nan 190 has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 98 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (1.02) | 18.7374 |
1990's | 66 (67.35) | 18.2507 |
2000's | 23 (23.47) | 29.6817 |
2010's | 8 (8.16) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Alonso-Cires, L; Corcóstegui, R; Labeaga, L; Orjales, A | 1 |
Berardi, F; Colabufo, NA; Fiorentini, F; Govoni, S; Olgiati, V; Perrone, R; Tortorella, V; Vanotti, E | 1 |
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL | 1 |
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B | 1 |
Beneitez, ME; Benhamú, B; Fuentes, JA; López-Rodríguez, ML; Manzanares, J; Morcillo, MJ; Orensanz, L; Rosado, ML; Sanz, AM | 1 |
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L | 1 |
Buck, LB; Petrascheck, M; Ye, X | 1 |
Barrett, JE; Gleeson, S; Seggel, MR; Weissman, BA | 1 |
Ahlgren, PC; Brännström, G; Fowler, CJ | 1 |
Dawson, IM; Hodgkiss, JP; Kelly, JS | 1 |
Dourish, CT; Williams, AR | 1 |
Barrett, JE; Gleeson, S | 1 |
Caldarola-Pastuszka, M; Montanez, S; Uphouse, L | 1 |
Ahlers, ST; Barrett, JE; Weissman, BA | 1 |
Glaser, T; Greuel, JM | 1 |
Moser, PC | 1 |
Durcan, MJ; Linnoila, M; Wozniak, KM | 1 |
Barrett, JE; Zhang, L | 1 |
Kelly, JS; Penington, NJ | 1 |
Budziszewska, B; Błaszczyńska, E; Chojnacka-Wójcik, E; Ismaiel, AM; Przegaliński, E; Tatarczyńska, E | 1 |
Glennon, RA; Lyon, RA; Naiman, NA; Pierson, ME; Titeler, M; Weisberg, E | 1 |
Empson, RM; Heinemann, U; Schmitz, D | 1 |
Deschaux, P; Ferriere, F; Khan, NA | 1 |
Jednak, MA; Judge, K; Ram, JL | 1 |
Cole, BJ; Jones, GH; Turner, JD | 1 |
Fornal, CA; Jacobs, BL; Marrosu, F; Metzler, CW; Tada, K | 1 |
Lucot, JB | 1 |
Olivier, B; Slangen, JL; Ybema, CE | 1 |
Amano, T; Kishimoto, T; Sasa, M; Todo, N; Yamanaka, T | 1 |
Bischoff, AM; Lalley, PM; Richter, DW | 1 |
Sillar, KT; Wedderburn, JF | 1 |
Azzaro, AJ; Johnson, EA; Shahan, YH; Tsai, CE | 1 |
Fozard, JR; Hoyer, D; McQuade, R; Sharp, T | 1 |
Kellar, KJ; Lumpkin, MD; Mulroney, SE; Shemer, A; Skudlarek, C | 1 |
Bole-Vunduk, B; Krisch, I | 1 |
Hiraga, Y; Ikeda, Y; Izumi, J; Miura, N; Washizuka, M | 1 |
Sakai, N; Tanaka, C | 1 |
Glass, JD; Rea, MA; Selim, M | 1 |
Moore, NA; Perrett, L; Rees, G; Sanger, G | 1 |
Bagdy, G; Kalogeras, KT | 1 |
Fozard, JR; Hoyer, D; Schoeffter, P; Seiler, MP; Siegl, H; Stoll, A | 1 |
Rabin, RA; Winter, JC | 1 |
de Vry, J; Schreiber, R | 1 |
Dunn, AJ; Farrar, GE; Saphier, D; Welch, JE | 1 |
Matsuyama, S; Nei, K; Tanaka, C | 2 |
Masson-Pévet, M; Pévet, P; Recio, J | 1 |
Belcheva, I; Belcheva, S; Hadjiivanova, C; Petkov, VD; Petkov, VV | 1 |
Bjørkum, AA; Ursin, R | 1 |
Fujii, T; Fujimoto, K; Kawashima, K; Nakai, K; Suzuki, T; Yoshizawa, M | 1 |
Helton, DR; Kallman, MJ; Rasmussen, K | 1 |
Ally, A; Asmundsson, G; Caringi, D; Ishide, T; Kobayashi, T; Mokler, DJ | 1 |
Draguhn, A; Empson, RM; Gloveli, T; Heinemann, U; Schmitz, D | 1 |
Nagaoka, I; Sasa, M; Yamawaki, S | 1 |
Pickard, GE; Rea, MA | 1 |
Gean, PW; Lu, KT | 1 |
Baker, GB; Bourin, M; Colombel, MC; Redrobe, JP | 2 |
Barros, DM; de Souza, MM; Izquierdo, I; Izquierdo, LA; Medina, JH; Mello e Souza, T | 1 |
Empson, RM; Gloveli, T; Heinemann, U; Schmitz, D | 1 |
Bagdy, G; Filakovszky, J; Gerber, K; Halasz, P | 1 |
Ardenghi, P; Bevilaqua, L; Bianchin, M; Bromberg, E; Izquierdo, I; Medina, JH; Quevedo, J; Schaeffer, E; Schmitz, PK; Schröder, N; Walz, R | 1 |
Bischoff, AM; Lalley, PM; Pierrefiche, O; Richter, DW; Schmidt-Garcon, P | 1 |
Darmani, NA; Zhao, W | 1 |
Cha, AE; Moerschbaecher, JM; Rodriguez, FH; Winsauer, PJ | 1 |
Honda, M; Ono, H | 1 |
Bult, H; Geerts, IS; Herman, AG; Matthys, KE | 1 |
Khan, NA; Poisson, JP | 1 |
Abe, K; Edagawa, Y; Saito, H | 1 |
Glennon, RA; Young, R | 1 |
Canto-de-Souza, A; da-Costa, M; Fornari, RV; Graeff, FG; Nunes-de-Souza, RL; Pelá, IR | 1 |
Akaike, N; Kishimoto, K; Koyama, S | 1 |
Moerschbaecher, JM; Winsauer, PJ | 1 |
Goodchild, AK; Miyawaki, T; Pilowsky, PM | 1 |
Gao, X; Wu, G; Yang, Z; Zhang, Y | 1 |
Beirlant, J; Engelborghs, Y; Hoebeke, J; Marot, C; Matthys, G; Strobbe, R; Van Craenenbroeck, E; Vercammen, J | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J | 1 |
