naltrexone and fentanyl

naltrexone has been researched along with fentanyl in 165 studies

Research

Studies (165)

TimeframeStudies, this research(%)All Research%
pre-199020 (12.12)18.7374
1990's50 (30.30)18.2507
2000's41 (24.85)29.6817
2010's36 (21.82)24.3611
2020's18 (10.91)2.80

Authors

AuthorsStudies
Bell, GI; Chen, Y; Kong, H; Raynor, K; Reisine, T; Yasuda, K; Yu, L1
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Jolivette, LJ; Ward, KW1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Brockmöller, J; Friesacher, HR; Meyer, MJ; Neumann, VE; Tzvetkov, MV; Zdrazil, B1
Burke, TF; Comer, SD; Lewis, JW; Woods, JH1
Crisp, T; Perni, VC; Stafinsky, JL; Uram, M1
Cometta-Morini, C; Kamal, J; Loew, G; Maguire, P; Tsai, N; Upton, C1
Malan, JH; Quandt, SK; Raath, JP1
Holtzman, SG; Paronis, CA1
France, CP; Medzihradsky, F; Rice, KC; Seggel, MR; Winger, G; Woods, JH1
Mjanger, E; Yaksh, TL1
Jang, Y; Yoburn, BC1
Botschev, C; Müller, N1
Sharpe, LG1
Ableitner, A; Ayesta, FJ; Emmett-Oglesby, MW; Herz, A; Shippenberg, TS1
Mueller, J; Quock, RM1
Gaumann, DM; Tyce, GM; Yaksh, TL1
Adams, JU; Holtzman, SG; Paronis, CA1
Beilin, B; Gale, RP; Liebeskind, JC; Martin, FC; Shavit, Y1
Blalock, JE; Carr, DJ; DeCosta, BR; Guarcello, V; Jacobson, AE; Kim, CH; Rice, KC1
Carino, MA; Chinn, C; Horita, A1
Abdelhamid, EM; Archer, S; Koolpe, GA; Michael, J; Michael, M; Nelson, WL; Simon, EJ1
Croughan, J; Sanders, K1
Bice, AN; Dannals, RF; Frost, JJ; Lee, MC; Tanada, S; Wagner, HN1
Dykstra, LA; Negus, SS1
Holtzman, SG3
Martin, WR; Wettstein, JG1
Harty, GJ; Onofrio, BM; Yaksh, TL1
Arendt, RM; Schulz, R; Vollmar, AM1
Hayes, AG; Stewart, BR1
Hayes, AG; Skingle, M; Tyers, MB1
Hynes, MD; Leander, JD; Reel, JK; Zimmerman, DM1
DiFazio, CA; Dixon, R; Gal, TJ1
DiFazio, CA; Gal, TJ1
Freye, E; Hartung, E; Kaliebe, S1
Herz, A; Schulz, R; Wüster, M1
Gioannini, T; Gorissen, H; Maryanoff, BE; Simon, EJ1
Cools, AR; Megens, AA1
Gates, CC; Haigh, JC1
Fujinami, T; Nishimura, M; Saeki, T; Sato, N; Watanabe, Y1
Bagley, JR; Brockunier, LL; Flynn, D; France, CP; Gerak, LR; Medzihradsky, F; Winger, GD; Woods, JH1
Gupta, SK; Hwang, SS; Southam, MA1
Carpenter, JW; Leith, DE; Shaw, ML1
Bagley, JR; Baker, ML; Brockunier, LL; Carr, DJ; France, CP; Holmes, C1
Bayer, BM; Flores, LR; Wahl, SM1
House, JD; Makhay, MM; Walker, EA; Young, AM1
Davis, T; Duttaroy, A; Shah, S; Yoburn, BC1
Osifchin, E; Veng-Pedersen, P; Waters, SJ; Wilhelm, JA; Zakszewski, TB2
Clyde, VL; Ramsay, EC; Sleeman, JM1
Lance, WR; Miller, MW; Wild, MA1
Butour, JL; Meunier, JC; Moisand, C; Mollereau, C; Parmentier, M1
Cook, CD; Morgan, D; Negus, SS; Picker, MJ1
Angel, F; Chevalier, E; Dahl, SG; Friese, N; Junien, JL; Pascaud, X; Riviere, PJ1
Coulais, Y; Francés, B; Goeldner, M; Guiraud, R; Hirth, C; Méjean-Galzi, A; Tafani, JA; Zajac, JM1
Rothe, KS; Stevens, CW1
Carter, W; Ramsay, EC; Sleeman, JM; Tobin, T1
Citino, SB; Heard, DJ; Schumacher, J; Young, L1
Civelek, AC; Dannals, RF; Dixon, RB; Joh, T; Kao, PF; Kim, S; Ravert, HT; Villemagne, VL; Wagner, HN1
Stevens, CW; Willenbring, S1
Bagley, JR; Brockunier, LL; France, CP; Gauthier, CA; Gerak, LR1
Brewer, C; Gastfriend, DR1
Bagley, JR; Brandt, MR; Brockunier, LL; France, CP; Gerak, LR; Landers, LK; Lelas, S1
Braselton, WE; Cook, RA; Dierenfeld, ES; House, C; Karesh, WB; Puche, H; Torres, A; Uhart, MM1
Cheung, P; Li, JG; Liu-Chen, LY; Raffa, RB; Tzeng, TB1
Morgan, D; Picker, MJ1
Bartok, RE; Craft, RM; Heideman, LM1
Cheng, CH; Naylor, RJ; Ngan, MP; Rudd, JA; Wai, MK1
Grech, DM; Platt, DM; Rowlett, JK; Spealman, RD1
Bagley, JR; Brockunier, LL; France, CP; Gerak, LR; Moerschbaecher, JM1
Sutherland, J; Walker, EA; Young, AM; Zhang, L1
Dougherty, TB; Porche, VH; Thall, PF1
Bagley, JR; Brockunier, LL; France, CP; Gauthier, CA1
Mama, KR; Steffey, EP; Withrow, SJ1
Akil, H; Bonner, G; Meng, F1
Kearns, KS; Ramsay, EC; Swenson, B1
Cebra, CK; Larsen, RS; Wild, MA1
Hales, TG; Law, PY; Piros, ET; Prather, PL; Song, L1
Breiter, H; D'Ambra, MN; Elman, I; Gastfriend, DR; Kane, M; Krause, S; Morris, R; Tuffy, L1
Holtzman, SG; White, DA1
Burns, MM; Chumpa, A; Kaplan, RL; Shannon, MW1
Bush, M; Citino, SB; Grobler, D; Lance, W1
Bu, H; Chen, YL; Halls, TD; Jiang, X; Naidong, W; Shou, WZ1
Imai, S; Itou, Y; Narita, M; Suzuki, T; Yajima, Y1
David Clark, J; Demirci, H; Gharagozlou, P; Lameh, J1
Barrett, AC; Picker, MJ; Smith, ES1
Ballachey, BE; McCormick, C; Monson, DH1
Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Adams, KA; Miller, BF; Miller, KV; Muller, LI; Osborn, DA; Ramsay, EC; Storms, TN; Warren, RJ1
Lance, WR; Miller, MW; Wolfe, LL1
Bares, R; Braus, DF; Braus, DH; Croissant, B; Dohmen, BM; Heinz, A; Hermann, D; Machulla, HJ; Mann, K; Mundle, G; Reimold, M; Schumann, G; Wrase, J1
Carpenter, JW; Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Aalto, S; Hagelberg, N; Hietala, J; Ingman, K; Juhakoski, A; Kallio, A; Karhuvaara, S; Någren, K; Oikonen, V; Scheinin, H1
Riters, LV; Schroeder, MB1
Darwish, M; Hellriegel, E; Jiang, JG; Kirby, M; Robertson, P1
Carpenter, JW; Cole, A; Dresser, BL; Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Buck, DJ; Davis, RL; Saffarian, N; Stevens, CW1
Dannals, RF; Frost, JJ; Kim, YK; Lee, JS; McCaul, ME; Wand, GS; Weerts, EM1
Greenwald, MK1
Butelman, ER; Chait, BT; Kreek, MJ; Mandau, M; Reed, B; Yuferov, V1
Virk, MS; Williams, JT1
Arastu, MF; Dean, RL; Deaver, DR; Dong, N; Gastfriend, DR; Kriksciukaite, K; O'Driscoll, K; Reitano, K; Todtenkopf, MS1
Martin, KK; Stahlheber, BW; Stevens, CW1
Bear, AE; Folk, JE; Negus, SS; Rice, KC1
Alonso, A; Darstein, C; Molenberghs, G; Renard, D1
Arout, C; Caldwell, M; Dahan, A; Kest, B; Waxman, AR1
Baud, FJ; Chevillard, L; Mégarbane, B; Risède, P1
Darwish, M; Kirby, M; Robertson, P; Tracewell, W; Xie, F1
Erickson, TB; George, AV; Lu, JJ; Metz, J; Pisano, MV1
Caulkett, NA; Shury, TK; Woodbury, MR1
Boyce, M; Eriksson, C; Kilborn, J; Lister, N; Tamaoka, M; Warrington, S1
Bührer, C; Degenhardt, P; Garten, L1
Beaver, J; Bullmore, ET; Bush, MA; Gunn, RN; Hill, S; Howard, J; Long, C; Makwana, A; Matthews, PM; Miller, SR; Nathan, PJ; Newbould, RD; Passchier, J; Rabiner, EA; Reiley, R; Searle, G1
Bihel, F; Bockel, F; Bourguignon, JJ; Elhabazi, K; Maldonado, R; Meziane, H; Mollereau, C; Moulédous, L; Petit-demoulière, B; Schmitt, M; Simonin, F; Trigo, JM; Zajac, JM1
Chateauraynaud, J; Gavello-Baudy, S; Laboureyras, E; Laulin, JP; Le Roy, C; Simonnet, G1
Moore, KT; Natarajan, J; Richarz, U; Sathyan, G; Vandenbossche, J1
Bobeck, EN; Haseman, RA; Hong, D; Ingram, SL; Morgan, MM1
Banks, ML; Lunzer, MM; Negus, SS; Portoghese, PS; Rice, KC; Yekkirala, AS1
Kellie, KA; Kreeger, TJ1
Chavan, A; Dillaha, L; Goskonda, V; Parikh, N1
Kalk, P; Moore, RP; Rainwater, KL; Sykes, JM; Valitutto, MT1
Bilsky, EJ; Cain, JP; Hruby, VJ; Hu, J; Kumirov, VK; Lee, YS; Podolsky, AT; Sandweiss, A; Vanderah, TW; Vardanyan, RS1
Dong, H; Gao, X; Gong, Z; Ma, W; Su, R; Yong, Z1
Herrero, JF; Herrero-Zorita, C; Ramos-Zepeda, GA1
Bell, RL; Gonzales, CR; Hart, JC; Lowe, SL; McKinzie, DL; McKinzie, JH; Mitch, CH; Need, AB; Rorick-Kehn, LM; Statnick, MA; Stoltz, RR; Suico, JG; Tauscher-Wisniewski, S; Weller, MA; Witcher, JW; Wong, CJ1
Cui, XL; Li, RP; Liao, X; Liu, GP; Sun, C; Wang, SY; Xu, YC; Xue, FS; Yang, GZ1
Lindsey, AM; Prinssen, EP; Rice, KC; Saccone, PA; Sulima, A; Wichmann, J; Woods, JH; Zelenock, KA1
Buck, RK; Fosgate, GT; Gerlach, C; Kästner, SBR; Kummrow, M; Meyer, LRC; Stegmann, GF; Zeiler, GE1
Batra, A; Hansson, AC; Hermann, D; Hirth, N; Hoffmann, S; Kiefer, F; la Fougère, C; Mann, K; Noori, HR; Reimold, M; Reischl, G; Smolka, MN; Sommer, WH; Spanagel, R1
Altshuler, D; Merchan, C; Papadopoulos, J1
Alexander-Scott, N; Boss, R; Brinkley-Rubinstein, L; Clarke, J; Green, TC; Marshall, BDL; Rich, JD1
Banks, ML; Negus, SS; Schwienteck, KL1
Abad-Santos, F; Alday, E; Belmonte, C; Hernández-Martínez, M; Herrador, C; Koller, D; Mejía, G; Ochoa, D; Román, M; Saiz-Rodríguez, M; Zubiaur, P1
Banks, ML; Blough, BE; Faunce, KE; Grim, TW; Negus, SS; Obeng, S; Rice, KC; Schwienteck, KL; Zhang, Y1
Heller, NM; Maher, DP; Walia, D1
Beeker, A; Berkhof, J; Neefjes, ECW; Rhodius, CA; Ten Oever, D; van den Berg, HP; van der Vliet, HJ; van der Vorst, MJDL; van der Wijngaart, H; Verheul, HMW1
Banks, ML; Blake, S; Bremer, PT; Faunce, KE; Hwang, CS; Janda, KD; Natori, Y; Townsend, EA; Zhou, B1
Banks, ML; Blake, S; Bremer, PT; Hwang, CS; Janda, KD; Poklis, JL; Tenney, RD; Zhou, B1
Banks, ML; Blake, S; Bremer, PT; Negus, SS; Poklis, JL; Schwienteck, KL; Townsend, EA1
McCranor, BJ; Pierce, SA; Racine, MC; Sciuto, AM; Tressler, J; Tuet, WY; Wong, B1
Bardo, MT; Beckmann, JS; Hammerslag, LR; Hofford, RS; Kang, Q; Kryscio, RJ1
Chen, Y; Fu, C; Hu, R; Huang, C; Jiang, H; Li, C; Sun, Y; Tang, D; Wang, H; Yan, J; Zhu, J1
Banks, ML; Bremer, PT; Faunce, KE; Janda, KD; Jaster, AM; Negus, SS; Robinson, HL; Townsend, EA1
Disney, A; France, CP; Gerak, LR; Husbands, SM; Javors, MA; Maguire, DR; Sanchez, JJ1
Freier, A; Lorch, U; Pierscionek, T; Spencer, CS; Täubel, J1
Baamonde, A; González-Rodríguez, S; Lastra, A; Machelska, H; Menéndez, L; Seitz, V; Stein, C1
Townsend, EA1
Gault, A; Wahl, G1
Flynn, SM; France, CP1
Baynard, C; Butelman, ER; Hedrick, SL; Horn, J; Jackson, K; Kaska, S; Kreek, MJ; Leggas, M; Luo, D; Niloy, KK; Prisinzano, TE; Sarma, R1
Cook, RR; Fanucchi, L; Foot, C; King, C; Korthuis, PT; Lucas, GM; Lum, PJ; Rodriguez, A; Tookes, H; Torralva, R; Vergara-Rodriguez, P; Waddell, EN1
Laks, J; Peterkin, A; Weinstein, ZM1
Schmitz, ZP; Soghoian, SE; Warstadt, NM1
Banks, ML; Negus, SS; Santos, EJ1
Marcus, MM; St Onge, CM; Taylor, KM; Townsend, EA1
Inomata, A; Makino, K; Moriyasu, T; Nakagawa, Y; Nakajima, J; Ono, Y; Sakamoto, M; Suzuki, J; Suzuki, T; Tada, Y; Takahashi, H; Tayama, K1
Bassman, JR; Beardsley, PM; Hassanien, SH; Holt, MC; Iula, DM; Layle, NK; Stevens, DL; Varshneya, NB1
Benner, JD; Cohen, SM; Fishman, M; Hollenbaugh, JA1

