naltrexone has been researched along with pentazocine in 37 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 15 (40.54) | 18.7374 |
1990's | 8 (21.62) | 18.2507 |
2000's | 7 (18.92) | 29.6817 |
2010's | 7 (18.92) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A | 1 |
Archer, S; Michne, WF | 1 |
Fennessy, MR; Laska, FJ | 1 |
Appel, JB; Hernandez, LL; Holohean, AM | 1 |
Bläsig, J; Herz, A; Höllt, V; Paschelke, G | 1 |
Misawa, M; Nagase, H; Narita, M; Suzuki, T | 2 |
Becketts, K; Nickel, B; Vaupel, DB | 1 |
Vaupel, DB | 1 |
Hamada, T; Kameyama, T; Nakayama, S; Ukai, M | 1 |
Holtzman, SG | 1 |
Brocklehurst, C; Devia, C; Moerschbaecher, JM | 1 |
Hameroff, SR | 1 |
Appel, JB; Hernández, LL | 1 |
Smith, AA; Wassef, NM | 1 |
Franklin, SR; Tang, AH | 1 |
Coale, EH; Hein, DW; Herling, S; Valentino, RJ; Woods, JH | 1 |
Holtzman, SG; White, JM | 1 |
Bigelow, GE; Preston, KL | 1 |
Iwamoto, Y; Kamei, J; Kasuya, Y; Misawa, M; Nagase, H | 1 |
Maity, R; Mukherjee, R; Skolnick, P | 1 |
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA | 1 |
Cheung, P; Li, JG; Liu-Chen, LY; Raffa, RB; Tzeng, TB | 1 |
Endoh, T; Izumimoto, N; Kamei, J; Mizoguchi, H; Nagase, H; Narita, M; Saitoh, A; Suzuki, T; Tajima, A; Tseng, LF | 1 |
Coles, JA; Iaizzo, PA; Sigg, DC | 1 |
Borgland, SL; Christie, MJ; Connor, M; Furness, JB; Osborne, PB | 1 |
Craft, RM; McNiel, DM | 1 |
Greene, JL; McClean, JM; Smith, MA | 1 |
Hiramatsu, M; Hoshino, T | 1 |
Chiba, S; Hayashida, M; Nishiyama, T; Shu, H; Yamada, Y; Yoshikawa, M | 1 |
Hayashi, SS; Kamei, J; Ohsawa, M | 1 |
Li, M; McMillan, DE; Wessinger, WD | 1 |
Horishita, T; Inagaki, H; Kawasaki, T; Obara, G; Sata, T; Takahashi, K; Toyohira, Y; Tsutsui, M; Ueno, S; Yanagihara, N | 1 |
Ise, Y; Itoh, T; Komiya, S; Masukawa, D; Mizuo, K; Mori, T; Saeki, T; Shibasaki, M; Suzuki, T; Yoshizawa, K | 1 |
Dou, Y; Huang, W; Li, Q; Lin, Y; Shu, H; Wang, Z; Xiao, X; Ye, F | 1 |
Haji, A; Kimura, S; Ohi, Y | 1 |
DiPetrillo, L; Ehrich, E; Kelsh, D; Nangia, N; Pathak, S; Puhl, MD; Setnik, B; Stanford, AD; Sun, L; Vince, B | 1 |
3 review(s) available for naltrexone and pentazocine
Article | Year |
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Recent progress in research on narcotic antagonists.
Topics: Animals; Benzomorphans; Chemical Phenomena; Chemistry; Cyclazocine; Humans; In Vitro Techniques; Models, Biological; Morphinans; Morphine Derivatives; Nalbuphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Receptors, Opioid; Structure-Activity Relationship; Substance-Related Disorders; Thebaine | 1976 |
Drug discrimination studies.
Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1985 |
Opiate receptor pharmacology: mixed agonist/antagonist narcotics.
Topics: Analgesics, Opioid; Buprenorphine; Butorphanol; Endorphins; Humans; Nalbuphine; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Opioid | 1983 |
1 trial(s) available for naltrexone and pentazocine
Article | Year |
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Differential naltrexone antagonism of hydromorphone and pentazocine effects in human volunteers.
Topics: Adult; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Humans; Hydromorphone; Male; Naltrexone; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1993 |
33 other study(ies) available for naltrexone and pentazocine
Article | Year |
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Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders | 1998 |
Acute effects of opiate agonists, partial agonists and antagonists on brain monoamines in the rat.
Topics: Animals; Behavior, Animal; Biogenic Amines; Brain Chemistry; Cyclazocine; Dextrorphan; Female; Levallorphan; Morphine; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Rats | 1979 |
Effects of opiates on the discriminative stimulus properties of dopamine agonists.