Akasu, T; Hasuo, H | 1 |
Gean, PW; Huang, YC; Lin, CH; Tsai, JJ | 1 |
Choi, H; Coitinho, A; Izquierdo, I; Mello e Souza, T; Rodrigues, C; Souza, MM; Vinadé, E | 1 |
Saifullah, AS; Tomioka, K | 1 |
Chandler, SH; Hsiao, CF; Wu, N | 1 |
Chen, R; Hamilton, R; Jordan, S; Kikuchi, T; Koprivica, V; Tottori, K; Whitehead, RE | 1 |
Djavadian, RL; Turlejski, K; Wielkopolska, E | 1 |
Egashira, N; Fujioka, M; Fujiwara, M; Ishigami, N; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Yano, A | 1 |
Fedotova, JO; Hartmann, G; Lénárd, L; Sapronov, NS | 2 |
Kaczyńska, K; Szereda-Przestaszewska, M | 1 |
Duffy-Whritenour, JE; Zelikoff, JT | 1 |
Glennon, RA; Khorana, N; Young, R | 1 |
Hu, Y; Huang, XY; Luo, CX; Wu, DL; Wu, HY; Ye, ML; Zhang, J; Zhou, QG; Zhu, DY; Zhu, LJ | 1 |
Charkhpour, M; Doustar, Y; Hassanzadeh, K; Nayebi, AR | 1 |
Fedotova, YO; Ordyan, NE | 1 |
Bakhtiari, A; Salari, AA; Solati, J | 1 |
Fedotova, IuO; Ordian, NÉ; Pivina, SG | 1 |
Adamczyk-Sowa, M; Misiolek, M; Namyslowski, G; Pierzchala, K; Sowa, P; Zwirska-Korczala, K | 1 |
Atzori, M; Dinh, L; Galindo-Charles, L; García-Oscos, F; Pérez Padilla, EA; Pineda, JC; Salgado, H; Torres-Ramírez, O | 1 |
Aguilar-Magaña, D; Atzori, M; Canto-Bustos, M; Cervantes-Ramírez, V; Góngora-Alfaro, JL; Pérez-Padilla, EA; Pineda, JC; Salgado, H | 1 |
1 review(s) available for nan 190 and 8-hydroxy-2-(di-n-propylamino)tetralin
Article | Year |
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Serotonergic innervation of the hypothalamic suprachiasmatic nucleus and photic regulation of circadian rhythms.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Afferent Pathways; Animals; Axons; Circadian Rhythm; Cricetinae; Light; Mammals; Mesocricetus; Mice; Photic Stimulation; Piperazines; Quipazine; Raphe Nuclei; Receptors, Serotonin; Retinal Ganglion Cells; Serotonin; Serotonin Receptor Agonists; Superior Colliculi; Suprachiasmatic Nucleus | 1997 |
97 other study(ies) available for nan 190 and 8-hydroxy-2-(di-n-propylamino)tetralin
Article | Year |
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New (2-methoxyphenyl)piperazine derivatives as 5-HT1A receptor ligands with reduced alpha 1-adrenergic activity. Synthesis and structure-affinity relationships.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Ligands; Male; Piperazines; Rabbits; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Structure-Activity Relationship | 1995 |
Mixed 5-HT1A/D-2 activity of a new model of arylpiperazines: 1-aryl-4-[3-(1,2-dihydronaphthalen-4-yl)-n-propyl]piperazines. 1. Synthesis and structure-activity relationships.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Membrane; Cerebral Cortex; Corpus Striatum; Ketanserin; Male; Molecular Structure; Naphthalenes; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Serotonin; Spiperone; Structure-Activity Relationship; Tritium | 1994 |
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution | 1993 |
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes | 1996 |
Synthesis and structure-activity relationships of a new model of arylpiperazines. 1. 2-[[4-(o-methoxyphenyl)piperazin-1-yl]methyl]-1, 3-dioxoperhydroimidazo[1,5-alpha]pyridine: a selective 5-HT1A receptor agonist.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Body Temperature; Cerebral Cortex; Kinetics; Mice; Piperazines; Raclopride; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Salicylamides; Serotonin Receptor Agonists; Social Behavior; Structure-Activity Relationship | 1996 |
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes | 1998 |
An antidepressant that extends lifespan in adult Caenorhabditis elegans.
Topics: Aging; Animals; Antidepressive Agents; Caenorhabditis elegans; Caloric Restriction; Humans; Longevity; Methiothepin; Mianserin; Octopamine; Receptors, Biogenic Amine; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Signal Transduction; Starvation | 2007 |
