Page last updated: 2024-09-05

nbi 27914 and r 121919

nbi 27914 has been researched along with r 121919 in 1 studies

Compound Research Comparison

Studies
(nbi 27914)
Trials
(nbi 27914)
Recent Studies (post-2010)
(nbi 27914)
Studies
(r 121919)
Trials
(r 121919)
Recent Studies (post-2010) (r 121919)
7602983432

Protein Interaction Comparison

ProteinTaxonomynbi 27914 (IC50)r 121919 (IC50)
Corticotropin-releasing factor receptor 1Homo sapiens (human)0.0321

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodbeck, R; De Lombaert, S; Doller, D; Fung, L; Ge, P; Gulianello, M; Hodgetts, KJ; Hoffman, D; Horvath, RF; Kehne, JH; Kieltyka, A; Krause, JE; Lee, Y; Maynard, GD; Yoon, T1

Other Studies

1 other study(ies) available for nbi 27914 and r 121919

ArticleYear
Discovery of N-(1-ethylpropyl)-[3-methoxy-5-(2-methoxy-4-trifluoromethoxyphenyl)-6-methyl-pyrazin-2-yl]amine 59 (NGD 98-2): an orally active corticotropin releasing factor-1 (CRF-1) receptor antagonist.
    Journal of medicinal chemistry, 2011, Jun-23, Volume: 54, Issue:12

    Topics: Adipose Tissue; Administration, Oral; Adrenocorticotropic Hormone; Animals; Biological Availability; Blood-Brain Barrier; Cell Line; Cerebral Cortex; Humans; In Vitro Techniques; Injections, Intraventricular; Male; Microsomes, Liver; Motor Activity; Pyrazines; Radioligand Assay; Rats; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Structure-Activity Relationship

2011