Page last updated: 2024-09-03

neurokinin a (4-10), beta-ala(8)- and neurokinin a

neurokinin a (4-10), beta-ala(8)- has been researched along with neurokinin a in 70 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), beta-ala(8)-)
Trials
(neurokinin a (4-10), beta-ala(8)-)
Recent Studies (post-2010)
(neurokinin a (4-10), beta-ala(8)-)
Studies
(neurokinin a)
Trials
(neurokinin a)
Recent Studies (post-2010) (neurokinin a)
71021,7653491

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), beta-ala(8)- (IC50)neurokinin a (IC50)
Substance-K receptorHomo sapiens (human)0.0017
Neuromedin-K receptorHomo sapiens (human)0.045
Substance-K receptorMesocricetus auratus (golden hamster)0.001

Research

Studies (70)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's43 (61.43)18.2507
2000's25 (35.71)29.6817
2010's2 (2.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brunelleschi, S; Ceni, E; Fantozzi, R; Giotti, A; Parenti, A1
Maggi, CA; Motta, A; Rovero, P; Saviano, G; Temussi, PA1
Maggi, CA; Patacchini, R; Quartara, L; Rovero, P; Santicioli, P1
Kodner, A; Mayer, EA; Regoli, M; Sachs, G; Sun, XP; Supplisson, S1
Abelli, L; Giachetti, A; Giuliani, S; Maggi, CA; Santicioli, P1
Abelli, L; Ballati, L; Giachetti, A; Giuliani, S; Maggi, CA; Manzini, S; Meli, A; Rovero, P1
Giuliani, S; Maggi, CA; Meini, S; Patacchini, R1
Barnes, PJ; Belvisi, MG; Maggi, CA; Patacchini, R1
Baranauskas, G; Fisher, ND; Nistri, A1
Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Giachetti, A; Giuliani, S; Maggi, CA; Meini, S; Patacchini, R; Potier, E; Quartara, L; Sisto, A1
Brugger, F; Evans, RH; Lepre, M; Olpe, HR1
Bowery, BJ; Hill, RG; Seabrook, GR1
Ballati, L; Boni, P; Evangelista, S1
Giachetti, A; Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Medeiros, MD; Turner, AJ1
Mak, JC; Meini, S; Rogers, DF; Rohde, JA1
Barnes, PJ; Hirayama, Y; Lei, YH; Rogers, DF1
Boden, PR; Norris, SK; Woodruff, GN1
Giachetti, A; Giuliani, S; Maggi, CA; Patacchini, R1
Bartho, L; Giuliani, S; Maggi, CA; Santicioli, P1
Humpel, C; Saria, A1
McKee, KT; Metters, KM; Millar, L; Rodger, IW1
Evangelista, S; Maggi, CA; Tramontana, M1
Basilisco, G; Phillips, SF1
Astolfi, M; Giachetti, A; Maggi, CA; Manzini, S; Meini, S; Treggiari, S1
Brideau, C; Chan, CC; Guevremont, D; Hale, JJ; MacCoss, M; Rodger, IW; Tousignant, C1
Astolfi, M; Goso, C; Manzini, S; Parlani, M1
Brunelleschi, S; Fantozzi, R; Guidotto, S; Tonso, E; Viano, I1
Cavero, I; Floch, A; Thiry, C1
Albera, C; Brunelleschi, S; Fantozzi, R; Ghio, P; Guidotto, S; Pozzi, E; Viano, I1
Fox, AJ; Naeem, S; Patel, IA; Urbán, L; Walpole, C1
Couture, R; Sgambato, V; Toma, N1
Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Baamonde, A; Hidalgo, A; Menéndez, L1
Evangelista, S; Giachetti, A; Manzini, S; Paoli, S1
Giuliani, S; Lazzeri, M; Maggi, CA; Patacchini, R; Quartara, L; Turini, A1
Bordin, G; Brunelleschi, S; Colangelo, D; Viano, I1
Criscuoli, M; Giuliani, S; Lecci, A; Lippi, A; Maggi, CA; Patacchini, R; Santicioli, P; Tramontana, M1
Ardell, JL; Armour, JA; Hoover, DB; Thompson, GW1
Petersen, M; Schaible, HG; Segond von Banchet, G1
Barnes, PJ; Elzinga, CR; Katsunuma, T; Mak, JC; Roffel, AF; Zaagsma, J1
Aggio, A; Onori, L; Taddei, G; Tonini, M1
Bialecki, R; Caccese, R; Graham, A1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L1
Albera, C; Brunelleschi, S; Gagliardi, L; Ghio, P; Lavagno, L; Nicali, R; Pozzi, E; Viano, I1
Catalioto, RM; Lecci, A; Maggi, CA; Tramontana, M1
Crane, LH; Hamlin, GP; Nimmo, AJ; Williams, MJ1
D'Agostino, G; Erbelding, D; Kilbinger, H1
Anderson, GP; Ball, HA; Bertrand, C; Gerspacher, M; Hauser, K; Mah, R; Subramanian, N; von Sprecher, A1
Cruwys, SC; Hood, VC; Kidd, BL; Urban, L1
Krysiak, PS; Preiksaitis, HG1
Cox, HM; Maggi, CA; Patacchini, R; Ståhl, S; Tough, IR1
Bordin, G; Brunelleschi, S; Colangelo, D; Lavagno, L; Viano, I1
Carini, F; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Bringas, A; Choppin, A; Dillon, MP; Groke, G; Stepan, G1
Hanesch, U; Nitz, C; Pawlak, M; Schmidt, RF1
Ogier, R; Raggenbass, M1
Smid, SD; Smith, AS1
Couture, R; Deschamps, K1
Juszczak, M1
Altamura, M; Catalani, C; Catalioto, RM; Cialdai, C; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Patacchini, R; Tramontana, M; Valenti, C1
de Groat, WC; Sculptoreanu, A1
Amato, A; Mulè, F; Serio, R1
Boczek-Leszczyk, E; Juszczak, M; Stempniak, B1
Emala, CW; Gallos, G; Goubaeva, F; Mizuta, F; Mizuta, K; Panettieri, RA; Xu, D; Yang, J; Zhu, D1
Aura Kullmann, F; de Groat, WC; Sculptoreanu, A1
Emala, CW; Gallos, G; Gleason, NR; Pak, SW; Sonett, JR; Yang, J; Zhang, Y1
Ikeda, M; Kojima, S; Tohei, A1
Anzai, N; Kojima, S; Tohei, A1