Neurochemical effects of 5-HT1 receptor ligands in pigeons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Brain; Columbidae; Hydroxyindoleacetic Acid; Indoles; Male; Methoxyhydroxyphenylglycol; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1992 |
GH4ZD10 cells expressing rat 5-HT1A receptors coupled to adenylyl cyclase are a model for the postsynaptic receptors in the rat hippocampus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Alprenolol; Animals; Cell Line; Cyclic AMP; Hippocampus; Piperazines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoactive Intestinal Peptide; Zinc | 1992 |
An intracellular study of the action of NAN-190 on neurons in the dorsal raphe nucleus of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Dose-Response Relationship, Drug; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurons; Piperazines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1992 |
Effects of the putative 5-HT1A receptor antagonist NAN-190 on free feeding and on feeding induced by the 5-HT1A receptor agonist 8-OH-DPAT in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Eating; Male; Motor Activity; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin Antagonists; Stereotyped Behavior | 1992 |
Discriminative stimulus effects of 8-OH-DPAT in pigeons: antagonism studies with the putative 5-HT1A receptor antagonists BMY 7378 and NAN-190.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Pindolol; Piperazines; Prazosin; Serotonin Antagonists | 1992 |
Intracerebral actions of the 5-HT1A agonists, 8-OH-DPAT and buspirone and of the 5-HT1A partial agonist/antagonist, NAN-190, on female sexual behavior.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Cerebral Ventricles; Dose-Response Relationship, Drug; Female; Injections; Injections, Intraperitoneal; Piperazines; Posture; Rats; Rats, Inbred F344; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus | 1992 |
Antagonism studies with BMY-7378 and NAN-190: effects on 8-hydroxy-2-(di-n-propylamino)tetralin-induced increases in punished responding of pigeons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Brain; Columbidae; Dose-Response Relationship, Drug; Drug Antagonism; Midazolam; Piperazines; Radioligand Assay; Serotonin Antagonists; Tetrahydronaphthalenes | 1992 |
The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Electrophysiology; In Vitro Techniques; Male; Piperazines; Propranolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tetrahydronaphthalenes | 1992 |
The effect of putative 5-HT1A receptor antagonists on 8-OH-DPAT-induced hypothermia in rats and mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dioxanes; Dose-Response Relationship, Drug; Hypothermia, Induced; Male; Mice; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Is NAN-190 an effective antagonist of the hypothermia and hyperglycemia induced by the 5-HT1A receptor agonist, 8-OH-DPAT?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hyperglycemia; Hypothermia, Induced; Male; Mice; Piperazines; Premedication; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Involvement of 5-HT1A activity in the discriminative stimulus effects of imipramine.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Columbidae; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Imipramine; Male; Piperazines; Prazosin; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Serotonin receptor activation reduces calcium current in an acutely dissociated adult central neuron.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium; Cell Membrane Permeability; Electric Conductivity; Membrane Potentials; Neurons; Piperazines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
The behavioural, but not the hypothermic or corticosterone, response to 8-hydroxy-2-(DI-n-propylamino)-tetralin, is antagonized by NAN-190 in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Body Temperature; Corticosterone; Male; Naphthalenes; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Reserpine; Serotonin Antagonists; Spiperone; Tetrahydronaphthalenes | 1990 |
NAN-190: an arylpiperazine analog that antagonizes the stimulus effects of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT).
