Page last updated: 2024-08-23

neurokinin b and piperidines

neurokinin b has been researched along with piperidines in 47 studies

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's26 (55.32)18.2507
2000's15 (31.91)29.6817
2010's6 (12.77)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bikker, J; Chung, FZ; Humblet, C; Lee, H; Pritchard, MC; Raphy, J; Suman-Chauhan, N; Tian, Y; Vartanian, MA; Wu, LH1
Couture, R; Picard, P; Regoli, D1
Chung, FZ; Grimson, P; Guard, S; Madden, Z; Pinnock, R; Suman-Chauhan, N; Watling, K; Woodruff, G1
Giuliani, S; Maggi, CA; Zagorodnyuk, V1
Andersson, KE; Ishizuka, O; Mattiasson, A1
Fukuhara, S; Mukai, H; Munekata, E1
Fong, TM; Huang, RR; Strader, CD; Vicario, PP1
Killingsworth, CR; Shore, SA1
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Pellegrini, CA1
Bichon, D; Ducoux, JP; Emonds-Alt, X; Heaulme, M; Miloux, B; Neliat, G; Poncelet, M; Proietto, V; Van Broeck, D; Vilain, P1
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Nakazato, P; Pellegrini, CA1
Chapman, RW; Danko, G; del Prado, M; Hey, JA1
Marchionni, D; Nisato, D; Roccon, A1
Inoue, H; Koshihara, Y; Nagata, N1
Hay, DW; Medhurst, AD; Parsons, AA; Roberts, JC1
Beaujouan, JC; Glowinski, J; Saffroy, M; Torrens, Y1
O'Grady, SM; Vetter, AE1
Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Parsons, AA1
MacNaughton, W; Moore, B; Vanner, S1
Jino, H; Kanda, M; Kurahashi, K; Murase, K; Nakamura, S; Shirahase, H; Usui, H1
Blanchet, F; Gauchy, C; Glowinski, J; Kemel, ML; Perez, S; Soubrié, P1
Guo, JZ; Otsuka, M; Yoshioka, K1
Bjorling, DE; Jerde, TJ; Nakada, SY; Saban, R1
Atherton, J; Chen, MH; Chung, FZ; Kuo, BS; Lee, HT; Roth, BD1
Bredenbröker, D; Fehmann, H; Klüber, D; Lange, A; Wagner, U; Wichert, P1
Calixto, JB; De Lima, TC; Ribeiro, SJ; Teixeira, RM1
Geraghty, DP; Mazzone, SB1
Chell, MJ; El-Fakahany, EE; Linden, DR; Seybold, VS1
Advenier, C; Daoui, S; Emonds-Alt, X; Lagente, V; Naline, E1
Coupar, IM; Kerr, KP; Thai, B1
Broccardo, M; Improta, G1
Krysiak, PS; Preiksaitis, HG1
Baird, AW; Goldhill, J; Moriarty, D; O'Donoghue, DP; Selve, N1
Advenier, C; Daoui, S; Emonds-Alt, X; Gueudet, C; Le Fur, G; Maffrand, JP; Michaud, JC; Naline, E; Oury-Donat, F; Pascal, M; Poncelet, M; Proietto, V; Soubrié, P; Steinberg, R; Vilain, P1
Akhtar, R; Brain, SD; Gerard, NP; Grant, AD1
Hirano, K; Kanaide, H; Naito, S; Nishimura, J; Takahashi, R1
Cvetkovic, V; Fellmann, D; Griffond, B; Poncet, F; Risold, PY1
de Francischi, JN; Lisboa, MC; Santos, JM; Tatsuo, MA; Turchetti-Maia, RM1
Morimoto, K; Mukaiyama, O; Nosaka, E; Takahashi, S; Yamashita, M1
Scott, CW; Tian, G; Wilkins, D1
Candenas, ML; Fernández-Sánchez, M; Orea, A; Pintado, CO; Pinto, FM; Ravina, CG; Seda, M1
Candenas, L; Cejudo-Román, A; Fernández-Sánchez, M; Garrido, N; Irazusta, J; Pinto, FM; Ravina, CG; Subiran, N1
Huston, JP; Schäble, S; Silva, MA1
Corboz, MR; Fernandez, X; Greenfeder, S; Rivelli, MA1
Boehm, U; de Croft, S; Herbison, AE1
Andero, R; Dias, BG; Ressler, KJ1
Dong, S; He, C; Wei, C; Yang, Q; Yang, Y; Zhou, L1