Topics: Amphetamine; Animals; Apomorphine; Discrimination, Psychological; Dopamine; Haloperidol; Male; Morphine; Naltrexone; Narcotics; Pentazocine; Rats; Time Factors | 1978 |
Comparison of withdrawal precipitating properties of various morphine antagonists and partial agonists in relation to their stereospecific binding to brain homogenates.
Topics: Benzomorphans; Binding Sites; Brain; Humans; Levallorphan; Morphine Dependence; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Drug; Sodium; Stereoisomerism; Subcellular Fractions; Substance Withdrawal Syndrome | 1976 |
Pentazocine-induced biphasic analgesia in mice.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Analgesics; Animals; Drug Administration Schedule; Drug Interactions; Drug Tolerance; Indoles; Injections, Intraventricular; Male; Mice; Morphinans; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Time Factors | 1991 |
Supraspinal analgesic action of pentazocine in mice.
Topics: Analgesics; Animals; Drug Tolerance; Indoles; Injections, Intraventricular; Male; Mice; Morphinans; Naltrexone; Pain Measurement; Pentazocine; Receptors, Opioid; Time Factors | 1990 |
Flupirtine antinociception in the dog is primarily mediated by nonopioid supraspinal mechanisms.
Topics: Aminopyridines; Analgesics; Animals; Decerebrate State; Dogs; Female; Naltrexone; Pentazocine; Reflex; Temperature; Time Factors | 1989 |
Interactions between pentazocine and tripelennamine on autonomic and nociceptive measures in the dog.
Topics: Animals; Autonomic Nervous System; Behavior, Animal; Body Temperature; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Female; Naltrexone; Nociceptors; Pentazocine; Pupil; Reflex; Time Factors; Tripelennamine | 1989 |
Discriminative stimulus properties of the mixed agonist-antagonist pentazocine in the rat using two-choice discrete-trial avoidance paradigm.
Topics: Animals; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Methamphetamine; Naltrexone; Narcotics; Pentazocine; Pentobarbital; Rats; Rats, Inbred Strains | 1989 |
Differential antagonism by naltrexone of the effects of opioids on a fixed-ratio discrimination in rats.
Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Rats | 1988 |
Effects of pentazocine and other opiates on shock detection in the rat: involvement of opiate and dopamine receptors.
Topics: Animals; Electroshock; Male; Morphine; Naltrexone; Narcotics; Pentazocine; Prejudice; Rats; Receptors, Dopamine; Receptors, Opioid; Reinforcement Schedule | 1980 |
Inhibition of growth in young mice treated with pentazocine: reversal by naltrexone.
Topics: Animals; Body Weight; Brain; Dose-Response Relationship, Drug; Growth; Liver; Mice; Muscle Proteins; Naloxone; Naltrexone; Pentazocine; Protein Biosynthesis; Receptors, Opioid | 1980 |
Acquisition of brightness discrimination in the rat is impaired by opiates with psychotomimetic properties.
Topics: Animals; Avoidance Learning; Cyclazocine; Discrimination Learning; Male; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Phenazocine; Photic Stimulation; Psychotropic Drugs; Rats; Rats, Inbred F344 | 1983 |
Narcotic discrimination in pigeons.
Topics: Animals; Clonidine; Codeine; Columbidae; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Ketamine; Meperidine; Morphine; Nalorphine; Naltrexone; Narcotics; Pentazocine; Pentobarbital; Species Specificity | 1980 |
Three-choice drug discrimination in the rat: morphine, cyclazocine and saline.
Topics: Animals; Cyclazocine; Dextroamphetamine; Discrimination Learning; Discrimination, Psychological; Generalization, Stimulus; Male; Morphine; Naltrexone; Pentazocine; Rats; Secobarbital; Sodium Chloride | 1981 |
Effects of diabetes on the antinociceptive effect of (+/-)pentazocine in mice.
Topics: Analgesics; Animals; Diabetes Mellitus, Experimental; Drug Synergism; Male; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptors; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1994 |
Stereoselective inhibition of natural killer activity by the sigma ligand (+)-pentazocine.
Topics: Animals; Cells, Cultured; Cyclohexylamines; Dose-Response Relationship, Drug; Immunosuppressive Agents; Killer Cells, Natural; Ligands; Mice; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship | 1996 |
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium | 1997 |
Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor.