Other Studies

70 other study(ies) available for neurokinin a (4-10), beta-ala(8)- and neurokinin a

ArticleYear
Enhanced responsiveness of ovalbumin-sensitized guinea-pig alveolar macrophages to tachykinins.
    British journal of pharmacology, 1992, Volume: 107, Issue:4

    Topics: Animals; Dinoprostone; Dose-Response Relationship, Drug; Glucuronidase; Guinea Pigs; Macrophages, Alveolar; Male; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin A; Ovalbumin; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Superoxides; Tachykinins; Thromboxane B2

1992
Conformation-activity relationship of tachykinin neurokinin A (4-10) and of some [Xaa8] analogues.
    Biochemistry, 1991, Oct-22, Volume: 30, Issue:42

    Topics: Amino Acid Sequence; Animals; Dimethyl Sulfoxide; Guinea Pigs; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Protein Conformation; Rabbits; Structure-Activity Relationship

1991
Tachykinin receptors in the guinea-pig isolated bronchi.
    European journal of pharmacology, 1991, May-17, Volume: 197, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Bronchi; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Neurokinin A; Oligopeptides; Peptide Fragments; Phenoxybenzamine; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins

1991
Neurokinin receptor-mediated regulation of [Ca]i and Ca-sensitive ion channels in mammalian colonic muscle.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Calcimycin; Calcium; Calcium Channels; Cells, Cultured; Colon; Membrane Potentials; Muscle, Smooth; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P

1991
Facilitation of reflex micturition by intravesical administration of [beta Ala8]-neurokinin A (4-10), a selective NK-2 tachykinin receptor agonist.
    The Journal of urology, 1991, Volume: 145, Issue:1

    Topics: Administration, Intravesical; Animals; Guinea Pigs; Male; Muscle Contraction; Neurokinin A; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Reflex; Stimulation, Chemical; Tachykinins; Urinary Bladder; Urination