Reviews

2 review(s) available for naltrexone and fentanyl

ArticleYear
Drug discrimination studies.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Analgesics, Opioid; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Generalization, Stimulus; Macaca mulatta; Morphine; Nalorphine; Naloxone; Naltrexone; Pentazocine; Phenazocine; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Current Best Practices for Acute and Chronic Management of Patients with Opioid Use Disorder.
    The Medical clinics of North America, 2022, Volume: 106, Issue:1

    Topics: Adult; Analgesics, Opioid; Buprenorphine; Comorbidity; Disease Management; Drug Overdose; Female; Fentanyl; Harm Reduction; Humans; Male; Mental Disorders; Methadone; Middle Aged; Naltrexone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Practice Guidelines as Topic; Prevalence

2022

Trials

18 trial(s) available for naltrexone and fentanyl

ArticleYear
Prolonged blockade of opioid effect with oral nalmefene.
    Clinical pharmacology and therapeutics, 1986, Volume: 40, Issue:5

    Topics: Administration, Oral; Adult; Analgesia; Clinical Trials as Topic; Double-Blind Method; Fentanyl; Humans; Male; Naltrexone; Narcotic Antagonists; Respiration; Time Factors

1986
Prolonged antagonism of opioid action with intravenous nalmefene in man.
    Anesthesiology, 1986, Volume: 64, Issue:2

    Topics: Adult; Drug Interactions; Fentanyl; Humans; Male; Muscle Rigidity; Naltrexone; Pain; Respiration; Tidal Volume; Time Factors

1986
Efficacy and safety of naltrexone hydrochloride for antagonizing carfentanil citrate immobilization in captive Rocky Mountain elk (Cervus elaphus nelsoni).
    Journal of wildlife diseases, 1996, Volume: 32, Issue:2

    Topics: Analgesics, Opioid; Animals; Deer; Female; Fentanyl; Immobilization; Male; Naltrexone; Narcotic Antagonists

1996
Longer occupancy of opioid receptors by nalmefene compared to naloxone as measured in vivo by a dual-detector system.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1997, Volume: 38, Issue:11

    Topics: Adult; Analgesics, Opioid; Brain; Carbon Radioisotopes; Cross-Over Studies; Female; Fentanyl; Humans; Male; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Time Factors; Tomography, Emission-Computed

1997
Maximum tolerated dose of nalmefene in patients receiving epidural fentanyl and dilute bupivacaine for postoperative analgesia.
    Anesthesiology, 2000, Volume: 92, Issue:4

    Topics: Adult; Aged; Analgesia, Epidural; Analgesics, Opioid; Anesthetics, Local; Bupivacaine; Female; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Pain, Postoperative

2000
Nalmefene for elective reversal of procedural sedation in children.
    The American journal of emergency medicine, 2001, Volume: 19, Issue:7

    Topics: Analgesics, Opioid; Anesthetics, Intravenous; Antidotes; Child; Child, Preschool; Emergency Medical Services; Female; Fentanyl; Humans; Infant; Male; Midazolam; Naltrexone; Narcotic Antagonists

2001
Prolonged central mu-opioid receptor occupancy after single and repeated nalmefene dosing.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:12

    Topics: Adolescent; Adult; Analgesics, Opioid; Area Under Curve; Caudate Nucleus; Electrocardiography; Fentanyl; Glucuronides; Humans; Male; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Prefrontal Cortex; Receptors, Opioid, mu; Thalamus

2005
Single-dose and steady-state pharmacokinetics of fentanyl buccal tablet in healthy volunteers.
    Journal of clinical pharmacology, 2007, Volume: 47, Issue:1

    Topics: Administration, Buccal; Adolescent; Adult; Chromatography, High Pressure Liquid; Drug Tolerance; Female; Fentanyl; Half-Life; Humans; Male; Middle Aged; Naltrexone; Tablets; Tandem Mass Spectrometry; Time Factors

2007
Dose proportionality of fentanyl buccal tablet in doses ranging from 600 to 1300 microg in healthy adult subjects: a randomized, open-label, four-period, crossover, single-centre study.
    Clinical drug investigation, 2010, Volume: 30, Issue:6

    Topics: Administration, Buccal; Adolescent; Adult; Analgesics, Opioid; Area Under Curve; Cross-Over Studies; Dose-Response Relationship, Drug; Female; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Time Factors; Young Adult

