naltrexone and pentazocine

naltrexone has been researched along with pentazocine in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-199015 (40.54)18.7374
1990's8 (21.62)18.2507
2000's7 (18.92)29.6817
2010's7 (18.92)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Archer, S; Michne, WF1
Fennessy, MR; Laska, FJ1
Appel, JB; Hernandez, LL; Holohean, AM1
Bläsig, J; Herz, A; Höllt, V; Paschelke, G1
Misawa, M; Nagase, H; Narita, M; Suzuki, T2
Becketts, K; Nickel, B; Vaupel, DB1
Vaupel, DB1
Hamada, T; Kameyama, T; Nakayama, S; Ukai, M1
Holtzman, SG1
Brocklehurst, C; Devia, C; Moerschbaecher, JM1
Hameroff, SR1
Appel, JB; Hernández, LL1
Smith, AA; Wassef, NM1
Franklin, SR; Tang, AH1
Coale, EH; Hein, DW; Herling, S; Valentino, RJ; Woods, JH1
Holtzman, SG; White, JM1
Bigelow, GE; Preston, KL1
Iwamoto, Y; Kamei, J; Kasuya, Y; Misawa, M; Nagase, H1
Maity, R; Mukherjee, R; Skolnick, P1
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA1
Cheung, P; Li, JG; Liu-Chen, LY; Raffa, RB; Tzeng, TB1
Endoh, T; Izumimoto, N; Kamei, J; Mizoguchi, H; Nagase, H; Narita, M; Saitoh, A; Suzuki, T; Tajima, A; Tseng, LF1
Coles, JA; Iaizzo, PA; Sigg, DC1
Borgland, SL; Christie, MJ; Connor, M; Furness, JB; Osborne, PB1
Craft, RM; McNiel, DM1
Greene, JL; McClean, JM; Smith, MA1
Hiramatsu, M; Hoshino, T1
Chiba, S; Hayashida, M; Nishiyama, T; Shu, H; Yamada, Y; Yoshikawa, M1
Hayashi, SS; Kamei, J; Ohsawa, M1
Li, M; McMillan, DE; Wessinger, WD1
Horishita, T; Inagaki, H; Kawasaki, T; Obara, G; Sata, T; Takahashi, K; Toyohira, Y; Tsutsui, M; Ueno, S; Yanagihara, N1
Ise, Y; Itoh, T; Komiya, S; Masukawa, D; Mizuo, K; Mori, T; Saeki, T; Shibasaki, M; Suzuki, T; Yoshizawa, K1
Dou, Y; Huang, W; Li, Q; Lin, Y; Shu, H; Wang, Z; Xiao, X; Ye, F1
Haji, A; Kimura, S; Ohi, Y1
DiPetrillo, L; Ehrich, E; Kelsh, D; Nangia, N; Pathak, S; Puhl, MD; Setnik, B; Stanford, AD; Sun, L; Vince, B1

Reviews

3 review(s) available for naltrexone and pentazocine

ArticleYear
Recent progress in research on narcotic antagonists.
    Progress in drug research. Fortschritte der Arzneimittelforschung. Progres des recherches pharmaceutiques, 1976, Volume: 20

    Topics: Animals; Benzomorphans; Chemical Phenomena; Chemistry; Cyclazocine; Humans; In Vitro Techniques; Models, Biological; Morphinans; Morphine Derivatives; Nalbuphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Receptors, Opioid; Structure-Activity Relationship; Substance-Related Disorders; Thebaine

1976
Drug discrimination studies.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Opiate receptor pharmacology: mixed agonist/antagonist narcotics.
    Contemporary anesthesia practice, 1983, Volume: 7

    Topics: Analgesics, Opioid; Buprenorphine; Butorphanol; Endorphins; Humans; Nalbuphine; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Opioid

1983

Trials

1 trial(s) available for naltrexone and pentazocine

ArticleYear
Differential naltrexone antagonism of hydromorphone and pentazocine effects in human volunteers.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Adult; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Humans; Hydromorphone; Male; Naltrexone; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu

1993

Other Studies

33 other study(ies) available for naltrexone and pentazocine

ArticleYear
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Acute effects of opiate agonists, partial agonists and antagonists on brain monoamines in the rat.
    Archives internationales de pharmacodynamie et de therapie, 1979, Volume: 238, Issue:1

    Topics: Animals; Behavior, Animal; Biogenic Amines; Brain Chemistry; Cyclazocine; Dextrorphan; Female; Levallorphan; Morphine; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Rats

1979
Effects of opiates on the discriminative stimulus properties of dopamine agonists.
    Pharmacology, biochemistry, and behavior, 1978, Volume: 9, Issue:4

    Topics: Amphetamine; Animals; Apomorphine; Discrimination, Psychological; Dopamine; Haloperidol; Male; Morphine; Naltrexone; Narcotics; Pentazocine; Rats; Time Factors