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Conditioning, Operant; Discrimination Learning; Naphthalenes; Piperazines; Prazosin; Rats; Serotonin Antagonists; Tetrahydronaphthalenes | 1988 |
Serotonin reduces inhibition via 5-HT1A receptors in area CA1 of rat hippocampal slices in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Electric Conductivity; Female; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Neurons; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission | 1995 |
Serotonin-induced calcium signaling via 5-HT1A receptors in human leukemia (K 562) cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium; Humans; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Signal Transduction; Tumor Cells, Cultured | 1995 |
Antagonists of cholinergic and serotonergic responses of Aplysia buccal muscle.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Aplysia; Atropine; Cholinergic Antagonists; Hexamethonium; In Vitro Techniques; Mecamylamine; Muscle Contraction; Muscle, Smooth; Piperazines; Pirenzepine; Serotonin Antagonists | 1994 |
5-HT1A receptor agonists improve the performance of normal and scopolamine-impaired rats in an operant delayed matching to position task.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Conditioning, Operant; Male; Memory, Short-Term; Piperazines; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Space Perception | 1994 |
Effects of the putative 5-hydroxytryptamine1A antagonists BMY 7378, NAN 190 and (-)-propranolol on serotonergic dorsal raphe unit activity in behaving cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Cats; Female; Male; Neurons; Piperazines; Propranolol; Raphe Nuclei; Serotonin; Serotonin Antagonists | 1994 |
Antiemetic effects of flesinoxan in cats: comparisons with 8-hydroxy-2-(di-n-propylamino)tetralin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antiemetics; Behavior, Animal; Cats; Dose-Response Relationship, Drug; Injections, Subcutaneous; Motion Sickness; Piperazines; Propranolol; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Vomiting; Xylazine | 1994 |
Discriminative stimulus effect of flesinoxan: effect of 5-HT1A antagonists and PCPA.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Discrimination Learning; Fenclonine; Male; Pindolol; Piperazines; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 1994 |
5-HT1A receptor-mediated inhibition of lateral vestibular nucleus neurons projecting to the abducens nucleus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Abducens Nerve; Animals; Brain; Cats; Electrophysiology; Female; Male; Neural Inhibition; Neurons; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Vestibular Nuclei | 1994 |
5-HT-1A receptor-mediated modulation of medullary expiratory neurones in the cat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Apnea; Cats; Electric Stimulation; Female; Hyperventilation; Injections, Intravenous; Iontophoresis; Male; Medulla Oblongata; Membrane Potentials; Neurons; Phrenic Nerve; Piperazines; Receptors, Serotonin; Respiratory Mechanics; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses | 1994 |
Modulation of rhythmic swimming activity in post-embryonic Xenopus laevis tadpoles by 5-hydroxytryptamine acting at 5HT1a receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Cyproheptadine; Ergolines; Ketanserin; Metamorphosis, Biological; Methysergide; Motor Activity; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming; Xenopus laevis | 1994 |
Serotonin 5-HT1A receptors mediate inhibition of tyrosine hydroxylation in rat striatum.