2010
Pharmacokinetics, safety, and tolerability of ascending doses of sublingual fentanyl, with and without naltrexone, in Japanese subjects.
    Journal of clinical pharmacology, 2011, Volume: 51, Issue:8

    Topics: Absorption; Administration, Sublingual; Adult; Analgesics, Opioid; Asian People; Blood Gas Monitoring, Transcutaneous; Dose-Response Relationship, Drug; Drug Interactions; Drug Monitoring; Female; Fentanyl; Half-Life; Humans; Japan; Male; Mouth Mucosa; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Respiratory Insufficiency; Tablets; Young Adult

2011
Pharmacological differentiation of opioid receptor antagonists by molecular and functional imaging of target occupancy and food reward-related brain activation in humans.
    Molecular psychiatry, 2011, Volume: 16, Issue:8

    Topics: Adult; Amygdala; Brain; Brain Mapping; Corpus Striatum; Dose-Response Relationship, Drug; Fentanyl; Food; Humans; Indans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Radioligand Assay; Radionuclide Imaging; Reward; Triazoles

2011
Randomized 5-treatment crossover study to assess the effects of external heat on serum fentanyl concentrations during treatment with transdermal fentanyl systems.
    Journal of clinical pharmacology, 2012, Volume: 52, Issue:8

    Topics: Administration, Cutaneous; Adolescent; Adult; Analgesics, Opioid; Area Under Curve; Combined Modality Therapy; Cross-Over Studies; Female; Fentanyl; Humans; Hyperthermia, Induced; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Young Adult

2012
Pharmacokinetics and dose proportionality of fentanyl sublingual spray: a single-dose 5-way crossover study.
    Clinical drug investigation, 2013, Volume: 33, Issue:6

    Topics: Administration, Sublingual; Adolescent; Adult; Analgesics, Opioid; Analysis of Variance; Area Under Curve; Biological Availability; Cross-Over Studies; Dose-Response Relationship, Drug; Female; Fentanyl; Humans; Hydrogen-Ion Concentration; Linear Models; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Single-Blind Method; Temperature; Young Adult

2013
Determining pharmacological selectivity of the kappa opioid receptor antagonist LY2456302 using pupillometry as a translational biomarker in rat and human.
    The international journal of neuropsychopharmacology, 2014, Oct-31, Volume: 18, Issue:2

    Topics: Adolescent; Adult; Animals; Benzamides; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Fentanyl; Humans; Male; Middle Aged; Miosis; Morphine; Mydriasis; Naltrexone; Narcotic Antagonists; Narcotics; Pupil; Pyrrolidines; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Young Adult

2014
Low μ-Opioid Receptor Status in Alcohol Dependence Identified by Combined Positron Emission Tomography and Post-Mortem Brain Analysis.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2017, Volume: 42, Issue:3

    Topics: Adult; Aged; Alcoholism; Analgesics, Opioid; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Receptors, Opioid, mu; Tissue Banks; Ventral Striatum

2017
Polymorphisms associated with fentanyl pharmacokinetics, pharmacodynamics and adverse effects.
    Basic & clinical pharmacology & toxicology, 2019, Volume: 124, Issue:3

    Topics: Adolescent; Adult; Analgesics, Opioid; ATP Binding Cassette Transporter, Subfamily B; Catechol O-Methyltransferase; Cross-Over Studies; Cytochrome P-450 Enzyme System; Female; Fentanyl; Gene Frequency; Genotype; Humans; Male; Middle Aged; Naltrexone; Pharmacogenetics; Polymorphism, Genetic; Receptors, Adrenergic, beta-1; Receptors, Opioid, mu; Young Adult

2019
Safety, Tolerability, and Dose Proportionality of a Novel Transdermal Fentanyl Matrix Patch and Bioequivalence With a Matrix Fentanyl Patch: Two Phase 1 Single-Center Open-Label, Randomized Crossover Studies in Healthy Japanese Volunteers.
    Clinical pharmacology in drug development, 2021, Volume: 10, Issue:3

    Topics: Administration, Cutaneous; Adult; Analgesics, Opioid; Area Under Curve; Biological Availability; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Compounding; Drug Delivery Systems; Drug Tolerance; Fentanyl; Healthy Volunteers; Humans; Japan; Naltrexone; Narcotic Antagonists; Reproducibility of Results; Safety; Therapeutic Equivalency; Transdermal Patch

2021
Associations between fentanyl use and initiation, persistence, and retention on medications for opioid use disorder among people living with uncontrolled HIV disease.
    Drug and alcohol dependence, 2021, 11-01, Volume: 228

    Topics: Buprenorphine; Delayed-Action Preparations; Fentanyl; HIV Infections; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders

2021

Other Studies

145 other study(ies) available for naltrexone and fentanyl

ArticleYear
Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:2

    Topics: Analgesics; Animals; Binding Sites; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Ligands; PC12 Cells; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Software

1994
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Extrapolation of human pharmacokinetic parameters from rat, dog, and monkey data: Molecular properties associated with extrapolative success or failure.
    Journal of pharmaceutical sciences, 2005, Volume: 94, Issue:7

    Topics: Algorithms; Animals; Dogs; Haplorhini; Humans; Pharmaceutical Preparations; Pharmacokinetics; Rats; Species Specificity; Tissue Distribution

2005
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Opioids as Substrates and Inhibitors of the Genetically Highly Variable Organic Cation Transporter OCT1.
    Journal of medicinal chemistry, 2019, 11-14, Volume: 62, Issue:21

    Topics: Analgesics, Opioid; HEK293 Cells; Humans; Inhibitory Concentration 50; Models, Molecular; Organic Cation Transporter 1; Permeability; Protein Conformation

2019
Clocinnamox: a novel, systemically-active, irreversible opioid antagonist.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Analgesia; Animals; Cinnamates; Dose-Response Relationship, Drug; Fentanyl; Male; Mice; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Receptors, Opioid

1992
The noradrenergic component contributing to spinal fentanyl-induced antinociception is supraspinally mediated.
    General pharmacology, 1992, Volume: 23, Issue:6

    Topics: Adrenergic Antagonists; Analgesics; Animals; Fentanyl; Injections, Intraventricular; Injections, Spinal; Male; Methysergide; Naltrexone; Norepinephrine; Pain Measurement; Phentolamine; Rats; Rats, Sprague-Dawley; Reaction Time; Serotonin Antagonists; Spinal Cord

1992
Pharmacological profiles of fentanyl analogs at mu, delta and kappa opiate receptors.
    European journal of pharmacology, 1992, Mar-24, Volume: 213, Issue:2

    Topics: Analgesics, Opioid; Animals; Benzeneacetamides; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Fentanyl; Guinea Pigs; Ileum; Male; Mice; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1992
Ostrich (Struthio camelus) immobilisation using carfentanil and xylazine and reversal with yohimbine and naltrexone.
    Journal of the South African Veterinary Association, 1992, Volume: 63, Issue:4

    Topics: Animals; Birds; Fentanyl; Immobilization; Naltrexone; Xylazine; Yohimbine

1992
Apparent pA2 value of naltrexone is not changed in rats following continuous exposure to morphine or naloxone.
    Life sciences, 1992, Volume: 50, Issue:19

    Topics: Analysis of Variance; Animals; Body Weight; Dose-Response Relationship, Drug; Drug Interactions; Fentanyl; Male; Morphine; Naloxone; Naltrexone; Pain Measurement; Rats; Rats, Inbred Strains

1992
Mirfentanil: pharmacological profile of a novel fentanyl derivative with opioid and nonopioid effects.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: Alfentanil; Analgesics; Animals; Columbidae; Discrimination Learning; Female; Fentanyl; In Vitro Techniques; Macaca mulatta; Male; Morphine; Naltrexone; Receptors, Opioid; Receptors, Opioid, mu; Respiration; Self Administration; Structure-Activity Relationship

1991
Characteristics of dose-dependent antagonism by beta-funaltrexamine of the antinociceptive effects of intrathecal mu agonists.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: Analgesics; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Fentanyl; Injections, Spinal; Male; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Spinal Cord; Sufentanil

1991
Evaluation of receptor mechanism mediating fentanyl analgesia and toxicity.
    European journal of pharmacology, 1991, May-17, Volume: 197, Issue:2-3

    Topics: Analgesics; Animals; Brain; Drug Tolerance; Fentanyl; Lethal Dose 50; Male; Mice; Morphine; Naloxone; Naltrexone; Receptors, Opioid

1991
Opiate receptor antagonists for delusions of parasitosis.
    Biological psychiatry, 1991, Sep-01, Volume: 30, Issue:5

    Topics: Delusions; Female; Fentanyl; Fluspirilene; Humans; Middle Aged; Myiasis; Naloxone; Naltrexone; Narcotic Antagonists

1991
Separate neural mechanisms mediate sufentanil-induced pupillary responses in the cat.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:3

    Topics: Analgesics, Opioid; Animals; Cats; Clonidine; Drug Interactions; Fentanyl; Male; Morphine; Mydriasis; Naltrexone; Pupil; Receptors, Opioid; Receptors, Opioid, mu; Sufentanil

1991
Paradoxical effect of chronic fentanyl treatment on naltrexone-induced supersensitivity and upregulation.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:1

    Topics: Analgesia; Animals; Autoradiography; Behavior, Animal; Discrimination Learning; Dose-Response Relationship, Drug; Drug Hypersensitivity; Drug Interactions; Fentanyl; Male; Naltrexone; Narcotics; Nociceptors; Rats; Rats, Inbred Strains; Time Factors; Up-Regulation

1992
Protection by U-50,488H against beta-chlornaltrexamine antagonism of nitrous oxide antinociception in mice.
    Brain research, 1991, May-17, Volume: 549, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Analgesics; Animals; Fentanyl; Male; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nitrous Oxide; Pain; Pyrrolidines; Sufentanil

1991
Effects of sufentanil and naltrexone on adrenal vein catecholamines and neuropeptides during splanchnic nerve stimulation in cats.
    Synapse (New York, N.Y.), 1990, Volume: 6, Issue:4

