Page last updated: 2024-09-05

neurokinin a (4-10), nle(10)- and substance p, sar(9)-met(o2)(11)-

neurokinin a (4-10), nle(10)- has been researched along with substance p, sar(9)-met(o2)(11)- in 10 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), nle(10)-)
Trials
(neurokinin a (4-10), nle(10)-)
Recent Studies (post-2010)
(neurokinin a (4-10), nle(10)-)
Studies
(substance p, sar(9)-met(o2)(11)-)
Trials
(substance p, sar(9)-met(o2)(11)-)
Recent Studies (post-2010) (substance p, sar(9)-met(o2)(11)-)
210315106

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), nle(10)- (IC50)substance p, sar(9)-met(o2)(11)- (IC50)
Substance-P receptorHomo sapiens (human)0.0006

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (60.00)18.2507
2000's1 (10.00)29.6817
2010's3 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Daniel, EE; Fox-Threlkeld, JE; Watson, EG1
Killingsworth, CR; Shore, SA1
Alberch, J; Arenas, E; Marsal, J; Pérez-Navarro, E1
Håkanson, R; Wang, ZY1
Brelière, JC; Emonds-Alt, X; Le Fur, G; Vilain, P1
Coupar, IM; Kerr, KP; Thai, B1

Other Studies

10 other study(ies) available for neurokinin a (4-10), nle(10)- and substance p, sar(9)-met(o2)(11)-

ArticleYear
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Tachykinin-mediated increase in motility acts independently of vasoactive intestinal polypeptide release in the canine ileum.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:2

    Topics: Animals; Dogs; Female; Gastrointestinal Motility; Ileum; Male; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasoactive Intestinal Peptide

1994
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
Selective resistance of tachykinin-responsive cholinergic neurons in the quinolinic acid lesioned neostriatum.
    Brain research, 1993, Feb-19, Volume: 603, Issue:2

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Microinjections; Neostriatum; Neurokinin A; Neurons; Peptide Fragments; Potassium Chloride; Quinolinic Acid; Rats; Rats, Sprague-Dawley; Substance P

1993
The rabbit iris sphincter contains NK1 and NK3 but not NK2 receptors: a study with selective agonists and antagonists.
    Regulatory peptides, 1993, Apr-08, Volume: 44, Issue:3

    Topics: Animals; Dactinomycin; Female; Iris; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Rabbits; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P

1993
Tachykinin-induced contractions of the guinea pig ileum longitudinal smooth muscle: tonic and phasic muscular activities.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Substance P; Tachykinins

1997
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000