naxagolide has been researched along with raclopride in 22 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (9.09) | 18.2507 |
2000's | 9 (40.91) | 29.6817 |
2010's | 11 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Nobrega, JN; Seeman, P | 1 |
Day, J; Fibiger, HC | 1 |
Ginovart, N; Houle, S; Hussey, D; Kapur, S; Seeman, P; Willeit, M; Wilson, AA | 1 |
Bloomfield, PM; Galineau, L; Ginovart, N; Houle, S; Kapur, S; Mizrahi, R; Seeman, P; Willeit, M; Wilson, AA | 1 |
Galineau, L; Garcia, A; Ginovart, N; Houle, S; Kapur, S; Wilson, AA | 1 |
Gmeiner, P; Kapur, S; Seeman, P; Wilson, A | 1 |
Guillin, O; Hwang, DR; Hwang, Y; Laruelle, M; Narendran, R; Rabiner, E; Reeder, S; Scher, E; Slifstein, M | 1 |
Ginovart, N; Graff-Guerrero, A; Kapur, S; Mamo, D; Mizrahi, R; Rusjan, P; Seeman, P; Vitcu, I; Willeit, M; Wilson, AA | 1 |
Kapur, S; McCormick, PN; Seeman, P; Wilson, AA | 1 |
Adams, JR; Boileau, I; Furukawa, Y; Guttman, M; Hornykiewicz, O; Houle, S; Kapur, S; Kish, SJ; Rusjan, P; Tong, J; Wilson, AA | 1 |
Barsoum, P; Graff-Guerrero, A; Houle, S; Kapur, S; Mamo, D; Marcon, H; Mizrahi, R; Rusjan, P; Shammi, CM; Wilson, AA | 1 |
Ahmad, R; Brickute, D; Egerton, A; Grasby, PM; Hirani, E; Howes, OD; Luthra, SK; Rosso, L; Turton, DR | 1 |
Ding, M; Dorff, P; Elmore, CS; Maier, D; Malmquist, J; Mrzljak, L; Peng, T; Ström, P; Tuke, D; Werkheiser, J; Widzowski, D; Zysk, J | 1 |
Ginovart, N; McCormick, PN; Wilson, AA | 1 |
Bobok, A; Horti, F; Kiss, B | 1 |
Abanades, S; Beaver, JD; Colasanti, A; Gunn, RN; Huiban, M; Laruelle, M; Miller, SR; Plisson, C; Rabiner, EA; Searle, GE; Shotbolt, P; Tziortzi, AC; van der Aart, J | 1 |
Carson, RE; Cosgrove, KP; Gallezot, JD; Huang, Y; Kloczynski, T; Labaree, D; Lim, K; Morris, ED; Pittman, B; Rabiner, EA; Ridler, K; Weinzimmer, D; Zheng, MQ | 1 |
Anderson, GM; Baldan, LC; Billingslea, E; Bloch, MH; Crowley, M; de Araujo, I; Ding, YS; Ercan-Sencicek, AG; Gallezot, JD; Gorczyca, R; Hughes, ZA; Krusong, K; Krystal, JH; Leventhal, BL; Loring, E; Mayes, L; Ohtsu, H; Panza, KE; Pittenger, C; Pogorelov, V; Rapanelli, M; State, MW; Wasylink, S; Williams, KA | 1 |
Alexoff, D; Carter, P; Fowler, JS; Kang, Y; Kim, D; Kim, SW; King, P; Logan, J; Muench, L; Shea, C; Skolnick, P; Volkow, ND | 1 |
Abi-Jaoude, E; Cho, SS; Houle, S; Lang, AE; Obeso, I; Rusjan, P; Sandor, P; Segura, B; Strafella, AP | 1 |
Boileau, I; Caravaggio, F; Chung, JK; Gerretsen, P; Graff-Guerrero, A; Houle, S; Mamo, DC; Nakajima, S; Plitman, E; Wilson, AA | 1 |
Boileau, I; Caravaggio, F; Chakravarty, MM; Gerretsen, P; Graff-Guerrero, A; Iwata, Y; Kim, J; Ku Chung, J; Patel, R; Plitman, E; Remington, G | 1 |
1 trial(s) available for naxagolide and raclopride
Article | Year |
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The effect of antipsychotics on the high-affinity state of D2 and D3 receptors: a positron emission tomography study With [11C]-(+)-PHNO.