1991
In vivo pharmacology of [beta Ala8]neurokinin A-(4-10), a selective NK-2 tachykinin receptor agonist.
    European journal of pharmacology, 1990, Feb-20, Volume: 177, Issue:1-2

    Topics: Anesthesia; Animals; Blood Pressure; Blood Proteins; Bronchi; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Salivation; Urinary Bladder

1990
Effect of longitudinal muscle-myenteric plexus removal and indomethacin on the response to tachykinin NK-2 and NK-3 receptor agonists in the circular muscle of the guinea-pig ileum.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:1

    Topics: Animals; Atropine; Calcium Channel Blockers; Guinea Pigs; Ileum; In Vitro Techniques; Indomethacin; Male; Muscle, Smooth; Myenteric Plexus; Neurokinin A; omega-Conotoxin GVIA; Peptide Fragments; Peptides; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tetrodotoxin

1994
Facilitatory effects of selective agonists for tachykinin receptors on cholinergic neurotransmission: evidence for species differences.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adult; Amino Acid Sequence; Animals; Bronchi; Capsaicin; Electric Stimulation; Guinea Pigs; Humans; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Parasympathetic Nervous System; Peptide Fragments; Rabbits; Receptors, Tachykinin; Substance P; Sulfones; Synaptic Transmission; Tachykinins

1994
Multiple types of tachykinin receptor mediate a slow excitation of rat spinal motoneurones in vitro.
    Neuroscience letters, 1994, Jan-03, Volume: 165, Issue:1-2

    Topics: Animals; Animals, Newborn; Female; In Vitro Techniques; Male; Membrane Potentials; Motor Neurons; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tetrodotoxin

1994
Different Ca2+ influx pathways mediate tachykinin receptor-induced contraction in circular muscle of guinea-pig colon.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: Action Potentials; Animals; Calcium Channels; Colon; Electrophysiology; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Sulfones

1994
Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones

1994
Physiological and pharmacological characterization of the spinal tachykinin NK2 receptor.
    European journal of pharmacology, 1994, Jun-02, Volume: 258, Issue:1-2

    Topics: Animals; Animals, Newborn; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Interactions; Ganglia, Spinal; Gerbillinae; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Oligopeptides; Peptide Fragments; Rats; Receptors, Neurokinin-2; Spinal Cord; Substance P; Tetrodotoxin

1994
Pharmacology of tachykinin receptors on neurones in the ventral tegmental area of rat brain slices.
    European journal of pharmacology, 1995, Jan-24, Volume: 273, Issue:1-2

    Topics: Action Potentials; Animals; Electrophysiology; In Vitro Techniques; Microelectrodes; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Ventral Tegmental Area

1995
Tachykinin NK1 and NK2 receptors mediate the non-cholinergic bronchospastic response to capsaicin and vagal stimulation in guinea-pigs.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:1

    Topics: Animals; Biphenyl Compounds; Bronchial Spasm; Capsaicin; Electric Stimulation; Guinea Pigs; Insufflation; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vagus Nerve

1995
Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic non-cholinergic excitation and contraction in the circular muscle of guinea-pig duodenum.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Action Potentials; Adenosine Diphosphate; Animals; Apamin; Arginine; Atropine; Dose-Response Relationship, Drug; Duodenum; Electric Stimulation; Guanethidine; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Nifedipine; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Suramin; Thionucleotides

1995
Metabolic stability of some tachykinin analogues to cell-surface peptidases: roles for endopeptidase-24.11 and aminopeptidase N.
    Peptides, 1995, Volume: 16, Issue:3

    Topics: Amino Acid Sequence; Animals; CD13 Antigens; Cell Membrane; Evaluation Studies as Topic; Hydrolysis; Kidney; Microvilli; Molecular Sequence Data; Neprilysin; Neurokinin A; Peptide Fragments; Swine; Tachykinins

1995
Tachykinin control of ferret airways: mucus secretion, bronchoconstriction and receptor mapping.
    Neuropeptides, 1993, Volume: 24, Issue:2

    Topics: Animals; Bronchoconstriction; Capsaicin; Ferrets; Male; Methacholine Chloride; Mucus; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Reproducibility of Results; Stimulation, Chemical; Substance P; Tachykinins; Trachea

