiazolo[2,3-a]isoindol-5(9bH)-ones and related compounds with anti-HIV-1 activity.
Topics: Animals; Antiviral Agents; Cells, Cultured; HIV Reverse Transcriptase; Indoles; Rats; Reverse Transcriptase Inhibitors; Stereoisomerism; Structure-Activity Relationship; Thiazoles | 1993 |
Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of PETT analogs.
Topics: Animals; Antiviral Agents; Cell Line; HIV-1; Humans; Isothiocyanates; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles; Thiourea | 1995 |
Pyrrolobenzothiazepinones and pyrrolobenzoxazepinones: novel and specific non-nucleoside HIV-1 reverse transcriptase inhibitors with antiviral activity.
Topics: Antiviral Agents; Cell Line; HIV Reverse Transcriptase; HIV-1; Humans; Models, Molecular; Molecular Structure; Oxazepines; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship; Thiazepines | 1996 |
Targeting delavirdine/atevirdine resistant HIV-1: identification of (alkylamino)piperidine-containing bis(heteroaryl)piperazines as broad spectrum HIV-1 reverse transcriptase inhibitors.
Topics: Animals; Anti-HIV Agents; Biological Availability; Cell Line; Delavirdine; Drug Resistance, Microbial; Drug Stability; HIV Reverse Transcriptase; HIV-1; Indoles; Molecular Structure; Piperazines; Piperidines; Pyridines; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 1996 |
Phenethylthiazolylthiourea (PETT) compounds as a new class of HIV-1 reverse transcriptase inhibitors. 2. Synthesis and further structure-activity relationship studies of PETT analogs.
Topics: Animals; Anti-HIV Agents; Cells, Cultured; HIV Reverse Transcriptase; Intercalating Agents; Structure-Activity Relationship; Thiazoles; Thiourea | 1996 |
Synthesis and anti-HIV activities of urea-PETT analogs belonging to a new class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Topics: Anti-HIV Agents; Blood Proteins; Cell Line; HIV-1; Humans; Microbial Sensitivity Tests; Protein Binding; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles; Triazoles | 1998 |
Novel 1,5-diphenylpyrazole nonnucleoside HIV-1 reverse transcriptase inhibitors with enhanced activity versus the delavirdine-resistant P236L mutant: lead identification and SAR of 3- and 4-substituted derivatives.
Topics: Anti-HIV Agents; Delavirdine; Drug Resistance, Microbial; HIV Reverse Transcriptase; Mutation; Pyrazoles; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 2000 |
HIV-1 reverse transcriptase plus-strand initiation exhibits preferential sensitivity to non-nucleoside reverse transcriptase inhibitors in vitro.
Topics: Alkynes; Anti-HIV Agents; Benzoxazines; Benzoxazoles; Cyclopropanes; DNA; Dose-Response Relationship, Drug; Drug Resistance, Viral; Enzyme Inhibitors; HIV Reverse Transcriptase; In Vitro Techniques; Inhibitory Concentration 50; Ligands; Models, Genetic; Oxazines; Pyridones; Reverse Transcriptase Inhibitors; Stochastic Processes; Transcription, Genetic; Virus Replication | 2007 |
Functional analysis of HIV-1 reverse transcriptase amino acids involved in resistance to multiple nonnucleoside inhibitors.
Topics: Amino Acid Sequence; Antiviral Agents; Azepines; Benzodiazepines; Benzoxazoles; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Nevirapine; Pyridines; Pyridones; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship | 1992 |
Mutational analysis of residue 190 of human immunodeficiency virus type 1 reverse transcriptase.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Delavirdine; DNA Mutational Analysis; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Indoles; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Pyridines; Pyridones; Quinoxalines; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Selection, Genetic; Structure-Activity Relationship | 1994 |
Enzymatic properties and sensitivity to inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase with Glu-138-->Arg and Tyr-188-->His mutations.
Topics: Amino Acids; Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Binding, Competitive; Deoxyguanine Nucleotides; Dideoxynucleotides; Foscarnet; HIV Reverse Transcriptase; Humans; Imidazoles; Kinetics; Molecular Sequence Data; Mutation; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sensitivity and Specificity | 1994 |
Simultaneous mutations at Tyr-181 and Tyr-188 in HIV-1 reverse transcriptase prevents inhibition of RNA-dependent DNA polymerase activity by the bisheteroarylpiperazine (BHAP) U-90152s.
Topics: Amino Acid Sequence; Antiviral Agents; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; HIV Reverse Transcriptase; HIV-1; HIV-2; Imidazoles; Indoles; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Point Mutation; Pyridines; Pyridones; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Tyrosine | 1995 |
A mutation in reverse transcriptase of bis(heteroaryl)piperazine-resistant human immunodeficiency virus type 1 that confers increased sensitivity to other nonnucleoside inhibitors.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; Drug Resistance; HIV Reverse Transcriptase; Imidazoles; Indoles; Molecular Sequence Data; Mutation; Nevirapine; Oligodeoxyribonucleotides; Piperazines; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1993 |