Topics: Adult; Antipsychotic Agents; Basal Ganglia; Benzodiazepines; Benzothiazoles; Binding, Competitive; Carbon Radioisotopes; Caudate Nucleus; Clozapine; Dopamine Agonists; Dopamine Antagonists; Double-Blind Method; Female; Globus Pallidus; Humans; Image Processing, Computer-Assisted; Male; Middle Aged; Olanzapine; Oxazines; Positron-Emission Tomography; Pramipexole; Putamen; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Risperidone; Schizophrenia | 2009 |
21 other study(ies) available for naxagolide and raclopride
Article | Year |
---|---|
Dopamine D2 receptors mapped in rat brain with [3H](+)PHNO.
Topics: Animals; Autoradiography; Brain; Brain Chemistry; Brain Mapping; Densitometry; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Ligands; Male; Oxazines; Raclopride; Rats; Rats, Wistar; Salicylamides; Spiperone | 1994 |
Dopaminergic regulation of cortical acetylcholine release: effects of dopamine receptor agonists.
Topics: Acetylcholine; Animals; Apomorphine; Benzazepines; Cerebral Cortex; Dialysis; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Indoles; Male; Nerve Endings; Oxazines; Phenanthridines; Quinpirole; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides | 1993 |
High-affinity states of human brain dopamine D2/3 receptors imaged by the agonist [11C]-(+)-PHNO.
Topics: Adult; Brain; Brain Mapping; Carbon Radioisotopes; Dopamine Antagonists; Female; Humans; Image Processing, Computer-Assisted; Magnetic Resonance Imaging; Male; Middle Aged; Oxazines; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2; Reference Values | 2006 |
Binding characteristics and sensitivity to endogenous dopamine of [11C]-(+)-PHNO, a new agonist radiotracer for imaging the high-affinity state of D2 receptors in vivo using positron emission tomography.
Topics: Amphetamine; Animals; Binding Sites; Binding, Competitive; Brain; Brain Chemistry; Carbon Radioisotopes; Cats; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Oxazines; Positron-Emission Tomography; Presynaptic Terminals; Raclopride; Receptors, Dopamine D2; Synaptic Transmission | 2006 |
In vivo characterization of the pharmacokinetics and pharmacological properties of [11C]-(+)-PHNO in rats using an intracerebral beta-sensitive system.
Topics: Amphetamine; Animals; Binding, Competitive; Brain; Brain Chemistry; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Male; Molecular Structure; Oxazines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2 | 2006 |
Dopamine D2 and D3 receptors in human putamen, caudate nucleus, and globus pallidus.
Topics: Animals; Binding, Competitive; Caudate Nucleus; CHO Cells; Cloning, Molecular; Cricetinae; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Globus Pallidus; Humans; In Vitro Techniques; Oxazines; Piperazines; Putamen; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Thiophenes | 2006 |
Dopamine (D2/3) receptor agonist positron emission tomography radiotracer [11C]-(+)-PHNO is a D3 receptor preferring agonist in vivo.
Topics: Animals; Binding, Competitive; Brain; Brain Mapping; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Down-Regulation; Female; Globus Pallidus; Male; Oxazines; Papio anubis; Piperazines; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Species Specificity; Time Factors | 2006 |
Brain region binding of the D2/3 agonist [11C]-(+)-PHNO and the D2/3 antagonist [11C]raclopride in healthy humans.
Topics: Adult; Binding, Competitive; Brain Mapping; Carbon Radioisotopes; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Globus Pallidus; Humans; Male; Neostriatum; Oxazines; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2; Substantia Nigra; Time Factors; Tissue Distribution | 2008 |
Dopamine D2 receptor radiotracers [(11)C](+)-PHNO and [(3)H]raclopride are indistinguishably inhibited by D2 agonists and antagonists ex vivo.
Topics: Animals; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Male; Oxazines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tritium | 2008 |
Decreased binding of the D3 dopamine receptor-preferring ligand [11C]-(+)-PHNO in drug-naive Parkinson's disease.
Topics: Aged; Binding, Competitive; Carbon Radioisotopes; Case-Control Studies; Corpus Striatum; Dopamine; Dopamine Antagonists; Female; Globus Pallidus; Humans; Male; Middle Aged; Oxazines; Parkinson Disease; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D3; Statistics, Nonparametric | 2009 |
Further evaluation of the carbon11-labeled D(2/3) agonist PET radiotracer PHNO: reproducibility in tracer characteristics and characterization of extrastriatal binding.