Other Studies

47 other study(ies) available for neurokinin b and piperidines

ArticleYear
Two classes of structurally different antagonists display similar species preference for the human tachykinin neurokinin3 receptor.
    Molecular pharmacology, 1995, Volume: 48, Issue:4

    Topics: Animals; Benzamides; Binding, Competitive; CHO Cells; Cricetinae; Dipeptides; Humans; Inositol Phosphates; Iodine Radioisotopes; Kinetics; Mutation; Neurokinin B; Phenylalanine; Piperidines; Radioligand Assay; Rats; Receptors, Neurokinin-3; Species Specificity; Structure-Activity Relationship

1995
Cardiovascular and behavioural effects of centrally administered tachykinins in the rat: characterization of receptors with selective antagonists.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Behavior, Animal; Benzamides; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Indoles; Injections, Intraventricular; Isoindoles; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Tachykinins

1994
Characterisation of [125I][MePhe7]neurokinin B binding to tachykinin NK3 receptors: evidence for interspecies variance.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: Amino Acid Sequence; Animals; Benzamides; Binding, Competitive; Cerebral Cortex; CHO Cells; Cricetinae; Cricetulus; Guinea Pigs; Humans; Molecular Sequence Data; Neurokinin B; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-3; Receptors, Tachykinin; Regression Analysis; Substance P

1994
Tachykinin NK3 receptor mediates NANC hyperpolarization and relaxation via nitric oxide release in the circular muscle of the guinea-pig colon.
    Regulatory peptides, 1994, Oct-21, Volume: 53, Issue:3

    Topics: Animals; Apamin; Arginine; Atropine; Colon; Dose-Response Relationship, Drug; Guanethidine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Neurokinin B; Nitric Oxide; Nitroarginine; Oligopeptides; Peptide Fragments; Piperidines; Quinuclidines; Receptors, Neurokinin-3; Stereoisomerism; Substance P; Tetrodotoxin

1994
Tachykinin effects on bladder activity in conscious normal rats.
    The Journal of urology, 1995, Volume: 154, Issue:1

    Topics: Administration, Intravesical; Animals; Benzamides; Female; Indoles; Injections, Intra-Arterial; Isoindoles; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Substance P; Urinary Bladder; Urination

1995
Pharmacological evidence for neurokinin receptors in murine neuroblastoma C1300 cells.
    Peptides, 1995, Volume: 16, Issue:2

    Topics: Animals; Benzamides; Calcium; Cell Line; Kinetics; Mice; Neuroblastoma; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; Substance P; Tumor Cells, Cultured

1995
Identification of residues involved in ligand binding to the neurokinin-2 receptor.
    Biochemistry, 1995, Aug-08, Volume: 34, Issue:31

    Topics: Amino Acid Sequence; Benzamides; Binding Sites; DNA Mutational Analysis; Dose-Response Relationship, Drug; Humans; Ligands; Molecular Sequence Data; Neurokinin A; Neurokinin B; Peptide Fragments; Phosphatidylinositols; Piperidines; Receptors, Neurokinin-2; Recombinant Proteins; Signal Transduction; Structure-Activity Relationship; Substance P; Tachykinins

1995
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
Tachykinins contract the circular muscle of the human esophageal body in vitro via NK2 receptors.
    Gastroenterology, 1993, Volume: 105, Issue:4

    Topics: Adolescent; Adult; Aged; Atropine; Benzamides; Biphenyl Compounds; Carbachol; Dose-Response Relationship, Drug; Esophagus; Glycopeptides; Humans; Isometric Contraction; Middle Aged; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; Substance P; Tachykinins; Tetrodotoxin

1993
SR 142801, the first potent non-peptide antagonist of the tachykinin NK3 receptor.
    Life sciences, 1995, Volume: 56, Issue:1

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; In Vitro Techniques; Neurokinin B; Piperidines; Rats; Receptors, Neurokinin-3; Vasoconstriction

1995
Tachykinins mediate contraction of the human lower esophageal sphincter in vitro via activation of NK2 receptors.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Benzamides; Biphenyl Compounds; Dose-Response Relationship, Drug; Esophagogastric Junction; Glycopeptides; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins

1993
Augmentation of neurally evoked cholinergic bronchoconstrictor responses by prejunctional NK2 receptors in the guinea-pig.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Bronchoconstriction; Bronchoconstrictor Agents; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Male; Medulla Oblongata; Methacholine Chloride; Muscle, Smooth; Neurokinin A; Neurokinin B; Piperidines; Substance P