Topics: 4-Butyrolactone; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Corpus Striatum; Dopamine; Dopamine D2 Receptor Antagonists; Hydroxylation; Male; Nerve Endings; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tyrosine 3-Monooxygenase | 1993 |
The novel 5-HT1A receptor antagonist, SDZ 216-525, decreases 5-HT release in rat hippocampus in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dialysis; Electrophysiology; GTP-Binding Proteins; Hippocampus; Indoles; Male; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Thiazoles | 1993 |
Tandospirone stimulates prolactin secretion in the rat by an action at serotonin-1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Dose-Response Relationship, Drug; Isoindoles; Male; Metergoline; Piperazines; Prolactin; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists | 1994 |
Behavioral studies on LEK-8804, a new ergoline derivative with potent 5-HT1A receptor agonist and 5-HT2 receptor antagonist activity.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Head; Kinetics; Lysergic Acid Diethylamide; Male; Mice; Movement; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists | 1994 |
Hippocampal serotonin 5-HT1A receptor enhances acetylcholine release in conscious rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Clomipramine; Hippocampus; Kinetics; Male; Physostigmine; Piperazines; Quinoxalines; Rats; Rats, Inbred F344; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1994 |
Inhibitory modulation of long-term potentiation via the 5-HT1A receptor in slices of the rat hippocampal dentate gyrus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Isoproterenol; Long-Term Potentiation; Male; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 1993 |
Modulation of light-induced C-Fos expression in the suprachiasmatic nuclei by 5-HT1A receptor agonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Biguanides; Cricetinae; Darkness; Female; Gene Expression; Light; Male; Mesocricetus; Piperazines; Proto-Oncogene Proteins c-fos; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus; Tryptophan | 1994 |
5-HT1A-mediated lower lip retraction: effects of 5-HT1A agonists and antagonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Lip; Male; Pindolol; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
Stimulation of 5-HT1A and 5-HT2/5-HT1C receptors induce oxytocin release in the male rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Buspirone; Male; Oxytocin; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
SDZ 216-525, a selective and potent 5-HT1A receptor antagonist.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Behavior, Animal; Brain; Dioxins; In Vitro Techniques; Indoles; Male; Phosphatidylinositols; Piperazines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine D2; Second Messenger Systems; Serotonin Antagonists; Spiro Compounds; Temperature; Thiazoles | 1993 |
Antagonism of the stimulus effects of yohimbine and 8-hydroxydipropylaminotetralin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Animals; Cerebral Cortex; Discrimination, Psychological; Hippocampus; Male; Pindolol; Piperazines; Radioligand Assay; Rats; Rats, Inbred F344; Receptors, Adrenergic, alpha; Serotonin; Serotonin Antagonists; Yohimbine | 1993 |
Studies on the neuronal circuits involved in the discriminative stimulus effects of 5-hydroxytryptamine1A receptor agonists in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Discrimination Learning; Hippocampus; Male; Methoxydimethyltryptamines; Neurons; Piperazines; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin | 1993 |
Central 5-HT1A receptors inhibit adrenocortical secretion.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenal Cortex; Anesthesia; Animals; Corticosterone; Injections, Intraventricular; Male; Paraventricular Hypothalamic Nucleus; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1993 |
Regulation of glutamate release via NMDA and 5-HT1A receptors in guinea pig dentate gyrus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dentate Gyrus; Dose-Response Relationship, Drug; Female; Glutamic Acid; Guinea Pigs; Male; Piperazines; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin Antagonists | 1996 |
Serotonergic modulation of photically induced increase in melatonin receptor density and Fos immunoreactivity in the suprachiasmatic nuclei of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Light; Male; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus | 1996 |
Behavorial responses to the 5-HT1A receptor antagonist NAN190 injected into rat CA1 hippocampal area.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Avoidance Learning; Functional Laterality; Hippocampus; Injections, Intraventricular; Male; Motor Activity; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists | 1997 |
Sleep/waking effects following intrathecal administration of the 5-HT(1A) Agonist 8-OH-DPAT alone and in combination with the putative 5-HT(1A) antagonist NAN-190 in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Electroencephalography; Injections, Spinal; Male; Piperazines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Serotonin Receptor Agonists; Sleep; Wakefulness | 1996 |
Regulation of GABA release via NMDA and 5-HT1A receptors in guinea pig dentate gyrus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium; Chromatography, High Pressure Liquid; Dentate Gyrus; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Glutamic Acid; Guinea Pigs; Magnesium; Male; N-Methylaspartate; Neurons; Piperazines; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin | 1997 |
Demonstration of the facilitatory role of 8-OH-DPAT on cholinergic transmission in the rat hippocampus using in vivo microdialysis.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Cholinesterase Inhibitors; Hippocampus; Locomotion; Male; Microdialysis; Physostigmine; Piperazines; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission | 1997 |
