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neurokinin a (4-10), nle(10)- and substance p

neurokinin a (4-10), nle(10)- has been researched along with substance p in 13 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), nle(10)-)
Trials
(neurokinin a (4-10), nle(10)-)
Recent Studies (post-2010)
(neurokinin a (4-10), nle(10)-)
Studies
(substance p)
Trials
(substance p)
Recent Studies (post-2010) (substance p)
210317,2892772,010

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), nle(10)- (IC50)substance p (IC50)
Substance-P receptorRattus norvegicus (Norway rat)0.0005
Substance-K receptorRattus norvegicus (Norway rat)0.2
Substance-K receptorHomo sapiens (human)0.2455
Substance-P receptorHomo sapiens (human)0.0011
Neuromedin-K receptorHomo sapiens (human)0.125
Substance-K receptorMesocricetus auratus (golden hamster)0.148

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (92.31)18.2507
2000's1 (7.69)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, FY; Lee, SD; Wang, PS; Yeh, GH1
Wong, TC; Zhang, M1
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Advenier, C; Gully, D; Martin, CA; Naline, E1
Daniel, EE; Fox-Threlkeld, JE; Watson, EG1
Killingsworth, CR; Shore, SA1
Advenier, C; Bétoin, F; Eschalier, A; Fardin, V; Lavarenne, J; Wilcox, G1
Alberch, J; Arenas, E; Marsal, J; Pérez-Navarro, E1
Håkanson, R; Wang, ZY1
Advenier, C; Crambes, O; Girard, V; Lundberg, JM; Malbezin, M; Malmström, RE; Naline, E1
Brelière, JC; Emonds-Alt, X; Le Fur, G; Vilain, P1
Advenier, C; Canet, E; Félétou, M; Girard, V1
Coupar, IM; Kerr, KP; Thai, B1

Other Studies

13 other study(ies) available for neurokinin a (4-10), nle(10)- and substance p

ArticleYear
The motor actions of natural neurokinins and their specific agonists on the gastrointestinal tract of the rat.
    The Chinese journal of physiology, 1992, Volume: 35, Issue:4

    Topics: Animals; Charcoal; Gastrointestinal Motility; Injections, Intraperitoneal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pilot Projects; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins

1992
Solution conformation study of substance P methyl ester and [Nle10]-neurokinin A (4-10) by NMR spectroscopy.
    Biopolymers, 1993, Volume: 33, Issue:12

    Topics: Amino Acid Sequence; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Protein Conformation; Solutions; Substance P

1993
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Neurotensin modulates cholinergic and noncholinergic neurotransmission in guinea-pig main bronchi in vitro.
    Neuropeptides, 1994, Volume: 26, Issue:3

    Topics: Acetylcholine; Animals; Autonomic Nervous System; Bronchi; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Neurotensin; Parasympathetic Nervous System; Peptide Fragments; Pyrazoles; Quinolines; Receptors, Neurotensin; Substance P; Synaptic Transmission

1994
Tachykinin-mediated increase in motility acts independently of vasoactive intestinal polypeptide release in the canine ileum.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:2

    Topics: Animals; Dogs; Female; Gastrointestinal Motility; Ileum; Male; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasoactive Intestinal Peptide

1994
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
In vitro and in vivo evidence for a tachykinin NK1 receptor antagonist effect of vapreotide, an analgesic cyclic analog of somatostatin.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Acetylcholine; Analgesics; Animals; Binding, Competitive; Brain; Bronchi; Capillary Permeability; Duodenum; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Injections, Spinal; Male; Mice; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Somatostatin; Substance P

1995
Selective resistance of tachykinin-responsive cholinergic neurons in the quinolinic acid lesioned neostriatum.
    Brain research, 1993, Feb-19, Volume: 603, Issue:2

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Microinjections; Neostriatum; Neurokinin A; Neurons; Peptide Fragments; Potassium Chloride; Quinolinic Acid; Rats; Rats, Sprague-Dawley; Substance P

1993
The rabbit iris sphincter contains NK1 and NK3 but not NK2 receptors: a study with selective agonists and antagonists.
    Regulatory peptides, 1993, Apr-08, Volume: 44, Issue:3

    Topics: Animals; Dactinomycin; Female; Iris; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Rabbits; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P

1993
Pre- and postjunctional inhibitory effects of fenspiride on guinea-pig bronchi.
    The European respiratory journal, 1997, Volume: 10, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchi; Bronchodilator Agents; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indomethacin; Lung; Nerve Fibers; Neurokinin A; Neuropeptides; Peptide Fragments; Propranolol; Spiro Compounds; Substance P

1997
Tachykinin-induced contractions of the guinea pig ileum longitudinal smooth muscle: tonic and phasic muscular activities.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Substance P; Tachykinins

1997
Effects of tachykinins and capsaicin on the mechanical and electrical activity of the guinea-pig isolated trachea.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Potassium Channel Blockers; Quinuclidines; Receptors, Neurokinin-2; Substance P; Tachykinins; Tetraethylammonium; Trachea

1997
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000