    Topics: Adrenal Glands; Analgesics; Animals; Blood Pressure; Catecholamines; Cats; Electric Stimulation; Fentanyl; Heart Rate; Naltrexone; Neuropeptides; Splanchnic Nerves; Sufentanil; Veins

1990
Assessment of relative intrinsic activity of mu-opioid analgesics in vivo by using beta-funaltrexamine.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Fentanyl; Levorphanol; Male; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Time Factors

1990
Suppression of natural killer cell activity by high-dose narcotic anesthesia in rats.
    Brain, behavior, and immunity, 1989, Volume: 3, Issue:2

    Topics: Anesthesia; Cytotoxicity Tests, Immunologic; Dose-Response Relationship, Drug; Fentanyl; Interferons; Killer Cells, Natural; Morphine; Naltrexone; Sufentanil; Time Factors

1989
Opioid receptors on cells of the immune system: evidence for delta- and kappa-classes.
    The Journal of endocrinology, 1989, Volume: 122, Issue:1

    Topics: Animals; Benzeneacetamides; Cell Line; Fentanyl; Indicators and Reagents; Macrophages; Mice; Mice, Inbred C57BL; Naltrexone; Pyrrolidines; Receptors, Opioid

1989
Fentanyl produces cholinergically-mediated analeptic and EEG arousal effects in rats.
    Neuropharmacology, 1989, Volume: 28, Issue:5

    Topics: Anesthesia; Animals; Atropine; Brain; Central Nervous System Stimulants; Choline; Electroencephalography; Fentanyl; Hippocampus; Injections; Male; Naltrexone; Parasympathetic Nervous System; Pentobarbital; Rats; Rats, Inbred Strains; Sleep; Stimulation, Chemical

1989
Chloroacryloyl amides and alpha-methylenelactones from naltrexone, oxymorphone and fentanyl.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Acrylates; Animals; Binding Sites; Brain; Chemical Phenomena; Chemistry; Fentanyl; Hydromorphone; In Vitro Techniques; Membranes; Naloxone; Naltrexone; Oxymorphone; Rats; Stereoisomerism

1985
Urine testing in impaired physicians.
    Missouri medicine, 1989, Volume: 86, Issue:6

    Topics: Fentanyl; Humans; Naltrexone; Opioid-Related Disorders; Patient Compliance; Physician Impairment

1989
Duration of occupancy of opiate receptors by naltrexone.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1988, Volume: 29, Issue:7

    Topics: Administration, Oral; Adult; Brain; Carbon Radioisotopes; Female; Fentanyl; Humans; Male; Naltrexone; Radionuclide Imaging; Receptors, Opioid; Receptors, Opioid, mu; Time Factors

1988
Kappa antagonist properties of buprenorphine in the shock titration procedure.
    European journal of pharmacology, 1988, Oct-26, Volume: 156, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Buprenorphine; Electroshock; Fentanyl; Male; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Saimiri

1988
An analysis of naltrexone and naloxone's possible agonistic actions in the dog.
    Drug and alcohol dependence, 1985, Volume: 15, Issue:4

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Dogs; Drug Synergism; Electroencephalography; Ethylketocyclazocine; Evoked Potentials; Female; Fentanyl; Morphine; Naloxone; Naltrexone; Reaction Time; Reflex; Reflex, Pupillary

1985
High dose of spinal morphine produce a nonopiate receptor-mediated hyperesthesia: clinical and theoretic implications.
    Anesthesiology, 1986, Volume: 64, Issue:5

    Topics: Anesthesia, Spinal; Animals; Blood Pressure; Cats; Drug Tolerance; Fentanyl; Hyperesthesia; Methadone; Morphine; Morphine Derivatives; Naltrexone; Rats; Receptors, Drug; Stimulation, Chemical; Strychnine; Sufentanil; Sulfates; Touch

1986
The effect of opioids on rat plasma atrial natriuretic peptide.
    European journal of pharmacology, 1987, Nov-17, Volume: 143, Issue:3

    Topics: Amino Acids; Animals; Atrial Natriuretic Factor; Chromatography, High Pressure Liquid; Clonidine; Dose-Response Relationship, Drug; Fentanyl; Male; Naltrexone; Narcotics; Radioimmunoassay; Rats; Rats, Inbred Strains

1987
Effect of mu and kappa opioid receptor agonists on rat plasma corticosterone levels.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Corticosterone; Dose-Response Relationship, Drug; Fentanyl; Male; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Reversal by beta-funaltrexamine of the antinociceptive effect of opioid agonists in the rat.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Buprenorphine; Cyclazocine; Ethylketocyclazocine; Fentanyl; Male; Naltrexone; Pain; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Biological Assay; Buprenorphine; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Etorphine; Fentanyl; Methadone; Mice; Morphine; Muscle Contraction; Nalbuphine; Nalorphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, mu

1987
Prevention of late fentanyl-induced respiratory depression after the injection of opiate antagonists naltrexone and S-20682: comparison with naloxone.
    British journal of anaesthesia, 1983, Volume: 55, Issue:1

    Topics: Animals; Carbon Dioxide; Depression, Chemical; Dogs; Electroencephalography; Fentanyl; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Oxygen; Partial Pressure; Respiration; Time Factors

1983
Receptor preference of dynorphin A fragments in the mouse vas deferens determined by different techniques.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Animals; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Fentanyl; Male; Mice; Naloxone; Naltrexone; Peptide Fragments; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1984
Potential affinity labels for the opiate receptor based on fentanyl and related compounds.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:8

    Topics: Affinity Labels; Animals; Chemical Phenomena; Chemistry; Fentanyl; In Vitro Techniques; Naloxone; Naltrexone; Rats; Rats, Inbred Strains; Receptors, Opioid

1982
Intraseptally injected opiate agents: effects on morphine-induced behaviour of cats.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:2

    Topics: Animals; Behavior, Animal; beta-Endorphin; Cats; Endorphins; Enkephalin, Methionine; Fentanyl; Morphine; Naloxone; Naltrexone; Narcotics; Receptors, Opioid; Septal Nuclei; Septum Pellucidum

1982
Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures.
    Journal of wildlife diseases, 1995, Volume: 31, Issue:1

    Topics: Analgesics, Opioid; Animals; Bison; Diprenorphine; Drug Combinations; Female; Fentanyl; Hypnotics and Sedatives; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Naloxone; Naltrexone; Narcotic Antagonists; Northwest Territories; Piperidines; Tranquilizing Agents; Xylazine

1995
Electrophysiological demonstration and activation of mu-opioid receptors in the rabbit sinoatrial node.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:1

    Topics: Action Potentials; Animals; Enkephalin, Leucine; Fentanyl; Microelectrodes; Naltrexone; Narcotic Antagonists; Narcotics; Patch-Clamp Techniques; Rabbits; Receptors, Opioid, mu; Sinoatrial Node

1995
Behavioral effects and receptor binding affinities of fentanyl derivatives in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:1

    Topics: Animals; Behavior, Animal; Fentanyl; Heart Rate; Macaca mulatta; Nalbuphine; Naltrexone; Receptors, Opioid, delta; Receptors, Opioid, mu; Respiration; Self Administration

1995
Evaluation of diurnal variation in fentanyl clearance.
    Journal of clinical pharmacology, 1995, Volume: 35, Issue:2

    Topics: Circadian Rhythm; Drug Administration Schedule; Fentanyl; Humans; Infusions, Intravenous; Male; Metabolic Clearance Rate; Naltrexone

1995
Complications with the use of carfentanil citrate and xylazine hydrochloride to immobilize domestic horses.
    Journal of the American Veterinary Medical Association, 1995, Mar-15, Volume: 206, Issue:6

    Topics: Analgesics, Opioid; Animals; Animals, Domestic; Fentanyl; Horse Diseases; Horses; Hypertension; Immobilization; Naloxone; Naltrexone; Pulmonary Edema; Tachycardia; Xylazine

1995
OHM3295: a fentanyl-related 4-heteroanilido piperidine with analgesic effects but not suppressive effects on splenic NK activity in mice.
    International journal of immunopharmacology, 1994, Volume: 16, Issue:10

    Topics: Analgesics; Animals; Fentanyl; Immunosuppressive Agents; Killer Cells, Natural; Male; Mice; Naltrexone; Spleen

1994
Mechanisms of morphine-induced immunosuppression: effect of acute morphine administration on lymphocyte trafficking.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:3

    Topics: Adrenalectomy; Animals; Cell Movement; Fentanyl; Immunosuppression Therapy; Leukocyte Count; Lymphocyte Activation; Lymphocyte Count; Lymphocytes; Male; Morphine; Naltrexone; Rats; Rats, Sprague-Dawley; T-Lymphocyte Subsets

1995
In vivo apparent pA2 analysis for naltrexone antagonism of discriminative stimulus and analgesic effects of opiate agonists in rats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: Analgesia; Animals; Benzomorphans; Buprenorphine; Discrimination, Psychological; Etorphine; Fentanyl; Male; Morphine; Nalbuphine; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu

1994
Opioid antagonist-induced receptor upregulation: effects of concurrent agonist administration.
    Brain research bulletin, 1994, Volume: 33, Issue:2

    Topics: Animals; Brain; Drug Combinations; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Fentanyl; Male; Mice; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Up-Regulation

1994
Duration of opioid antagonism by nalmefene and naloxone in the dog: an integrated pharmacokinetic/pharmacodynamic comparison.
    Journal of pharmaceutical sciences, 1995, Volume: 84, Issue:9

    Topics: Animals; Blood Gas Monitoring, Transcutaneous; Dogs; Female; Fentanyl; Infusions, Intravenous; Models, Biological; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Respiration

1995
Duration of opioid antagonism by nalmefene and naloxone in the dog. A nonparametric pharmacodynamic comparison based on generalized cross-validated spline estimation.
    International journal of clinical pharmacology and therapeutics, 1995, Volume: 33, Issue:10