Serotonin-1A antagonists attenuate the effects of nicotine withdrawal on the auditory startle response.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Auditory Perception; Male; Nicotine; Piperazines; Pyridines; Rats; Reflex, Startle; Serotonin Antagonists; Substance Withdrawal Syndrome | 1997 |
Extracellular serotonin changes in VLM during muscle contraction: effects of 5-HT1A-receptor activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Electric Stimulation; Heart Rate; Kinetics; Male; Medulla Oblongata; Microdialysis; Muscle Contraction; Neuromuscular Junction; Paralysis; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tibial Nerve | 1997 |
Serotonin reduces synaptic excitation in the superficial medial entorhinal cortex of the rat via a presynaptic mechanism.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Entorhinal Cortex; Excitatory Postsynaptic Potentials; Female; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Male; Patch-Clamp Techniques; Piperazines; Potassium Channels; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Synapses; Synaptic Transmission; Tetrodotoxin | 1998 |
5-HT1A receptor-mediated inhibition of nucleus accumbens neurons activated by stimulation of parafascicular nucleus of thalamus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Electric Stimulation; Iontophoresis; Male; Neurons; Nucleus Accumbens; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thalamic Nuclei | 1998 |
Endogenous serotonin inhibits epileptiform activity in rat hippocampal CA1 neurons via 5-hydroxytryptamine1A receptor activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Barium; Epilepsy; Excitatory Postsynaptic Potentials; Fluoxetine; Hippocampus; In Vitro Techniques; Ketanserin; Male; Membrane Potentials; Metergoline; Neurons; Oxadiazoles; Picrotoxin; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Tryptamines | 1998 |
Dose-dependent noradrenergic and serotonergic properties of venlafaxine in animal models indicative of antidepressant activity.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Second-Generation; Cyclohexanols; Male; Mice; Motor Activity; Pindolol; Piperazines; Selective Serotonin Reuptake Inhibitors; Venlafaxine Hydrochloride | 1998 |
Short- and long-term memory are differentially regulated by monoaminergic systems in the rat brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Avoidance Learning; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Entorhinal Cortex; Hippocampus; Male; Memory; Memory, Short-Term; Models, Neurological; Norepinephrine; Parietal Lobe; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Biogenic Amine; Receptors, Dopamine D1; Receptors, Serotonin; Serotonin Antagonists; Statistics, Nonparametric; Timolol | 1998 |
Serotonin reduces polysynaptic inhibition via 5-HT1A receptors in the superficial entorhinal cortex.
Topics: 2-Amino-5-phosphonovalerate; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Entorhinal Cortex; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radical Scavengers; Membrane Potentials; Neural Inhibition; Organ Culture Techniques; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses | 1998 |
The 5-HT1A agonist 8-OH-DPAT increases the number of spike-wave discharges in a genetic rat model of absence epilepsy.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Epilepsy, Absence; Genetic Predisposition to Disease; Injections, Intraperitoneal; Injections, Intraventricular; Piperazines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Serotonin Receptor Agonists | 1998 |
Drugs acting upon the cyclic adenosine monophosphate/protein kinase A signalling pathway modulate memory consolidation when given late after training into rat hippocampus but not amygdala.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Amygdala; Animals; Avoidance Learning; Benzazepines; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Dopamine Antagonists; Hippocampus; Indoles; Male; Memory; Norepinephrine; Piperazines; Pyrroles; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Dopamine D1; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Time Factors; Timolol | 1997 |
Neurotransmitters and neuromodulators controlling the hypoxic respiratory response in anaesthetized cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenosine; Anesthesia, General; Animals; Cats; Cell Membrane; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Glutamic Acid; Hypoxia; Medulla Oblongata; Microdialysis; Microinjections; Phrenic Nerve; Piperazines; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Respiratory Mechanics; Serotonin; Serotonin Antagonists | 1999 |
Production of serotonin syndrome by 8-OH DPAT in Cryptotis parva.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Fluorobenzenes; Injections, Intraperitoneal; Male; Phenols; Piperazines; Propranolol; Serotonin Antagonists; Serotonin Receptor Agonists; Serotonin Syndrome; Shrews | 1998 |
Full and partial 5-HT1A receptor agonists disrupt learning and performance in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Learning; Male; Piperazines; Psychomotor Performance; Rats; Rats, Long-Evans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
Psychopharmacological profile of the selective serotonin reuptake inhibitor, paroxetine: implication of noradrenergic and serotonergic mechanisms.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amines; Animals; Antidepressive Agents; Apomorphine; Brain; Clonidine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Hypothermia; Indoles; Male; Mice; Motor Activity; Norepinephrine; Paroxetine; Pindolol; Piperazines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 1998 |
Differential effects of (R)- and (S)-8-hydroxy-2-(di-n-propylamino)tetralin on the monosynaptic spinal reflex in rats.