1996
Study of SR 142801, a new potent non-peptide NK3 receptor antagonist on cardiovascular responses in conscious guinea-pig.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Analysis of Variance; Animals; Blood Pressure; Dose-Response Relationship, Drug; Guinea Pigs; Heart Rate; Injections, Intravenous; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Substance P

1996
Involvement of tachykinin receptors in oedema formation and plasma extravasation induced by substance P, neurokinin A, and neurokinin B in mouse ear.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:7

    Topics: Animals; Capillary Permeability; Edema; Glycopeptides; Male; Mice; Neurokinin A; Neurokinin B; Piperidines; Quinuclidines; Receptors, Tachykinin; Substance P

1996
Characterization of NK3 receptors in rabbit isolated iris sphincter muscle.
    British journal of pharmacology, 1997, Volume: 120, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Benzamides; Electric Stimulation; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle, Smooth; Neurokinin B; Peptide Fragments; Phenoxybenzamine; Piperidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1997
Substance P(6-11) and natural tachykinins interact with septide-sensitive tachykinin receptors coupled to a phospholipase C in the rat urinary bladder.
    Neuropeptides, 1997, Volume: 31, Issue:3

    Topics: Analgesics; Animals; Benzamides; Binding Sites; Inositol Phosphates; Male; Neurokinin A; Neurokinin B; Neuropeptides; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Tachykinins; Tritium; Type C Phospholipases; Urinary Bladder

1997
Mechanisms of electrolyte transport across the endometrium. II. Regulation by GRP and substance P.
    The American journal of physiology, 1997, Volume: 273, Issue:1 Pt 1

    Topics: Amiloride; Animals; Biological Transport; Cell Membrane Permeability; Electrolytes; Female; Gastrin-Releasing Peptide; Gastrointestinal Hormones; Ionomycin; Kinetics; Membrane Potentials; Models, Biological; Mucous Membrane; Myometrium; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptides; Piperidines; Potassium; Substance P; Swine; Thapsigargin

1997
In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Animals; In Vitro Techniques; Iris; Male; Miosis; Muscle Contraction; Muscle, Smooth; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Substance P

1997
Cellular pathways mediating tachykinin-evoked secretomotor responses in guinea pig ileum.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Capsaicin; Electric Stimulation; Evoked Potentials; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Mucosa; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins

1997
[Tachykinin receptor subtypes involved in endothelium-dependent and -independent responses in rabbit intrapulmonary arteries].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1997, Volume: 110 Suppl 1

    Topics: Animals; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Pulmonary Artery; Rabbits; Receptors, Tachykinin; Substance P

1997
Distinct modifications by neurokinin1 (SR140333) and neurokinin2 (SR48968) tachykinin receptor antagonists of the N-methyl-D-aspartate-evoked release of acetylcholine in striosomes and matrix of the rat striatum.
    Neuroscience, 1998, Volume: 85, Issue:4

    Topics: Acetylcholine; Animals; Benzamides; Dopamine; Excitatory Amino Acid Agonists; In Vitro Techniques; Male; N-Methylaspartate; Neostriatum; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-2; Stimulation, Chemical; Substance P

1998
Effects of a tachykinin NK3 receptor antagonist, SR 142801, studied in isolated neonatal rat spinal cord.
    Neuropeptides, 1998, Volume: 32, Issue:6

    Topics: Animals; Animals, Newborn; Capsaicin; Electrophysiology; Female; In Vitro Techniques; Male; Membrane Potentials; Neurokinin B; Neurons, Afferent; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Spinal Cord; Spinal Nerve Roots; Substance P

1998
NK-2 is the predominant tachykinin receptor subtype in the swine ureter.
    BJU international, 1999, Volume: 83, Issue:3

    Topics: Animals; Benzamides; Dose-Response Relationship, Drug; Neurokinin A; Neurokinin B; Piperidines; Receptors, Neurokinin-2; Swine; Ureter

1999
Syntheses and biological activities of chiral piperidines-tachykinin NK3 antagonists.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:3

    Topics: Animals; Area Under Curve; Intestinal Absorption; Male; Neurokinin B; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship

1999
Effects of selective tachykinin-receptor antagonists on tachykinin-induced airway mucus secretion in the rat.
    Neuropeptides, 1999, Volume: 33, Issue:1

    Topics: Animals; Benzamides; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mucosa; Substance P; Tachykinins; Trachea

1999
Tachykinin NK(3)receptor involvement in anxiety.
    Neuropeptides, 1999, Volume: 33, Issue:2

    Topics: Animals; Anxiety; Cerebral Ventricles; Injections, Intraventricular; Male; Maze Learning; Mice; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins

1999
Respiratory actions of tachykinins in the nucleus of the solitary tract: characterization of receptors using selective agonists and antagonists.
    British journal of pharmacology, 2000, Volume: 129, Issue:6

    Topics: Animals; Benzamides; Indoles; Isoindoles; Male; Microinjections; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mechanics; Solitary Nucleus; Substance P; Tachykinins; Tidal Volume

2000
Neurokinin(3) receptors couple to the activation of neuronal nitric-oxide synthase in stably transfected Chinese hamster ovary cells.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:2

    Topics: Animals; Calcium; Calcium Signaling; Cell Line; CHO Cells; Citrulline; Cricetinae; Cyclic GMP; Enzyme Activation; Guanylate Cyclase; Humans; Immunohistochemistry; Inositol Phosphates; Neurokinin B; Neurons; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Piperidines; Rats; Receptors, Neurokinin-3; Transfection

2000
Neurokinin B- and specific tachykinin NK(3) receptor agonists-induced airway hyperresponsiveness in the guinea-pig.
    British journal of pharmacology, 2000, Volume: 130, Issue:1

    Topics: Acetylcholine; Animals; Bronchi; Bronchoconstrictor Agents; Female; Guinea Pigs; Male; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins; Vasodilator Agents

2000
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000
Effects of supraspinal administration of PG-SPI and PG-KII, two amphibian tachykinin peptides, on nociception in the rat.
    Peptides, 2000, Volume: 21, Issue:11

    Topics: Analgesia; Animals; Dose-Response Relationship, Drug; Hot Temperature; Indoles; Male; Naloxone; Narcotic Antagonists; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Oligopeptides; Pain Measurement; Pain Threshold; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins; Time Factors

2000
Tachykinins contribute to nerve-mediated contractions in the human esophagus.
    Gastroenterology, 2001, Volume: 120, Issue:1

    Topics: Atropine; Autonomic Nervous System; Benzamides; Dose-Response Relationship, Drug; Esophagus; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Parasympatholytics; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Substance P; Tachykinins

2001
Human colonic anti-secretory activity of the potent NK(1) antagonist, SR140333: assessment of potential anti-diarrhoeal activity in food allergy and inflammatory bowel disease.
    British journal of pharmacology, 2001, Volume: 133, Issue:8

    Topics: Animals; Antidiarrheals; Capsaicin; Colitis, Ulcerative; Colon; Crohn Disease; Epithelial Cells; Food Hypersensitivity; Guinea Pigs; Humans; Immunoglobulin E; Inflammatory Bowel Diseases; Male; Mast Cells; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Receptors, Neurokinin-1; Species Specificity; Substance P; Tachykinins

2001
Biochemical and pharmacological activities of SSR 146977, a new potent nonpeptide tachykinin NK3 receptor antagonist.
    Canadian journal of physiology and pharmacology, 2002, Volume: 80, Issue:5

    Topics: Animals; CHO Cells; Cricetinae; Gerbillinae; Guinea Pigs; Humans; Methylurea Compounds; Motor Activity; Neurokinin B; Peptide Fragments; Piperidines; Rabbits; Rats; Receptors, Neurokinin-3; Substance P

2002
Neurokinin B induces oedema formation in mouse lung via tachykinin receptor-independent mechanisms.
    The Journal of physiology, 2002, Sep-15, Volume: 543, Issue:Pt 3

    Topics: Animals; Antipsychotic Agents; Benzamides; Cyclooxygenase Inhibitors; Edema; Enzyme Inhibitors; Extravascular Lung Water; Female; Indomethacin; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Piperidines; Plasma; Pulmonary Edema; Receptors, Neurokinin-1; Substance P

2002
The mechanisms for tachykinin-induced contractions of the rabbit corpus cavernosum.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Animals; Benzamides; Calcium; Dose-Response Relationship, Drug; Glycopeptides; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Penis; Permeability; Piperidines; Quinuclidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Type C Phospholipases

2002
Diencephalic neurons producing melanin-concentrating hormone are influenced by local and multiple extra-hypothalamic tachykininergic projections through the neurokinin 3 receptor.
    Neuroscience, 2003, Volume: 119, Issue:4

    Topics: Animals; Brain; Colchicine; Feeding Behavior; Hypothalamic Hormones; Hypothalamus; Interneurons; Male; Melanins; Neural Pathways; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Organ Culture Techniques; Peptide Fragments; Piperidines; Pituitary Hormones; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-3; RNA, Messenger; Sexual Behavior; Substance P; Tachykinins