    Topics: Analysis of Variance; Animals; Carbon Dioxide; Computer Simulation; Cross-Over Studies; Dogs; Drug Tolerance; Fentanyl; Injections, Intravenous; Male; Models, Statistical; Naloxone; Naltrexone; Narcotic Antagonists; Respiratory Insufficiency; Time Factors

1995
Immobilization of black bears (Ursus americanus) with orally administered carfentanil citrate.
    Journal of wildlife diseases, 1995, Volume: 31, Issue:3

    Topics: Administration, Oral; Analgesics, Opioid; Animals; Diazepam; Female; Fentanyl; Immobilization; Male; Muscle Relaxants, Central; Muscle, Skeletal; Naltrexone; Narcotic Antagonists; Oxygen; Respiration; Ursidae

1995
Replacement of Gln280 by His in TM6 of the human ORL1 receptor increases affinity but reduces intrinsic activity of opioids.
    FEBS letters, 1996, Oct-14, Volume: 395, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Diprenorphine; Dynorphins; Etorphine; Fentanyl; Glutamine; Histamine; Humans; Kinetics; Ligands; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid

1996
Effects of the delta opioid against BW373U86 in pigeons trained to discriminate fentanyl, bremazocine and water in a three-choice drug discrimination procedure.
    Psychopharmacology, 1996, Volume: 126, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Columbidae; Discrimination, Psychological; Female; Fentanyl; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Piperazines; Receptors, Opioid, delta

1996
Reversal by kappa-agonists of peritoneal irritation-induced ileus and visceral pain in rats.
    Life sciences, 1997, Volume: 60, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetic Acid; Analgesics; Animals; Benzofurans; Benzomorphans; Cyclazocine; Fentanyl; Gastric Emptying; Intestinal Pseudo-Obstruction; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Peritoneum; Pyrroles; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thiophenes

1997
In vivo binding of [125I]NH2-carfentanil to mu opioid receptors in mouse brain.
    Nuclear medicine and biology, 1994, Volume: 21, Issue:2

    Topics: Animals; Autoradiography; Brain; Fentanyl; Injections, Intraperitoneal; Iodine Radioisotopes; Logistic Models; Mice; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Radioligand Assay; Receptors, Opioid, mu

1994
Antagonism of morphine-like discriminative effects by beta-funaltrexamine.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 57, Issue:4

    Topics: Analgesics, Opioid; Animals; Buprenorphine; Cisterna Magna; Discrimination Learning; Fentanyl; Injections; Male; Meperidine; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

1997
Supraspinal administration of opioids with selectivity for mu-, delta- and kappa-opioid receptors produces analgesia in amphibians.
    European journal of pharmacology, 1997, Jul-16, Volume: 331, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzofurans; Dose-Response Relationship, Drug; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Female; Fentanyl; Injections, Intraventricular; Male; Morphine; Naltrexone; Narcotics; Pyrrolidines; Rana pipiens; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1997
Immobilization of domestic goats (Capra hircus) using orally administered carfentanil citrate and detomidine hydrochloride.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1997, Volume: 28, Issue:2

    Topics: Absorption; Administration, Oral; Adrenergic alpha-Antagonists; Analgesics; Analgesics, Opioid; Animals; Blood Pressure; Body Temperature; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Female; Fentanyl; Goats; Heart Rate; Hypnotics and Sedatives; Imidazoles; Immobilization; Naltrexone; Narcotic Antagonists; Respiration; Saponins; Yohimbine

1997
Cardiopulmonary effects of carfentanil in dama gazelles (Gazella dama).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1997, Volume: 28, Issue:2

    Topics: Analgesics, Opioid; Animals; Animals, Zoo; Antelopes; Blood Gas Analysis; Blood Pressure; Carbon Dioxide; Female; Fentanyl; Heart Rate; Immobilization; Male; Naltrexone; Narcotic Antagonists; Oximetry; Oxygen; Pregnancy; Reproducibility of Results; Respiration

1997
Spinal mu, delta and kappa opioids alter chemical, mechanical and thermal sensitivities in amphibians.
    Life sciences, 1997, Volume: 61, Issue:22

    Topics: Analgesics, Opioid; Animals; Drug Interactions; Enkephalin, Leucine-2-Alanine; Fentanyl; Injections, Spinal; Morphine; Naltrexone; Narcotic Antagonists; Nociceptors; Pain Measurement; Pain Threshold; Rana pipiens; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sensitivity and Specificity; Spinal Cord

1997
The rate-decreasing effects of fentanyl derivatives in pigeons before, during and after chronic morphine treatment.
    Psychopharmacology, 1998, Volume: 137, Issue:1

    Topics: Analgesics; Animals; Columbidae; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Tolerance; Fentanyl; Morphine; Naltrexone

1998
Rapid opioid detoxification.
    JAMA, 1998, Jun-17, Volume: 279, Issue:23

    Topics: Adult; Drug Implants; Fentanyl; Humans; Male; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders

1998
Pharmacological profile of a deuterium-substituted mirfentanil derivative, OHM10579, in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Deuterium; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Fentanyl; Macaca mulatta; Male; Nalbuphine; Naltrexone; Narcotic Antagonists; Pain Measurement; Respiratory Mechanics

1998
Health evaluation of free-ranging guanaco (Lama guanicoe).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1998, Volume: 29, Issue:2

    Topics: Analgesics, Opioid; Anesthetics; Animals; Animals, Domestic; Animals, Wild; Antibodies; Antidotes; Blood Chemical Analysis; Camelids, New World; Communicable Diseases; Drug Combinations; Enzymes; Female; Fentanyl; Flumazenil; Health Status; Immobilization; Male; Minerals; Naltrexone; Narcotic Antagonists; Physical Examination; Reference Values; Sheep; Tiletamine; Vitamins; Zolazepam

1998
Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor.
    European journal of pharmacology, 1998, Aug-07, Volume: 354, Issue:2-3

    Topics: Analgesics; Animals; Binding, Competitive; CHO Cells; Cricetinae; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Ligands; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Peptide Fragments; Peptides; Radioligand Assay; Rats; Receptors, Opioid, mu; Somatostatin; Sufentanil; Thermodynamics; Time Factors

1998
The mu opioid irreversible antagonist beta-funaltrexamine differentiates the discriminative stimulus effects of opioids with high and low efficacy at the mu opioid receptor.
    Psychopharmacology, 1998, Volume: 140, Issue:1

    Topics: Animals; Buprenorphine; Butorphanol; Columbidae; Discrimination Learning; Female; Fentanyl; Levallorphan; Methadone; Morphine; Nalbuphine; Nalorphine; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu

1998
Effect of gonadectomy on discriminative stimulus effects of morphine in female versus male rats.
    Drug and alcohol dependence, 1999, Jan-07, Volume: 53, Issue:2

    Topics: Animals; Buprenorphine; Castration; Discrimination Learning; Female; Fentanyl; Gonadal Steroid Hormones; Injections; Male; Morphine; Nalbuphine; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptors; Rats; Rats, Sprague-Dawley; Sex Characteristics

1999
Modulation of emesis by fentanyl and opioid receptor antagonists in Suncus murinus (house musk shrew).
    European journal of pharmacology, 1999, Jun-11, Volume: 374, Issue:1

    Topics: Animals; Antiemetics; Female; Fentanyl; Male; Naloxone; Naltrexone; Narcotic Antagonists; Nicotine; Receptors, Opioid; Shrews; Vomiting

1999
Discriminative stimulus effects of morphine in squirrel monkeys: stimulants, opioids, and stimulant-opioid combinations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Amphetamine; Analgesics, Opioid; Anesthetics, Local; Animals; Anti-Anxiety Agents; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Combinations; Fentanyl; Male; Morphine; Naltrexone; Narcotic Antagonists; Piperazines; Receptors, Opioid; Saimiri; Selective Serotonin Reuptake Inhibitors

1999
Effects of a novel fentanyl derivative on drug discrimination and learning in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 64, Issue:2

    Topics: Analgesics, Opioid; Animals; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Fentanyl; Macaca mulatta; Naltrexone; Narcotic Antagonists; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule

1999
Discriminative stimulus effects of two doses of fentanyl in rats: pharmacological selectivity and effect of training dose on agonist and antagonist effects of mu opioids.
    Psychopharmacology, 2000, Volume: 148, Issue:2

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Operant; Dextroamphetamine; Dose-Response Relationship, Drug; Fentanyl; Male; Methadone; Morphine; Nalbuphine; Nalorphine; Naltrexone; Narcotic Antagonists; Narcotics; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu

2000
Daily mirfentanil induces (cross-) tolerance to the rate-decreasing effects of morphine and not mirfentanil.
    Behavioural pharmacology, 1999, Volume: 10, Issue:5

    Topics: Analgesics; Animals; Arousal; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Tolerance; Fentanyl; Ketamine; Morphine; Naltrexone

1999
Use of orally administered carfentanil prior to isoflurane-induced anesthesia in a Kodiak brown bear.
    Journal of the American Veterinary Medical Association, 2000, Aug-15, Volume: 217, Issue:4

    Topics: Acid-Base Equilibrium; Administration, Oral; Analgesics, Opioid; Anesthetics, Inhalation; Animals; Blood Gas Analysis; Blood Pressure; Fentanyl; Fibrosarcoma; Forelimb; Heart Rate; Isoflurane; Male; Naltrexone; Narcotic Antagonists; Preanesthetic Medication; Respiration; Soft Tissue Neoplasms; Ursidae

2000
Selectivity of mu-opioid receptor determined by interfacial residues near third extracellular loop.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Amino Acid Substitution; Animals; Benzamides; Benzomorphans; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Morphine; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Peptides; Piperazines; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid, mu; Signal Transduction; Sulfur Radioisotopes

2000
Oral induction of anesthesia with droperidol and transmucosal carfentanil citrate in chimpanzees (Pan troglodytes).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2000, Volume: 31, Issue:2