1978
Comparison of withdrawal precipitating properties of various morphine antagonists and partial agonists in relation to their stereospecific binding to brain homogenates.
    Psychopharmacologia, 1976, Volume: 46, Issue:1

    Topics: Benzomorphans; Binding Sites; Brain; Humans; Levallorphan; Morphine Dependence; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Drug; Sodium; Stereoisomerism; Subcellular Fractions; Substance Withdrawal Syndrome

1976
Pentazocine-induced biphasic analgesia in mice.
    Life sciences, 1991, Volume: 48, Issue:19

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Analgesics; Animals; Drug Administration Schedule; Drug Interactions; Drug Tolerance; Indoles; Injections, Intraventricular; Male; Mice; Morphinans; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Time Factors

1991
Supraspinal analgesic action of pentazocine in mice.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Analgesics; Animals; Drug Tolerance; Indoles; Injections, Intraventricular; Male; Mice; Morphinans; Naltrexone; Pain Measurement; Pentazocine; Receptors, Opioid; Time Factors

1990
Flupirtine antinociception in the dog is primarily mediated by nonopioid supraspinal mechanisms.
    European journal of pharmacology, 1989, Mar-29, Volume: 162, Issue:3

    Topics: Aminopyridines; Analgesics; Animals; Decerebrate State; Dogs; Female; Naltrexone; Pentazocine; Reflex; Temperature; Time Factors

1989
Interactions between pentazocine and tripelennamine on autonomic and nociceptive measures in the dog.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:1

    Topics: Animals; Autonomic Nervous System; Behavior, Animal; Body Temperature; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Female; Naltrexone; Nociceptors; Pentazocine; Pupil; Reflex; Time Factors; Tripelennamine

1989
Discriminative stimulus properties of the mixed agonist-antagonist pentazocine in the rat using two-choice discrete-trial avoidance paradigm.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:2

    Topics: Animals; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Methamphetamine; Naltrexone; Narcotics; Pentazocine; Pentobarbital; Rats; Rats, Inbred Strains

1989
Differential antagonism by naltrexone of the effects of opioids on a fixed-ratio discrimination in rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Rats

1988
Effects of pentazocine and other opiates on shock detection in the rat: involvement of opiate and dopamine receptors.
    Psychopharmacology, 1980, Volume: 67, Issue:2

    Topics: Animals; Electroshock; Male; Morphine; Naltrexone; Narcotics; Pentazocine; Prejudice; Rats; Receptors, Dopamine; Receptors, Opioid; Reinforcement Schedule

1980
Inhibition of growth in young mice treated with pentazocine: reversal by naltrexone.
    European journal of pharmacology, 1980, Aug-29, Volume: 66, Issue:2-3

    Topics: Animals; Body Weight; Brain; Dose-Response Relationship, Drug; Growth; Liver; Mice; Muscle Proteins; Naloxone; Naltrexone; Pentazocine; Protein Biosynthesis; Receptors, Opioid

1980
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:6

    Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344

1983
Narcotic discrimination in pigeons.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 214, Issue:1

    Topics: Animals; Clonidine; Codeine; Columbidae; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Ketamine; Meperidine; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Pentobarbital; Species Specificity

1980
Three-choice drug discrimination in the rat: morphine, cyclazocine and saline.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 217, Issue:2

    Topics: Animals; Cyclazocine; Dextroamphetamine; Discrimination Learning; Discrimination, Psychological; Generalization, Stimulus; Male; Morphine; Naltrexone; Pentazocine; Rats; Secobarbital; Sodium Chloride

1981
Effects of diabetes on the antinociceptive effect of (+/-)pentazocine in mice.
    Research communications in chemical pathology and pharmacology, 1994, Volume: 84, Issue:1

    Topics: Analgesics; Animals; Diabetes Mellitus, Experimental; Drug Synergism; Male; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptors; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu

1994
Stereoselective inhibition of natural killer activity by the sigma ligand (+)-pentazocine.
    Journal of neuroimmunology, 1996, Volume: 70, Issue:1

    Topics: Animals; Cells, Cultured; Cyclohexylamines; Dose-Response Relationship, Drug; Immunosuppressive Agents; Killer Cells, Natural; Ligands; Mice; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship

1996
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
    Journal of neuroimmunology, 1997, Volume: 72, Issue:1

    Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium

1997
Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor.
    European journal of pharmacology, 1998, Aug-07, Volume: 354, Issue:2-3

    Topics: Analgesics; Animals; Binding, Competitive; CHO Cells; Cricetinae; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Ligands; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Peptide Fragments; Peptides; Radioligand Assay; Rats; Receptors, Opioid, mu; Somatostatin; Sufentanil; Thermodynamics; Time Factors

1998
TRK-820, a selective kappa-opioid agonist, produces potent antinociception in cynomolgus monkeys.
    Japanese journal of pharmacology, 2001, Volume: 85, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Behavior, Animal; Macaca fascicularis; Morphinans; Morphine; Naloxone; Naltrexone; Pain Measurement; Pentazocine; Pentobarbital; Receptors, Opioid, kappa; Spiro Compounds