Topics: 5,6-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Male; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Reflex, Monosynaptic; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Spiro Compounds; Stereoisomerism | 1999 |
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction | 1999 |
5-HT3 receptor-channels coupled with Na+ influx in human T cells: role in T cell activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium Signaling; Cell Cycle; Enzyme Activation; Granisetron; Humans; Ion Channel Gating; Ion Transport; Jurkat Cells; Lymphocyte Activation; Metoclopramide; Neoplasm Proteins; Phytohemagglutinins; Piperazines; Protein Kinase C; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Ryanodine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sodium Channels; T-Lymphocytes; Thapsigargin | 1999 |
The serotonin 5-HT2 receptor-phospholipase C system inhibits the induction of long-term potentiation in the rat visual cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Bicuculline; Electrophysiology; Estrenes; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Long-Term Potentiation; Male; Phosphodiesterase Inhibitors; Piperazines; Pyrrolidinones; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Type C Phospholipases; Visual Cortex | 2000 |
MDMA stimulus generalization to the 5-HT(1A) serotonin agonist 8-hydroxy-2- (di-n-propylamino)tetralin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Drug Interactions; Male; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Anxiety-induced antinociception in mice: effects of systemic and intra-amygdala administration of 8-OH-DPAT and midazolam.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amygdala; Analgesia; Animals; Anti-Anxiety Agents; Anxiety; Male; Mice; Microinjections; Midazolam; Naloxone; Narcotic Antagonists; Pain Measurement; Piperazines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Presynaptic modulation of synaptic gamma-aminobutyric acid transmission by tandospirone in rat basolateral amygdala.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Amygdala; Animals; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Isoindoles; Neurons; Piperazines; Presynaptic Terminals; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission | 2000 |
Differential effects of 5-HT agonists and antagonists on the repeated acquisition and performance of response sequences in monkeys.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Amphetamines; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ergolines; Learning; Macaca fascicularis; Macaca mulatta; Piperazines; Pyridines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Rostral ventral medulla 5-HT1A receptors selectively inhibit the somatosympathetic reflex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Baroreflex; Chemoreceptor Cells; Functional Laterality; Male; Medulla Oblongata; Microinjections; Neurons; Piperazines; Pressoreceptors; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Sympathetic Nervous System | 2001 |
The role of 5-hydroxytryptamine1A and 5-hydroxytryptamine1B receptors in modulating spinal nociceptive transmission in normal and carrageenan-injected rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Carrageenan; Electric Stimulation; Electrophysiology; Female; Male; Neurons, Afferent; Nociceptors; Pain; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission | 2001 |
Heuristic statistical analysis of fluorescence fluctuation data with bright spikes: application to ligand binding to the human serotonin receptor expressed in Escherichia coli cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Benzopyrans; Data Interpretation, Statistical; Escherichia coli; Fluorescence; Humans; Ligands; Models, Statistical; Normal Distribution; Oxadiazoles; Piperazines; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spectrometry, Fluorescence | 2001 |
Differential effect of serotonin 5-HT(1A) receptor antagonists on the secretion of corticotropin and prolactin.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Cyclohexylamines; Male; Piperazines; Prolactin; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Restraint, Physical; Serotonin; Serotonin Antagonists; Stress, Physiological | 2001 |
5-Hydroxytryptamine facilitates spatiotemporal propagation of optical signals in the hippocampal-septal pathway.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Bicuculline; Electric Stimulation; Electronic Data Processing; Excitatory Amino Acid Antagonists; Fornix, Brain; GABA Antagonists; Hippocampus; Male; Neural Conduction; Neurons; Phosphinic Acids; Piperazines; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Tetrodotoxin | 2001 |
Modulation of voltage-dependent calcium currents by serotonin in acutely isolated rat amygdala neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylate Cyclase Toxin; Adenylyl Cyclases; Amygdala; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Enzyme Inhibitors; Ethylmaleimide; GTP-Binding Proteins; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Neurons; Nimodipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Patch-Clamp Techniques; Pertussis Toxin; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sympathomimetics; Thionucleotides; Virulence Factors, Bordetella | 2001 |
Involvement of the serotonergic type 1A (5-HT1A) receptor in the agranular insular cortex in the consolidation of memory for inhibitory avoidance in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Avoidance Learning; Injections; Male; Memory; Piperazines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
5-HT(7)-like receptors mediate serotonergic modulation of photo-responsiveness of the medulla bilateral neurons in the cricket, Gryllus bimaculatus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Clozapine; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Gryllidae; Ketanserin; Light; Neurons; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Visual Pathways | 2003 |