    Topics: Administration, Oral; Analgesics, Opioid; Anesthetics, Combined; Anesthetics, Dissociative; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Benzodiazepines; Blood Gas Analysis; Body Temperature; Droperidol; Female; Fentanyl; Heart Rate; Least-Squares Analysis; Male; Mouth Mucosa; Naltrexone; Oximetry; Pan troglodytes; Tiletamine; Zolazepam

2000
Diagnosis and treatment of obstructive urolithiasis in a captive Rocky Mountain wapiti (Cervus elaphus nelsoni).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2000, Volume: 31, Issue:2

    Topics: Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Deer; Fentanyl; Hematuria; Hydrogen-Ion Concentration; Male; Naltrexone; Penis; Phenylbutazone; Specific Gravity; Urethra; Urethral Obstruction; Urinary Bladder; Urinary Calculi

2000
delta-Opioid receptors are more efficiently coupled to adenylyl cyclase than to L-type Ca(2+) channels in transfected rat pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alkylating Agents; Analgesics, Opioid; Animals; Barium; Calcium Channels, L-Type; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Heterotrimeric GTP-Binding Proteins; Ion Channels; Naltrexone; Pituitary Gland; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Transfection; Virulence Factors, Bordetella

2000
Ultrarapid opioid detoxification: effects on cardiopulmonary physiology, stress hormones and clinical outcomes.
    Drug and alcohol dependence, 2001, Jan-01, Volume: 61, Issue:2

    Topics: Adrenocorticotropic Hormone; Adult; Analgesics, Opioid; Analysis of Variance; Anesthesia, General; Blood Pressure; Female; Fentanyl; Follow-Up Studies; Heart Rate; Humans; Hydrocortisone; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Respiration; Statistics, Nonparametric; Substance Withdrawal Syndrome

2001
Acute opioid pretreatment potentiates naltrexone-induced drinking suppression in water-deprived rats.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Analgesics, Opioid; Animals; Area Under Curve; Discrimination, Psychological; Dose-Response Relationship, Drug; Drinking; Fentanyl; Male; Meperidine; Morphine; Naltrexone; Narcotic Antagonists; Pain Measurement; Rats; Rats, Sprague-Dawley; Water Deprivation

2001
Anesthesia of boma-captured Lichtenstein's hartebeest (Sigmoceros lichtensteinii) with a combination of thiafentanil, medetomidine, and ketamine.
    Journal of wildlife diseases, 2002, Volume: 38, Issue:2

    Topics: Adrenergic alpha-Agonists; Anesthesia; Anesthetics, Combined; Anesthetics, Dissociative; Animals; Antelopes; Drug Synergism; Female; Fentanyl; Ketamine; Male; Medetomidine; Naltrexone; Narcotic Antagonists

2002
Simultaneous development of six LC-MS-MS methods for the determination of multiple analytes in human plasma.
    Journal of pharmaceutical and biomedical analysis, 2002, Jun-15, Volume: 28, Issue:6

    Topics: Albuterol; Chromatography, Liquid; Clonidine; Fentanyl; Humans; Loratadine; Mass Spectrometry; Naltrexone; Pharmaceutical Preparations; Ritonavir; Technology, Pharmaceutical

2002
Possible involvement of mu1-opioid receptors in the fentanyl- or morphine-induced antinociception at supraspinal and spinal sites.
    Life sciences, 2002, Apr-05, Volume: 70, Issue:20

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Injections, Intraventricular; Injections, Spinal; Injections, Subcutaneous; Male; Mice; Mice, Inbred C57BL; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Pain Measurement; Receptors, Opioid, mu; Spinal Cord

2002
Activity of opioid ligands in cells expressing cloned mu opioid receptors.
    BMC pharmacology, 2003, Jan-04, Volume: 3

    Topics: Azocines; beta-Endorphin; Binding, Competitive; Butorphanol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Hydromorphone; Ligands; Morphine; Naltrexone; Phenazocine; Radioligand Assay; Receptors, Opioid, mu; Tritium

2003
Discrimination of a single dose of morphine followed by naltrexone: substitution of other agonists for morphine and other antagonists for naltrexone in a rat model of acute dependence.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:3

    Topics: Acute Disease; Analgesics, Opioid; Animals; Disease Models, Animal; Fentanyl; Male; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

2003
Use of irreversible antagonists to determine the relative efficacy of mu-opioids in a pigeon drug discrimination procedure: comparison of beta-funaltrexamine and clocinnamox.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:3

    Topics: Animals; Cinnamates; Columbidae; Female; Fentanyl; Methadone; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Narcotics; Reaction Time; Receptors, Opioid, mu; Sufentanil

2003
Chemical anesthesia of northern sea otters (Enhydra lutris): results of past field studies.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2001, Volume: 32, Issue:2

    Topics: Anesthesia; Anesthetics, Combined; Anesthetics, Intravenous; Animals; Azaperone; Body Temperature; Diazepam; Female; Fentanyl; Heart Rate; Hypnotics and Sedatives; Immobilization; Logistic Models; Male; Naloxone; Naltrexone; Narcotic Antagonists; Otters; Respiration; Seizures; Time Factors; Tremor

2001
Extraction and quantitation of carfentanil and naltrexone in goat plasma with liquid chromatography-mass spectrometry.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2003, Aug-15, Volume: 793, Issue:2

    Topics: Analgesics, Opioid; Animals; Chromatography, Liquid; Fentanyl; Goats; Naltrexone; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization

2003
A comparison of carfentanil/xylazine and Telazol/xylazine for immobilization of white-tailed deer.
    Journal of wildlife diseases, 2003, Volume: 39, Issue:4

    Topics: Adrenergic alpha-Agonists; Anesthetics; Animals; Deer; Dose-Response Relationship, Drug; Drug Combinations; Female; Fentanyl; Heart Rate; Immobilization; Injections, Intramuscular; Male; Naltrexone; Random Allocation; Respiration; Safety; Tiletamine; Time Factors; Xylazine; Yohimbine; Zolazepam

2003
Immobilization of mule deer with thiafentanil (A-3080) or thiafentanil plus xylazine.
    Journal of wildlife diseases, 2004, Volume: 40, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthetics, Combined; Animals; Cross-Over Studies; Deer; Dose-Response Relationship, Drug; Female; Fentanyl; Immobilization; Male; Naltrexone; Narcotic Antagonists; Random Allocation; Respiration; Time Factors; Xylazine; Yohimbine

2004
Correlation of stable elevations in striatal mu-opioid receptor availability in detoxified alcoholic patients with alcohol craving: a positron emission tomography study using carbon 11-labeled carfentanil.
    Archives of general psychiatry, 2005, Volume: 62, Issue:1

    Topics: Adult; Alcohol Drinking; Alcoholism; Basal Ganglia; Behavior, Addictive; Carbon Radioisotopes; Fentanyl; Hospitalization; Humans; Male; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Psychiatric Status Rating Scales; Receptors, Opioid, mu; Severity of Illness Index; Temperance

2005
Pharmacokinetics of carfentanil and naltrexone in domestic goats (Capra hircus).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2004, Volume: 35, Issue:4

    Topics: Absorption; Analgesics, Opioid; Animals; Cross-Over Studies; Female; Fentanyl; Gas Chromatography-Mass Spectrometry; Goats; Half-Life; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Metabolic Clearance Rate; Naltrexone; Narcotic Antagonists; Random Allocation

2004
Pharmacological manipulations of dopamine and opioids have differential effects on sexually motivated song in male European starlings.
    Physiology & behavior, 2006, Jul-30, Volume: 88, Issue:4-5

    Topics: Analgesics, Opioid; Animals; Dopamine Agents; Dopamine Uptake Inhibitors; Drug Implants; Female; Fentanyl; Male; Motivation; Naltrexone; Narcotic Antagonists; Orchiectomy; Piperazines; Receptors, Dopamine D1; Receptors, Opioid; Reward; Sexual Behavior, Animal; Starlings; Testosterone; Vocalization, Animal

2006
Pharmacokinetics and pharmacodynamics of carfentanil and naltrexone in female common eland (Taurotragus oryx).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2006, Volume: 37, Issue:3

    Topics: Analgesics, Opioid; Animals; Antelopes; Area Under Curve; Body Temperature; Female; Fentanyl; Gas Chromatography-Mass Spectrometry; Half-Life; Heart Rate; Immobilization; Injections, Intramuscular; Metabolic Clearance Rate; Naltrexone; Narcotic Antagonists; Random Allocation; Respiration

2006
The opioid antagonist, beta-funaltrexamine, inhibits chemokine expression in human astroglial cells.
    Journal of neuroimmunology, 2007, Volume: 186, Issue:1-2

    Topics: Analysis of Variance; Astrocytes; Astrocytoma; Cell Line, Tumor; Cell Survival; Chemokine CXCL10; Chemokines; Chemokines, CXC; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme-Linked Immunosorbent Assay; Fentanyl; Humans; Morphine; Naltrexone; Narcotic Antagonists; Narcotics

2007
Differences in delta- and mu-opioid receptor blockade measured by positron emission tomography in naltrexone-treated recently abstinent alcohol-dependent subjects.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:3

    Topics: Adult; Alcoholism; Analgesics, Opioid; Data Interpretation, Statistical; Female; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Opioid, delta; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Temperance

2008
Behavioral economic analysis of drug preference using multiple choice procedure data.
    Drug and alcohol dependence, 2008, Jan-11, Volume: 93, Issue:1-2

    Topics: Choice Behavior; Economics; Fentanyl; Fluoxetine; Hallucinogens; Humans; Hydromorphone; Injections, Intramuscular; Methadone; Models, Psychological; Motivation; N-Methyl-3,4-methylenedioxyamphetamine; Naltrexone; Narcotics; Psychotropic Drugs; Recreation; Selective Serotonin Reuptake Inhibitors; Substance Abuse, Intravenous; Substance-Related Disorders