1993
Effects of two novel tachykinin antagonists, FK224 and FK888, on neurogenic airway plasma exudation, bronchoconstriction and systemic hypotension in guinea-pigs in vivo.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Blood Pressure; Bronchoconstriction; Capsaicin; Dipeptides; Electric Stimulation; Evans Blue; Exudates and Transudates; Guinea Pigs; Hypotension; Indoles; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Platelet Activating Factor; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Respiratory Mechanics; Smoking; Substance P; Vagus Nerve

1993
Agonists selective for tachykinin NK1 and NK3 receptors excite subpopulations of neurons in the rat medial habenula nucleus in vitro.
    European journal of pharmacology, 1993, Apr-06, Volume: 234, Issue:2-3

    Topics: Animals; Electrophysiology; Extracellular Space; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins; Thalamic Nuclei

1993
In vivo and in vitro activity of SR 48,968, a non-peptide tachykinin NK-2 receptor antagonist.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Blood Pressure; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Rats; Receptors, Neurokinin-2; Saliva; Substance P; Sulfones; Urinary Bladder

1993
Tachykinin NK-1 and NK-2 receptors in the circular muscle of the guinea-pig proximal colon.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Benzamides; Biphenyl Compounds; Colon; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones; Tetrodotoxin

1993
Intranigral injection of selective neurokinin-1 and neurokinin-3 but not neurokinin-2 receptor agonists biphasically modulate striatal dopamine metabolism but not striatal preprotachykinin-A mRNA in the rat.
    Neuroscience letters, 1993, Jul-23, Volume: 157, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Dopamine; Female; Gene Expression Regulation; Injections; Neurokinin A; Neurokinin B; Peptide Fragments; Protein Precursors; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Substantia Nigra; Tachykinins

1993
Identification of both NK1 and NK2 receptors in guinea-pig airways.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Animals; Benzamides; Chromatography, High Pressure Liquid; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Lung; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory System; Substance P; Trachea

1993
Spasmolytic effect of the NK2-receptor-selective antagonist MEN 10,627 in rat small intestine.
    Japanese journal of pharmacology, 1994, Volume: 65, Issue:3

    Topics: Amino Acid Sequence; Animals; Carbachol; Dose-Response Relationship, Drug; Gastric Emptying; Gastrointestinal Transit; Injections, Intravenous; Intestine, Small; Male; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2

1994
A selective NK-2 antagonist blocks the increase of canine colonic tone and ileal contractions induced by the NK-2 selective receptor agonist, [beta Ala8] neurokinin A-(4-10).
    Alimentary pharmacology & therapeutics, 1994, Volume: 8, Issue:5

    Topics: Animals; Benzamides; Colon; Dogs; Female; Gastrointestinal Motility; Ileum; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-2

1994
Characterization of the tachykinin NK2 receptor in the human bronchus: influence of amastatin-sensitive metabolic pathways.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: Amino Acid Sequence; Anti-Bacterial Agents; Bronchi; Bronchial Spasm; Female; Humans; In Vitro Techniques; Male; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Peptides; Peptides, Cyclic; Receptors, Neurokinin-2; Tachykinins

1994
NK2 receptors mediate plasma extravasation in guinea-pig lower airways.
    British journal of pharmacology, 1993, Volume: 108, Issue:2

    Topics: Animals; Benzamides; Blood Proteins; Bronchi; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Iodine Radioisotopes; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter

1993
[3H][beta-Ala8]neurokinin A-(4-10): a novel, selective radioligand for the tachykinin NK2 receptor.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Animals; Benzamides; Binding, Competitive; Cricetinae; In Vitro Techniques; Kinetics; Ligands; Male; Membranes; Mesocricetus; Muscle Contraction; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Urinary Bladder

1995
Modulation by protein kinase C of the enhanced responsiveness to tachykinins in ovalbumin-sensitized guinea pig alveolar macrophages.
    Neuropeptides, 1996, Volume: 30, Issue:3