Topics: Animals; Binding, Competitive; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine Agonists; Male; Oxazines; Positron-Emission Tomography; Protein Binding; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reproducibility of Results; Tissue Distribution | 2010 |
D2 receptor occupancy in conscious rat brain is not significantly distinguished with [3H]-MNPA, [3H]-(+)-PHNO, and [3H]-raclopride.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Brain; CHO Cells; Cricetinae; Cricetulus; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Male; Oxazines; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, G-Protein-Coupled | 2010 |
Isoflurane anaesthesia differentially affects the amphetamine sensitivity of agonist and antagonist D2/D3 positron emission tomography radiotracers: implications for in vivo imaging of dopamine release.
Topics: Amphetamine; Anesthesia; Animals; Cats; Cerebellum; Dopamine; Dopamine D2 Receptor Antagonists; Isoflurane; Male; Neostriatum; Oxazines; Positron-Emission Tomography; Raclopride; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Time Factors | 2011 |
In vitro and in vivo comparison of [³H](+)-PHNO and [³H]raclopride binding to rat striatum and lobes 9 and 10 of the cerebellum: a method to distinguish dopamine D₃ from D₂ receptor sites.
Topics: Animals; Binding, Competitive; Cerebellum; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ligands; Male; Oxazines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Staining and Labeling; Tissue Culture Techniques; Tritium | 2011 |
Within-subject comparison of [(11)C]-(+)-PHNO and [(11)C]raclopride sensitivity to acute amphetamine challenge in healthy humans.
Topics: Adult; Amphetamine; Binding, Competitive; Brain; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Ligands; Male; Middle Aged; Oxazines; Positron-Emission Tomography; Protein Binding; Raclopride; Radioligand Assay; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Sensitivity and Specificity | 2012 |
Imaging nicotine- and amphetamine-induced dopamine release in rhesus monkeys with [(11)C]PHNO vs [(11)C]raclopride PET.
Topics: Amphetamine; Animals; Brain; Central Nervous System Stimulants; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Macaca mulatta; Magnetic Resonance Imaging; Nicotine; Nicotinic Agonists; Oxazines; Positron-Emission Tomography; Protein Binding; Raclopride | 2014 |
Histidine decarboxylase deficiency causes tourette syndrome: parallel findings in humans and mice.
Topics: Adolescent; Adult; Amphetamine; Animals; Brain; Child; Dopamine Agonists; Dopamine Antagonists; Exploratory Behavior; Female; Histidine Decarboxylase; Humans; Male; Maze Learning; Mice; Mice, Knockout; Middle Aged; Mutation; Oxazines; Raclopride; Radionuclide Imaging; Stereotyped Behavior; Time Factors; Tourette Syndrome; Tryptophan; Young Adult | 2014 |
Therapeutic doses of buspirone block D3 receptors in the living primate brain.
Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Benzazepines; Benzofurans; Buspirone; Corpus Striatum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Functional Neuroimaging; Globus Pallidus; Injections, Intramuscular; Mesencephalon; Oxazines; Papio anubis; Positron-Emission Tomography; Raclopride; Radioligand Assay; Receptors, Dopamine D3 | 2014 |
Similar striatal D2/D3 dopamine receptor availability in adults with Tourette syndrome compared with healthy controls: A [(11) C]-(+)-PHNO and [(11) C]raclopride positron emission tomography imaging study.
Topics: Adolescent; Adult; Corpus Striatum; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Female; Humans; Male; Middle Aged; Oxazines; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Severity of Illness Index; Tourette Syndrome; Young Adult | 2015 |
Lack of age-dependent decrease in dopamine D3 receptor availability: a [(11)C]-(+)-PHNO and [(11)C]-raclopride positron emission tomography study.
Topics: Adolescent; Adult; Aged; Aging; Binding, Competitive; Brain; Brain Chemistry; Carbon Radioisotopes; Caudate Nucleus; Corpus Striatum; Dopamine Agonists; Female; Globus Pallidus; Healthy Volunteers; Humans; Image Processing, Computer-Assisted; Male; Middle Aged; Oxazines; Positron-Emission Tomography; Putamen; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D3; Young Adult | 2015 |
The relationship between subcortical brain volume and striatal dopamine D
Topics: Adult; Corpus Striatum; Female; Hippocampus; Humans; Magnetic Resonance Imaging; Male; Organ Size; Oxazines; Positron-Emission Tomography; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Thalamus | 2017 |