Page last updated: 2024-09-05

neurokinin a (4-10), nle(10)- and somatostatin

neurokinin a (4-10), nle(10)- has been researched along with somatostatin in 3 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), nle(10)-)
Trials
(neurokinin a (4-10), nle(10)-)
Recent Studies (post-2010)
(neurokinin a (4-10), nle(10)-)
Studies
(somatostatin)
Trials
(somatostatin)
Recent Studies (post-2010) (somatostatin)
210329011

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), nle(10)- (IC50)somatostatin (IC50)
Somatostatin receptor type 5Mus musculus (house mouse)0.0001
Protein-lysine 6-oxidaseHomo sapiens (human)0.01
Somatostatin receptor type 1Homo sapiens (human)0.0012
Somatostatin receptor type 1Mus musculus (house mouse)0.0001
Somatostatin receptor type 2Homo sapiens (human)0.0007
Somatostatin receptor type 2Mus musculus (house mouse)0.0002
Somatostatin receptor type 3Mus musculus (house mouse)0.0001
Somatostatin receptor type 5Rattus norvegicus (Norway rat)0.0009
Somatostatin receptor type 4Homo sapiens (human)0.0012
Somatostatin receptor type 3Homo sapiens (human)0.002
Delta-type opioid receptorRattus norvegicus (Norway rat)2
Mu-type opioid receptorRattus norvegicus (Norway rat)0.006
Somatostatin receptor type 5Homo sapiens (human)0.003
Somatostatin receptor type 4 Mus musculus (house mouse)0.0001

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1

Other Studies

3 other study(ies) available for neurokinin a (4-10), nle(10)- and somatostatin

ArticleYear
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017