2008
Limited effects of beta-endorphin compared to loperamide or fentanyl in a neuroendocrine biomarker assay in non-human primates.
    Psychoneuroendocrinology, 2008, Volume: 33, Issue:3

    Topics: Analgesics, Opioid; Animals; Antidiarrheals; beta-Endorphin; Biomarkers; Biotransformation; Dose-Response Relationship, Drug; Fentanyl; Injections, Intravenous; Loperamide; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Neurosecretory Systems; Polymorphism, Single Nucleotide; Receptors, Opioid, mu; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2008
Agonist-specific regulation of mu-opioid receptor desensitization and recovery from desensitization.
    Molecular pharmacology, 2008, Volume: 73, Issue:4

    Topics: Analgesics, Opioid; Animals; Down-Regulation; Electrophysiology; Enkephalins; Etorphine; Fentanyl; In Vitro Techniques; Male; Naltrexone; Oxymorphone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2008
Overriding the blockade of antinociceptive actions of opioids in rats treated with extended-release naltrexone.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 89, Issue:4

    Topics: Alcoholism; Analgesics, Opioid; Animals; Delayed-Action Preparations; Drug Interactions; Fentanyl; Humans; Hydrocodone; Male; Morphine; Motor Activity; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Plethysmography, Whole Body; Rats; Rats, Sprague-Dawley; Respiration

2008
Nociceptin produces antinociception after spinal administration in amphibians.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 91, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetic Acid; Analgesics; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Interactions; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Injections, Spinal; Naltrexone; Nociceptin; Opioid Peptides; Pain Threshold; Peptide Fragments; Rana pipiens

2009
Role of delta opioid efficacy as a determinant of mu/delta opioid interactions in rhesus monkeys.
    European journal of pharmacology, 2009, Jan-05, Volume: 602, Issue:1

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Interactions; Fentanyl; Hot Temperature; Ligands; Macaca mulatta; Naltrexone; Pain; Pain Measurement; Receptors, Opioid, delta; Receptors, Opioid, mu

2009
Evaluation of biomarkers for pharmacological activity.
    Journal of biopharmaceutical statistics, 2009, Volume: 19, Issue:2

    Topics: Adult; Algorithms; Analgesics, Opioid; Biomarkers; Computer Simulation; Cross-Over Studies; Fentanyl; Hormones; Humans; Longitudinal Studies; Male; Multivariate Analysis; Naltrexone; Narcotic Antagonists; Pharmacology, Clinical; Research Design

2009
Acute and chronic fentanyl administration causes hyperalgesia independently of opioid receptor activity in mice.
    Neuroscience letters, 2009, Oct-02, Volume: 462, Issue:1

    Topics: Analysis of Variance; Animals; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Fentanyl; Hot Temperature; Hyperalgesia; Male; Mice; Mice, Knockout; Naltrexone; Narcotic Antagonists; Narcotics; Pain; Pain Measurement; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Time Factors

2009
Characteristics and comparative severity of respiratory response to toxic doses of fentanyl, methadone, morphine, and buprenorphine in rats.
    Toxicology letters, 2009, Dec-15, Volume: 191, Issue:2-3

    Topics: Animals; Blood Gas Analysis; Buprenorphine; Catheterization; Fentanyl; Lactic Acid; Male; Methadone; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Narcotics; Plethysmography, Whole Body; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Respiratory Insufficiency; Respiratory Mechanics

2009
Carfentanil--an ultra potent opioid.
    The American journal of emergency medicine, 2010, Volume: 28, Issue:4

    Topics: Accidents, Occupational; Adult; Analgesics, Opioid; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Veterinarians

2010
Intranasal naltrexone and atipamezole for reversal of white-tailed deer immobilized with carfentanil and medetomidine.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2010, Volume: 51, Issue:5

    Topics: Administration, Intranasal; Adrenergic alpha-Antagonists; Animals; Cross-Over Studies; Deer; Dose-Response Relationship, Drug; Drug Combinations; Female; Fentanyl; Imidazoles; Immobilization; Injections, Intramuscular; Medetomidine; Naltrexone; Narcotic Antagonists; Random Allocation

2010
Resolution of opioid-induced postoperative ileus in a newborn infant after methylnaltrexone.
    Journal of pediatric surgery, 2011, Volume: 46, Issue:3

    Topics: Aortic Arch Syndromes; Coronary Disease; Extracorporeal Membrane Oxygenation; Fatal Outcome; Female; Fentanyl; Humans; Infant, Newborn; Intestinal Pseudo-Obstruction; Naltrexone; Narcotic Antagonists; Narcotics; Pain, Postoperative; Postoperative Complications; Quaternary Ammonium Compounds; Remission Induction

2011
Involvement of neuropeptide FF receptors in neuroadaptive responses to acute and chronic opiate treatments.
    British journal of pharmacology, 2012, Volume: 165, Issue:2

    Topics: Adamantane; Analgesics, Opioid; Animals; Behavior, Animal; Conditioning, Classical; Dipeptides; Drug Tolerance; Fentanyl; Hot Temperature; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Motor Activity; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Pain; Receptors, Neuropeptide; Substance Withdrawal Syndrome

2012
Endogenous opioids released during non-nociceptive environmental stress induce latent pain sensitization Via a NMDA-dependent process.
    The journal of pain, 2011, Volume: 12, Issue:10

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Carrageenan; Disease Models, Animal; Excitatory Amino Acid Antagonists; Fentanyl; Hyperalgesia; Inflammation; Ketamine; Male; Naltrexone; Narcotic Antagonists; Opioid Peptides; Pain Measurement; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Stress, Psychological; Swimming; Time Factors

2011
Differential development of antinociceptive tolerance to morphine and fentanyl is not linked to efficacy in the ventrolateral periaqueductal gray of the rat.
    The journal of pain, 2012, Volume: 13, Issue:8

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Fentanyl; Male; Microinjections; Morphine; Naltrexone; Narcotic Antagonists; Pain Measurement; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Reaction Time

2012
Clinically employed opioid analgesics produce antinociception via μ-δ opioid receptor heteromers in Rhesus monkeys.
    ACS chemical neuroscience, 2012, Sep-19, Volume: 3, Issue:9

    Topics: Analgesics; Analgesics, Opioid; Animals; Calcium Signaling; Data Interpretation, Statistical; Female; Fentanyl; HEK293 Cells; Humans; Injections, Spinal; Macaca mulatta; Male; Methadone; Mice; Naltrexone; Narcotic Antagonists; Pain Measurement; Receptors, Opioid, delta; Receptors, Opioid, mu

2012
Sufentanil citrate immobilization of Alaskan moose calves.
    Journal of wildlife diseases, 2012, Volume: 48, Issue:4

    Topics: Alaska; Anesthesia Recovery Period; Animals; Animals, Newborn; Animals, Wild; Deer; Dose-Response Relationship, Drug; Female; Fentanyl; Immobilization; Male; Naltrexone; Narcotics; Oxygen; Respiration; Sufentanil; Time Factors; Tolazoline; Xylazine

2012
Comparison of two injectable immobilization combinations in Himalayan tahr (Hemitragus jemlahicus): medetomidine, ketamine, and atipamezole versus carfentanil, xylazine, naltrexone, and atipamezole.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2013, Volume: 44, Issue:3

    Topics: Animals; Fentanyl; Hypnotics and Sedatives; Imidazoles; Ketamine; Medetomidine; Naltrexone; Ruminants; Xylazine

2013
Novel fentanyl-based dual μ/δ-opioid agonists for the treatment of acute and chronic pain.
    Life sciences, 2013, Dec-18, Volume: 93, Issue:25-26

    Topics: Acute Pain; Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Chronic Pain; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Enkephalins; Fentanyl; Male; Mice; Mice, Inbred ICR; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu

2013
Nalmefene reverses carfentanil-induced loss of righting reflex and respiratory depression in rats.
    European journal of pharmacology, 2014, Sep-05, Volume: 738

    Topics: Analgesics, Opioid; Animals; Blood Gas Analysis; Dose-Response Relationship, Drug; Fentanyl; Male; Naltrexone; Rats; Rats, Sprague-Dawley; Reflex, Righting; Respiratory Insufficiency; Time Factors

2014
Interaction of the adenosine A1 receptor agonist N6-cyclopentyladenosine and κ-opioid receptors in rat spinal cord nociceptive reflexes.
    Behavioural pharmacology, 2014, Volume: 25, Issue:8

    Topics: Adenosine; Animals; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Fentanyl; Inflammation; Male; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Rats; Rats, Wistar; Receptors, Opioid, kappa; Reflex; Spinal Cord

2014
κ-Opioid receptors are involved in enhanced cardioprotection by combined fentanyl and limb remote ischemic postconditioning.
    Journal of anesthesia, 2015, Volume: 29, Issue:4

    Topics: Animals; Extremities; Fentanyl; Ischemic Postconditioning; Male; Myocardial Reperfusion Injury; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2015
Characterization of the Discriminative Stimulus Effects of a NOP Receptor Agonist Ro 64-6198 in Rhesus Monkeys.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Analgesics, Opioid; Animals; Benzimidazoles; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Fentanyl; GABA Modulators; Imidazoles; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Pain Measurement; Piperidines; Receptors, Opioid; Spiro Compounds

2016
Propofol-medetomidine-ketamine total intravenous anaesthesia in thiafentanil-medetomidine-immobilized impala (Aepyceros melampus).
    Veterinary anaesthesia and analgesia, 2017, Volume: 44, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Anesthesia, Intravenous; Anesthetics, Combined; Animals; Antelopes; Female; Fentanyl; Heart Rate; Hypnotics and Sedatives; Imidazoles; Ketamine; Medetomidine; Naltrexone; Narcotic Antagonists; Propofol; Prospective Studies; Respiratory Rate

2017
Methylnaltrexone Versus Naloxone for Opioid-Induced Constipation in the Medical Intensive Care Unit.
    The Annals of pharmacotherapy, 2017, Volume: 51, Issue:3