Topics: Analgesics; Animals; Binding, Competitive; CHO Cells; Cricetinae; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Ligands; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Peptide Fragments; Peptides; Radioligand Assay; Rats; Receptors, Opioid, mu; Somatostatin; Sufentanil; Thermodynamics; Time Factors | 1998 |
TRK-820, a selective kappa-opioid agonist, produces potent antinociception in cynomolgus monkeys.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Behavior, Animal; Macaca fascicularis; Morphinans; Morphine; Naloxone; Naltrexone; Pain Measurement; Pentazocine; Pentobarbital; Receptors, Opioid, kappa; Spiro Compounds | 2001 |
Role of kappa-opioid receptor activation in pharmacological preconditioning of swine.
Topics: Animals; Arrhythmias, Cardiac; Coronary Circulation; Enkephalin, Leucine-2-Alanine; Hemodynamics; Ischemic Preconditioning, Myocardial; Morphine; Myocardial Infarction; Myocardial Ischemia; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Receptors, Opioid, kappa; Swine | 2003 |
Opioid agonists have different efficacy profiles for G protein activation, rapid desensitization, and endocytosis of mu-opioid receptors.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Electric Conductivity; Endocytosis; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GTP-Binding Proteins; Methadone; Mice; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Neuroblastoma; Pentazocine; Pituitary Neoplasms; Receptors, Opioid, mu; Transfection; Tumor Cells, Cultured | 2003 |
Agonist/antagonist properties of nalbuphine, butorphanol and (-)-pentazocine in male vs. female rats.
Topics: Animals; Benzeneacetamides; Butorphanol; Diuresis; Diuretics; Dose-Response Relationship, Drug; Female; Male; Nalbuphine; Naltrexone; Narcotic Antagonists; Pentazocine; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sex Characteristics; Urination | 2003 |
Enhanced sensitivity to the antinociceptive effects of kappa opioids in naltrexone-treated rats: dose- and time-dependent effects.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Animals; Dose-Response Relationship, Drug; Drug Administration Schedule; Male; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Pentazocine; Pyrrolidines; Rats; Rats, Long-Evans; Receptors, Opioid, kappa | 2003 |
Improvement of memory impairment by (+)- and (-)-pentazocine via sigma, but not kappa opioid receptors.
Topics: Acetic Acid; Analgesics, Opioid; Analysis of Variance; Animals; Anisoles; Antipsychotic Agents; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Exploratory Behavior; Isomerism; Male; Maze Learning; Memory Disorders; Mice; Naltrexone; Narcotic Antagonists; Pain Measurement; Pentazocine; Propylamines; Receptors, Opioid, kappa; Receptors, sigma; Scopolamine | 2005 |
Inhibitory effect of low-dose pentazocine on the development of antinociceptive tolerance to morphine.
Topics: Analgesics, Opioid; Animals; Cinnamates; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Mice, Inbred ICR; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Pain Measurement; Pentazocine; Pressure; Receptors, Opioid, kappa | 2009 |
Effect of acute topical application of +-pentazocine on the mechanical allodynia in diabetic mice.
Topics: Administration, Topical; Animals; Diabetes Complications; Ethylenediamines; Male; Mice; Mice, Inbred ICR; Naltrexone; Nitric Oxide; Pentazocine; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor | 2010 |
Drug discrimination in pigeons trained to discriminate among morphine, U50488, a combination of these drugs, and saline.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Butorphanol; Columbidae; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule; Sodium Chloride | 2011 |
Pentazocine inhibits norepinephrine transporter function by reducing its surface expression in bovine adrenal medullary cells.
Topics: Adrenal Medulla; Analgesics, Opioid; Animals; Cattle; Cell Line; Cell Membrane; Cells, Cultured; Ethylenediamines; Fluoxetine; Gene Expression; Humans; Naltrexone; Narcotic Antagonists; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Pentazocine; Radionuclide Imaging | 2013 |
Involvement of μ- and δ-opioid receptor function in the rewarding effect of (±)-pentazocine.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Isomerism; Male; Naloxone; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Pain; Pentazocine; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Reward | 2015 |
High-dose pentazocine antagonizes the antinociception induced by high-dose morphine.
Topics: Analgesics, Opioid; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred C57BL; Morphine; Naltrexone; Pain; Pentazocine; Receptors, Opioid, kappa | 2015 |
Mechanisms of pentazocine-induced ventilatory depression and antinociception in anesthetized rats.
Topics: Analgesics; Anesthesia; Animals; Male; Naltrexone; Pentazocine; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiratory Insufficiency | 2016 |
Abuse Potential of Samidorphan: A Phase I, Oxycodone-, Pentazocine-, Naltrexone-, and Placebo-Controlled Study.
Topics: Adult; Analgesics, Opioid; Cross-Over Studies; Double-Blind Method; Female; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Oxycodone; Pentazocine; Placebos | 2019 |