2003
Leukocyte recruitment to peritoneal cavity of rats following formalin injection: role of tachykinin receptors.
    Journal of pharmacological sciences, 2004, Volume: 94, Issue:4

    Topics: Animals; Benzamides; Cell Movement; Dose-Response Relationship, Drug; Female; Formaldehyde; Injections, Intraperitoneal; Leukocytes; Models, Biological; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peritoneal Cavity; Peritoneal Lavage; Piperidines; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Time Factors

2004
Involvement of enhanced neurokinin NK3 receptor expression in the severe asthma guinea pig model.
    European journal of pharmacology, 2004, Sep-13, Volume: 498, Issue:1-3

    Topics: Animals; Asthma; Benzamides; Binding, Competitive; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Bronchoconstrictor Agents; Disease Models, Animal; Dose-Response Relationship, Drug; Eosinophils; Guinea Pigs; Lung; Male; Methacholine Chloride; Neurokinin B; Ovalbumin; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tritium

2004
Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition.
    Molecular pharmacology, 2007, Volume: 71, Issue:3

    Topics: Animals; Binding, Competitive; Calcium; CHO Cells; Cricetinae; Cricetulus; Kinetics; Neurokinin B; Piperidines; Quinolines; Receptors, Neurokinin-3

2007
A role for tachykinins in the regulation of human sperm motility.
    Human reproduction (Oxford, England), 2007, Volume: 22, Issue:6

    Topics: Benzamides; Humans; Immunohistochemistry; Male; Neurokinin A; Neurokinin B; Piperidines; Quinuclidines; Receptors, Tachykinin; Sperm Motility; Spermatozoa; Substance P; Tachykinins

2007
Autocrine regulation of human sperm motility by tachykinins.
    Reproductive biology and endocrinology : RB&E, 2010, Aug-26, Volume: 8

    Topics: Adolescent; Adult; Antidepressive Agents; Antipsychotic Agents; Autocrine Communication; Benzamides; Drug Evaluation, Preclinical; Humans; Male; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; RNA, Messenger; Sperm Motility; Spermatozoa; Tachykinins; Young Adult

2010
Neurokinin2-R in medial septum regulate hippocampal and amygdalar ACh release induced by intraseptal application of neurokinins A and B.
    Hippocampus, 2012, Volume: 22, Issue:5

    Topics: Acetylcholine; Amygdala; Analysis of Variance; Animals; Benzamides; Cholinergic Neurons; Frontal Lobe; Hippocampus; Male; Memory; Neurokinin A; Neurokinin B; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Septal Nuclei; Septum of Brain

2012
Neuromodulation mediated by the tachykinin NK3-receptor agonist [MePhe7]-neurokinin B in the isolated perfused lung of nonsensitized nonchallenged and ovalbumin-sensitized and -challenged guinea pig.
    Experimental lung research, 2012, Volume: 38, Issue:5

    Topics: Animals; Bronchoconstriction; Electrodes; Guinea Pigs; Lung; Male; Neurokinin A; Neurokinin B; Neurotransmitter Agents; Ovalbumin; Piperidines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Vagus Nerve; Vagus Nerve Stimulation

2012
Neurokinin B activates arcuate kisspeptin neurons through multiple tachykinin receptors in the male mouse.
    Endocrinology, 2013, Volume: 154, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Arcuate Nucleus of Hypothalamus; Dynorphins; Green Fluorescent Proteins; Kisspeptins; Male; Membrane Potentials; Mice; Mice, Transgenic; Neurokinin B; Neurons; Oligopeptides; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Opioid, kappa; Receptors, Tachykinin; Substance P

2013
A role for Tac2, NkB, and Nk3 receptor in normal and dysregulated fear memory consolidation.
    Neuron, 2014, Jul-16, Volume: 83, Issue:2

    Topics: Amygdala; Animals; Conditioning, Classical; Fear; Male; Memory; Mice; Neurokinin B; Neurons; Piperidines; Protein Precursors; Receptors, Neurokinin-3; Tachykinins

2014
Interaction of endokinin A/B and (Mpa(6))-γ2-MSH-6-12 in pain regulation in mice.
    Neuropeptides, 2015, Volume: 53

    Topics: Animals; Dose-Response Relationship, Drug; gamma-MSH; Hyperalgesia; Injections, Intraventricular; Injections, Spinal; Male; Mice; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Pain; Pain Measurement; Piperidines; Receptors, Neurokinin-3; Tropanes

2015