Voltage-dependent calcium currents in trigeminal motoneurons of early postnatal rats: modulation by 5-HT receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Analysis of Variance; Animals; Animals, Newborn; Calcium Channel Blockers; Calcium Channels; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; In Vitro Techniques; Ketanserin; Membrane Potentials; Motor Neurons; Neural Inhibition; Patch-Clamp Techniques; Piperazines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nuclei | 2005 |
In vitro profile of the antidepressant candidate OPC-14523 at rat and human 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Autoradiography; Binding, Competitive; Buspirone; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Frontal Lobe; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Male; Middle Aged; Pindolol; Piperazines; Pyridines; Quinolones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfur Radioisotopes | 2005 |
Postnatal treatment with NAN-190 but not with 5-HT1A receptor agonists retards growth of the rat brain.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Buspirone; Cerebral Cortex; Drug Administration Schedule; Immunologic Techniques; Piperazines; Rats; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Staining and Labeling; Vibrissae | 2005 |
Investigation of mechanisms mediating 8-OH-DPAT-induced impairment of spatial memory: involvement of 5-HT1A receptors in the dorsal hippocampus in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Interactions; Hippocampus; Male; Maze Learning; Memory Disorders; Microinjections; Phenols; Piperazines; Prazosin; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Sulfonamides | 2006 |
Effects of 5-HT1A receptor agonist and antagonist on anxiety in intact and ovariectomized female rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Estradiol; Female; Ovariectomy; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Involvement of 5-HT1A receptors in passive avoidance learning in intact and ovariectomized female rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Avoidance Learning; Estradiol; Female; Ovariectomy; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Peripheral 5-HT1A receptors are not essential for increased ventilation evoked by systemic 8-OH-DPAT challenge in anaesthetized rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Blood Pressure; Male; Nodose Ganglion; Piperazines; Pulmonary Ventilation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists; Tidal Volume; Vagotomy | 2007 |
Relationship between serotonin and the immune system in a teleost model.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Fenclonine; Immune System; Models, Animal; Neuroimmunomodulation; Perciformes; Piperazines; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spleen | 2008 |
Effect of 8-hydroxy-2-(N,N-di-n-propylamino)tetralin and MDMA on the discriminative stimulus effects of the classical hallucinogen DOM in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Discrimination Learning; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Drug Synergism; Generalization, Stimulus; Hallucinogens; Isomerism; Male; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Serotonin Receptor Agonists | 2009 |
Neuronal nitric oxide synthase alteration accounts for the role of 5-HT1A receptor in modulating anxiety-related behaviors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Anxiety Disorders; CREB-Binding Protein; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Exploratory Behavior; Feeding Behavior; Fluoxetine; Gene Expression Regulation, Enzymologic; Hippocampus; Indazoles; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitric Oxide Synthase Type I; Phosphorylation; Piperazines; Reaction Time; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2010 |
8-OH-DPAT prevents morphine-induced apoptosis in rat dorsal raphe nucleus: a possible mechanism for attenuating morphine tolerance.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics, Opioid; Animals; Apoptosis; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Tolerance; Hot Temperature; In Situ Nick-End Labeling; Injections, Intraperitoneal; Male; Morphine; Pain; Pain Measurement; Piperazines; Raphe Nuclei; Rats; Rats, Wistar; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2010 |
Effects of 8-OH-DPAT and NAN-190 on anxious-depressive-like behavior of female rats during the estrous cycle.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Anxiety Disorders; Depression; Estrous Cycle; Female; Maze Learning; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists | 2010 |
5HT(1A) and 5HT(1B) receptors of medial prefrontal cortex modulate anxiogenic-like behaviors in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anxiety; Exploratory Behavior; Male; Microinjections; Piperazines; Piperidones; Prefrontal Cortex; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds | 2011 |
[Analysis of 8-OH-DPAT and NAN-190 effects in young prenatally stressed rats under experimental estrogen deficiency conditions].
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Behavior, Animal; Estrogens; Female; Male; Ovariectomy; Piperazines; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Serotonin Receptor Agonists; Stress, Physiological | 2012 |
The role of serotonergic 5-HT1A receptors in central cardiovascular regulation in haemorrhagic shock in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Heart Rate; Male; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Shock, Hemorrhagic | 2013 |
Activation of 5-HT receptors inhibits GABAergic transmission by pre-and post-synaptic mechanisms in layer II/III of the juvenile rat auditory cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Auditory Cortex; GABA Agonists; GABAergic Neurons; Inhibitory Postsynaptic Potentials; Miniature Postsynaptic Potentials; Muscimol; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Receptor Agonists; Synapses | 2015 |
Citalopram reduces glutamatergic synaptic transmission in the auditory cortex via activation of 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Auditory Cortex; Citalopram; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Piperazines; Pyramidal Cells; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission | 2019 |