    Topics: Animals; Bordetella pertussis; Cytochrome c Group; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Guinea Pigs; Immunization; Macrophages, Alveolar; Male; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin A; Ovalbumin; Peptide Fragments; Protein Kinase C; Receptors, Tachykinin; Staurosporine; Substance P; Superoxides; Tachykinins; Tetradecanoylphorbol Acetate

1996
Pharmacological evidence that NK-2 tachykinin receptors mediate hypotension in the guinea pig but not in the rat.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Animals; Benzamides; Blood Pressure; Guinea Pigs; Hypotension; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1996
Tachykinin activation of human alveolar macrophages in tobacco smoke and sarcoidosis: a phenotypical and functional study.
    Neuropeptides, 1996, Volume: 30, Issue:5

    Topics: Adult; Bronchoalveolar Lavage Fluid; Female; Humans; Immunophenotyping; Macrophage Activation; Macrophages, Alveolar; Male; Middle Aged; Neurokinin A; Peptide Fragments; Peptidyl-Dipeptidase A; Receptors, Neurokinin-2; Respiratory Burst; Sarcoidosis, Pulmonary; Smoking; Substance P; Superoxides; Tachykinins

1996
Receptors mediating tachykinin-evoked depolarisations of neurons in the neonatal rat spinal cord.
    Acta biologica Hungarica, 1996, Volume: 47, Issue:1-4

    Topics: Animals; Animals, Newborn; Biphenyl Compounds; Evoked Potentials; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins

1996
Effect of angiotensin II on a spinal nociceptive reflex in the rat: receptor and mechanism of action.
    Life sciences, 1997, Volume: 61, Issue:5

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Interactions; Hot Temperature; Imidazoles; Injections, Spinal; Losartan; Male; Naloxone; Neurokinin A; Neurokinin B; Nociceptors; Peptide Fragments; Rats; Rats, Sprague-Dawley; Reflex; Spinal Cord; Substance P; Tetrazoles

1997
Role of tachykinin NK1 and NK2 receptors on colonic motility in anesthetized rats: effect of agonists.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:6

    Topics: Anesthesia; Animals; Benzamides; Colon; Gastrointestinal Motility; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1997
Spinal calmodulin inhibitors reduce N-methyl-D-aspartate- and septide-induced nociceptive behavior.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Enzyme Inhibitors; Imidazoles; Injections, Intraventricular; Male; N-Methylaspartate; Neurokinin A; Pain; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P; Sulfonamides

1997
Involvement of tachykinin NK1 receptors in plasma protein extravasation induced by tachykinins in the guinea pig upper airways.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Animals; Antigens; Blood Proteins; Capsaicin; Dextrans; Dipeptides; Extravasation of Diagnostic and Therapeutic Materials; Fluorescein-5-isothiocyanate; Glycopeptides; Guinea Pigs; Indoles; Male; Nasal Mucosa; Neurokinin A; Neurokinin-1 Receptor Antagonists; Olfactory Receptor Neurons; Peptide Fragments; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Rhinitis; Substance P

1997
Effect of several bicyclic peptide and cyclic pseudopeptide tachykinin NK2 receptor antagonists in the human isolated ileum and colon.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Animals; Colon; Cricetinae; Drug Interactions; Female; Humans; Ileum; Male; Mesocricetus; Middle Aged; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Pulmonary Artery; Rabbits; Receptors, Neurokinin-2; Trachea

1997
Tachykinin receptors are present on human monocytes and play a role in rheumatoid arthritis.
    Journal of chemotherapy (Florence, Italy), 1998, Volume: 10, Issue:2

    Topics: Aged; Arthritis, Rheumatoid; Cell Separation; Female; Humans; Male; Middle Aged; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Superoxides; Tetradecanoylphorbol Acetate

1998
Characterization of the antibronchoconstrictor activity of MEN 11420, a tachykinin NK2 receptor antagonist, in guinea-pigs.
    European journal of pharmacology, 1998, Jul-10, Volume: 352, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Atropine; Benzamides; Bronchi; Bronchoconstriction; Bronchodilator Agents; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1998
Canine intrinsic cardiac neurons involved in cardiac regulation possess NK1, NK2, and NK3 receptors.
    The American journal of physiology, 1998, Volume: 275, Issue:5

