naltrexone and ly 255582

naltrexone has been researched along with ly 255582 in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (33.33)18.2507
2000's4 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantrell, BE; Johnson, BG; Leander, JD; Mendelsohn, LG; Mitch, CH; Reel, JK; Shaw, WN; Snoddy, JD; Takemori, AE; Wong, DT1
Cantrell, BE; Carroll, FI; Dersch, CM; Mascarella, SW; McCullough, KB; Partilla, JS; Rothman, RB; Thomas, JB; Xu, H; Zimmerman, DM1
Carroll, FI1
Carroll, FI; Chaudhari, S; Deschamps, J; Gigstad, KM; Mascarella, SW; Navarro, HA; Thomas, JB1
Emmerson, PJ; Holloway, WG; Matt, JE; McKinzie, JH; Mitch, CH; Siegel, MG; Statnick, MA; Surface, PL; Suter, TM; Takeuchi, K; Thomas, EM; Wolfe, CN1
Emmerson, PJ; Holloway, WG; McKinzie, JH; Mitch, CH; Quimby, SJ; Siegel, MG; Statnick, MA; Surface, PL; Suter, TM; Takeuchi, K; Thomas, EM1

Reviews

1 review(s) available for naltrexone and ly 255582

ArticleYear
2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Animals; Biogenic Monoamines; Biological Transport; Carrier Proteins; Cocaine; Fluorescent Dyes; Humans; Isoquinolines; Ligands; Morphinans; Narcotic Antagonists; Piperidines; Protein Binding; Radioisotopes; Receptors, Opioid; Structure-Activity Relationship; Substance-Related Disorders

2003

Other Studies

5 other study(ies) available for naltrexone and ly 255582

ArticleYear
3,4-Dimethyl-4-(3-hydroxyphenyl)piperidines: opioid antagonists with potent anorectant activity.
    Journal of medicinal chemistry, 1993, Oct-01, Volume: 36, Issue:20

    Topics: Analgesia; Animals; Appetite Depressants; Cyclohexanes; Diuresis; Eating; Endorphins; Guinea Pigs; Male; Mice; Molecular Structure; Piperidines; Rats; Rats, Sprague-Dawley; Rats, Zucker; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship

1993
Investigation of the N-substituent conformation governing potency and mu receptor subtype-selectivity in (+)-(3R, 4R)-dimethyl-4-(3-hydroxyphenyl)piperidine opioid antagonists.
    Journal of medicinal chemistry, 1998, May-21, Volume: 41, Issue:11

    Topics: Animals; Brain; Crystallography, X-Ray; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; In Vitro Techniques; Molecular Conformation; Narcotic Antagonists; Piperidines; Rats; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1998
N-substituted cis-4a-(3-hydroxyphenyl)-8a-methyloctahydroisoquinolines are opioid receptor pure antagonists.
    Journal of medicinal chemistry, 2005, Dec-29, Volume: 48, Issue:26

    Topics: Animals; Benzeneacetamides; CHO Cells; Cricetinae; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Isoquinolines; Models, Molecular; Molecular Conformation; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2005
Structure-activity relationship studies of carboxamido-biaryl ethers as opioid receptor antagonists (OpRAs). Part 1.
    Bioorganic & medicinal chemistry letters, 2007, Oct-01, Volume: 17, Issue:19

    Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Drug Design; Ethers; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Molecular Conformation; Narcotic Antagonists; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship

2007
Structure activity relationship studies of carboxamido-biaryl ethers as opioid receptor antagonists (OpRAs). Part 2.
    Bioorganic & medicinal chemistry letters, 2007, Dec-15, Volume: 17, Issue:24

    Topics: Acrylic Resins; Amides; Carboxylic Acids; Ethers; Molecular Structure; Narcotic Antagonists; Receptors, Opioid; Structure-Activity Relationship

2007