Page last updated: 2024-09-05

neurokinin a (4-10), nle(10)- and sr 48968

neurokinin a (4-10), nle(10)- has been researched along with sr 48968 in 5 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), nle(10)-)
Trials
(neurokinin a (4-10), nle(10)-)
Recent Studies (post-2010)
(neurokinin a (4-10), nle(10)-)
Studies
(sr 48968)
Trials
(sr 48968)
Recent Studies (post-2010) (sr 48968)
2103338213

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), nle(10)- (IC50)sr 48968 (IC50)
Substance-K receptorHomo sapiens (human)0.0001
Substance-P receptorHomo sapiens (human)0.8

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Killingsworth, CR; Shore, SA1
Brelière, JC; Emonds-Alt, X; Gueudet, C; Le Fur, G; Poncelet, M; Soubrié, P1
Advenier, C; Canet, E; Félétou, M; Girard, V1
Coupar, IM; Kerr, KP; Thai, B1

Other Studies

5 other study(ies) available for neurokinin a (4-10), nle(10)- and sr 48968

ArticleYear
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Tachykinin receptors mediating contraction of guinea pig lung strips.
    Regulatory peptides, 1995, May-30, Volume: 57, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; Biphenyl Compounds; Dipeptides; Guinea Pigs; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Trachea

1995
Turning behavior induced in mice by a neurokinin A receptor agonist: stereoselective blockade by SR 48968, a non-peptide receptor antagonist.
    Neuroscience letters, 1993, Jan-04, Volume: 149, Issue:1

    Topics: Animals; Behavior, Animal; Benzamides; Corpus Striatum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Injections; Injections, Intraperitoneal; Mice; Mice, Inbred Strains; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spiperone; Stereoisomerism; Stereotyped Behavior

1993
Effects of tachykinins and capsaicin on the mechanical and electrical activity of the guinea-pig isolated trachea.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Potassium Channel Blockers; Quinuclidines; Receptors, Neurokinin-2; Substance P; Tachykinins; Tetraethylammonium; Trachea

1997
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000