    Topics: Animals; Dogs; Heart; Myocardial Contraction; Neurokinin A; Neurons, Afferent; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1998
Expression of neurokinin-1 receptors on cultured dorsal root ganglion neurons from the adult rat.
    Neuroscience, 1999, Volume: 90, Issue:2

    Topics: Animals; Cells, Cultured; Ganglia, Spinal; Kinetics; Male; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Time Factors

1999
beta(2)-adrenoceptor agonist-induced upregulation of tachykinin NK(2) receptor expression and function in airway smooth muscle.
    American journal of respiratory cell and molecular biology, 1999, Volume: 21, Issue:3

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Animals; Anti-Inflammatory Agents; Cattle; Dexamethasone; Dose-Response Relationship, Drug; Fenoterol; Muscle, Smooth; Neurokinin A; Organ Culture Techniques; Peptide Fragments; Receptors, Neurokinin-2; RNA, Messenger; Time Factors; Trachea; Up-Regulation

1999
Contribution of NK(2) tachykinin receptors to propulsion in the rabbit distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 278, Issue:1

    Topics: Animals; Benzamides; Colon; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Rabbits; Receptors, Neurokinin-2; Time Factors

2000
Pharmacological characterization of mucin secretion from CHO-K1-hNK(1)R cells.
    Neuropeptides, 1999, Volume: 33, Issue:3

    Topics: Angiotensin II; Animals; Benzamides; Biological Transport; CHO Cells; Cricetinae; Endothelin-1; Glucosamine; Humans; Methacholine Chloride; Mucins; Muscarinic Agonists; Neurokinin A; Peptide Fragments; Phenylephrine; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Serotonin; Substance P; Transfection; Tritium; Vasoconstrictor Agents

1999
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium

2000
Tachykinin activation of human monocytes from patients with interstitial lung disease, healthy smokers or healthy volunteers.
    Neuropeptides, 2000, Volume: 34, Issue:1

    Topics: Adult; Aged; Cells, Cultured; Female; Humans; Lung Diseases, Interstitial; Male; Middle Aged; Monocytes; Neurokinin A; Peptide Fragments; Pulmonary Fibrosis; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Reference Values; Sarcoidosis; Smoking; Substance P; Superoxides; Tachykinins

2000
Role of prostanoids in the contraction induced by a tachykinin NK2 receptor agonist in the hamster urinary bladder.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 361, Issue:4

    Topics: Animals; Cricetinae; Cyclooxygenase Inhibitors; Dinoprostone; Imidazoles; In Vitro Techniques; Ketoprofen; Male; Mesocricetus; Muscle Contraction; Muscle, Smooth; Neurokinin A; Nifedipine; Peptide Fragments; Prostaglandins; Receptors, Neurokinin-2; Stereoisomerism; Urinary Bladder

2000
Hormonal variation of rat uterine contractile responsiveness to selective neurokinin receptor agonists.
    Biology of reproduction, 2000, Volume: 62, Issue:6

    Topics: Animals; Diestrus; Estrogens; Estrus; Female; Metestrus; Neurokinin A; Ovariectomy; Peptide Fragments; Piperidines; Proestrus; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Uterine Contraction

2000
Tachykinin NK(2) receptors facilitate acetylcholine release from guinea-pig isolated trachea.
    European journal of pharmacology, 2000, May-12, Volume: 396, Issue:1

    Topics: Acetylcholine; Animals; Benzamides; Capsaicin; Choline; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Trachea

2000
N-[(R,R)-(E)-1-(4-chloro-benzyl)-3-(2-oxo-azepan-3-ylcarbamoyl)-allyl]-N-methyl-3,5-bis-trifluoromethyl-benzamide: an orally active neurokinin NK1/NK2 antagonist.
    Bioorganic & medicinal chemistry letters, 2000, Jul-03, Volume: 10, Issue:13

    Topics: Administration, Oral; Animals; Anti-Asthmatic Agents; Aza Compounds; Benzamides; Bronchoconstriction; Drug Design; Guinea Pigs; Molecular Structure; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-2; Stereoisomerism; Substance P

2000
Differential role of neurokinin receptors in human lymphocyte and monocyte chemotaxis.
    Regulatory peptides, 2000, Dec-22, Volume: 96, Issue:1-2