    Topics: Adult; Analgesics, Opioid; Constipation; Critical Illness; Electronic Health Records; Female; Fentanyl; Heart Rate; Humans; Intensive Care Units; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Prospective Studies; Quaternary Ammonium Compounds; Retrospective Studies

2017
Postincarceration Fatal Overdoses After Implementing Medications for Addiction Treatment in a Statewide Correctional System.
    JAMA psychiatry, 2018, 04-01, Volume: 75, Issue:4

    Topics: Adolescent; Adult; Buprenorphine; Cause of Death; Drug Overdose; Female; Fentanyl; Health Plan Implementation; Humans; Male; Methadone; Middle Aged; Naltrexone; Odds Ratio; Opioid-Related Disorders; Patient Discharge; Prisoners; Prisons; Retrospective Studies; Rhode Island; Transitional Care; Young Adult

2018
Sex differences in the effectiveness of buprenorphine to decrease rates of responding in rhesus monkeys.
    Behavioural pharmacology, 2019, Volume: 30, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Buprenorphine; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Macaca mulatta; Male; Naltrexone; Receptors, Opioid, mu; Sex Factors

2019
Effectiveness comparisons of G-protein biased and unbiased mu opioid receptor ligands in warm water tail-withdrawal and drug discrimination in male and female rats.
    Neuropharmacology, 2019, 05-15, Volume: 150

    Topics: Analgesics, Opioid; Animals; Discrimination Learning; Female; Fentanyl; Male; Morphine; Naltrexone; Narcotic Antagonists; Nociception; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Spiro Compounds; Thiophenes

2019
Suppression of Human Natural Killer Cells by Different Classes of Opioids.
    Anesthesia and analgesia, 2019, Volume: 128, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Anesthesia; Buprenorphine; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Fluoresceins; Humans; Immunosuppression Therapy; K562 Cells; Killer Cells, Natural; Loperamide; Methadone; Morphinans; Morphine; Naloxone; Naltrexone; Succinimides; Toll-Like Receptor 4; Tramadol

2019
Optimal treatment of opioid induced constipation in daily clinical practice - an observational study.
    BMC palliative care, 2019, Mar-29, Volume: 18, Issue:1

    Topics: Aged; Analgesics, Opioid; Constipation; Female; Fentanyl; Humans; Laxatives; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Neoplasms; Oxycodone; Pain Management; Prospective Studies; Quaternary Ammonium Compounds; Retrospective Studies; Surveys and Questionnaires

2019
Conjugate vaccine produces long-lasting attenuation of fentanyl vs. food choice and blocks expression of opioid withdrawal-induced increases in fentanyl choice in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:10

    Topics: Adrenergic alpha-2 Receptor Agonists; Analgesics, Opioid; Animals; Behavior, Animal; Choice Behavior; Clonidine; Drug-Seeking Behavior; Feeding Behavior; Female; Fentanyl; Food; Male; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Rats; Reinforcement, Psychology; Self Administration; Substance Withdrawal Syndrome; Tetanus Toxoid; Vaccines, Conjugate

2019
Vaccine blunts fentanyl potency in male rhesus monkeys.
    Neuropharmacology, 2019, 11-01, Volume: 158

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Fentanyl; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Nociception; Oxycodone; Receptors, Opioid, mu; Tetanus Toxoid; Vaccines; Vaccines, Conjugate

2019
Effectiveness and selectivity of a heroin conjugate vaccine to attenuate heroin, 6-acetylmorphine, and morphine antinociception in rats: Comparison with naltrexone.
    Drug and alcohol dependence, 2019, 11-01, Volume: 204

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Administration Routes; Female; Fentanyl; Heroin; Male; Morphine; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Rats; Tetanus Toxoid; Vaccination

2019
Changes in murine respiratory dynamics induced by aerosolized carfentanil inhalation: Efficacy of naloxone and naltrexone.
    Toxicology letters, 2019, Volume: 316

    Topics: Administration, Inhalation; Aerosols; Analgesics, Opioid; Animals; Computer Simulation; Dose-Response Relationship, Drug; Fentanyl; Humans; Lung; Male; Mice; Models, Biological; Naloxone; Naltrexone; Narcotic Antagonists; Plethysmography, Whole Body; Respiration; Respiratory Insufficiency; Risk Assessment

2019
Changes in fentanyl demand following naltrexone, morphine, and buprenorphine in male rats.
    Drug and alcohol dependence, 2020, 02-01, Volume: 207

    Topics: Animals; Buprenorphine; Dose-Response Relationship, Drug; Drug Interactions; Fentanyl; Male; Morphine; Naltrexone; Rats; Receptors, Opioid; Receptors, Opioid, mu; Reinforcement Schedule; Self Administration

2020
GluN2A-selective positive allosteric modulator-nalmefene-flumazenil reverses ketamine-fentanyl-dexmedetomidine-induced anesthesia and analgesia in rats.
    Scientific reports, 2020, 03-24, Volume: 10, Issue:1

    Topics: Adjuvants, Anesthesia; Allosteric Regulation; Analgesia; Anesthesia; Animals; Delayed Emergence from Anesthesia; Dexmedetomidine; Drug Combinations; Drug Evaluation, Preclinical; Female; Fentanyl; Flumazenil; GABA-A Receptor Antagonists; Ketamine; Male; Maze Learning; Naltrexone; Narcotic Antagonists; Nociception; Pain Measurement; Rats; Receptors, N-Methyl-D-Aspartate; Reflex, Righting; Rotarod Performance Test

2020
Evaluation of a Dual Fentanyl/Heroin Vaccine on the Antinociceptive and Reinforcing Effects of a Fentanyl/Heroin Mixture in Male and Female Rats.
    ACS chemical neuroscience, 2020, 05-06, Volume: 11, Issue:9

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Female; Fentanyl; Heroin; Male; Naltrexone; Rats; Vaccines

2020
Effects of acute and repeated treatment with methocinnamox, a mu opioid receptor antagonist, on fentanyl self-administration in rhesus monkeys.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2020, Volume: 45, Issue:12

    Topics: Analgesics, Opioid; Animals; Cinnamates; Dose-Response Relationship, Drug; Fentanyl; Macaca mulatta; Morphine Derivatives; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Self Administration

2020
A low pKa ligand inhibits cancer-associated pain in mice by activating peripheral mu-opioid receptors.
    Scientific reports, 2020, 10-29, Volume: 10, Issue:1

    Topics: Analgesics, Opioid; Animals; Bone Neoplasms; Cancer Pain; Cell Line, Tumor; Fentanyl; Hydrogen-Ion Concentration; Hyperalgesia; Ligands; Male; Melanoma, Experimental; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Piperidines; Receptors, Opioid, mu

2020
Effects of kappa opioid receptor agonists on fentanyl vs. food choice in male and female rats: contingent vs. non-contingent administration.
    Psychopharmacology, 2021, Volume: 238, Issue:4

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Female; Fentanyl; Male; Morphinans; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Reinforcement, Psychology; Spiro Compounds

2021
Reversal of ingested fentanyl patch toxicity with oral naltrexone in remote Australia: case report.
    Clinical toxicology (Philadelphia, Pa.), 2021, Volume: 59, Issue:9

    Topics: Administration, Oral; Adult; Analgesics, Opioid; Australia; Fentanyl; Humans; Male; Naltrexone; Opioid-Related Disorders; Out-of-Hospital Cardiac Arrest; Rural Population; Transdermal Patch; Treatment Outcome

2021
Discriminative stimulus effects of carfentanil in rats discriminating fentanyl: Differential antagonism by naltrexone.
    Drug and alcohol dependence, 2021, 04-01, Volume: 221

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Fentanyl; Heroin; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2021
Design, synthesis, and preliminary evaluation of a potential synthetic opioid rescue agent.
    Journal of biomedical science, 2021, Sep-09, Volume: 28, Issue:1

    Topics: Analgesics, Opioid; Animals; Drug Design; Fentanyl; Male; Mice; Mice, Inbred C57BL; Naltrexone; Narcotic Antagonists

2021
Olanzapine/samidorphan precipitated opioid withdrawal in a patient taking transdermal fentanyl.
    Clinical toxicology (Philadelphia, Pa.), 2022, Volume: 60, Issue:7

    Topics: Administration, Cutaneous; Analgesics, Opioid; Fentanyl; Humans; Naltrexone; Olanzapine; Substance Withdrawal Syndrome

2022
Role of Efficacy as a Determinant of Locomotor Activation by Mu Opioid Receptor Ligands in Female and Male Mice.
    The Journal of pharmacology and experimental therapeutics, 2022, Volume: 382, Issue:1

    Topics: Analgesics, Opioid; Animals; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Female; Fentanyl; Ligands; Male; Mice; Naltrexone; Rats; Receptors, Opioid, mu

2022
Sensitivity of a fentanyl-vs.-social interaction choice procedure to environmental and pharmacological manipulations.
    Pharmacology, biochemistry, and behavior, 2022, Volume: 221

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Female; Fentanyl; Humans; Male; Naltrexone; Opioid-Related Disorders; Rats; Self Administration; Social Interaction

2022
Hepatic and renal toxicities and metabolism of fentanyl analogues in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2023, Volume: 396, Issue:1

    Topics: Analgesics, Opioid; Animals; Fentanyl; Liver; Naltrexone; Narcotic Antagonists; Rats

2023
Fentanyl analog structure-activity relationships demonstrate determinants of diverging potencies for antinociception and respiratory depression.
    Pharmacology, biochemistry, and behavior, 2023, Volume: 226

    Topics: Analgesics, Opioid; Animals; Fentanyl; Hypoventilation; Male; Mice; Morphine; Naltrexone; Receptors, Opioid, mu

2023
Fentanyl-induced respiratory depression in rodents is inhibited by bioabsorbable, subcutaneous naltrexone implants at 3.5 months.
    Addiction biology, 2023, Volume: 28, Issue:12

    Topics: Absorbable Implants; Animals; Fentanyl; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Respiratory Insufficiency; Rodentia

2023