Page last updated: 2024-09-03

neurokinin a (4-10), beta-ala(8)- and atropine

neurokinin a (4-10), beta-ala(8)- has been researched along with atropine in 6 studies

Compound Research Comparison

Studies
(neurokinin a (4-10), beta-ala(8)-)
Trials
(neurokinin a (4-10), beta-ala(8)-)
Recent Studies (post-2010)
(neurokinin a (4-10), beta-ala(8)-)
Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010) (atropine)
710226,7111,2591,697

Protein Interaction Comparison

ProteinTaxonomyneurokinin a (4-10), beta-ala(8)- (IC50)atropine (IC50)
cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)21.41
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.012
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0067
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.0007
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.0009
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.0015
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.0021
Alpha-1D adrenergic receptorHomo sapiens (human)1.354
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.012

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's3 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Giuliani, S; Maggi, CA; Meini, S; Patacchini, R1
Giachetti, A; Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Criscuoli, M; Giuliani, S; Lecci, A; Lippi, A; Maggi, CA; Patacchini, R; Santicioli, P; Tramontana, M1
Krysiak, PS; Preiksaitis, HG1
Carini, F; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
Amato, A; Mulè, F; Serio, R1

Other Studies

6 other study(ies) available for neurokinin a (4-10), beta-ala(8)- and atropine

ArticleYear
Effect of longitudinal muscle-myenteric plexus removal and indomethacin on the response to tachykinin NK-2 and NK-3 receptor agonists in the circular muscle of the guinea-pig ileum.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:1

    Topics: Animals; Atropine; Calcium Channel Blockers; Guinea Pigs; Ileum; In Vitro Techniques; Indomethacin; Male; Muscle, Smooth; Myenteric Plexus; Neurokinin A; omega-Conotoxin GVIA; Peptide Fragments; Peptides; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tetrodotoxin

1994
Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic non-cholinergic excitation and contraction in the circular muscle of guinea-pig duodenum.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Action Potentials; Adenosine Diphosphate; Animals; Apamin; Arginine; Atropine; Dose-Response Relationship, Drug; Duodenum; Electric Stimulation; Guanethidine; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Nifedipine; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Suramin; Thionucleotides

1995
Characterization of the antibronchoconstrictor activity of MEN 11420, a tachykinin NK2 receptor antagonist, in guinea-pigs.
    European journal of pharmacology, 1998, Jul-10, Volume: 352, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Atropine; Benzamides; Bronchi; Bronchoconstriction; Bronchodilator Agents; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1998
Tachykinins contribute to nerve-mediated contractions in the human esophagus.
    Gastroenterology, 2001, Volume: 120, Issue:1

    Topics: Atropine; Autonomic Nervous System; Benzamides; Dose-Response Relationship, Drug; Esophagus; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Parasympatholytics; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Substance P; Tachykinins

2001
Tachykinin NK(2) receptors and enhancement of cholinergic transmission in the inflamed rat colon: an in vivo motility study.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Acetic Acid; Animals; Atropine; Cholinergic Fibers; Colon; Enzyme Inhibitors; Gastrointestinal Motility; Hexamethonium; Inflammation; Male; Muscarinic Antagonists; Neurokinin A; NG-Nitroarginine Methyl Ester; Peptide Fragments; Peptides, Cyclic; Rats; Rats, Wistar; Receptors, Neurokinin-2; Synaptic Transmission; Time Factors

2001
Role for NK(1) and NK(2) receptors in the motor activity in mouse colon.
    European journal of pharmacology, 2007, Sep-10, Volume: 570, Issue:1-3

    Topics: Animals; Atropine; Colon; Electric Stimulation; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sodium Channel Blockers; Substance P; Tetrodotoxin

2007