    Topics: Chemotaxis, Leukocyte; Dose-Response Relationship, Drug; Humans; Indoles; Inflammation; Monocytes; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; T-Lymphocytes

2000
Tachykinins contribute to nerve-mediated contractions in the human esophagus.
    Gastroenterology, 2001, Volume: 120, Issue:1

    Topics: Atropine; Autonomic Nervous System; Benzamides; Dose-Response Relationship, Drug; Esophagus; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Parasympatholytics; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Substance P; Tachykinins

2001
Tachykinin NK(2) receptor mediates contraction and ion transport in rat colon by different mechanisms.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Colon; Indomethacin; Intestinal Mucosa; Ion Transport; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Rats; Rats, Wistar; Receptors, Neurokinin-2; Substance P

2001
Tachykinin activation of human monocytes from patients with rheumatoid arthritis: in vitro and ex-vivo effects of cyclosporin A.
    Neuropeptides, 2001, Volume: 35, Issue:2

    Topics: Arthritis, Rheumatoid; Carcinogens; Cells, Cultured; Cyclosporine; Humans; Immunosuppressive Agents; In Vitro Techniques; Monocytes; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Burst; Substance P; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha

2001
Tachykinin NK(2) receptors and enhancement of cholinergic transmission in the inflamed rat colon: an in vivo motility study.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Acetic Acid; Animals; Atropine; Cholinergic Fibers; Colon; Enzyme Inhibitors; Gastrointestinal Motility; Hexamethonium; Inflammation; Male; Muscarinic Antagonists; Neurokinin A; NG-Nitroarginine Methyl Ester; Peptide Fragments; Peptides, Cyclic; Rats; Rats, Wistar; Receptors, Neurokinin-2; Synaptic Transmission; Time Factors

2001
Effect of YM-44781, YM-44778 and YM-49598, novel tachykinin antagonists, in a drug-induced bladder contraction model.
    Pharmacology, 2002, Volume: 65, Issue:2

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dipeptides; Female; Indoles; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spiro Compounds; Transfection; Urinary Bladder

2002
The neurokinin-2 receptor is not involved in the sensitization of primary afferents of the rat knee joint.
    Neuroscience letters, 2002, Jun-28, Volume: 326, Issue:2

    Topics: Animals; Knee Joint; Male; Mechanoreceptors; Nerve Fibers; Neurokinin A; Neurons, Afferent; Pain; Peptide Fragments; Physical Stimulation; Rats; Rats, Wistar; Receptors, Neurokinin-2; Rotation; Substance P

2002
Action of tachykinins in the rat hippocampus: modulation of inhibitory synaptic transmission.
    The European journal of neuroscience, 2003, Volume: 17, Issue:12

    Topics: Animals; Animals, Newborn; Bicuculline; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuropeptides; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Time Factors

2003
Impaired capsaicin and neurokinin-evoked colonic motility in inflammatory bowel disease.
    Journal of gastroenterology and hepatology, 2005, Volume: 20, Issue:5

    Topics: Adult; Aged; Aged, 80 and over; Capsaicin; Case-Control Studies; Colon; Electric Stimulation; Gastrointestinal Motility; Humans; Inflammatory Bowel Diseases; Middle Aged; Neurokinin A; Neuromuscular Junction; Peptide Fragments; Stimulation, Chemical; Synaptic Transmission; Tissue Culture Techniques

2005
The ventral tegmental area as a putative target for tachykinins in cardiovascular regulation.
    British journal of pharmacology, 2005, Volume: 145, Issue:6

    Topics: Acetates; Adrenergic beta-Antagonists; Animals; Atenolol; Behavior, Animal; Benzamides; Benzazepines; Blood Pressure; Dopamine D2 Receptor Antagonists; Glutamic Acid; Heart Rate; Indoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Ventral Tegmental Area

2005
Vasopressin release from the rat hypothalamo-neurohypophysial system: effects of tachykinin NK-1 and NK-2 receptors agonists and antagonists.
    Neuro endocrinology letters, 2005, Volume: 26, Issue:4

    Topics: Animals; Hypothalamo-Hypophyseal System; In Vitro Techniques; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasopressins

2005
MEN15596, a novel nonpeptide tachykinin NK2 receptor antagonist.
    European journal of pharmacology, 2006, Nov-07, Volume: 549, Issue:1-3

    Topics: Aged; Animals; Binding, Competitive; Bronchoconstriction; Cell Membrane; CHO Cells; Colon; Cricetinae; Cricetulus; Dipeptides; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; In Vitro Techniques; Male; Mice; Middle Aged; Muscle Contraction; Neurokinin A; Peptide Fragments; Rabbits; Radioligand Assay; Rats; Rats, Wistar; Receptors, Neurokinin-2; Swine; Thiophenes; Vasoconstriction

2006
Neurokinins enhance excitability in capsaicin-responsive DRG neurons.
    Experimental neurology, 2007, Volume: 205, Issue:1

    Topics: Action Potentials; Animals; Capsaicin; Electric Stimulation; Enzyme Activation; Ganglia, Spinal; Intracellular Membranes; Male; Neurokinin A; Neurons, Afferent; Patch-Clamp Techniques; Peptide Fragments; Potassium Channel Blockers; Potassium Channels; Protein Kinase C; Protein Kinase Inhibitors; Rats; Receptors, Neurokinin-2; Signal Transduction; Substance P; Tachykinins

2007
Role for NK(1) and NK(2) receptors in the motor activity in mouse colon.
    European journal of pharmacology, 2007, Sep-10, Volume: 570, Issue:1-3

    Topics: Animals; Atropine; Colon; Electric Stimulation; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sodium Channel Blockers; Substance P; Tetrodotoxin

2007
Effect of melatonin on the vasopressin secretion as influenced by tachykinin NK-1 receptor agonist and antagonist: in vivo and in vitro studies.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2007, Volume: 58, Issue:4

    Topics: Analysis of Variance; Animals; Hypothalamo-Hypophyseal System; In Vitro Techniques; Male; Melatonin; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Peptide Fragments; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Vasopressins

2007
Expression and coupling of neurokinin receptor subtypes to inositol phosphate and calcium signaling pathways in human airway smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 294, Issue:3

    Topics: Boron Compounds; Calcium Signaling; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate; Muscle, Smooth; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Trachea

2008
Neurokinin 2 receptor-mediated activation of protein kinase C modulates capsaicin responses in DRG neurons from adult rats.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Age Factors; Animals; Calcium; Capsaicin; Carcinogens; Cells, Cultured; Ganglia, Spinal; Male; Neurokinin A; Neurokinin B; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Peptide Fragments; Phorbol Esters; Phosphorylation; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Sensory System Agents; Signal Transduction; Substance P; TRPV Cation Channels

2008
Activation of endogenous GABAA channels on airway smooth muscle potentiates isoproterenol-mediated relaxation.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 295, Issue:6

    Topics: Acetylcholine; Adenosine Triphosphatases; Adrenergic beta-Agonists; Animals; Bronchoconstriction; Dose-Response Relationship, Drug; GABA Antagonists; Guinea Pigs; Humans; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Neurokinin A; Organ Culture Techniques; Peptide Fragments; Peptides; Pyridazines; Receptors, GABA-A; Trachea; Vasodilator Agents

2008
Melatonin inhibits tachykinin NK₂ receptor-triggered 5-HT release from guinea pig isolated colonic mucosa.
    British journal of pharmacology, 2011, Volume: 162, Issue:5

    Topics: Animals; Colon; Guinea Pigs; Hydroxyindoleacetic Acid; In Vitro Techniques; Intestinal Mucosa; Melatonin; Neurokinin A; Peptide Fragments; Prazosin; Receptors, Melatonin; Receptors, Neurokinin-2; Serotonin; Tryptamines

2011
A role for endogenous peptide YY in tachykinin NK(2) receptor-triggered 5-HT release from guinea pig isolated colonic mucosa.
    British journal of pharmacology, 2012, Volume: 167, Issue:6

    Topics: Animals; Colon; Guinea Pigs; In Vitro Techniques; Intestinal Mucosa; Male; Neurokinin A; Peptide Fragments; Peptide YY; Receptors, Neurokinin-2; Serotonin

2012