2001
Role of kappa-opioid receptor activation in pharmacological preconditioning of swine.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:6

    Topics: Animals; Arrhythmias, Cardiac; Coronary Circulation; Enkephalin, Leucine-2-Alanine; Hemodynamics; Ischemic Preconditioning, Myocardial; Morphine; Myocardial Infarction; Myocardial Ischemia; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Receptors, Opioid, kappa; Swine

2003
Opioid agonists have different efficacy profiles for G protein activation, rapid desensitization, and endocytosis of mu-opioid receptors.
    The Journal of biological chemistry, 2003, May-23, Volume: 278, Issue:21

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Electric Conductivity; Endocytosis; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GTP-Binding Proteins; Methadone; Mice; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Neuroblastoma; Pentazocine; Pituitary Neoplasms; Receptors, Opioid, mu; Transfection; Tumor Cells, Cultured

2003
Agonist/antagonist properties of nalbuphine, butorphanol and (-)-pentazocine in male vs. female rats.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 75, Issue:1

    Topics: Animals; Benzeneacetamides; Butorphanol; Diuresis; Diuretics; Dose-Response Relationship, Drug; Female; Male; Nalbuphine; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sex Characteristics; Urination

2003
Enhanced sensitivity to the antinociceptive effects of kappa opioids in naltrexone-treated rats: dose- and time-dependent effects.
    Behavioural pharmacology, 2003, Volume: 14, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Animals; Dose-Response Relationship, Drug; Drug Administration Schedule; Male; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Pentazocine; Pyrrolidines; Rats; Rats, Long-Evans; Receptors, Opioid, kappa

2003
Improvement of memory impairment by (+)- and (-)-pentazocine via sigma, but not kappa opioid receptors.
    Brain research, 2005, Sep-28, Volume: 1057, Issue:1-2

    Topics: Acetic Acid; Analgesics, Opioid; Analysis of Variance; Animals; Anisoles; Antipsychotic Agents; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Exploratory Behavior; Isomerism; Male; Maze Learning; Memory Disorders; Mice; Naltrexone; Narcotic Antagonists; Pain Measurement; Pentazocine; Propylamines; Receptors, Opioid, kappa; Receptors, sigma; Scopolamine

2005
Inhibitory effect of low-dose pentazocine on the development of antinociceptive tolerance to morphine.
    Journal of anesthesia, 2009, Volume: 23, Issue:1

    Topics: Analgesics, Opioid; Animals; Cinnamates; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Mice, Inbred ICR; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Pain Measurement; Pentazocine; Pressure; Receptors, Opioid, kappa

2009
Effect of acute topical application of +-pentazocine on the mechanical allodynia in diabetic mice.
    European journal of pharmacology, 2010, Sep-01, Volume: 641, Issue:1

    Topics: Administration, Topical; Animals; Diabetes Complications; Ethylenediamines; Male; Mice; Mice, Inbred ICR; Naltrexone; Nitric Oxide; Pentazocine; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor

2010
Drug discrimination in pigeons trained to discriminate among morphine, U50488, a combination of these drugs, and saline.
    Behavioural pharmacology, 2011, Volume: 22, Issue:5-6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Butorphanol; Columbidae; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule; Sodium Chloride

2011
Pentazocine inhibits norepinephrine transporter function by reducing its surface expression in bovine adrenal medullary cells.
    Journal of pharmacological sciences, 2013, Volume: 121, Issue:2

    Topics: Adrenal Medulla; Analgesics, Opioid; Animals; Cattle; Cell Line; Cell Membrane; Cells, Cultured; Ethylenediamines; Fluoxetine; Gene Expression; Humans; Naltrexone; Narcotic Antagonists; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Pentazocine; Radionuclide Imaging

2013
Involvement of μ- and δ-opioid receptor function in the rewarding effect of (±)-pentazocine.
    Addiction biology, 2015, Volume: 20, Issue:4

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Isomerism; Male; Naloxone; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Pain; Pentazocine; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Reward

2015
High-dose pentazocine antagonizes the antinociception induced by high-dose morphine.
    Life sciences, 2015, Jun-01, Volume: 130

    Topics: Analgesics, Opioid; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred C57BL; Morphine; Naltrexone; Pain; Pentazocine; Receptors, Opioid, kappa

2015
Mechanisms of pentazocine-induced ventilatory depression and antinociception in anesthetized rats.
    Journal of pharmacological sciences, 2016, Volume: 130, Issue:3

    Topics: Analgesics; Anesthesia; Animals; Male; Naltrexone; Pentazocine; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiratory Insufficiency

2016
Abuse Potential of Samidorphan: A Phase I, Oxycodone-, Pentazocine-, Naltrexone-, and Placebo-Controlled Study.
    Journal of clinical pharmacology, 2019, Volume: 59, Issue:2

    Topics: Adult; Analgesics, Opioid; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Oxycodone; Pentazocine; Placebos

2019